Page last updated: 2024-09-04

glucagon and trifluoperazine

glucagon has been researched along with trifluoperazine in 14 studies

Compound Research Comparison

Studies
(glucagon)
Trials
(glucagon)
Recent Studies (post-2010)
(glucagon)
Studies
(trifluoperazine)
Trials
(trifluoperazine)
Recent Studies (post-2010) (trifluoperazine)
26,0391,4983,0543,696157198

Protein Interaction Comparison

ProteinTaxonomyglucagon (IC50)trifluoperazine (IC50)
Genome polyprotein 0.7
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Bile salt export pumpHomo sapiens (human)10
Lysozyme C-1Rattus norvegicus (Norway rat)9
Beta-glucuronidaseRattus norvegicus (Norway rat)7.8
ATP-dependent translocase ABCB1Homo sapiens (human)6.75
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)6.226
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.35
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.35
Pleiotropic ABC efflux transporter of multiple drugsSaccharomyces cerevisiae S288C1.4
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.35
D(2) dopamine receptorRattus norvegicus (Norway rat)0.016
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)6.226
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)6.226
WD repeat-containing protein 48Homo sapiens (human)8

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-199011 (78.57)18.7374
1990's3 (21.43)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Papadimituiou, JM; Sforcina, D1
Aprille, JR; Dransfield, DT; Nosek, MT1
Cheng, PY; Kanasawa, Y; Katori, T; Kume, S; Oka, H; Sawada, S; Suzuki, S; Yamaguchi, K; Yasuda, H1
Kurokawa, K; Takaichi, K1
Hii, CS; Howell, SL1
Marshall, L; Steiner, RF1
Jones, AB; Wolff, J1
Chick, WL; Hales, CN; Hutton, JC; Naber, SP; Sopwith, AM1
Evanson, T; Kelley, DS; Potter, VR1
Exton, JH; Morgan, NG; Shipp, CC1
Harano, Y; Kashiwagi, A; Kosugi, K; Nakano, T; Shigeta, Y; Suzuki, M1
Kimura, S; Koide, Y; Kugai, N; Tada, R; Yamashita, K1
He, LP; Kitasato, H1
Atwater, I; He, LP; Kitasato, H; Mears, D1

Other Studies

14 other study(ies) available for glucagon and trifluoperazine

ArticleYear
The effects of drugs on monocytic fusion in vivo.
    Experimental cell research, 1975, Mar-15, Volume: 91, Issue:2

    Topics: Adenosine Triphosphatases; Animals; Calcium; Cell Fusion; Cell Membrane; Cortisone; Cyclic AMP; Diphenhydramine; Edetic Acid; Glucagon; Insulin; Isoproterenol; Lidocaine; Lysosomes; Male; Mice; Mice, Inbred C57BL; Monocytes; Ouabain; Pyrilamine; Tetracaine; Trifluoperazine; Verapamil

1975
Calcium stimulates ATP-Mg/Pi carrier activity in rat liver mitochondria.
    The Journal of biological chemistry, 1990, May-25, Volume: 265, Issue:15

    Topics: Adenine Nucleotides; Adenosine Triphosphate; Animals; Calcium Chloride; Calmodulin; Carrier Proteins; Cells, Cultured; Chlorpromazine; Egtazic Acid; Glucagon; Imidazoles; Kinetics; Liver; Magnesium; Male; Mitochondria, Liver; Neomycin; Phosphates; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine; Vasopressins

1990
Stimulative effects of TMB-8 and trifluoperazine on pancreatic hormone release.
    Diabetes research and clinical practice, 1989, Apr-01, Volume: 6, Issue:3

    Topics: Animals; Calcium Channel Blockers; Gallic Acid; Glucagon; Hydroxydopamines; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Oxidopamine; Rats; Rats, Inbred Strains; Somatostatin; Trifluoperazine

1989
AVP-sensitive cAMP production is dependent on calmodulin in both MTAL and MCT.
    The American journal of physiology, 1988, Volume: 255, Issue:5 Pt 2

    Topics: Adenylyl Cyclases; Animals; Arginine Vasopressin; Calmodulin; Colforsin; Cyclic AMP; Enzyme Activation; Glucagon; Kidney Tubules; Kidney Tubules, Collecting; Loop of Henle; Mice; Sulfonamides; Trifluoperazine

1988
Role of second messengers in the regulation of glucagon secretion from isolated rat islets of Langerhans.
    Molecular and cellular endocrinology, 1987, Volume: 50, Issue:1-2

    Topics: Animals; Arginine; Calcimycin; Calcium; Colforsin; Cyclic AMP; Diglycerides; Drug Interactions; Glucagon; Glycerides; Islets of Langerhans; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Trifluoperazine

1987
Sites of interaction of calmodulin with trifluoperazine and glucagon.
    Archives of biochemistry and biophysics, 1985, Volume: 240, Issue:1

    Topics: Amino Acids; Animals; Binding Sites; Binding, Competitive; Calmodulin; Cattle; Chemical Phenomena; Chemistry; Circular Dichroism; Energy Transfer; Glucagon; Male; Mathematics; Models, Chemical; Peptide Fragments; Protein Binding; Spectrometry, Fluorescence; Testis; Trifluoperazine; Tyrosine

1985
Inhibition of hormone-sensitive adenyl cyclase by phenothiazines.
    Proceedings of the National Academy of Sciences of the United States of America, 1970, Volume: 65, Issue:2

    Topics: Adenine Nucleotides; Adenylyl Cyclase Inhibitors; Adrenal Glands; Adrenocorticotropic Hormone; Animals; Cattle; Cell Membrane; Chlorpromazine; Enzyme Inhibitors; Epinephrine; Fluorides; Glucagon; Kidney; Liver; Phenothiazines; Pituitary Hormones, Anterior; Prochlorperazine; Prostaglandin Antagonists; Stimulation, Chemical; Thymol; Thyroid Gland; Thyrotropin; Trifluoperazine

1970
Insulin secretion by a transplantable rat islet cell tumour.
    Diabetologia, 1981, Volume: 21, Issue:3

    Topics: Adenoma, Islet Cell; Animals; Colchicine; Epinephrine; Glucagon; Glucose; Insulin; Insulin Secretion; Insulinoma; Kinetics; Neoplasms, Experimental; Pancreatic Neoplasms; Rats; Rats, Inbred Strains; Somatostatin; Theophylline; Trifluoperazine; Vinblastine

1981
Calcium-dependent hormonal regulation of amino acid transport and cyclic AMP accumulation in rat hepatocyte monolayer cultures.
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:10

    Topics: Aminoisobutyric Acids; Animals; Biological Transport, Active; Calcimycin; Calcium; Cells, Cultured; Cyclic AMP; Glucagon; Liver; Rats; Trifluoperazine

1980
Studies on the mechanism of inhibition of hepatic cAMP accumulation by vasopressin.
    FEBS letters, 1983, Nov-14, Volume: 163, Issue:2

    Topics: Adenylyl Cyclases; Animals; Calcium; Calmodulin; Chlorpromazine; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Enzyme Activation; Glucagon; In Vitro Techniques; Liver; Male; Rats; Rats, Inbred Strains; Trifluoperazine; Vasopressins

1983
Mechanism of adrenergic stimulation of hepatic ketogenesis.
    Metabolism: clinical and experimental, 1983, Volume: 32, Issue:11

    Topics: Animals; Catecholamines; Epinephrine; Glucagon; In Vitro Techniques; Insulin; Ketone Bodies; Liver; Liver Glycogen; Male; Norepinephrine; Palmitates; Rats; Rats, Inbred Strains; Sympatholytics; Sympathomimetics; Trifluoperazine

1983
Inhibition by trifluoperazine of glycogenolytic effects of phenylephrine, vasopressin, and angiotensin II.
    Endocrinologia japonica, 1982, Volume: 29, Issue:3

    Topics: Angiotensin II; Animals; Calcium; Glucagon; Glucose; Liver Glycogen; Male; Phentolamine; Phenylephrine; Phosphorylase a; Rats; Rats, Inbred Strains; Trifluoperazine; Vasopressins

1982
Glucagon induces Ca2+-dependent increase of reduced pyridine nucleotides in mouse pancreatic beta-cells.
    Biochimica et biophysica acta, 1996, Feb-29, Volume: 1310, Issue:3

    Topics: Animals; Calcium; Calmodulin; Cell Membrane; Cells, Cultured; Chlorpromazine; Dose-Response Relationship, Drug; Fura-2; Glucagon; Glucose; Islets of Langerhans; Kinetics; Membrane Potentials; Mice; Mice, Inbred ICR; NAD; NADP; Sulfonamides; Trifluoperazine

1996
Glucagon induces suppression of ATP-sensitive K+ channel activity through a Ca2+/calmodulin-dependent pathway in mouse pancreatic beta-cells.
    The Journal of membrane biology, 1998, Dec-01, Volume: 166, Issue:3

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Bucladesine; Calcium Signaling; Calmodulin; Chlorpromazine; Glucagon; Glucose; Ion Channel Gating; Ion Transport; Islets of Langerhans; Membrane Potentials; Mice; Mice, Inbred ICR; Patch-Clamp Techniques; Photolysis; Potassium; Potassium Channel Blockers; Potassium Channels; Sulfonamides; Trifluoperazine

1998