Page last updated: 2024-09-04

glucagon and prazosin

glucagon has been researched along with prazosin in 32 studies

Compound Research Comparison

Studies
(glucagon)
Trials
(glucagon)
Recent Studies (post-2010)
(glucagon)
Studies
(prazosin)
Trials
(prazosin)
Recent Studies (post-2010) (prazosin)
26,0391,4983,0547,914713682

Protein Interaction Comparison

ProteinTaxonomyglucagon (IC50)prazosin (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)5.87
Interstitial collagenaseHomo sapiens (human)4.036
Alpha-2A adrenergic receptorHomo sapiens (human)2.638
Matrix metalloproteinase-9Homo sapiens (human)6.963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0008
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)0.0078
Alpha-2B adrenergic receptorHomo sapiens (human)0.29
Alpha-2C adrenergic receptorHomo sapiens (human)0.647
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0008
Alpha-1D adrenergic receptorHomo sapiens (human)0.0007
Bromodomain-containing protein 2Homo sapiens (human)0.0009
Alpha-1A adrenergic receptorHomo sapiens (human)0.0006
Alpha-1B adrenergic receptorHomo sapiens (human)0.0006
5-hydroxytryptamine receptor 2BHomo sapiens (human)4.118
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0008
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.5849
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.6

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-199020 (62.50)18.7374
1990's10 (31.25)18.2507
2000's2 (6.25)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kneer, NM; Lardy, HA; Wagner, MJ1
Gross, R; Hillaire-Buys, D; Loubatières-Mariani, MM; Ribes, G; Roye, M1
Oda, S; Ohneda, A; Sasaki, Y; Tsuda, T1
Faulkner, A; Pollock, HT1
Swindell, AC; Valentine, JJ1
Ganas, L; Studer, RK1
Gotoh, M; Iguchi, A; Matsunaga, H; Miura, H; Sakamoto, N; Satake, T; Tamagawa, T; Uemura, K; Yatomi, A1
Hashimoto, K; Kato, K; Tsujimoto, A; Tsujimoto, G1
Dileepan, KN; Wagle, SR1
Blackmore, PF; Charest, R; Exton, JH; Lynch, CJ1
Talesnik, J; Youngson, BJ1
Bertrand, G; Gross, R; Loubatières-Mariani, MM; Ribes, G1
Jungermann, K; Nath, A; Püschel, GP1
Adams, JH; Irving, G; Koeslag, JH; Lochner, JD; Sandell, RC; Wilkinson, C1
Dileepan, KN; Khawaja, AM; Wagle, SR1
Crane, D; Graf, P; Sies, H1
Carrà, G; Damante, G; Del Campo, F; Di Vincenzo, S; Ferlito, S; Puleo, F1
Knudtzon, J1
Greenberg, ML; Malbon, CC1
Corvera, S; García-Sáinz, JA; Pushpendran, CK1
Birnbaumer, L; Dighe, RR; Garber, AJ; Rojas, FJ1
Ichihara, A; Kato, S; Nakamura, T1
Bygrave, FL; Reinhart, PH; Taylor, WM1
Bogoyevitch, MA; Fuller, SJ; Sugden, PH1
Belahsen, R; Deshaies, Y1
Alvarez, C; Bladé, C; Cartañà, J1
Pittner, RA; Spitzer, JA1
Hirose, H; Ito, K; Kido, K; Koyama, K; Maruyama, H; Saruta, T1
Hernández, ML; Martínez, MJ; Ochoa, B; Ruiz, JI1
Brechet, S; Chayvialle, JA; Claustre, J; Cuber, JC; Plaisancie, P1
Aarnio, P; Dela, F; Lauritsen, T1
Hemmings, SJ; Wilson, TR1

Reviews

1 review(s) available for glucagon and prazosin

ArticleYear
Somatostatin: a metabolic regulator.
    Life sciences, 1985, Dec-23, Volume: 37, Issue:25

    Topics: Adrenocorticotropic Hormone; Animals; Bicarbonates; Bile; Blood Glucose; Calcium; Cyclic AMP; Digestive System Physiological Phenomena; Glucagon; Gluconeogenesis; Glycogen; Growth Hormone; Homeostasis; Humans; Insulin; Insulin Secretion; Kidney Cortex; Liver; Pancreas; Pituitary Gland; Prazosin; Prolactin; Pyruvates; Pyruvic Acid; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Somatostatin; Thyrotropin; Yohimbine

1985

Trials

1 trial(s) available for glucagon and prazosin

ArticleYear
Effect of alpha-1-blockade by prazosin on blood sugar, insulin and glucagon levels in normals and non-insulin dependent diabetics.
    Journal of endocrinological investigation, 1983, Volume: 6, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adult; Blood Glucose; Diabetes Mellitus; Female; Glucagon; Glucose Tolerance Test; Humans; Insulin; Middle Aged; Prazosin; Quinazolines

1983

Other Studies

30 other study(ies) available for glucagon and prazosin

ArticleYear
Regulation by calcium of hormonal effects on gluconeogenesis.
    The Journal of biological chemistry, 1979, Dec-10, Volume: 254, Issue:23

    Topics: Animals; Calcimycin; Calcium; Dihydroxyacetone; Dose-Response Relationship, Drug; Ethanol; Fructose; Glucagon; Gluconeogenesis; Hydroxybutyrates; In Vitro Techniques; Kinetics; Lactates; Liver; Male; Norepinephrine; Prazosin; Propranolol; Rats

1979
Adrenergic inhibition of insulin secretion involves pertussis toxin-sensitive and -insensitive mechanisms.
    European journal of pharmacology, 1992, Aug-06, Volume: 218, Issue:2-3

    Topics: Analysis of Variance; Animals; Epinephrine; Glucagon; GTP-Binding Proteins; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pertussis Toxin; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella; Yohimbine

1992
Glucagon and insulin responses to alpha-adrenergic subtype receptor blockade in sheep.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1990, Volume: 96, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Epinephrine; Glucagon; Infusions, Intravenous; Insulin; Insulin Secretion; Male; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Sheep; Yohimbine

1990
Effects of glucagon and alpha- and beta-agonists on glycogenolysis and gluconeogenesis in isolated ovine hepatocytes.
    Biochimica et biophysica acta, 1990, Apr-09, Volume: 1052, Issue:1

    Topics: Animals; Bucladesine; Cells, Cultured; Glucagon; Gluconeogenesis; Isoproterenol; Kinetics; Liver; Liver Glycogen; Phenylephrine; Prazosin; Sheep; Vasopressins; Yohimbine

1990
Interactions of doxazosin with insulin or glucagon in the ob/ob mouse.
    Journal of cardiovascular pharmacology, 1989, Volume: 13 Suppl 2

    Topics: 3-Hydroxybutyric Acid; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Cholesterol; Doxazosin; Fatty Acids, Nonesterified; Glucagon; Glycerol; Hydroxybutyrates; Insulin; Lactates; Lactic Acid; Male; Mice; Mice, Obese; Prazosin; Triglycerides

1989
Effect of diabetes on hormone-stimulated and basal hepatocyte calcium metabolism.
    Endocrinology, 1989, Volume: 125, Issue:5

    Topics: Animals; Arginine Vasopressin; Calcium; Cells, Cultured; Diabetes Mellitus, Experimental; Epinephrine; Glucagon; Inositol 1,4,5-Trisphosphate; Kinetics; Liver; Male; Phentolamine; Phosphorylases; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reference Values

1989
Central nervous system-mediated glucagon secretion is enhanced by alpha 2-adrenoreceptor activation.
    Endocrinology, 1989, Volume: 125, Issue:3

    Topics: Adrenalectomy; Adrenergic alpha-Antagonists; Animals; Blood Glucose; Cerebral Ventricles; Glucagon; Hexamethonium; Hexamethonium Compounds; Injections, Intraventricular; Male; Neostigmine; Norepinephrine; Phentolamine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reference Values; Yohimbine

1989
In vivo desensitization of glycogenolysis to Ca2+-mobilizing hormones in rat liver cells.
    The Journal of clinical investigation, 1988, Volume: 82, Issue:6

    Topics: Adrenal Gland Neoplasms; Angiotensin II; Animals; Arginine Vasopressin; Bucladesine; Calcimycin; Calcium; Colforsin; Glucagon; Hormones; Liver Glycogen; Male; Norepinephrine; Phenoxybenzamine; Phenylephrine; Pheochromocytoma; Phosphorylases; Prazosin; Rats; Receptors, Adrenergic, alpha; Second Messenger Systems

1988
Studies on the hepatic alpha 1-adrenergic receptor. Modulation of guanine nucleotide effects by calcium, temperature, and age.
    The Journal of biological chemistry, 1985, Feb-10, Volume: 260, Issue:3

    Topics: Aging; Animals; Calcium; Cell Membrane; Cold Temperature; Egtazic Acid; Glucagon; Guanine Nucleotides; Guanylyl Imidodiphosphate; Liver; Male; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Cell Surface; Receptors, Glucagon

1985
Modulation of positive inotropy and metabolic coronary dilatation by myocardial alpha-adrenoceptors.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:12

    Topics: Animals; Calcium Chloride; Catecholamines; Coronary Vessels; Dobutamine; Electric Stimulation; Glucagon; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Muscle, Smooth, Vascular; Myocardial Contraction; Norepinephrine; Phenoxybenzamine; Phentolamine; Phenylephrine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tyramine; Vasodilation

1985
Alpha 2-adrenergic potentiation of adenosine-stimulating effect on glucagon secretion.
    Endocrinology, 1987, Volume: 121, Issue:2

    Topics: Adenosine; Animals; Clonidine; Drug Synergism; Epinephrine; Glucagon; Male; Pancreas; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1987
Increase of urate formation by stimulation of sympathetic hepatic nerves, circulating noradrenaline and glucagon in the perfused rat liver.
    FEBS letters, 1987, Jul-13, Volume: 219, Issue:1

    Topics: Allopurinol; Animals; Glucagon; Glucose; Insulin; Lactates; Lactic Acid; Liver; Male; Nitroprusside; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Uric Acid

1987
Beta-adrenergic blockade restores glucose's antiketogenic activity after exercise in carbohydrate-depleted athletes.
    The Journal of physiology, 1987, Volume: 386

    Topics: 3-Hydroxybutyric Acid; Autonomic Nervous System; Blood Glucose; Fatty Acids, Nonesterified; Female; Glucagon; Glucose; Humans; Hydroxybutyrates; Insulin; Ketone Bodies; Male; Physical Exertion; Prazosin; Propantheline; Propranolol; Running; Time Factors

1987
Studies on the mechanism of action of somatostatin on renal gluconeogenesis: evidence for the involvement of alpha 1-adrenergic stimuli.
    Archives of biochemistry and biophysics, 1982, Volume: 213, Issue:1

    Topics: Animals; Calcium; Glucagon; Gluconeogenesis; Insulin; Kidney Cortex; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Reserpine; Somatostatin; Yohimbine

1982
Decreased flux through pyruvate dehydrogenase during calcium ion movements induced by vasopressin, alpha-adrenergic agonists and the ionophore A23187 in perfused rat liver.
    The Biochemical journal, 1983, May-15, Volume: 212, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Anti-Bacterial Agents; Calcimycin; Calcium; Glucagon; In Vitro Techniques; Liver; Male; Perfusion; Prazosin; Pyruvate Dehydrogenase Complex; Pyruvates; Pyruvic Acid; Rats; Rats, Inbred Strains; Vasopressins

1983
Adrenergic effects on plasma levels of glucagon, insulin, glucose and free fatty acids in rabbits--influences of selective blocking drugs.
    Acta physiologica Scandinavica, 1984, Volume: 120, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Glucose; Epinephrine; Fatty Acids, Nonesterified; Female; Glucagon; Insulin; Isoproterenol; Metoprolol; Prazosin; Propanolamines; Rabbits; Yohimbine

1984
3,3',5-triiodothyronine administration in vivo modulates the hormone-sensitive adenylate cyclase system of rat hepatocytes.
    The Journal of clinical investigation, 1982, Volume: 69, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzyl Alcohols; Cholera Toxin; Cyclic AMP; Epinephrine; Female; Glucagon; Guanosine Triphosphate; Hormones; Hyperthyroidism; Isoproterenol; Liver; Pindolol; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Triiodothyronine; Triiodothyronine, Reverse

1982
Effect of pertussis toxin on hormonal responsiveness of rat hepatocytes.
    FEBS letters, 1983, Aug-22, Volume: 160, Issue:1-2

    Topics: Adenylate Cyclase Toxin; Animals; Bacterial Toxins; Cyclic AMP; Epinephrine; Female; Glucagon; In Vitro Techniques; Isoproterenol; Kinetics; Liver; Pertussis Toxin; Phosphatidylinositols; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Urea; Virulence Factors, Bordetella

1983
Glucagon-stimulable adenylyl cyclase in rat liver. The impact of streptozotocin-induced diabetes mellitus.
    The Journal of clinical investigation, 1984, Volume: 73, Issue:4

    Topics: Adenylyl Cyclases; Animals; Cell Membrane; Diabetes Mellitus, Experimental; Enzyme Activation; Female; Glucagon; Insulin; Kinetics; Liver; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Cell Surface; Receptors, Glucagon

1984
Glucagon and glucose as major regulators of glycogen metabolism in primary cultured rat hepatocytes.
    Journal of biochemistry, 1984, Volume: 95, Issue:6

    Topics: Animals; Cells, Cultured; Glucagon; Glucose; Glycogen Synthase; Insulin; Kinetics; Liver; Liver Glycogen; Male; Phenoxybenzamine; Phenylephrine; Phosphorylases; Prazosin; Rats; Rats, Inbred Strains

1984
Studies on alpha-adrenergic-induced respiration and glycogenolysis in perfused rat liver.
    The Journal of biological chemistry, 1982, Feb-25, Volume: 257, Issue:4

    Topics: Animals; Antimycin A; Dinitrophenols; Female; Glucagon; Kinetics; Liver; Liver Glycogen; Oxygen Consumption; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Rotenone; Yohimbine

1982
cAMP and protein synthesis in isolated adult rat heart preparations.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Adenine Nucleotides; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Energy Metabolism; Epinephrine; Glucagon; Heart; Hypertension; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Perfusion; Phenylephrine; Phosphocreatine; Prazosin; Propranolol; Protein Biosynthesis; Rats; Rats, Sprague-Dawley; Yohimbine

1993
Alpha-1 adrenergic blockade interacts with dietary carbohydrates on triacylglycerol metabolism in rats.
    The Journal of nutrition, 1993, Volume: 123, Issue:3

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic alpha-Antagonists; Animals; Dietary Carbohydrates; Glucagon; Insulin; Lipoprotein Lipase; Liver; Male; Prazosin; Rats; Rats, Sprague-Dawley; Starch; Sucrose; Triglycerides

1993
Alpha 2-adrenergic blockade prevents hyperglycemia and hepatic glutathione depletion in nickel-injected rats.
    Toxicology and applied pharmacology, 1993, Volume: 121, Issue:1

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Female; Glucagon; Glutathione; Hyperglycemia; Insulin; Liver; Nickel; Phentolamine; Prazosin; Propranolol; Rats; Rats, Wistar; Yohimbine

1993
Shift from alpha- to beta-type adrenergic receptor-mediated responses in chronically endotoxemic rats.
    The American journal of physiology, 1993, Volume: 264, Issue:4 Pt 1

    Topics: Angiotensin II; Animals; Cells, Cultured; Chlorides; Endotoxins; Escherichia coli; Glucagon; Inositol Phosphates; Kinetics; Lithium; Lithium Chloride; Liver; Male; Norepinephrine; Phosphorylase a; Prazosin; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Shock, Septic; Vasopressins

1993
Adrenoceptor antagonists, but not guanethidine, reduce glucopenia-induced glucagon secretion from perfused rat pancreas.
    Diabetes research and clinical practice, 1995, Volume: 30, Issue:3

    Topics: Adrenergic Agents; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Drug Combinations; Glucagon; Glucose; Guanethidine; Insulin; Insulin Secretion; Male; Norepinephrine; Pancreas; Perfusion; Prazosin; Propranolol; Rats; Rats, Wistar; Time Factors; Tyramine; Yohimbine

1995
Stimulation of microsomal cholesterol ester hydrolase by glucagon, cyclic AMP analogues, and vasopressin in isolated rat hepatocytes.
    Lipids, 1996, Volume: 31, Issue:3

    Topics: Animals; Bucladesine; Cholesterol Esters; Colforsin; Cyclic AMP; Diglycerides; Glucagon; Microsomes, Liver; Particle Size; Prazosin; Rats; Sterol Esterase; Thionucleotides; Vasopressins

1996
Stimulatory effect of beta-adrenergic agonists on ileal L cell secretion and modulation by alpha-adrenergic activation.
    The Journal of endocrinology, 1999, Volume: 162, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Clonidine; Epinephrine; Glucagon; Glucagon-Like Peptide 1; Isoproterenol; Peptide Fragments; Peptide YY; Phenylephrine; Prazosin; Protein Precursors; Rats; Rats, Wistar

1999
Insulin secretion and glucose kinetics during exercise with and without pharmacological alpha(1)- and alpha(2)-receptor blockade.
    Diabetes, 2001, Volume: 50, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Blood Glucose; Blood Pressure; C-Peptide; Cross-Over Studies; Epinephrine; Exercise; Fatty Acids, Nonesterified; Glucagon; Glycerol; Heart Rate; Hemodynamics; Humans; Insulin; Insulin Secretion; Kinetics; Lactates; Male; Physical Exertion; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Time Factors; Tritium; Yohimbine

2001
Lymphosarcoma-induced alterations in hepatic adrenergic receptors: implications to the hypoglycemia of cancer cachexia.
    Molecular and cellular biochemistry, 2003, Volume: 250, Issue:1-2

    Topics: Alanine Transaminase; Animals; Blood Glucose; Cachexia; Cell Line, Tumor; Cell Membrane; Female; gamma-Glutamyltransferase; Glucagon; Hypoglycemia; Kinetics; Liver; Lymphoma, Non-Hodgkin; Prazosin; Protein Binding; Radioimmunoassay; Rats; Rats, Inbred F344; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Thyroid Hormones; Time Factors

2003