Page last updated: 2024-09-04

glucagon and pirenzepine

glucagon has been researched along with pirenzepine in 9 studies

Compound Research Comparison

Studies
(glucagon)
Trials
(glucagon)
Recent Studies (post-2010)
(glucagon)
Studies
(pirenzepine)
Trials
(pirenzepine)
Recent Studies (post-2010) (pirenzepine)
26,0391,4983,0543,812587140

Protein Interaction Comparison

ProteinTaxonomyglucagon (IC50)pirenzepine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.6891
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.5856
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.6134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.6222
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.6227
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.6227
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.3406
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.6281
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.0291
Muscarinic acetylcholine receptor M1Mus musculus (house mouse)0.75
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.9556
Muscarinic acetylcholine receptor M4Mus musculus (house mouse)0.75
Muscarinic acetylcholine receptor M5Mus musculus (house mouse)0.75
Muscarinic acetylcholine receptor M3Mus musculus (house mouse)0.75
Muscarinic acetylcholine receptor M2Mus musculus (house mouse)0.51

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19905 (55.56)18.7374
1990's4 (44.44)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bianconi, L; Capretti, L; Coiro, V; Davoli, C; Fagnoni, F; Gardini, E; Maffei, ML; Passeri, M; Speroni, G; Volpi, R1
Atiea, JA; Creagh, F; Owens, DR; Page, M; Peters, JR; Scanlon, MF1
Butturini, U; Camellini, L; Chiodera, P; Coiro, V; d'Amato, L; Pignatti, D; Rossi, G; Volpi, R1
Giordano, G; Pasquali, C; Ragazzi, E; Scandellari, C; Valentini, P; Zaccaria, M; Zeviani, M1
Adrian, TE; Baron, JH; Bloom, SR; El-Sabbagh, HN; Prinz, RA; Welbourn, RB1
Delitala, G; Frulio, T; Maioli, M; Pacifico, A1
Hanai, H; Kajimura, M; Kaneko, E; Kodaira, M; Lin, S; Takeuchi, K1
Gil, MJ; Goñi, F; Goñi, MJ; Moncada, E; Monreal, M; Salvador, J; Sopena, M1
Joye, F; Marion, F; Michoux, I; Orrillard, M; Parisot, R1

Trials

2 trial(s) available for glucagon and pirenzepine

ArticleYear
The effect of pirenzepine on meal-stimulated gastrointestinal hormones.
    Scandinavian journal of gastroenterology. Supplement, 1980, Volume: 66

    Topics: Adult; Benzodiazepinones; Eating; Gastric Inhibitory Polypeptide; Gastrins; Gastrointestinal Hormones; Glucagon; Glucagon-Like Peptides; Humans; Insulin; Neurotensin; Pancreatic Polypeptide; Piperazines; Pirenzepine; Somatostatin; Vasoactive Intestinal Peptide

1980
Effects of cholinergic blockade on nocturnal thyrotropin and growth hormone (GH) secretion in type I diabetes mellitus: further evidence supporting somatostatin's involvement in GH suppression.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:11

    Topics: Administration, Oral; Adult; Blood Glucose; Circadian Rhythm; Cohort Studies; Diabetes Mellitus, Type 1; Double-Blind Method; Female; Glucagon; Growth Hormone-Releasing Hormone; Human Growth Hormone; Humans; Hydrocortisone; Insulin-Like Growth Factor I; Male; Muscarinic Antagonists; Pirenzepine; Somatostatin; Thyrotropin

1997

Other Studies

7 other study(ies) available for glucagon and pirenzepine

ArticleYear
Reduced sensitivity to pirenzepine-induced blockade of growth hormone responses to arginine, exercise, and growth hormone-releasing hormone in type I diabetic subjects.
    Metabolism: clinical and experimental, 1990, Volume: 39, Issue:7

    Topics: Adolescent; Adult; Arginine; Blood Glucose; Child; Child, Preschool; Diabetes Mellitus, Type 1; Exercise; Glucagon; Growth Hormone; Growth Hormone-Releasing Hormone; Humans; Kinetics; Muscarinic Antagonists; Pirenzepine; Receptors, Muscarinic

1990
Early morning hyperglycemia in insulin-dependent diabetes: acute and sustained effects of cholinergic blockade.
    The Journal of clinical endocrinology and metabolism, 1989, Volume: 69, Issue:2

    Topics: Adult; Blood Glucose; Circadian Rhythm; Diabetes Mellitus, Type 1; Glucagon; Growth Hormone; Humans; Hydrocortisone; Hyperglycemia; Insulin; Male; Parasympatholytics; Pirenzepine

1989
Muscarinic cholinergic modulation of insulin response to an intravenous glucose tolerance test in normal man.
    Journal of endocrinological investigation, 1986, Volume: 9, Issue:1

    Topics: Adult; Benzodiazepinones; Blood Glucose; Female; Glucagon; Glucose Tolerance Test; Humans; Injections, Intravenous; Insulin; Male; Pirenzepine; Receptors, Muscarinic

1986
Effects of pirenzepine on plasma insulin, glucagon and pancreatic polypeptide levels in normal man.
    European journal of clinical pharmacology, 1985, Volume: 27, Issue:6

    Topics: Adult; Arginine; Benzodiazepinones; Blood Glucose; Glucagon; Glucose Tolerance Test; Humans; Insulin; Pancreatic Polypeptide; Pirenzepine; Radioimmunoassay; Time Factors

1985
Participation of cholinergic muscarinic receptors in glucagon- and arginine-mediated growth hormone secretion in man.
    The Journal of clinical endocrinology and metabolism, 1982, Volume: 55, Issue:6

    Topics: Adult; Arginine; Benzodiazepinones; Glucagon; Growth Hormone; Humans; Male; Parasympatholytics; Pirenzepine; Prolactin; Receptors, Cholinergic; Receptors, Muscarinic

1982
Expression of muscarinic receptor subtypes in rat gastric smooth muscle: effect of M3 selective antagonist on gastric motility and emptying.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:5

    Topics: Animals; Atropine; Butylscopolammonium Bromide; Dioxoles; Gastric Emptying; Gastrointestinal Motility; Glucagon; Male; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Pirenzepine; Polymerase Chain Reaction; Rats; Receptors, Muscarinic; Stomach

1997
[Severe intoxication probably from olanzapine (Zyprexa). Beneficial effect of glucagon].
    Annales francaises d'anesthesie et de reanimation, 1999, Volume: 18, Issue:6

    Topics: Adult; Alprazolam; Antipsychotic Agents; Benzodiazepines; Bradycardia; Carbamazepine; Disseminated Intravascular Coagulation; Drug Therapy, Combination; Gastrointestinal Agents; Glucagon; Humans; Hypothermia; Infusions, Intravenous; Male; Methotrimeprazine; Olanzapine; Pirenzepine; Schizophrenia; Shock

1999