gliclazide has been researched along with glyburide in 158 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 20 (12.66) | 18.7374 |
1990's | 43 (27.22) | 18.2507 |
2000's | 56 (35.44) | 29.6817 |
2010's | 32 (20.25) | 24.3611 |
2020's | 7 (4.43) | 2.80 |
Authors | Studies |
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Ahmad, P; Kumar, A; Pathak, SR; Ray, S; Srivastava, AK; Tewari, P | 1 |
Chander, R; Chaturvedi, D; Ray, S; Srivastava, AK | 1 |
Ahmad, P; Kumar, A; Maurya, RA; Singh, AB; Srivastava, AK | 1 |
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Ahmad, P; Kumar, A; Maurya, RA; Sharma, S; Singh, AB; Srivastava, AK; Tamrakar, AK | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Campillo, NE; Guerra, A; Páez, JA | 1 |
Barber, J; Dawson, S; Kenna, JG; Paul, N; Stahl, S | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Jackson, WP; Jacobs, P; Kernoff, L; Klaff, LJ; Malan, E; Vinik, AI | 1 |
Dubecz, E; Pogátsa, G | 1 |
De Vigan, C; Delporte, MP; Perrault, M; Thomas, M | 1 |
Balabolkin, MI; Danilova, TI; Ol'shanskaia, AA; Timofeev, AV; Zhuleva, LIu | 1 |
Ambrosi, F; Cristallini, S; Filipponi, P; Gregorio, F; Pedetti, M; Santeusanio, F | 1 |
Friedberg, SJ; Pugh, JA; Ramirez, G; Sawyer, J; Tuley, M; Wagner, ML | 1 |
Nakano, S; Naruto, S; Noguchi, H; Tomita, N | 1 |
Kume, S; Ozaki, Y; Yatomi, Y | 1 |
Harrower, AD | 2 |
Aranyi, Z; Ballagi-Pordány, G; Koltai, MZ; Köszeghy, A; Pogátsa, G | 1 |
Katsumata, K; Katsumata, Y | 1 |
Boutagy, JS; Shenfield, GM; Webb, C | 1 |
Doi, K | 1 |
Harrower, AD; Wong, C | 1 |
Brasseur, R; Deleers, M | 1 |
Godfrey, H; Jerums, G; Larkins, RG; Martin, TJ; Smith, IL; Taft, JL | 1 |
Caravaggio, V; Cortinovis, A; Crippa, A; Crippa, M; Sciacca, V | 1 |
Barnett, AH; Florkowski, CM; Jennings, PE; Jones, AF; Le Guen, C; Lunec, J; O'Donnell, MJ; Richardson, MR | 1 |
Balabolkin, MI; Nedosugova, LV | 1 |
Malaisse, WJ; Malaisse-Lagae, F; Mathias, PC; Sener, A | 1 |
Hatao, K; Kaku, K; Kaneko, T; Matsuda, M; Tsuchiya, M | 1 |
Furman, BL; Musbah, MO | 1 |
Chan, TK; Chan, V; Teng, CS; Yeung, RT | 1 |
Deleers, M; Gelbcke, M; Malaisse, WJ | 2 |
Baba, S; Fukui, I; Goto, Y; Maezawa, H; Nakagawa, S; Sakamoto, N; Takebe, K; Takeda, R | 1 |
Abe, M; Ikeda, Y; Minami, N | 1 |
Frolova, AI; Saltykov, BB; Shubina, IO; Velikov, VK | 1 |
Jackson, WP; Jacobs, P; Kernoff, L; Klaff, LJ; Vinik, AI | 1 |
Enzmann, F; Gastpar, H; Weissgerber, PW; Zoltobrocki, M | 1 |
Chow, CC; Cockram, CS; Sorensen, JP; Tsang, LW | 1 |
Akkan, AG; Malaisse, WJ; Sener, A | 1 |
Abiru, N; Akazawa, S; Ishibasi, M; Kawasaki, E; Matsumoto, K; Matsuo, H; Uotani, S; Yamamoto, H; Yamasaki, H; Yano, M | 1 |
Fantus, IG; Klip, A; Leiter, LA; Ramlal, T; Tsiani, E | 1 |
Jennings, PE | 1 |
Bravo, G; Dawson, K; Meneilly, GS; Tessier, D; Tétrault, JP | 1 |
Balabolkin, MI; Maksumova, MA; Orekhov, AN; Slavina, ES; Sobenin, IA | 1 |
Inoue, S; Kobayashi, M; Koizumi, T; Ohnota, H; Sato, F; Tsutsumi, N | 1 |
Kruseman, AC; Menheere, PP; Müller, PG; Nijst, L; Sels, JP; Wolffenbuttel, BH | 1 |
Katsumata, K; Katsumata, Y; Ozawa, T | 1 |
König, E; Limmer, J; Rupprecht, E | 1 |
Akaoka, L; Funato, H; Kawasaki, T; Miyashita, H; Ogata, N; Sekino, N; Tagaya, T; Yamanouchi, T | 1 |
Gross, AS; Rieutord, A; Shenfield, GM; Stupans, I | 1 |
Geisen, K; Krause, E; Papp, JG; Végh, A | 1 |
Selvaag, E | 1 |
Gagliardino, JJ; García, ME; Rossi, PF | 1 |
Delaey, C; Van de Voorde, J | 1 |
Mori, A; Noda, Y; Packer, L | 1 |
Abenhaim, L; Monette, J; van Staa, T | 1 |
Ambrosi, F; Filipponi, P; Gregorio, F; Manfrini, S; Santucci, A | 1 |
Desfaits, AC; Renier, G; Serri, O | 2 |
Koyama, H; Mori, S; Nakajima, K; Sugioka, N; Uno, A | 1 |
Kaneko, T; Sakamoto, N | 1 |
Luo, M; O'Brien, RC | 1 |
Bouskela, E; Conde, CM; Cyrino, FZ; Garcia, AA | 1 |
Bataille, D; Blache, P; Gros, L; Salazar, G; Virsolvy, A | 1 |
Furman, BL; Tanira, MO | 1 |
Fukuzawa, M; Ikehata, F; Miyaguchi, S; Nakazawa, T; Ohta, S; Qiang, X; Sakata, Y; Satoh, J; Toyota, T | 1 |
Courtois, P; Herbaut, C; Malaisse, WJ; Sener, A; Turc, A | 1 |
Ambrosi, F; Carle, F; Filipponi, P; Gregorio, F; Manfrini, S; Merante, D; Testa, R; Velussi, M | 1 |
Gomis, R; Jones, NP; Patwardhan, RN; Squatrito, S; Wolffenbuttel, BH | 1 |
Cossins, E; Mori, A; Noda, Y; Packer, L | 1 |
Belch, JJ; Jennings, PE | 2 |
de Smet, PA; Fischer, HR | 1 |
Heine, RJ; van der Wal, PS | 1 |
Brunelli, C; Cordera, R; Cordone, S; Olivotti, L; Rossettin, P; Schiavo, M; Spallarossa, P | 1 |
Iwamoto, Y; Ohta, M; Wasada, T; Yano, T; Yui, N | 1 |
Chugh, K; Chugh, SN; Dhawan, R; Kishore, K; Sharma, A | 1 |
Ashcroft, SJ; Mikhailov, MV; Mikhailova, EA | 1 |
Cassone-Faldetta, M; De Luca, O; De Mattia, G; Fava, D; Ghiselli, A; Laurenti, O | 1 |
Abe, Y; Matsumoto, K; Miyake, S; Sera, Y; Tominaga, T; Ueki, Y | 1 |
Farouque, HM; Meredith, IT | 1 |
Auclair, J; Bouskela, E; Félétou, M; Levens, N; Néliat, G; Ravel, D | 1 |
Chow, WH; Davies, C; Jiang, J; Li, GW; Pan, CY; Shi, HL; Sun, XC; Tian, H; Yang, WY; Zhu, XX | 1 |
Antić, S; Bogicević, M; Milojković, M; Mitić-Zlatković, M; Stefanović, V; Stojiljković, S; Vlahović, P | 1 |
Fujita, T; Goto, A; Onozato, ML; Tojo, A | 1 |
Abe, Y; Matsumoto, K; Miyake, S; Sera, Y; Tominaga, T; Yeki, Y | 1 |
Crawford, BA; Perera, C | 1 |
Maddock, HL; Siedlecka, SM; Yellon, DM | 1 |
Bae, JH; Cho, CH; Han, J; Jang, BC; Kim, SP; Kim, SS; Lee, HY; Lim, JG; Park, JW; Park, MJ; Song, DK; Suh, SI; Yun, JE | 1 |
Hayaishi-Okano, R; Hori, M; Kaneto, H; Katakami, N; Kosugi, K; Matsuhisa, M; Ohtoshi, K; Yamasaki, Y | 1 |
Boes, U; Wascher, TC | 1 |
Aburuz, S; McElnay, J; Millership, J | 1 |
Fowler, A; Galiñanes, M; Loubani, M; Standen, NB | 1 |
Awata, T; Inukai, K; Kashiwabara, H; Katayama, S; Kurihara, S; Nakashima, Y; Sawa, T; Suzuki, M; Takata, N; Tanaka, M; Watanabe, M; Yokota, K | 1 |
Hinokio, Y; Hirai, M; Ishihara, H; Katagiri, H; Oka, Y; Satoh, J; Suzuki, S; Takahashi, K; Takizawa, Y; Tsuji, I | 1 |
Harata, N; Kinukawa, J; Shimura, M; Tamai, M | 1 |
Kardas, P | 1 |
Choudhury, H; Harisudhan, T; Mullangi, R; Srinivas, NR; Venkatesh, P | 1 |
Chang, NC; Huang, CL; Lee, TM; Lin, MS; Pan, NH | 1 |
Boggi, U; Bugliani, M; Del Chiaro, M; Del Guerra, S; Del Prato, S; Grupillo, M; Lupi, R; Marchetti, P; Masini, M; Mosca, F; Torri, S; Vistoli, F | 1 |
Chalikias, G; Floros, D; Hatseras, D; Kortsaris, A; Maltezos, E; Papadopoulou, E; Papanas, N; Souliou, E; Symeonidis, G; Trypsianis, G; Tziakas, D | 1 |
Aishima, M; Ito, Y; Naito, S; Nakano, T; Seki, N; Sueishi, K; Teramoto, N; Tomoda, T; Yonemitsu, Y; Yunoki, T | 1 |
Buithieu, J; Mamputu, JC; Räkel, A; Renier, G; Roussin, A; Serri, O | 1 |
Balzi, D; Barchielli, A; Buiatti, E; Lamanna, C; Mannucci, E; Marchionni, N; Masotti, G; Monami, M | 1 |
Jin, SH; Li, ZR; Shi, YQ; Yao, J | 1 |
Kimura, T; Kita, M; Suzuma, K; Takagi, H; Watanabe, D; Yoshimura, N | 1 |
Bilinska, M; Korzeniowska-Kubacka, I; Piotrowicz, R; Potocka, J | 1 |
Ishida, H; Kimoto, K; Kizaki, T; Miyazawa, N; Nakano, N; Ohno, H; Sakurai, T; Suzuki, K; Takahashi, K; Takahashi, M | 1 |
Li, J; Wang, L; Wu, GT; Zhu, WZ | 1 |
Gupta, A; Jain, S; Kumar, N; Tiwary, AK | 1 |
Fujii, M; Inoguchi, T; Kobayashi, K; Maeda, Y; Morinaga, H; Nomura, M; Sasaki, S; Sawada, F; Takayanagi, R; Tsubouchi, H | 1 |
Futami-Suda, S; Kigawa, Y; Nakano, H; Norose, J; Oba, K; Ouchi, M; Suzuki, K; Suzuki, T; Watanabe, K; Yasuoka, H | 1 |
Balzi, D; Lamanna, C; Mannucci, E; Marchionni, N; Monami, M | 1 |
Argaud, L; Couture-Lepetit, E; Garrier, O; Gateau-Roesch, O; Gomez, L; Loufouat, J; Ovize, M; Robert, D | 1 |
Hayakawa, M; Matsuyama-Yokono, A; Nakano, R; Shibasaki, M; Shiraki, K; Someya, Y; Tahara, A | 1 |
Boggi, U; Bugliani, M; D'Aleo, V; Del Guerra, S; Filipponi, F; Lupi, R; Marchetti, P; Masini, M | 1 |
Khalangot, M; Kovtun, V; Kravchenko, V; Tronko, M | 1 |
Ee, JW; Kwon, SW; Lee, J; Lee, WJ; Park, JH; Shaodong, J | 1 |
Hamaguchi, T; Hasegawa, Y; Ishikawa, T; Kakishita, E; Katsuno, T; Kohri, K; Konya, H; Miuchi, M; Miyagawa, J; Namba, M; Satani, K; Suehiro, A; Umehara, A | 1 |
Arai, K; Hirao, K; Kanamori, A; Matoba, K; Matsuba, I; Mori, H; Takai, M; Takeda, H; Terauchi, Y; Yamauchi, M | 1 |
Chan, JC; Chow, CC; Ko, GT; Kong, AP; Luk, AO; Ma, RC; Ng, VW; Ozaki, R; So, WY; Tong, PC; Yang, X; Yu, LW | 1 |
Buhl, ES; Bøtker, HE; Flyvbjerg, A; Kristiansen, SB; Løfgren, B; Nielsen, JM; Nielsen, TT; Nielsen-Kudsk, JE; Rungby, J; Støttrup, NB | 1 |
Abdelmoneim, AS; Brocks, DR; Hasenbank, SE; Light, PE; Seubert, JM; Simpson, SH | 1 |
Fatehi, M; Lang, VY; Light, PE | 1 |
Lim, PC; Lim, SL; Oiyammaal, C | 1 |
Dyrskjøt, L; Grimm, D; Magnusson, NE; Pietsch, J; Rungby, J; Wehland, M | 1 |
Gomes, T; Juurlink, DN; Mamdani, MM; Shah, BR | 1 |
Binz, TM; Neels, H; Schneider, S; Villani, N | 1 |
Bo, S; Castiglione, A; Cavallo-Perin, P; Ciccone, G; Durazzo, M; Gentile, L; Ghigo, E | 1 |
Kimura, H; Masuda, S; Sato, D; Sato, Y | 1 |
Abdelmoneim, AS; Eurich, DT; Gamble, JM; Johnson, JA; Qiu, W; Seubert, JM; Simpson, SH | 1 |
Khalangot, M; Kovtun, V | 1 |
Buranphalin, S; Doomkaew, A; Prapatpong, P; Suntornsuk, L; Vander Heyden, Y | 1 |
Andersson, C; Fosbøl, EL; Gislason, G; Køber, L; Mogensen, UM; Scheller, NM; Schramm, TK; Torp-Pedersen, C; Vaag, A | 1 |
Abdelmoneim, AS; Huang, Y; Light, P; Qiu, W; Simpson, SH | 1 |
Clemens, KK; Dixon, SN; Fleet, JL; Garg, AX; Hramiak, I; McArthur, E | 1 |
Chan, SP; Colagiuri, S | 1 |
Abdelmoneim, AS; Eurich, DT; Qiu, W; Senthilselvan, A; Simpson, SH | 1 |
Feng, YG; Fu, XH; Jiang, ZA; Li, LH; Li, LZ; Zheng, M | 1 |
Ashcroft, FM; Haythorne, E; Kramer, H; Proks, P | 1 |
Dong, J; Liao, L; Shen, X; Xie, T; Xu, C; Zhang, R; Zhou, X; Zou, Z | 1 |
Cordiner, RLM; Pearson, ER | 1 |
Huang, HK; Yeh, JI | 1 |
Bell, C; Shah, AJ; Singh, A; Zhao, K | 1 |
Ramazani, Z; Rashidi, H; Saberi, A; Saberi, M | 1 |
Hage, DS; Li, Z; Matsuda, R; Rodriguez, EL; Sun, Z; Tao, P; Woolfork, AG | 1 |
Chiriac, FL; Iancu, VI; Radu, GL; Scutariu, RE | 1 |
Hussain, F; Khan, M; Parvez, M | 1 |
Gayakvad, B; Kothari, C; Patel, C; Patel, R; Solanki, R; Wadhwana, P | 1 |
Bakulin, DA; Ivanova, OV; Kolosov, YA; Krysanov, IS; Kudrin, RA; Kurkin, DV; Makarova, EV; Robertus, AI | 1 |
Hiley, CR; White, R | 1 |
Fujiwara, H; Hashikawa-Hobara, N; Kawasaki, H; Kitamura, Y; Makino, K; Takatori, S; Wake, Y; Zamami, Y | 1 |
7 review(s) available for gliclazide and glyburide
Article | Year |
---|---|
Is combination sulfonylurea and insulin therapy useful in NIDDM patients? A metaanalysis.
Topics: Blood Glucose; C-Peptide; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; MEDLINE; Meta-Analysis as Topic; Middle Aged; Periodicals as Topic; Sulfonylurea Compounds; Tolazamide; Treatment Outcome; United States | 1992 |
Sulfonylureas and platelet function.
Topics: Adenosine Diphosphate; Blood Glucose; Blood Platelets; Collagen; Diabetes Mellitus; Diabetic Angiopathies; Epinephrine; Gliclazide; Glyburide; Humans; Platelet Aggregation; Sulfonylurea Compounds | 1981 |
[Clinical efficacy of glimepiride].
Topics: Blood Glucose; Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Sulfonylurea Compounds; Vascular Resistance | 1997 |
[Timing of administration of sulfonyl urea derivatives].
Topics: Biological Availability; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Drug Administration Schedule; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Tolbutamide | 2000 |
Variations in tissue selectivity amongst insulin secretagogues: a systematic review.
Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Cardiovascular Diseases; Cricetinae; Cyclohexanes; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Ischemic Preconditioning, Myocardial; Isoindoles; Mice; Muscle, Smooth, Vascular; Myocytes, Cardiac; Nateglinide; Phenylalanine; Piperidines; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Risk Factors; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide | 2012 |
Systematic review and meta-analysis of the efficacy and hypoglycemic safety of gliclazide versus other insulinotropic agents.
Topics: Adult; Aged; Aged, 80 and over; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemia; Hypoglycemic Agents; Metformin; Middle Aged; Randomized Controlled Trials as Topic; Sulfonylurea Compounds; Treatment Outcome; Young Adult | 2015 |
Reflections on the sulphonylurea story: A drug class at risk of extinction or a drug class worth reviving?
Topics: Diabetes Mellitus; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glucagon-Like Peptide-1 Receptor; Glyburide; History, 20th Century; History, 21st Century; Humans; Hypoglycemic Agents; Insulin Secretion; Insulin-Secreting Cells; Metformin; Sodium-Glucose Transporter 2 Inhibitors; Sulfonylurea Compounds; Treatment Failure | 2019 |
35 trial(s) available for gliclazide and glyburide
Article | Year |
---|---|
Effects of the sulphonylurea drugs gliclazide and glibenclamide on blood glucose control and platelet function.
Topics: Adult; Aged; Blood Glucose; Diabetes Mellitus; Female; Gliclazide; Glyburide; Humans; Male; Middle Aged; Platelet Aggregation; Sulfonylurea Compounds | 1979 |
Is combination sulfonylurea and insulin therapy useful in NIDDM patients? A metaanalysis.
Topics: Blood Glucose; C-Peptide; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; MEDLINE; Meta-Analysis as Topic; Middle Aged; Periodicals as Topic; Sulfonylurea Compounds; Tolazamide; Treatment Outcome; United States | 1992 |
Efficacy of gliclazide in comparison with other sulphonylureas in the treatment of NIDDM.
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Diet, Diabetic; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Tolbutamide | 1991 |
Comparison of secondary failure rate between three second generation sulphonylureas.
Topics: Blood Glucose; Diabetes Mellitus, Type 2; Diet, Diabetic; Follow-Up Studies; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Random Allocation | 1990 |
Lack of effect of gliclazide on platelet aggregation in insulin-treated and non-insulin-treated diabetes: a two-year controlled study.
Topics: Clinical Trials as Topic; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Double-Blind Method; Gliclazide; Glyburide; Humans; Platelet Aggregation; Random Allocation; Sulfonylurea Compounds | 1988 |
Comparison of diabetic control in type 2 (non-insulin dependent) diabetic patients treated with different sulphonylureas.
Topics: Aged; Chlorpropamide; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Middle Aged; Random Allocation; Sulfonylurea Compounds | 1985 |
[Effects of gliclazide and glibenclamide on platelet function, fibrinolysis and metabolic control in diabetic patients with retinopathy (author's transl)].
Topics: Blood Glucose; Diabetic Retinopathy; Fibrinolysis; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Middle Aged; Platelet Aggregation; Sulfonylurea Compounds | 1982 |
Comparison of gliclazide and glibenclamide treatment in non-insulin-dependent diabetes.
Topics: Adult; Aged; Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Double-Blind Method; Female; Fundus Oculi; Gliclazide; Glyburide; Humans; Lipids; Male; Middle Aged; Platelet Adhesiveness; Platelet Aggregation; Random Allocation; Sulfonylurea Compounds | 1983 |
Comparison of insulin with or without continuation of oral hypoglycemic agents in the treatment of secondary failure in NIDDM patients.
Topics: Analysis of Variance; Biomarkers; Blood Glucose; Body Mass Index; C-Peptide; Cholesterol; Cholesterol, HDL; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Fructosamine; Gliclazide; Glipizide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Hypoglycemic Agents; Insulin; Male; Metformin; Middle Aged; Treatment Failure; Triglycerides | 1995 |
Insulin response after treatment depends on fasting plasma glucose level in NIDDM.
Topics: Adult; Blood Glucose; Body Mass Index; C-Peptide; Diabetes Mellitus, Type 2; Diet, Diabetic; Fasting; Female; Gliclazide; Glucagon; Glucose Tolerance Test; Glyburide; Humans; Insulin; Male; Middle Aged | 1994 |
The potential of gliclazide, a sulphonylurea to influence the oxidative processes within the pathogenesis of diabetic vascular disease.
Topics: Adult; Aged; Analysis of Variance; Animals; Blood Glucose; Diabetic Angiopathies; Free Radical Scavengers; Gliclazide; Glyburide; Glycated Hemoglobin; Glycosylation; Humans; Lipid Peroxides; Male; Middle Aged; Oxidative Stress; Platelet Aggregation; Protein Processing, Post-Translational; Serum Albumin; Superoxide Dismutase | 1994 |
Glibenclamide vs gliclazide in type 2 diabetes of the elderly.
Topics: Aged; Blood Glucose; Diabetes Mellitus, Type 2; Female; Gliclazide; Glyburide; Humans; Hypoglycemia; Male | 1994 |
Effects of a new oral hypoglycaemic agent, repaglinide, on metabolic control in sulphonylurea-treated patients with NIDDM.
Topics: Aged; Blood Glucose; Carbamates; Diabetes Mellitus, Type 2; Female; Fructosamine; Gliclazide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Hypoglycemic Agents; Lipids; Male; Middle Aged; Piperidines; Tolbutamide | 1993 |
Clinical usefulness of serum 1,5-anhydroglucitol in monitoring glycaemic control.
Topics: Biomarkers; Blood Glucose; Deoxyglucose; Diabetes Mellitus, Type 2; Drug Administration Schedule; Evaluation Studies as Topic; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Isomerism; Male; Middle Aged; Prospective Studies; Sensitivity and Specificity; Time Factors | 1996 |
Meformin, plasma glucose and free fatty acids in type II diabetic out-patients: results of a clinical study.
Topics: Blood Glucose; Body Constitution; Body Mass Index; C-Peptide; Cholesterol; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Fasting; Fatty Acids, Nonesterified; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Lipoprotein(a); Male; Metformin; Middle Aged; Regression Analysis; Sex Characteristics | 1997 |
Poorly controlled elderly Type 2 diabetic patients: the effects of increasing sulphonylurea dosages or adding metformin.
Topics: Aged; Aging; Antithrombin III; Blood Glucose; Blood Platelets; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Female; Fibrinolysis; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Metformin; Thrombin | 1999 |
Addition of low-dose rosiglitazone to sulphonylurea therapy improves glycaemic control in Type 2 diabetic patients.
Topics: Adult; Aged; Blood Glucose; C-Peptide; Cholesterol; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Therapy, Combination; Europe; Female; Fructosamine; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Rosiglitazone; Safety; Thiazoles; Thiazolidinediones; Triglycerides | 2000 |
Free radical scavenging activity of sulfonylureas: a clinical assessment of the effect of gliclazide.
Topics: Adult; Aged; Blood Platelets; Collagen; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Therapy, Combination; Free Radical Scavengers; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Oxidation-Reduction; Sulfonylurea Compounds | 2000 |
Characteristics of pancreatic beta-cell secretion in Type 2 diabetic patients treated with gliclazide and glibenclamide.
Topics: Aged; Blood Glucose; Cross-Over Studies; Diabetes Mellitus, Type 2; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Male; Middle Aged; Reference Values; Sulfonylurea Compounds | 2001 |
Sulfonylurea treatment of type 2 diabetic patients does not reduce the vasodilator response to ischemia.
Topics: Aged; Aged, 80 and over; Blood Pressure; Brachial Artery; Diabetes Mellitus, Type 2; Diet, Diabetic; Female; Forearm; Gliclazide; Glyburide; Humans; Hyperlipidemias; Hypertension; Hypoglycemic Agents; Ischemia; Male; Metformin; Middle Aged; Reference Values; Regional Blood Flow; Sulfonylurea Compounds; Ultrasonography | 2001 |
[Free radical scavenging activity of sulfonylureas: a clinical assessment of the effectiveness of gliclazide].
Topics: Adult; Aged; Blood Glucose; Diabetes Mellitus, Type 2; Follow-Up Studies; Free Radical Scavengers; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Lipid Peroxidation; Male; Middle Aged; Myocardial Ischemia; Oxidative Stress; Time Factors | 2001 |
Glibenclamide vs gliclazide in reducing oxidative stress in patients of noninsulin dependent diabetes mellitus--a double blind randomized study.
Topics: Diabetes Mellitus, Type 2; Double-Blind Method; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Oxidative Stress | 2001 |
Gliclazide improves anti-oxidant status and nitric oxide-mediated vasodilation in Type 2 diabetes.
Topics: Adult; Aged; Antioxidants; Arginine; Blood Pressure; Diabetes Mellitus, Type 2; Free Radicals; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Injections, Intravenous; Lipid Peroxides; Male; Middle Aged; Nitric Oxide; Oxidative Stress; Vasodilation | 2002 |
Combination therapy of alpha-glucosidase inhibitor and a sulfonylurea compound prolongs the duration of good glycemic control.
Topics: Blood Glucose; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Enzyme Inhibitors; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Glycoside Hydrolase Inhibitors; Humans; Inositol; Male; Middle Aged; Sulfonylurea Compounds; Survival Analysis; Time Factors | 2002 |
Addition of rosiglitazone to existing sulfonylurea treatment in chinese patients with type 2 diabetes and exposure to hepatitis B or C.
Topics: Adult; Asian People; Blood Glucose; China; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Therapy, Combination; Environmental Exposure; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Hepatitis B; Hepatitis C; Humans; Hypoglycemic Agents; Insulin; Male; Middle Aged; Rosiglitazone; Sulfonylurea Compounds; Thiazoles; Thiazolidinediones | 2003 |
Metformin or gliclazide, rather than glibenclamide, attenuate progression of carotid intima-media thickness in subjects with type 2 diabetes.
Topics: Carotid Arteries; Carotid Artery Diseases; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Follow-Up Studies; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Lipids; Male; Metformin; Middle Aged; Multivariate Analysis; Tunica Intima; Tunica Media | 2004 |
Forearm vascular reactivity is differentially influenced by gliclazide and glibenclamide in chronically treated type 2 diabetic patients.
Topics: Adult; Analysis of Variance; Cross-Over Studies; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Forearm; Gliclazide; Glyburide; Humans; Hyperemia; Hypoglycemic Agents; Ischemia; Male; Middle Aged; Plethysmography; Regional Blood Flow; Time Factors; Vasodilation | 2005 |
Efficacy of glimepiride in Japanese type 2 diabetic subjects.
Topics: Aged; Asian People; Body Mass Index; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Homeostasis; Humans; Hypoglycemic Agents; Insulin Resistance; Logistic Models; Male; Middle Aged; Obesity; Retreatment; Sulfonylurea Compounds; Treatment Outcome | 2005 |
Secondary sulfonylurea failure: comparison of period until insulin treatment between diabetic patients treated with gliclazide and glibenclamide.
Topics: Age of Onset; Databases, Factual; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Middle Aged; Sulfonylurea Compounds; Time Factors; Treatment Failure | 2005 |
The DIACOM study (effect of DosIng frequency of oral Antidiabetic agents on the COMpliance and biochemical control of type 2 diabetes).
Topics: Adult; Aged; Anthropometry; Blood Glucose; Diabetes Mellitus, Type 2; Drug Administration Schedule; Drug Monitoring; Female; Gliclazide; Glyburide; Hemoglobins, Abnormal; Humans; Hypoglycemic Agents; Male; Middle Aged; Patient Compliance | 2005 |
Association of gliclazide and left ventricular mass in type 2 diabetic patients.
Topics: Aged; Body Mass Index; Diabetes Mellitus, Type 2; Electrocardiography; Female; Gliclazide; Glyburide; Heart Ventricles; Humans; Hypoglycemic Agents; Male; Middle Aged; Oxidative Stress; Prospective Studies; Ventricular Function, Left | 2006 |
Gliclazide treatment lowers serum ICAM-1 levels in poorly controlled type 2 diabetic patients.
Topics: Adult; Blood Glucose; Diabetes Mellitus, Type 2; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Intercellular Adhesion Molecule-1; Male; Middle Aged; Reference Values; Vascular Cell Adhesion Molecule-1 | 2006 |
Beneficial effects of gliclazide modified release compared with glibenclamide on endothelial activation and low-grade inflammation in patients with type 2 diabetes.
Topics: Adult; Aged; Diabetes Mellitus, Type 2; Double-Blind Method; Endothelium, Vascular; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Inflammation; Male; Middle Aged | 2007 |
'Warm-up' phenomenon in diabetic patients with stable angina treated with diet or sulfonylureas.
Topics: Angina Pectoris; Blood Pressure; Diabetes Mellitus, Type 2; Exercise; Gliclazide; Glyburide; Heart Rate; Humans; Hypoglycemic Agents; Ischemic Preconditioning, Myocardial; Male; Middle Aged; Sulfonylurea Compounds | 2007 |
Daily blood glucose profiles of glibenclamide and gliclazide taken once or twice daily in elderly type 2 diabetic patients.
Topics: Aged; Aged, 80 and over; Blood Glucose; Circadian Rhythm; Diabetes Mellitus, Type 2; Drug Administration Schedule; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Treatment Outcome | 2008 |
117 other study(ies) available for gliclazide and glyburide
Article | Year |
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Novel substituted naphthalen-1-yl-methanone derivatives as anti-hyperglycemic agents.
Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Hypoglycemic Agents; Male; Naphthalenes; Rats; Rats, Sprague-Dawley; Streptozocin | 2006 |
Omega-(2-Naphthyloxy) amino alkanes as a novel class of anti-hyperglycemic and lipid lowering agents.
Topics: Alkanes; Alkylation; Amination; Animals; Hypoglycemic Agents; Hypolipidemic Agents; Lipid Metabolism; Male; Molecular Structure; Naphthalenes; PPAR gamma; Rats; Structure-Activity Relationship | 2008 |
Novel 2-aryl-naphtho[1,2-d]oxazole derivatives as potential PTP-1B inhibitors showing antihyperglycemic activities.
Topics: Animals; Diabetes Mellitus, Experimental; Enzyme Inhibitors; Hypoglycemic Agents; Lipids; Mice; Oxazoles; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Rats; Structure-Activity Relationship; Triglycerides | 2009 |
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship | 2008 |
Design and synthesis of 3,5-diarylisoxazole derivatives as novel class of anti-hyperglycemic and lipid lowering agents.
Topics: Animals; Blood Glucose; Cholesterol; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Hypoglycemic Agents; Hypolipidemic Agents; Isoxazoles; Male; Mice; Mice, Inbred C57BL; PPAR gamma; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Rats; Rats, Sprague-Dawley; Rats, Wistar; Streptozocin; Sucrose; Triglycerides | 2009 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical | 2010 |
In vitro inhibition of the bile salt export pump correlates with risk of cholestatic drug-induced liver injury in humans.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Cholestasis; Drug-Related Side Effects and Adverse Reactions; Humans; Insecta; Rats; Risk Factors | 2012 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
The direct effect of hypoglycaemic sulphonylureas on myocardial contractile force and arterial blood pressure.
Topics: Adrenalectomy; Animals; Blood Pressure; Carbutamide; Cardiac Output; Dogs; Female; Gliclazide; Glyburide; Heart Rate; Hematocrit; Male; Myocardial Contraction; Oxygen; Pancreatectomy; Sulfonylurea Compounds | 1977 |
[Hypoglycemic complications of oral drug therapy of diabetes mellitus. 21 cases].
Topics: Age Factors; Aged; Diabetes Mellitus; Diabetic Coma; Drug Interactions; Female; Gliclazide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Kidney Failure, Chronic; Liver Diseases; Male; Middle Aged; Neurologic Manifestations; Sulfonamides | 1976 |
[The insulin-secreting and proliferative activity of established islet cells in the presence of sulfonylurea].
Topics: Animals; Cell Division; Cell Line; Cell Line, Transformed; Cells, Cultured; Cricetinae; Gliclazide; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Sulfonylurea Compounds; Time Factors; Tolbutamide | 1992 |
Therapeutical concentrations of tolbutamide, glibenclamide, gliclazide and gliquidone at different glucose levels: in vitro effects on pancreatic A- and B-cell function.
Topics: Animals; Blood Glucose; Dose-Response Relationship, Drug; Gliclazide; Glucagon; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Perfusion; Rats; Rats, Sprague-Dawley; Sulfonylurea Compounds; Time Factors; Tolbutamide | 1992 |
Determination of gliclazide in serum by high-performance liquid chromatography using solid-phase extraction.
Topics: Chromatography, High Pressure Liquid; Gliclazide; Glyburide; Humans; Reference Standards; Reproducibility of Results; Spectrophotometry, Ultraviolet | 1992 |
Effects of oral hypoglycaemic agents on platelet functions.
Topics: Arachidonic Acid; Calcium; Dose-Response Relationship, Drug; Fura-2; Gliclazide; Glyburide; Humans; Ionomycin; Platelet Activation; Platelet Aggregation Inhibitors; Sulfonylurea Compounds | 1992 |
Divergent cardiac effects of the first and second generation hypoglycemic sulfonylurea compounds.
Topics: Animals; Arrhythmias, Cardiac; Blood Glucose; Carbutamide; Dose-Response Relationship, Drug; Electrocardiography; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Male; Myocardial Infarction; Potassium; Rats; Rats, Inbred Strains; Reference Values; Structure-Activity Relationship; Tolbutamide | 1990 |
The potentiating effect of the simultaneous administration of tolbutamide, glibenclamide, and gliclazide on the development of alloxan-induced diabetes in rats.
Topics: Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Drug Synergism; Gliclazide; Glucose Tolerance Test; Glyburide; Insulin; Male; Pancreas; Rats; Rats, Inbred Strains; Sulfonylurea Compounds; Tolbutamide | 1990 |
A screening test for detecting sulfonylureas in plasma.
Topics: Aged; Aged, 80 and over; Chlorpropamide; Chromatography, High Pressure Liquid; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Male; Middle Aged; Sulfonylurea Compounds; Tolbutamide | 1990 |
[New oral antidiabetic agents].
Topics: Animals; Cyclohexanols; Diabetes Mellitus; Drug Evaluation; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Imidazoles; Insulin; Insulin Secretion; Molecular Structure; Pyrrolidines; Stimulation, Chemical; Sulfonylurea Compounds | 1990 |
Protonophoretic activity of hypoglycemic sulfonylureas in black lipid membranes.
Topics: Biological Transport; Calcium; Cell Membrane; Chemical Phenomena; Chemistry, Physical; Gliclazide; Glyburide; Glycerol; Hypoglycemic Agents; In Vitro Techniques; Ionophores; Membrane Lipids; Membranes, Artificial; Protons; Sulfonylurea Compounds | 1986 |
[Hemorheologic, metabolic and blood coagulation changes in diabetics in treatment with sulfanyl ureas].
Topics: Blood Coagulation; Blood Viscosity; Diabetes Mellitus, Type 2; Erythrocyte Deformability; Gliclazide; Glyburide; Humans; Rheology; Sulfonylurea Compounds | 1988 |
Effect of gliclazide on thromboxane B2, parameters of haemostasis, fluorescent IgG and lipid peroxides in non-insulin dependent diabetes mellitus.
Topics: Aged; Blood Proteins; Diabetes Mellitus, Type 2; Female; Fructosamine; Gliclazide; Glyburide; Glycated Hemoglobin; Hexosamines; Humans; Immunoglobulin G; Lipid Peroxides; Male; Platelet Aggregation; Sulfonylurea Compounds; Thromboxane B2 | 1988 |
[Effect of long-term therapy with sulfanylurea preparations on the relation of insulin secretion and the insulin-binding capacity of its receptors].
Topics: Blood Glucose; Chlorpropamide; Diabetes Mellitus, Type 2; Drug Evaluation; Female; Gliclazide; Glucose Tolerance Test; Glyburide; Glycosuria; Humans; Hypoglycemic Agents; Insulin; Insulin Antibodies; Insulin Secretion; Leukocytes; Male; Middle Aged; Receptor, Insulin; Sulfonylurea Compounds | 1988 |
Suppression by 2-ketoisocaproate of the insulinotropic action of hypoglycemic sulfonylureas.
Topics: Animals; Calcium; Gliclazide; Glucose; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Insulin; Insulin Secretion; Ionophores; Keto Acids; Oxidation-Reduction; Rats; Sulfonylurea Compounds; Tolbutamide | 1985 |
Sulfonylurea stimulates liver fructose-2,6-bisphosphate formation in proportion to its hypoglycemic action.
Topics: Acetohexamide; Animals; Buformin; Chlorpropamide; Fructosediphosphates; Gliclazide; Gluconeogenesis; Glyburide; Glycolysis; Hexosediphosphates; In Vitro Techniques; Liver; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulfamethoxazole; Sulfonylurea Compounds; Tolbutamide | 1985 |
In vitro metabolic effects of gliclazide and glibenclamide in the rat.
Topics: Adipose Tissue; Animals; Gliclazide; Glucose; Glyburide; Glycogen; In Vitro Techniques; Insulin; Male; Metabolism; Muscle, Smooth; Oxidation-Reduction; Rats; Sulfonylurea Compounds | 1980 |
Transport of Pr3+ by hypoglycemic sulfonylureas across liposomal membranes.
Topics: Biological Transport; Gliclazide; Glyburide; Ionophores; Kinetics; Liposomes; Magnetic Resonance Spectroscopy; Models, Biological; Molecular Conformation; Praseodymium; Pulmonary Surfactants; Sulfonylurea Compounds | 1983 |
Gliclazide- and glibenclamide-mediated transport of Pr3+ across an artificial lipid membrane.
Topics: Biological Transport, Active; Gliclazide; Glyburide; Liposomes; Magnetic Resonance Spectroscopy; Membranes, Artificial; Praseodymium; Sulfonylurea Compounds | 1983 |
Preventive and therapeutic effects of gliclazide on diabetic retinopathy: comparison with glibenclamide treatment.
Topics: Adult; Aged; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Female; Gliclazide; Glyburide; Humans; Male; Middle Aged; Platelet Adhesiveness; Sulfonylurea Compounds | 1983 |
[Experience with diamicron treatment of diabetics].
Topics: Adult; Aged; Chronic Disease; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Drug Evaluation; Drug Therapy, Combination; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfanilamides; Sulfonylurea Compounds; Time Factors | 1984 |
The inhibition of cancer cell stickiness, a model for investigation of platelet aggregation inhibitors in vivo. Effect of the sulfonyl urea derivatives, glibenclamide, gliclazide, and HB180, as well as the carboxylic acid derivative, meglitinide.
Topics: Animals; Benzamides; Carcinoma 256, Walker; Cell Aggregation; Diabetes Mellitus; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Platelet Aggregation; Platelet Count; Rats; Rats, Inbred Strains; Sulfonylurea Compounds | 1982 |
Standardized procedure for the assay and identification of hypoglycemic sulfonylureas in human plasma.
Topics: Chromatography, High Pressure Liquid; Diabetes Mellitus, Type 2; Drug Monitoring; Forensic Medicine; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Reproducibility of Results; Sensitivity and Specificity; Sulfonylurea Compounds | 1995 |
Stimulation of glucose uptake and increased plasma membrane content of glucose transporters in L6 skeletal muscle cells by the sulfonylureas gliclazide and glyburide.
Topics: Animals; Biological Transport, Active; Cell Line; Cell Membrane; Cycloheximide; Deoxyglucose; Dose-Response Relationship, Drug; Gliclazide; Glucose; Glyburide; Insulin; Kinetics; Monosaccharide Transport Proteins; Muscle, Skeletal; Rats; Tissue Distribution | 1995 |
Sulfonylureas induce cholesterol accumulation in cultured human intimal cells and macrophages.
Topics: Adult; Animals; Cells, Cultured; Cholesterol; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Humans; Macrophages, Peritoneal; Male; Mice; Mice, Inbred BALB C; Middle Aged; Muscle, Smooth, Vascular; Sulfonylurea Compounds; Tunica Intima | 1994 |
Novel rapid- and short-acting hypoglycemic agent, a calcium(2s)-2-benzyl-3-(cis-hexahydro-2-isoindolinylcarbonyl) propionate (KAD-1229) that acts on the sulfonylurea receptor: comparison of effects between KAD-1229 and gliclazide.
Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Biological Transport; Cells, Cultured; Dogs; Gliclazide; Glyburide; Hypoglycemic Agents; Indoles; Insulin; Insulin Secretion; Islets of Langerhans; Isoindoles; Male; Mice; Mice, Inbred ICR; Microsomes; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rubidium; Sulfonylurea Receptors | 1994 |
Potentiating effects of combined usage of three sulfonylurea drugs on the occurrence of alloxan diabetes in rats.
Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Drug Combinations; Drug Synergism; Gliclazide; Glyburide; Hypoglycemic Agents; Rats; Rats, Wistar; Sulfonylurea Compounds; Tolbutamide | 1993 |
[Clinical evaluation of gliquidone--short acting sulfonylurea derivative--comparison with glibenclamide and gliclazide].
Topics: Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Sulfonylurea Compounds | 1993 |
Gliclazide hydroxylation by rat liver microsomes.
Topics: Animals; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2D6; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Gliclazide; Glipizide; Glyburide; Hydroxylation; Hypoglycemic Agents; Kinetics; Male; Microsomes, Liver; Mixed Function Oxygenases; Rats; Rats, Sprague-Dawley; Tolbutamide | 1995 |
Cardiovascular effects of conventional sulfonylureas and glimepiride.
Topics: Animals; Blood Pressure; Cardiovascular System; Coronary Vessels; Diabetes Mellitus, Experimental; Dogs; Electrocardiography; Female; Gliclazide; Glyburide; Hypoglycemic Agents; Male; Myocardial Ischemia; Potassium Channels; Rats; Rats, Wistar; Sulfonylurea Compounds | 1996 |
Photohemolytic potency of oral antidiabetic drugs in vitro: effects of antioxidants and a nitrogen atmosphere.
Topics: Antioxidants; Ascorbic Acid; Carbutamide; Chlorpropamide; Dose-Response Relationship, Drug; Gliclazide; Glipizide; Glyburide; Hemolysis; Humans; Hypoglycemic Agents; Nitrogen; Radiation-Sensitizing Agents; Reactive Oxygen Species; Sulfonamides; Sulfonylurea Compounds; Superoxide Dismutase; Tolazamide; Tolbutamide; Ultraviolet Rays; Vitamin E | 1996 |
Inhibitory effect of sulfonylureas on protein phosphatase activity in rat pancreatic islets.
Topics: Animals; Cytosol; Gliclazide; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kinetics; Male; Okadaic Acid; Phosphoprotein Phosphatases; Rats; Rats, Wistar; Sulfonylurea Compounds; Tolbutamide | 1997 |
Heterogeneity of the inhibitory influence of sulfonylureas on prostanoid-induced smooth muscle contraction.
Topics: Animals; Aorta, Thoracic; Arteries; Bronchi; Cattle; Drug Interactions; Female; Gliclazide; Glyburide; Guinea Pigs; Humans; Hypoglycemic Agents; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Prostaglandins; Rats; Rats, Wistar; Species Specificity; Tolazamide; Trachea | 1997 |
Gliclazide scavenges hydroxyl, superoxide and nitric oxide radicals: an ESR study.
Topics: Dose-Response Relationship, Drug; Electron Spin Resonance Spectroscopy; Free Radical Scavengers; Free Radicals; Gliclazide; Glyburide; Hypoglycemic Agents; Nitric Oxide; Oxidative Stress; Superoxides | 1997 |
Rates of hypoglycemia in users of sulfonylureas.
Topics: Adult; Aged; Chlorpropamide; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Incidence; Male; Middle Aged; Poisson Distribution; Risk; Risk Factors; Sulfonylurea Compounds; Surveys and Questionnaires; Time Factors; Tolbutamide | 1997 |
Gliclazide decreases cell-mediated low-density lipoprotein (LDL) oxidation and reduces monocyte adhesion to endothelial cells induced by oxidatively modified LDL.
Topics: Animals; Aorta; Cattle; Cell Adhesion; Cell Survival; Cells, Cultured; Copper Sulfate; Endothelium, Vascular; Gliclazide; Glyburide; Humans; In Vitro Techniques; Lipoproteins, LDL; Monocytes; Oxidation-Reduction; Thiobarbituric Acid Reactive Substances | 1997 |
Effects of glycosylation of hypoglycaemic drug binding to serum albumin.
Topics: Acetohexamide; Binding Sites; Binding, Competitive; Gliclazide; Glyburide; Glycated Serum Albumin; Glycation End Products, Advanced; Glycosylation; Humans; Hypoglycemic Agents; Metformin; Serum Albumin; Spectrometry, Fluorescence; Structure-Activity Relationship; Tolbutamide | 1997 |
The effects of gliclazide and other sulfonylureas on low-density lipoprotein oxidation in vitro.
Topics: Administration, Oral; Adult; Antioxidants; Ascorbic Acid; Coronary Artery Disease; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Lipoproteins, LDL; Male; Middle Aged; Oxidation-Reduction; Sulfonylurea Compounds; Tolbutamide | 1997 |
Microvascular permeability with sulfonylureas in normal and diabetic hamsters.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Capillary Permeability; Cricetinae; Dextrans; Diabetes Mellitus, Experimental; Diazoxide; Disease Models, Animal; Dose-Response Relationship, Drug; Fluorescein-5-isothiocyanate; Gliclazide; Glyburide; Histamine; Hypoglycemic Agents; Insulin; Macromolecular Substances; Male; Mesocricetus; Nifedipine; Potassium Channels; Reperfusion Injury; Streptozocin; Sulfonylurea Compounds | 1997 |
Normalization of plasma lipid peroxides, monocyte adhesion, and tumor necrosis factor-alpha production in NIDDM patients after gliclazide treatment.
Topics: Animals; Aorta; Arteriosclerosis; Cattle; Cell Adhesion; Cell Adhesion Molecules; Cells, Cultured; Cytokines; Diabetes Mellitus, Type 2; E-Selectin; Endothelium, Vascular; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Intercellular Adhesion Molecule-1; Interleukin-1; Interleukin-6; Lipid Peroxides; Lipopolysaccharides; Monocytes; Reference Values; Treatment Failure; Tumor Necrosis Factor-alpha; Vascular Cell Adhesion Molecule-1 | 1998 |
Characterization of low-affinity binding sites for glibenclamide on the Kir6.2 subunit of the beta-cell KATP channel.
Topics: Animals; ATP-Binding Cassette Transporters; Binding Sites; Blotting, Northern; Cell Line; Cell Membrane; COS Cells; Gliclazide; Glipizide; Glyburide; Islets of Langerhans; Kinetics; Organelles; Phentolamine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, Drug; Recombinant Fusion Proteins; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide; Transfection | 1999 |
The in vivo interaction between gliclazide and glibenclamide and insulin on glucose disposal in the rat.
Topics: Animals; Biomarkers; Blood Glucose; Diabetes Mellitus, Experimental; Drug Interactions; Fatty Acids, Nonesterified; Gliclazide; Glucose; Glucose Tolerance Test; Glyburide; Hypoglycemic Agents; Insulin; Male; Rats; Rats, Wistar | 1999 |
Glimepiride: new preparation. Just another hypoglycaemic sulphonylurea agent.
Topics: Blood Glucose; Clinical Trials as Topic; Diabetes Mellitus, Type 2; Double-Blind Method; Drug Evaluation; Europe; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemia; Hypoglycemic Agents; Sulfonylurea Compounds; Treatment Outcome; United States | 1998 |
Inhibition of tumor necrosis factor-alpha with anti-diabetic agents.
Topics: Animals; Biological Assay; Cells, Cultured; Chromans; Enzyme-Linked Immunosorbent Assay; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Interleukin-1; Interleukin-6; Male; Mice; Mice, Inbred BALB C; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1999 |
Pharmacokinetics of gliquidone, glibenclamide, gliclazide and glipizide in middle-aged and aged subjects.
Topics: Aged; Female; Gliclazide; Glipizide; Glyburide; Half-Life; Humans; Hypoglycemic Agents; Male; Middle Aged; Sulfonylurea Compounds | 1999 |
Gliclazide scavenges hydroxyl and superoxide radicals: an electron spin resonance study.
Topics: Electron Spin Resonance Spectroscopy; Free Radical Scavengers; Gliclazide; Glyburide; Hydroxyl Radical; Hypoglycemic Agents; Superoxides | 2000 |
ATP-Sensitive potassium channels modulate glucose transport in cultured human skeletal muscle cells.
Topics: 3-O-Methylglucose; Adenosine Triphosphate; Benzopyrans; Biological Transport; Cells, Cultured; Cyclopentanes; Deoxyglucose; Enzyme Activation; Gliclazide; Glucose; Glyburide; Humans; Hypoglycemic Agents; Insulin; Ion Channel Gating; Muscle, Skeletal; Nicorandil; Potassium Channel Blockers; Potassium Channels; Protein Kinase C; Tetradecanoylphorbol Acetate | 2001 |
A novel simple method for the investigation of drug binding to the K(ATP) channel sulfonylurea receptor.
Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Gliclazide; Glyburide; Hypoglycemic Agents; Kinetics; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Rats; Receptors, Drug; Spodoptera; Sulfonylurea Receptors; Tolbutamide | 2002 |
Effects of inhibition of ATP-sensitive potassium channels on metabolic vasodilation in the human forearm.
Topics: Adenosine Triphosphate; Adult; Dose-Response Relationship, Drug; Female; Forearm; Gliclazide; Glyburide; Humans; Hyperemia; Male; Muscle, Skeletal; Plethysmography; Potassium Channel Blockers; Potassium Channels; Regional Blood Flow; Vasodilation | 2003 |
Differential effects of sulphonylureas on the vasodilatory response evoked by K(ATP) channel openers.
Topics: Adenosine Triphosphate; Animals; Aorta, Thoracic; Cricetinae; Cromakalim; Diazoxide; Drug Interactions; Gliclazide; Glyburide; Guinea Pigs; Hypoglycemic Agents; In Vitro Techniques; Ion Channel Gating; Male; Potassium Channels; Rats; Rats, Wistar; Species Specificity; Sulfonylurea Compounds; Vasodilation; Vasodilator Agents | 2003 |
Urinary PC-1 and N-acetyl-beta-D-glucosaminidase activity in patients with type 2 diabetes treated with metformin, gliclazide or glibenclamide.
Topics: Acetylglucosaminidase; Administration, Oral; Adult; Aged; Creatinine; Diabetes Mellitus, Type 2; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Obesity; Phosphoric Diester Hydrolases; Pyrophosphatases | 2003 |
Radical scavenging effect of gliclazide in diabetic rats fed with a high cholesterol diet.
Topics: Animals; Blood Pressure; Cholesterol, Dietary; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Free Radical Scavengers; Gliclazide; Glyburide; Glycated Hemoglobin; Hypoglycemic Agents; Intercellular Adhesion Molecule-1; Kidney; Macrophages; Male; NADPH Oxidases; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitrites; Oxidative Stress; Rats; Rats, Sprague-Dawley; Superoxide Dismutase | 2004 |
Metformin attenuates progression of carotid arterial wall thickness in patients with type 2 diabetes.
Topics: Arteriosclerosis; Carotid Arteries; Carotid Artery Diseases; Chronic Disease; Diabetes Mellitus, Type 2; Diet Therapy; Drug Administration Schedule; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Japan; Male; Metformin; Middle Aged; Prospective Studies; Sulfonylurea Compounds; Time Factors; Tunica Intima; Tunica Media | 2004 |
Octreotide treatment for sulfonylurea-induced hypoglycaemia.
Topics: Aged; Blood Glucose; Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Octreotide; Sulfonylurea Compounds; Treatment Outcome | 2004 |
Myocardial protection from either ischaemic preconditioning or nicorandil is not blocked by gliclazide.
Topics: Animals; Anti-Arrhythmia Agents; Gliclazide; Glyburide; Hypoglycemic Agents; Ischemic Preconditioning; Male; Membrane Potentials; Mitochondria, Heart; Myocardial Infarction; Nicorandil; Rats; Rats, Sprague-Dawley | 2004 |
Taurine block of cloned ATP-sensitive K+ channels with different sulfonylurea receptor subunits expressed in Xenopus laevis oocytes.
Topics: Animals; ATP-Binding Cassette Transporters; Carbamates; Drug Interactions; Female; Gene Expression; Gliclazide; Glyburide; Hypoglycemic Agents; Membrane Proteins; Mice; Oocytes; Piperidines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Subunits; Rats; Receptors, Drug; Sulfonylurea Receptors; Taurine; Tolbutamide; Xenopus laevis | 2004 |
The development and validation of liquid chromatography method for the simultaneous determination of metformin and glipizide, gliclazide, glibenclamide or glimperide in plasma.
Topics: Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Metformin; Reference Standards; Sensitivity and Specificity | 2005 |
The effect of gliclazide and glibenclamide on preconditioning of the human myocardium.
Topics: Algorithms; Atrial Appendage; Creatine Kinase; Dose-Response Relationship, Drug; Enzyme Activation; Gliclazide; Glyburide; Heart; Humans; Hypoglycemic Agents; In Vitro Techniques; Ischemic Preconditioning, Myocardial; Muscle, Smooth, Vascular; Myocardium; p38 Mitogen-Activated Protein Kinases; Potassium Channels; Protein Kinase C; Signal Transduction | 2005 |
Gliclazide attenuates the intracellular Ca2+ changes induced in vitro by ischemia in the retinal slices of rats with streptozotocin-induced diabetes.
Topics: Aniline Compounds; Animals; Calcium; Diabetes Mellitus, Experimental; Diabetic Retinopathy; Gliclazide; Glyburide; Hypoglycemic Agents; Ionomycin; Ionophores; Ischemia; Microscopy, Confocal; Rats; Rats, Sprague-Dawley; Retina; Streptozocin; Xanthenes | 2005 |
Simultaneous estimation of six anti-diabetic drugs--glibenclamide, gliclazide, glipizide, pioglitazone, repaglinide and rosiglitazone: development of a novel HPLC method for use in the analysis of pharmaceutical formulations and its application to human p
Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Molecular Structure; Pioglitazone; Piperidines; Reproducibility of Results; Rosiglitazone; Thiazolidinediones | 2006 |
Gliclazide protects human islet beta-cells from apoptosis induced by intermittent high glucose.
Topics: Antioxidants; Apoptosis; Cells, Cultured; Female; Gliclazide; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Male; Microscopy, Electron; Middle Aged; Tyrosine | 2007 |
Actions of ZD0947, a novel ATP-sensitive K+ channel opener, on membrane currents in human detrusor myocytes.
Topics: ATP-Binding Cassette Transporters; Carbachol; Diazoxide; Dihydropyridines; Dose-Response Relationship, Drug; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Gliclazide; Glyburide; Humans; Immunochemistry; In Vitro Techniques; Membrane Potentials; Muscle Relaxation; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors; Urinary Bladder | 2006 |
Are sulphonylureas all the same? A cohort study on cardiovascular and cancer-related mortality.
Topics: Aged; Cardiovascular Diseases; Cohort Studies; Diabetes Mellitus, Type 2; Female; Follow-Up Studies; Gliclazide; Glyburide; Heart Diseases; Humans; Hypoglycemic Agents; Incidence; Male; Middle Aged; Neoplasms; Retrospective Studies; Sulfonylurea Compounds | 2007 |
Development of a RP-HPLC method for screening potentially counterfeit anti-diabetic drugs.
Topics: Carbamates; Chromatography, High Pressure Liquid; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Molecular Structure; Piperidines; Reproducibility of Results; Sulfonylurea Compounds | 2007 |
Comparisons between the beneficial effects of different sulphonylurea treatments on ischemia-induced retinal neovascularization.
Topics: Acetylcysteine; Animals; Blood Glucose; Female; Gliclazide; Glyburide; Ischemia; Mice; Oxidative Stress; Oxygen; Retina; Retinal Neovascularization; RNA, Messenger; Sulfonylurea Compounds; Vascular Endothelial Growth Factor A | 2007 |
Gliclazide inhibits proliferation but stimulates differentiation of white and brown adipocytes.
Topics: Adipocytes, Brown; Adipocytes, White; Animals; Blotting, Western; Cell Differentiation; Cell Line; Cell Proliferation; Diazoxide; Epidermal Growth Factor; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Gliclazide; Glyburide; Hypoglycemic Agents; Mice; Phosphorylation; PPAR gamma; Signal Transduction; Sulfonylurea Compounds | 2007 |
Effects of glibenclamide, glimepiride, and gliclazide on ischemic preconditioning in rat heart.
Topics: Animals; Gliclazide; Glyburide; Heart; Ischemic Preconditioning; Male; Rats; Rats, Sprague-Dawley; Sulfonylurea Compounds | 2007 |
Spermicidal activity of sulfonylureas and meglitinide analogues: role of intrasperm Ca2+ elevation.
Topics: Adult; Benzamides; Calcium; Carbamates; Cross-Over Studies; Dose-Response Relationship, Drug; Gliclazide; Glyburide; Homeostasis; Humans; Hypoglycemic Agents; KATP Channels; Male; Piperidines; Sperm Motility; Spermatocidal Agents; Spermatozoa; Sulfonylurea Compounds; Time Factors | 2008 |
Differential effect of sulfonylureas on production of reactive oxygen species and apoptosis in cultured pancreatic beta-cell line, MIN6.
Topics: Animals; Apoptosis; Cell Line; Cyclohexanes; Fluoresceins; Gliclazide; Glyburide; Hypoglycemic Agents; In Situ Nick-End Labeling; Insulin-Secreting Cells; Mice; Mice, Inbred C57BL; Microscopy, Fluorescence; NADPH Oxidases; Nateglinide; Phenylalanine; Protein Kinase C; Reactive Oxygen Species; Sulfonylurea Compounds | 2008 |
Sulphonylureas and cancer: a case-control study.
Topics: Aged; Case-Control Studies; Diabetes Mellitus, Type 2; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Neoplasms; Risk Factors; Sulfonylurea Compounds | 2009 |
Second-generation sulfonylureas preserve inhibition of mitochondrial permeability transition by the mitochondrial K+(ATP) opener nicorandil in experimental myocardial infarction.
Topics: Animals; Calcium; Gliclazide; Glyburide; Hemodynamics; Male; Mitochondria; Myocardial Infarction; Nicorandil; Potassium Channel Blockers; Potassium Channels; Rabbits; Sulfonylurea Compounds | 2009 |
Antidiabetic effects of dipeptidyl peptidase-IV inhibitors and sulfonylureas in streptozotocin-nicotinamide-induced mildly diabetic mice.
Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Gliclazide; Glucagon-Like Peptide 1; Glucose Intolerance; Glyburide; Hypoglycemic Agents; Insulin; Male; Mice; Mice, Inbred ICR; Niacinamide; Piperidines; Pyrrolidines; Sulfonylurea Compounds | 2009 |
Effects of exposure of human islet beta-cells to normal and high glucose levels with or without gliclazide or glibenclamide.
Topics: Aged; Analysis of Variance; Cells, Cultured; Female; Gliclazide; Glucose; Glyburide; Homeodomain Proteins; Humans; Hyperglycemia; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; Ki-67 Antigen; Male; Middle Aged; Pancreas; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tissue Donors; Trans-Activators | 2009 |
Glibenclamide-related excess in total and cardiovascular mortality risks: data from large Ukrainian observational cohort study.
Topics: Blood Glucose; Blood Pressure; Body Mass Index; Cardiovascular Diseases; Cohort Studies; Cross-Sectional Studies; Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Middle Aged; Patient Selection; Proportional Hazards Models; Risk Factors; Sulfonylurea Compounds; Ukraine | 2009 |
Comparison of ultraviolet detection, evaporative light scattering detection and charged aerosol detection methods for liquid-chromatographic determination of anti-diabetic drugs.
Topics: Aerosols; Chromatography, High Pressure Liquid; Chromatography, Reverse-Phase; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Light; Reproducibility of Results; Scattering, Radiation; Spectrophotometry, Ultraviolet; Sulfonylurea Compounds | 2010 |
Effects of gliclazide on platelet aggregation and the plasminogen activator inhibitor type 1 level in patients with type 2 diabetes mellitus.
Topics: Aged; alpha-2-Antiplasmin; Antithrombin III; Azides; Blood Glucose; Body Mass Index; Deoxyuracil Nucleotides; Diabetes Mellitus, Type 2; Female; Fibrinolysin; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Middle Aged; Peptide Hydrolases; Plasminogen Activator Inhibitor 1; Platelet Aggregation | 2010 |
Present status of sulfonylurea treatment for type 2 diabetes in Japan: second report of a cross-sectional survey of 15,652 patients.
Topics: Aged; Blood Glucose; Cross-Sectional Studies; Diabetes Mellitus, Type 2; Family Practice; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Japan; Middle Aged; Practice Patterns, Physicians'; Sulfonylurea Compounds; Treatment Outcome | 2010 |
Use of sulphonylurea and cancer in type 2 diabetes-The Hong Kong Diabetes Registry.
Topics: Aged; Asian People; Cohort Studies; Diabetes Mellitus, Type 2; Female; Gliclazide; Glipizide; Glyburide; Hong Kong; Humans; Male; Middle Aged; Neoplasms; Proportional Hazards Models; Prospective Studies; Registries; Risk Factors; Sulfonylurea Compounds | 2010 |
Comparison of two sulfonylureas with high and low myocardial K(ATP) channel affinity on myocardial infarct size and metabolism in a rat model of type 2 diabetes.
Topics: Animals; Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Glycogen; Lactic Acid; Male; Myocardial Infarction; Myocardium; Potassium Channels; Rats; Rats, Wistar; Sulfonylurea Compounds | 2011 |
Pharmacogenomic analysis of ATP-sensitive potassium channels coexpressing the common type 2 diabetes risk variants E23K and S1369A.
Topics: ATP-Binding Cassette Transporters; Chlorpropamide; Cyclohexanes; Diabetes Mellitus, Type 2; Gene Expression Regulation; Gliclazide; Glyburide; Haplotypes; Homozygote; Humans; Isoindoles; Nateglinide; Patch-Clamp Techniques; Phenylalanine; Polymorphism, Single Nucleotide; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Structure-Activity Relationship; Sulfonylurea Compounds; Sulfonylurea Receptors; Tolbutamide | 2012 |
Glycaemic control and cost analysis when changing from gliclazide co-administered with metformin to pre-combined glibenclamide-metformin tablets in type 2 diabetes mellitus.
Topics: Blood Glucose; Costs and Cost Analysis; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glyburide; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Retrospective Studies; Tablets | 2012 |
Gene networks modified by sulphonylureas in beta cells: a pathway-based analysis of insulin secretion and cell death.
Topics: Animals; Cell Death; Cell Line; Cluster Analysis; Diabetes Mellitus, Type 2; Gene Regulatory Networks; Gliclazide; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Insulin-Secreting Cells; Microarray Analysis; Rats; Sulfonylurea Compounds; Up-Regulation | 2012 |
Adverse cardiovascular events during treatment with glyburide (glibenclamide) or gliclazide in a high-risk population.
Topics: Aged; Angioplasty, Balloon, Coronary; Cohort Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Incidence; Ischemic Preconditioning; Male; Myocardial Infarction; Myocardium; Ontario; Risk Factors; Sulfonylurea Compounds; Treatment Outcome | 2012 |
Rapid extraction, identification and quantification of oral hypoglycaemic drugs in serum and hair using LC-MS/MS.
Topics: Acetonitriles; Chromatography, Liquid; Female; Forensic Toxicology; Gliclazide; Glipizide; Glyburide; Hair; Humans; Hypoglycemic Agents; Limit of Detection; Male; Mass Spectrometry; Metformin; Methanol; Middle Aged; Molecular Structure; Solvents; Sulfonylurea Compounds | 2012 |
Mortality outcomes of different sulphonylurea drugs: the results of a 14-year cohort study of type 2 diabetic patients.
Topics: Adult; Aged; Cardiovascular Diseases; Cause of Death; Cohort Studies; Confounding Factors, Epidemiologic; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Kaplan-Meier Estimate; Male; Metformin; Middle Aged; Neoplasms; Odds Ratio; Proportional Hazards Models; Research Design; Retrospective Studies; Risk Assessment; Risk Factors; Sulfonylurea Compounds; Tolbutamide | 2013 |
Effects of a sitagliptin safety alert on prescription behaviour for oral antihyperglycaemic drugs: a propensity score-matched cohort study of prescription receipt data in Japan.
Topics: Aged; Cohort Studies; Female; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Japan; Logistic Models; Male; Middle Aged; Patient Safety; Practice Patterns, Physicians'; Propensity Score; Pyrazines; Sitagliptin Phosphate; Sulfonylurea Compounds; Triazoles | 2013 |
Risk of acute coronary events associated with glyburide compared with gliclazide use in patients with type 2 diabetes: a nested case-control study.
Topics: Acute Coronary Syndrome; Aged; Alberta; Case-Control Studies; Cohort Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Odds Ratio; Risk Assessment; Risk Factors; Sulfonylurea Compounds; Treatment Outcome | 2014 |
Evaluation approach can significantly influence oral glucose-lowering drugs total mortality risks in retrospective cohorts of type 2 diabetes mellitus patients.
Topics: Diabetes Mellitus, Type 2; Gliclazide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Metformin; Registries; Retrospective Studies; Risk Factors; Treatment Outcome; Ukraine | 2014 |
Fast and Simultaneous Analysis of Combined Anti-Diabetic Drugs by Capillary Zone Electrophoresis.
Topics: Drug Combinations; Electrophoresis, Capillary; Gliclazide; Glyburide; Hypoglycemic Agents; Limit of Detection; Linear Models; Metformin; Reproducibility of Results; Tablets | 2015 |
Metformin in combination with various insulin secretagogues in type 2 diabetes and associated risk of cardiovascular morbidity and mortality--a retrospective nationwide study.
Topics: Aged; Carbamates; Cardiovascular Diseases; Denmark; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Male; Metformin; Middle Aged; Morbidity; Myocardial Infarction; Piperidines; Registries; Retrospective Studies; Risk Factors; Stroke; Sulfonylurea Compounds; Tolbutamide | 2015 |
Comparative cardiovascular safety of insulin secretagogues following hospitalization for ischemic heart disease among type 2 diabetes patients: a cohort study.
Topics: Aged; Aged, 80 and over; Alberta; Blue Cross Blue Shield Insurance Plans; Carbamates; Cardiovascular Diseases; Cohort Studies; Databases, Factual; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Diabetic Cardiomyopathies; Female; Gliclazide; Glyburide; Hospitalization; Humans; Hypoglycemic Agents; Male; Myocardial Ischemia; Piperidines; Proportional Hazards Models; Retrospective Studies; Risk; Universal Health Insurance | 2015 |
The Hypoglycemic Risk of Glyburide (Glibenclamide) Compared with Modified-Release Gliclazide.
Topics: Aged; Aged, 80 and over; Cohort Studies; Delayed-Action Preparations; Diabetes Mellitus, Type 2; Female; Gliclazide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Ontario; Population Surveillance; Retrospective Studies; Risk Factors | 2015 |
Dose-response relationship between sulfonylureas and major adverse cardiovascular events in elderly patients with type 2 diabetes.
Topics: Aged; Aged, 80 and over; Cardiovascular Diseases; Cohort Studies; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Follow-Up Studies; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Male; Propensity Score; Proportional Hazards Models; Retrospective Studies; Sulfonylurea Compounds; Time Factors | 2016 |
[Effects of different sulfonylureas on the warm-up phenomenon in diabetes patients with coronary artery disease].
Topics: Angina Pectoris; Coronary Angiography; Coronary Artery Disease; Diabetes Complications; Diabetes Mellitus; Electrocardiography; Exercise Test; Gliclazide; Glyburide; Humans; Hypoglycemic Agents | 2017 |
Binding of sulphonylureas to plasma proteins - A KATP channel perspective.
Topics: Animals; Cattle; Cells, Cultured; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin-Secreting Cells; KATP Channels; Mice; Mice, Inbred C57BL; Oocytes; Patch-Clamp Techniques; Protein Binding; Recombinant Proteins; Serum Albumin; Serum Albumin, Bovine; Xenopus laevis | 2018 |
Different sulfonylureas induce the apoptosis of proximal tubular epithelial cell differently via closing K
Topics: Apoptosis; Cell Line; Epithelial Cells; Gliclazide; Glyburide; Humans; KATP Channels; Kidney Tubules, Proximal; Sulfonylurea Compounds | 2018 |
Comparison of mortality and cardiovascular event risk associated with various insulin secretagogues: A nationwide real-world analysis.
Topics: Aged; Carbamates; Cardiovascular Diseases; Cohort Studies; Diabetes Mellitus, Type 2; Diabetic Angiopathies; Female; Follow-Up Studies; Gliclazide; Glipizide; Glyburide; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Male; Middle Aged; Mortality; Piperidines; Secretagogues; Sulfonylurea Compounds; Taiwan | 2019 |
Effect of berberine on in vitro metabolism of sulfonylureas: A herb-drug interactions study.
Topics: Animals; Berberine; Chromatography, Liquid; Cytochrome P-450 Enzyme System; Female; Gliclazide; Glyburide; Herb-Drug Interactions; Male; Mass Spectrometry; Microsomes, Liver; Rats; Sulfonylurea Compounds | 2020 |
The Effect of CYP2C9 Genotype Variants in Type 2 Diabetes on the Pharmacological Effectiveness of Sulfonylureas, Diabetic Retinopathy, and Nephropathy.
Topics: Biomarkers; Blood Glucose; Cytochrome P-450 CYP2C9; Diabetes Mellitus, Type 2; Diabetic Nephropathies; Diabetic Retinopathy; Female; Gene Frequency; Gliclazide; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Male; Middle Aged; Pharmacogenomic Variants; Risk Factors; Treatment Outcome | 2020 |
Studies of binding by sulfonylureas with glyoxal- and methylglyoxal-modified albumin by immunoextraction using affinity microcolumns.
Topics: Adsorption; Antibodies; Chromatography, Affinity; Drug Interactions; Gliclazide; Glyburide; Glycation End Products, Advanced; Glycosylation; Glyoxal; Humans; Kinetics; Protein Binding; Protein Stability; Pyruvaldehyde; Serum Albumin, Human; Sulfonylurea Compounds; Warfarin | 2021 |
Sensitive detection of antidiabetic compounds and one degradation product in wastewater samples by a new SPE-LC-MS/MS method.
Topics: Chromatography, Liquid; Environmental Monitoring; Gliclazide; Glipizide; Glyburide; Hypoglycemic Agents; Metformin; Reproducibility of Results; Solid Phase Extraction; Sulfonylurea Compounds; Tandem Mass Spectrometry; Wastewater; Water Pollutants, Chemical | 2021 |
Crude extract from
Topics: Alloxan; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Euphorbia; Gliclazide; Glyburide; Hypoglycemic Agents; Insulin; Metformin; Plant Extracts; Rats | 2023 |
Analytical Method Capable of Quantifying Eight Nitrosamine Impurities from Five Different Commercially Available Metformin Formulations with Glipizide, Glibenclamide, Gliclazide, Evogliptin, and Glimepiride by Ultra High Performance Liquid Chromatography
Topics: Chromatography, High Pressure Liquid; Chromatography, Liquid; Diabetes Mellitus, Type 2; Gliclazide; Glipizide; Glyburide; Humans; Metformin; Nitrosamines; Pharmaceutical Preparations; Tandem Mass Spectrometry | 2023 |
[Characteristics of purchases of hypoglycemic agents in pharmacy retail sector in 2016-2020 years dynamics].
Topics: Dipeptidyl Peptidase 4; Gliclazide; Glyburide; Humans; Hypoglycemic Agents; Metformin; Pharmacies; Pharmacy | 2023 |
Hyperpolarisation of rat mesenteric endothelial cells by ATP-sensitive K(+) channel openers.
Topics: Adenosine Triphosphate; Animals; Apamin; Barium Compounds; Benzimidazoles; Carbachol; Charybdotoxin; Chlorides; Cromakalim; Dose-Response Relationship, Drug; Electrophysiology; Endothelium, Vascular; Glyburide; Glycyrrhetinic Acid; In Vitro Techniques; Male; Membrane Potentials; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Ouabain; Potassium Channels; Rats; Rats, Wistar; Vasodilator Agents | 2000 |
Endothelium-derived relaxing factor-mediated vasodilation in mouse mesenteric vascular beds.
Topics: Acetylcholine; Animals; Biological Factors; Calcimycin; Calcium Ionophores; Cyclooxygenase Inhibitors; Endothelium-Dependent Relaxing Factors; Endothelium, Vascular; Enzyme Inhibitors; Gap Junctions; Glyburide; Glycyrrhetinic Acid; Indomethacin; Male; Mesenteric Arteries; Mice; Mice, Inbred C57BL; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitroprusside; Potassium Channel Blockers; Tetraethylammonium; Vasodilation; Vasodilator Agents | 2012 |