Page last updated: 2024-08-23

gestrinone and tetrahydrogestrinone

gestrinone has been researched along with tetrahydrogestrinone in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's25 (92.59)29.6817
2010's2 (7.41)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kondro, W1
Knight, J1
Czap, A1
Ashley, S1
Death, AK; Handelsman, DJ; Kazlauskas, R; McGrath, KC1
Ahrens, BD; Catlin, DH; Chang, YC; Hatton, CK; Sekera, MH; Starcevic, B1
Foster, ZJ; Housner, JA1
Belleau, P; Calvo, E; Cloutier, J; Gauthier, S; Labrie, C; Labrie, F; Lévesque, MH; Luu-The, V; Martel, C; Morissette, J1
Berthelette, C; Chauret, N; Lévesque, JF; Templeton, E; Trimble, L1
Erickson, BE1
Artaza, JN; Baker, M; Bhasin, S; Catlin, DH; Chandsawangbhuwana, C; Chang, YC; Datta, G; Herbst, KL; Jasuja, R; Miller, A; Sarkissian, A; Singh, R; Starcevic, B1
Armsey, TD; Malvey, TC1
Dhar, R; Estes, NA; Homoud, MK; Link, MS; Stout, CW; Weinstock, J1
Diel, P; Friedel, A; Geyer, H; Kamber, M; Laudenbach-Leschowsky, U; Schänzer, W; Thevis, M; Vollmer, G; Zierau, O1
Bovee, TF; Hamers, AR; Hoogenboom, LR; Nielen, MW; Rutgers, P; van Engelen, MC; van Rhijn, JH1
Blanchet, J; Breton, R; Cantin, L; Côté, PL; Labrie, F; Pereira de Jésus-Tran, K1
Calvo, E; Chernomoretz, A; Labrie, C; Labrie, F; Luu-The, V; Martel, C; Morissette, J1
de Aquino Neto, FR; Marques, MA; Padilha, MC; Pereira, HM1
Georgakopoulus, C; Nielen, MW; Touber, ME; van Engelen, MC; van Rhijn, JA1
Marco, MP; Salvador, JP; Sanchez-Baeza, F1
Bolt, HM; Degen, GH; Diel, P; Dorn, SB; Thevis, M1
Diel, P; Lehmann, S; Schänzer, W; Vollmer, G; Zierau, O1
Düe, M; Gerlach, M; Guddat, S; Kietzmann, M; Machnik, M; Niedorf, F; Schänzer, W; Schenk, I; Thevis, M1
Georgakopoulus, C; Nielen, MW; Peters, RJ; Touber, ME; van Engelen, MC1
Neto, FR; Padilha, MC; Pereira, HM1
Kim, SH; Moon, HY; Ryu, SH; Suh, PG1
Miller, S1

Reviews

2 review(s) available for gestrinone and tetrahydrogestrinone

ArticleYear
Anabolic-androgenic steroids and testosterone precursors: ergogenic aids and sport.
    Current sports medicine reports, 2004, Volume: 3, Issue:4

    Topics: Anabolic Agents; Androgens; Androstenedione; Animals; Body Composition; Dietary Supplements; Doping in Sports; Gestrinone; Humans; Muscle, Skeletal; Substance Abuse Detection

2004
Cardiovascular toxicities of performance-enhancing substances in sports.
    Mayo Clinic proceedings, 2005, Volume: 80, Issue:10

    Topics: Androstenedione; Caffeine; Cardiovascular System; Central Nervous System Stimulants; Dietary Supplements; Doping in Sports; Ephedra; Gestrinone; Humans; Male

2005

Other Studies

25 other study(ies) available for gestrinone and tetrahydrogestrinone

ArticleYear
Athletes' "designer steroid" leads to widening scandal.
    Lancet (London, England), 2003, Nov-01, Volume: 362, Issue:9394

    Topics: Anabolic Agents; Crime; Designer Drugs; Dietary Supplements; Doping in Sports; Fraud; Gestrinone; Humans; Male; Substance Abuse Detection

2003
Drugs in sport: no dope.
    Nature, 2003, Nov-13, Volume: 426, Issue:6963

    Topics: Doping in Sports; Gestrinone; Humans; Mass Spectrometry; Urinalysis

2003
"Fish on Steroids"?
    Alternative medicine review : a journal of clinical therapeutic, 2003, Volume: 8, Issue:4

    Topics: California; Dietary Supplements; Gestrinone; Humans; Legislation, Food; Sports

2003
Doping by design.
    Scientific American, 2004, Volume: 290, Issue:2

    Topics: Doping in Sports; Gestrinone; Humans; Substance Abuse Detection

2004
Tetrahydrogestrinone is a potent androgen and progestin.
    The Journal of clinical endocrinology and metabolism, 2004, Volume: 89, Issue:5

    Topics: Androgens; Biological Assay; Dose-Response Relationship, Drug; Gestrinone; Humans; Nandrolone; Progestins; Receptors, Androgen; Receptors, Estrogen; Receptors, Progesterone; Transcriptional Activation; Trenbolone Acetate; Yeasts

2004
Tetrahydrogestrinone: discovery, synthesis, and detection in urine.
    Rapid communications in mass spectrometry : RCM, 2004, Volume: 18, Issue:12

    Topics: Animals; Doping in Sports; Gas Chromatography-Mass Spectrometry; Gestrinone; Humans; Magnetic Resonance Spectroscopy; Male; Papio; Spectrometry, Mass, Electrospray Ionization; Spectrum Analysis

2004
Tetrahydrogestrinone induces a genomic signature typical of a potent anabolic steroid.
    The Journal of endocrinology, 2005, Volume: 184, Issue:2

    Topics: Anabolic Agents; Animals; Binding, Competitive; Cell Line; Dihydrotestosterone; Doping in Sports; Gene Expression; Gene Expression Profiling; Gestrinone; Humans; Kidney; Male; Metribolone; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Oligonucleotide Array Sequence Analysis; Prostate; Protein Binding; Random Allocation; Receptors, Androgen; Testosterone

2005
Discovery, biosynthesis, and structure elucidation of metabolites of a doping agent and a direct analogue, tetrahydrogestrinone and gestrinone, using human hepatocytes.
    Analytical chemistry, 2005, May-15, Volume: 77, Issue:10

    Topics: Anabolic Agents; Biomarkers; Chromatography, High Pressure Liquid; Doping in Sports; Gestrinone; Glucuronic Acid; Glycoconjugates; Hepatocytes; Humans; Hydroxylation; Magnetic Resonance Spectroscopy; Mass Spectrometry; Oxidation-Reduction; Receptors, Antigen, T-Cell

2005
Detecting doping.
    Analytical chemistry, 2005, Jun-01, Volume: 77, Issue:11

    Topics: Doping in Sports; Ephedrine; Filtration; Gestrinone; Hepatocytes; Humans; Membranes, Artificial; Sensitivity and Specificity

2005
Tetrahydrogestrinone is an androgenic steroid that stimulates androgen receptor-mediated, myogenic differentiation in C3H10T1/2 multipotent mesenchymal cells and promotes muscle accretion in orchidectomized male rats.
    Endocrinology, 2005, Volume: 146, Issue:10

    Topics: Animals; Cell Differentiation; Cells, Cultured; Gestrinone; Male; Mesoderm; Mice; Muscle, Skeletal; Orchiectomy; Rats; Receptors, Androgen

2005
Tetrahydrogestrinone: the discovery of a designer steroid.
    Current sports medicine reports, 2005, Volume: 4, Issue:4

    Topics: Anabolic Agents; Designer Drugs; Doping in Sports; Gestrinone; History, 21st Century; Humans; Sports Medicine; United States

2005
Tetrahydrogestrinone is a potent but unselective binding steroid and affects glucocorticoid signalling in the liver.
    Toxicology letters, 2006, Jun-20, Volume: 164, Issue:1

    Topics: Anabolic Agents; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Gene Expression; Gestrinone; Humans; Liver; Male; Molecular Structure; Muscle, Smooth; Orchiectomy; Organ Size; Prostate; Radioligand Assay; Rats; Rats, Wistar; Receptors, Androgen; Receptors, Glucocorticoid; Seminal Vesicles; Signal Transduction; Yeasts

2006
Urine testing for designer steroids by liquid chromatography with androgen bioassay detection and electrospray quadrupole time-of-flight mass spectrometry identification.
    Analytical chemistry, 2006, Jan-15, Volume: 78, Issue:2

    Topics: Anabolic Agents; Androgens; Biological Assay; Chromatography, Liquid; Designer Drugs; Doping in Sports; Female; Gestrinone; Humans; Male; Spectrometry, Mass, Electrospray Ionization; Substance Abuse Detection

2006
Comparison of crystal structures of human androgen receptor ligand-binding domain complexed with various agonists reveals molecular determinants responsible for binding affinity.
    Protein science : a publication of the Protein Society, 2006, Volume: 15, Issue:5

    Topics: Androgen Antagonists; Androgens; Binding Sites; Crystallization; Crystallography, X-Ray; Dihydrotestosterone; Gestrinone; Humans; Hydrogen Bonding; Ligands; Molecular Structure; Multiprotein Complexes; Protein Binding; Protein Structure, Tertiary; Receptors, Androgen; Testosterone

2006
Dehydroepiandrosterone (DHEA) is an anabolic steroid like dihydrotestosterone (DHT), the most potent natural androgen, and tetrahydrogestrinone (THG).
    The Journal of steroid biochemistry and molecular biology, 2006, Volume: 100, Issue:1-3

    Topics: Anabolic Agents; Androgens; Animals; Animals, Outbred Strains; Crosses, Genetic; Dehydroepiandrosterone; Dihydrotestosterone; Dose-Response Relationship, Drug; Gene Expression Profiling; Genome; Gestrinone; Male; Mice; Mice, Inbred C57BL; Models, Biological; Oligonucleotide Array Sequence Analysis; Orchiectomy; Organ Size; Prostate; Seminal Vesicles; Time Factors

2006
Analysis of synthetic 19-norsteroids trenbolone, tetrahydrogestrinone and gestrinone by gas chromatography-mass spectrometry.
    Journal of chromatography. A, 2007, May-25, Volume: 1150, Issue:1-2

    Topics: Adult; Female; Gas Chromatography-Mass Spectrometry; Gestrinone; Humans; Molecular Structure; Reproducibility of Results; Trenbolone Acetate

2007
Multi-detection of corticosteroids in sports doping and veterinary control using high-resolution liquid chromatography/time-of-flight mass spectrometry.
    Analytica chimica acta, 2007, Mar-14, Volume: 586, Issue:1-2

    Topics: Adrenal Cortex Hormones; Animals; Cattle; Chromatography, Liquid; Designer Drugs; Doping in Sports; Ethanolamines; Formoterol Fumarate; Gestrinone; Humans; Mass Spectrometry; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Substance Abuse Detection; Urinalysis; Veterinary Medicine

2007
Preparation of antibodies for the designer steroid tetrahydrogestrinone and development of an enzyme-linked immunosorbent assay for human urine analysis.
    Analytical chemistry, 2007, May-15, Volume: 79, Issue:10

    Topics: Antibodies; Gestrinone; Haptens; Humans; Sensitivity and Specificity; Urinalysis

2007
Induction of micronuclei in V79 cells by the anabolic doping steroids tetrahydrogestrinone and trenbolone.
    Archives of toxicology, 2008, Volume: 82, Issue:4

    Topics: Anabolic Agents; Animals; Cell Cycle; Cell Line; Cell Survival; Cricetinae; Dose-Response Relationship, Drug; Gestrinone; Micronuclei, Chromosome-Defective; Micronucleus Tests; Trenbolone Acetate

2008
Detection of anabolic steroid abuse using a yeast transactivation system.
    Steroids, 2008, Volume: 73, Issue:11

    Topics: Anabolic Agents; Androgens; beta-Galactosidase; Biological Assay; Designer Drugs; Dihydrotestosterone; Dose-Response Relationship, Drug; Genes, Reporter; Gestrinone; Humans; Male; Norpregnenes; Receptors, Androgen; Saccharomyces cerevisiae; Sensitivity and Specificity; Substance Abuse Detection; Testosterone; Transcriptional Activation

2008
Detection and pharmacokinetics of tetrahydrogestrinone in horses.
    Journal of veterinary pharmacology and therapeutics, 2009, Volume: 32, Issue:2

    Topics: Animals; Doping in Sports; Gas Chromatography-Mass Spectrometry; Gestrinone; Half-Life; Horses; Male; Substance Abuse Detection; Tandem Mass Spectrometry

2009
Searching for in silico predicted metabolites and designer modifications of (cortico)steroids in urine by high-resolution liquid chromatography/time-of-flight mass spectrometry.
    Rapid communications in mass spectrometry : RCM, 2009, Volume: 23, Issue:15

    Topics: Chromatography, Liquid; Gestrinone; Glucocorticoids; Humans; Mass Spectrometry; Software; Substance Abuse Detection

2009
Tetrahydrogestrinone analysis and designer steroids revisited.
    Bioanalysis, 2009, Volume: 1, Issue:8

    Topics: Anabolic Agents; Chemistry Techniques, Analytical; Designer Drugs; Dietary Supplements; Doping in Sports; Gestrinone; Humans; Substance Abuse Detection; Veterinary Drugs

2009
The androgenic anabolic steroid tetrahydrogestrinone produces dioxin-like effects via the aryl hydrocarbon receptor.
    Toxicology in vitro : an international journal published in association with BIBRA, 2012, Volume: 26, Issue:7

    Topics: Azo Compounds; Cytochrome P-450 CYP1A1; Dioxins; Gene Expression Regulation, Enzymologic; Genes, Reporter; Gestrinone; Hep G2 Cells; Hepatocytes; Humans; Luciferases; Pyrazoles; Receptors, Aryl Hydrocarbon; Response Elements; RNA, Messenger

2012
New ELISA bulks up detection ability of steroid screening methods.
    Bioanalysis, 2012, Volume: 4, Issue:10

    Topics: Anabolic Agents; Androgens; Doping in Sports; Enzyme-Linked Immunosorbent Assay; Gestrinone; Humans; Limit of Detection; Serum; Stanozolol; Steroids; Testosterone; Time Factors

2012