Page last updated: 2024-08-23

gepirone and kampirone

gepirone has been researched along with kampirone in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19909 (56.25)18.7374
1990's5 (31.25)18.2507
2000's2 (12.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA; Lyon, RA; Naiman, NA; Titeler, M1
Balster, RL1
Engel, JA; Hjorth, S; Söderpalm, B1
Dixon, V; Gage-White, D; Guthrie, D; Matheson, GK; Rhoades, J; White, G1
Eison, MS; Matheson, GK1
Caccia, S; Fong, MH; Guiso, G1
Le Moal, M; Louilot, A; Simon, H1
Bianchi, G; Caccia, S; Della Vedova, F; Garattini, S1
Bianchi, G; Caccia, S1
Skolnick, P; Weissman, BA; Youdim, MB1
Cullen, WK; Rowan, MJ1
Farmen, RH; Pittman, KA; Sciacca, MA; Sostrin, MB; Tay, LK1
Fabre, LF; Fogelman, SM; Granda, BW; Grassi, JM; Greenblatt, DJ; Harmatz, JS; Kramer, SJ; Shader, RI; von Moltke, LL1
Olivares, E; Tripathi, B; Turek, FW; Van Reeth, O; Zhang, Y1
Garteiz, DA; Giancarlo, GM; Greenblatt, DJ; Von Moltke, LL1
Sitsen, JM; Timmer, CJ1

Reviews

1 review(s) available for gepirone and kampirone

ArticleYear
Abuse potential of buspirone and related drugs.
    Journal of clinical psychopharmacology, 1990, Volume: 10, Issue:3 Suppl

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Clinical Trials as Topic; Double-Blind Method; Drug Evaluation, Preclinical; Euphoria; Humans; Product Surveillance, Postmarketing; Pyrimidines; Rats; Substance-Related Disorders

1990

Trials

3 trial(s) available for gepirone and kampirone

ArticleYear
Abuse potential of buspirone and related drugs.
    Journal of clinical psychopharmacology, 1990, Volume: 10, Issue:3 Suppl

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Clinical Trials as Topic; Double-Blind Method; Drug Evaluation, Preclinical; Euphoria; Humans; Product Surveillance, Postmarketing; Pyrimidines; Rats; Substance-Related Disorders

1990
Effect of food on the bioavailability of gepirone in humans.
    Journal of clinical pharmacology, 1993, Volume: 33, Issue:7

    Topics: Administration, Oral; Adolescent; Adult; Anti-Anxiety Agents; Antidepressive Agents; Biological Availability; Buspirone; Fasting; Food; Humans; Male; Pyrimidines

1993
Pharmacokinetic evaluation of gepirone immediate-release capsules and gepirone extended-release tablets in healthy volunteers.
    Journal of pharmaceutical sciences, 2003, Volume: 92, Issue:9

    Topics: Adult; Area Under Curve; Biological Availability; Buspirone; Capsules; Cross-Over Studies; Delayed-Action Preparations; Half-Life; Humans; Intestinal Absorption; Male; Pyrimidines; Serotonin Receptor Agonists; Tablets; Time Factors

2003

Other Studies

13 other study(ies) available for gepirone and kampirone

ArticleYear
Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:10

    Topics: Animals; Chemical Phenomena; Chemistry; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Structure-Activity Relationship

1988
Effects of 5-HT1A receptor agonists and L-5-HTP in Montgomery's conflict test.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:1

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Buspirone; Conflict, Psychological; Male; Motor Activity; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tetrahydronaphthalenes

1989
The effects of gepirone and 1-(2-pyrimidinyl)-piperazine on levels of corticosterone in rat plasma.
    Neuropharmacology, 1989, Volume: 28, Issue:4

    Topics: Animals; Buspirone; Circadian Rhythm; Corticosterone; Dose-Response Relationship, Drug; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pyrimidines; Rats; Rats, Inbred Strains; Stress, Physiological

1989
The effects of buspirone, BMY-13805 and 1-(2-pyrimidinyl)-piperazine on cat spinal reflexes.
    Methods and findings in experimental and clinical pharmacology, 1985, Volume: 7, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Cats; Female; Ganglia, Spinal; Male; Piperazines; Pyrimidines; Reflex; Reflex, Monosynaptic; Spinal Cord

1985
Disposition of the psychotropic drugs buspirone, MJ-13805 and piribedil, and of their common active metabolite 1-(2-pyrimidinyl)-piperazine in the rat.
    Xenobiotica; the fate of foreign compounds in biological systems, 1985, Volume: 15, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Blood Proteins; Brain; Buspirone; Kinetics; Male; Piperazines; Piribedil; Protein Binding; Pyrimidines; Rats; Rats, Inbred Strains

1985
A study of the effects of buspirone, BMY 13805, and 1-PP on dopaminergic metabolism in the nucleus accumbens using in vivo voltammetry in freely moving rats.
    Life sciences, 1986, Aug-25, Volume: 39, Issue:8

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anti-Anxiety Agents; Buspirone; Dopamine; Electrochemistry; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Nucleus Accumbens; Piperazines; Pyrimidines; Rats; Rats, Inbred Strains; Septal Nuclei

1986
The alpha 2-adrenoceptor antagonist activity of ipsapirone and gepirone is mediated by their common metabolite 1-(2-pyrimidinyl)-piperazine (PmP).
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Animals; Anti-Anxiety Agents; Buspirone; Chromatography, High Pressure Liquid; Clonidine; Drug Interactions; Gastrointestinal Transit; Injections, Intravenous; Male; Pyrimidines; Rats

1988
Simultaneous determination of buspirone, gepirone, ipsapirone and their common metabolite 1-(2-pyrimidinyl)piperazine in rat plasma and brain by high-performance liquid chromatography.
    Journal of chromatography, 1988, Oct-14, Volume: 431, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Brain Chemistry; Buspirone; Male; Pyrimidines; Rats; Spectrophotometry, Ultraviolet

1988
Monoaminergic involvement in the pharmacological actions of buspirone.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Apomorphine; Behavior, Animal; Brain; Buspirone; Dopamine; Ketanserin; Male; Methoxydimethyltryptamines; Monoamine Oxidase; p-Chloroamphetamine; Piperazines; Piperidines; Psychotropic Drugs; Pyrimidines; Rats; Serotonin

1985
Gepirone and 1-(2-pyrimidinyl)-piperazine-induced reduction of aversively evoked ultrasonic vocalisation in the rat.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Buspirone; Darkness; Electroshock; Light; Male; Motor Activity; Proadifen; Pyrimidines; Rats; Rats, Wistar; Ultrasonics; Vocalization, Animal

1994
Gepirone and 1-(2-pyrimidinyl)-piperazine in vitro: human cytochromes mediating transformation and cytochrome inhibitory effects.
    Psychopharmacology, 1998, Volume: 140, Issue:3

    Topics: Antidepressive Agents; Biotransformation; Buspirone; Cytochrome P-450 Enzyme System; Drug Interactions; Humans; Ketoconazole; Microsomes, Liver; Pyrimidines

1998
Chronobiotic effects of gepirone, a potential antidepressant with 5HT1A receptor partial agonist properties.
    Behavioural pharmacology, 1999, Volume: 10, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Buspirone; Circadian Rhythm; Cricetinae; Darkness; Light; Male; Mesocricetus; Motor Activity; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1999
Human cytochromes mediating gepirone biotransformation at low substrate concentrations.
    Biopharmaceutics & drug disposition, 2003, Volume: 24, Issue:2

    Topics: Biotransformation; Buspirone; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Gas Chromatography-Mass Spectrometry; Humans; In Vitro Techniques; Microsomes, Liver; Piperidones; Pyrimidines; Serotonin Receptor Agonists

2003