Page last updated: 2024-09-03

gefitinib and xav939

gefitinib has been researched along with xav939 in 2 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(xav939)
Trials
(xav939)
Recent Studies (post-2010) (xav939)
5,2315662,9191860179

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)xav939 (IC50)
Chain A, Tankyrase-1Homo sapiens (human)0.011
Chain A, Tankyrase-1Homo sapiens (human)0.011
Poly [ADP-ribose] polymerase tankyrase-1Homo sapiens (human)0.0656
Poly [ADP-ribose] polymerase 1Homo sapiens (human)0.9968
Protein Wnt-3aMus musculus (house mouse)0.078
Protein Wnt-3aHomo sapiens (human)0.078
Protein mono-ADP-ribosyltransferase PARP14Homo sapiens (human)5.8942
Vesicular acetylcholine transporterRattus norvegicus (Norway rat)0.015
Poly [ADP-ribose] polymerase tankyrase-2Homo sapiens (human)0.052
Poly [ADP-ribose] polymerase 2Homo sapiens (human)0.0792
Protein mono-ADP-ribosyltransferase PARP4Homo sapiens (human)4.3776
Protein mono-ADP-ribosyltransferase PARP3Homo sapiens (human)0.8354

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Fang, D; Li, HY; Liang, C; Liu, FY; Niu, J; Sun, H; Wang, X; Xie, SQ; Zhang, YD1

Other Studies

2 other study(ies) available for gefitinib and xav939

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Suppression of epidermal growth factor receptor-mediated β-catenin nuclear accumulation enhances the anti-tumor activity of phosphoinositide 3-kinase inhibitor in breast cancer.
    Cell biology international, 2019, Volume: 43, Issue:8

    Topics: Antineoplastic Combined Chemotherapy Protocols; beta Catenin; Breast Neoplasms; Cell Proliferation; Chromones; Drug Resistance, Neoplasm; ErbB Receptors; Female; Gefitinib; Heterocyclic Compounds, 3-Ring; Humans; MCF-7 Cells; Morpholines; Phosphoinositide-3 Kinase Inhibitors

2019