Page last updated: 2024-09-03

gefitinib and su 6656

gefitinib has been researched along with su 6656 in 3 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(su 6656)
Trials
(su 6656)
Recent Studies (post-2010) (su 6656)
5,2315662,919154073

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)su 6656 (IC50)
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.1
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)0.15
Tyrosine-protein kinase FynHomo sapiens (human)0.17
Tyrosine-protein kinase YesHomo sapiens (human)0.02
Tyrosine-protein kinase LynHomo sapiens (human)0.13
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)0.77
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.1765
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)8.7
Serine/threonine-protein kinase 3Homo sapiens (human)0.11
Serine/threonine-protein kinase BRSK2Homo sapiens (human)0.1
Aurora kinase BHomo sapiens (human)0.019
ALK tyrosine kinase receptorHomo sapiens (human)0.85
Aurora kinase CHomo sapiens (human)0.017

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Lin, J; Shen, W; Sun, J; Xue, J; Zhang, C; Zhang, X1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

3 other study(ies) available for gefitinib and su 6656

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Novel oxazolo[4,5-g]quinazolin-2(1H)-ones: dual inhibitors of EGFR and Src protein tyrosine kinases.
    European journal of medicinal chemistry, 2012, Volume: 55

    Topics: Cell Line, Tumor; Cell Proliferation; ErbB Receptors; Humans; Molecular Docking Simulation; Protein Conformation; Protein Kinase Inhibitors; Quinazolines; src-Family Kinases

2012
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013