Page last updated: 2024-09-03

gefitinib and rabeprazole

gefitinib has been researched along with rabeprazole in 3 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(rabeprazole)
Trials
(rabeprazole)
Recent Studies (post-2010) (rabeprazole)
5,2315662,9191,073446405

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)rabeprazole (IC50)
Adenosine receptor A3Homo sapiens (human)3.219
Urease subunit alphaHelicobacter pylori 266950.29
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)3.219
Alpha-2B adrenergic receptorHomo sapiens (human)1.737
D(3) dopamine receptorHomo sapiens (human)2.326
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)3.219
WD repeat-containing protein 5Homo sapiens (human)0.49
Urease subunit betaHelicobacter pylori 266950.29
Histone-lysine N-methyltransferase 2AHomo sapiens (human)0.49
NAD(+) hydrolase SARM1Homo sapiens (human)3.25
Cytosolic endo-beta-N-acetylglucosaminidaseHomo sapiens (human)4.47
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)8.5

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Delabio, LC; Dutra, JP; Hembecker, M; Kita, DH; Moure, VR; Pereira, GDS; Scheiffer, G; Valdameri, G; Zattoni, IF1

Reviews

2 review(s) available for gefitinib and rabeprazole

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators.
    European journal of medicinal chemistry, 2022, Jul-05, Volume: 237

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Breast Neoplasms; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Neoplasm Proteins; Neoplastic Stem Cells

2022

Other Studies

1 other study(ies) available for gefitinib and rabeprazole

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008