Page last updated: 2024-09-03

gefitinib and oxadiazoles

gefitinib has been researched along with oxadiazoles in 4 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(oxadiazoles)
Trials
(oxadiazoles)
Recent Studies (post-2010) (oxadiazoles)
5,2315662,9196,0572572,359

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Ding, K; Han, C; Huang, Z; Ji, H; Lai, Y; Peng, S; Wan, L; Zhang, Y1
He, C; He, J; Wei, S; Xie, M1
An, YJ; Choi, SY; Im, JH; Jeong, BH; Kang, KW; Kim, SY; Kim, YG; Lee, JS; Park, S1
Altelaar, M; Iskit, S; Peeper, DS; Rontogianni, S; van Doorn, S1

Other Studies

4 other study(ies) available for gefitinib and oxadiazoles

ArticleYear
Synthesis and evaluation of 2-anilinopyrimidines bearing 3-aminopropamides as potential epidermal growth factor receptor inhibitors.
    European journal of medicinal chemistry, 2014, Apr-22, Volume: 77

    Topics: Antineoplastic Agents; Cell Line; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; ErbB Receptors; Gefitinib; Humans; Molecular Structure; Nitric Oxide; Oxadiazoles; Pyrimidines; Quinazolines; Signal Transduction; Structure-Activity Relationship

2014
γ Secretase inhibitor BMS-708163 reverses resistance to EGFR inhibitor via the PI3K/Akt pathway in lung cancer.
    Journal of cellular biochemistry, 2015, Volume: 116, Issue:6

    Topics: Amyloid Precursor Protein Secretases; Animals; Apoptosis; Cell Line, Tumor; Cell Survival; ErbB Receptors; Female; Gefitinib; Immunohistochemistry; Lung Neoplasms; Mice; Mice, Inbred BALB C; Oxadiazoles; Phosphatidylinositol 3-Kinases; Proto-Oncogene Proteins c-akt; Quinazolines; Sulfonamides

2015
GPR119 agonist enhances gefitinib responsiveness through lactate-mediated inhibition of autophagy.
    Journal of experimental & clinical cancer research : CR, 2018, Nov-29, Volume: 37, Issue:1

    Topics: Animals; Autophagy; Breast Neoplasms; Cell Line, Tumor; Drug Synergism; Female; Gefitinib; Humans; Lactic Acid; MCF-7 Cells; Mesylates; Mice, Inbred BALB C; Mice, Nude; Oxadiazoles; Receptors, G-Protein-Coupled; Tetrazoles; Thiazoles; Transfection

2018
Combined EGFR and ROCK Inhibition in Triple-negative Breast Cancer Leads to Cell Death Via Impaired Autophagic Flux.
    Molecular & cellular proteomics : MCP, 2020, Volume: 19, Issue:2

    Topics: Antineoplastic Agents; Autophagy; Cell Death; Cell Line, Tumor; ErbB Receptors; Female; Gefitinib; Humans; Imidazoles; Mass Spectrometry; Oxadiazoles; Protein Kinase Inhibitors; Proteomics; rho-Associated Kinases; Triple Negative Breast Neoplasms

2020