Page last updated: 2024-09-03

gefitinib and npi 2358

gefitinib has been researched along with npi 2358 in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(npi 2358)
Trials
(npi 2358)
Recent Studies (post-2010) (npi 2358)
5,2315662,91936431

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)npi 2358 (IC50)
Tubulin alpha-1A chainSus scrofa (pig)1.8
Tubulin beta chainSus scrofa (pig)1.8
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)8.9
Mitogen-activated protein kinase 10Rattus norvegicus (Norway rat)6.8
Tubulin beta-2B chainBos taurus (cattle)2.4
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)2.4
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)2.4

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cheng, H; Deng, M; Ding, Z; Dou, G; Hou, Y; Li, F; Li, W; Ma, M; Zhao, J1

Other Studies

1 other study(ies) available for gefitinib and npi 2358

ArticleYear
In vitro and in vivo pharmacokinetic and pharmacodynamic study of MBRI-001, a deuterium-substituted plinabulin derivative as a potent anti-cancer agent.
    Bioorganic & medicinal chemistry, 2018, 09-01, Volume: 26, Issue:16

    Topics: Animals; Antineoplastic Agents; Blood Proteins; Cell Line, Tumor; Cytochrome P-450 Enzyme System; Deuterium; Diketopiperazines; Female; Half-Life; Humans; Inhibitory Concentration 50; Male; Mice; Mice, Inbred BALB C; Microsomes, Liver; Neoplasms; Protein Binding; Rats; Rats, Wistar; Tissue Distribution

2018