Page last updated: 2024-09-03

gefitinib and nafamostat

gefitinib has been researched along with nafamostat in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(nafamostat)
Trials
(nafamostat)
Recent Studies (post-2010) (nafamostat)
5,2315662,91964054198

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)nafamostat (IC50)
Ubiquitin-like modifier activating enzyme 2Homo sapiens (human)7.47
SUMO1 activating enzyme subunit 1Homo sapiens (human)7.47
ubiquitin-like modifier-activating enzyme 1Homo sapiens (human)14
SUMO-conjugating enzyme UBC9Homo sapiens (human)7.47
ubiquitin-conjugating enzyme E2 NHomo sapiens (human)14
ubiquitin-conjugating enzyme E2 variant 1 isoform aHomo sapiens (human)14
ProthrombinHomo sapiens (human)1.9
Complement C1r subcomponentHomo sapiens (human)0.8
PlasminogenHomo sapiens (human)2.9
Cationic trypsinBos taurus (cattle)0.017
Serine protease hepsinHomo sapiens (human)0.005
Trypsin-1Homo sapiens (human)0.017
Complement C1s subcomponentHomo sapiens (human)0.029
Hepatocyte growth factor activatorHomo sapiens (human)0.15

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Damalanka, VC; Janetka, JW; Klampfer, L; Li, S; Mahoney, MW; Primeau, T; Voss, JJLP1

Other Studies

1 other study(ies) available for gefitinib and nafamostat

ArticleYear
Macrocyclic Inhibitors of HGF-Activating Serine Proteases Overcome Resistance to Receptor Tyrosine Kinase Inhibitors and Block Lung Cancer Progression.
    Journal of medicinal chemistry, 2021, 12-23, Volume: 64, Issue:24

    Topics: Animals; Carcinoma, Non-Small-Cell Lung; Disease Progression; Drug Discovery; Hepatocyte Growth Factor; Humans; Lung Neoplasms; Macrocyclic Compounds; Mice; Receptor Protein-Tyrosine Kinases; Serine Proteinase Inhibitors; Structure-Activity Relationship

2021