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gefitinib and n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea

gefitinib has been researched along with n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea in 2 studies

Compound Research Comparison

Studies (gefitinib)	Trials (gefitinib)	Recent Studies (post-2010) (gefitinib)	Studies (n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea)	Trials (n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea)	Recent Studies (post-2010) (n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea)
5,231	566	2,919	94	0	61

Protein Interaction Comparison

Protein	Taxonomy	n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea (IC50)
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	0.104
Glycogen synthase kinase-3 beta	Homo sapiens (human)	0.1269
Glycogen synthase kinase-3 beta	Mus musculus (house mouse)	0.1
Cysteine protease ATG4B	Homo sapiens (human)	1.6

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	1 (50.00)	29.6817
2010's	1 (50.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M	1
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB	1

Other Studies

2 other study(ies) available for gefitinib and n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea

Article	Year
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases. Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51 Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases	2007
Navigating the kinome. Nature chemical biology, 2011, Volume: 7, Issue:4 Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology	2011

Article

Year

A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.

Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007

Navigating the kinome.

Nature chemical biology, 2011, Volume: 7, Issue:4

Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011