Page last updated: 2024-09-03

gefitinib and incb3619

gefitinib has been researched along with incb3619 in 2 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(incb3619)
Trials
(incb3619)
Recent Studies (post-2010) (incb3619)
5,2315662,919905

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)incb3619 (IC50)
Disintegrin and metalloproteinase domain-containing protein 10Homo sapiens (human)0.0312
Disintegrin and metalloproteinase domain-containing protein 17Sus scrofa (pig)0.014
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.068
72 kDa type IV collagenaseHomo sapiens (human)0.037
Stromelysin-1Homo sapiens (human)3.78
Matrix metalloproteinase-9Homo sapiens (human)0.366
Macrophage metalloelastaseHomo sapiens (human)0.017
Matrix metalloproteinase-14Homo sapiens (human)0.772
Disintegrin and metalloproteinase domain-containing protein 8Homo sapiens (human)1
Disintegrin and metalloproteinase domain-containing protein 17Homo sapiens (human)0.507
Disintegrin and metalloproteinase domain-containing protein 33Homo sapiens (human)1.026

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dreymuller, D; Fields, GB; Fridman, R; Giulianotti, M; Golubkov, V; Houghten, RA; Knapinska, AM; LaVoi, TM; Ludwig, A; Minond, D; Smith, L; Sohail, A1
Baribaud, F; Caudler, E; Fridman, JS; Friedman, SM; Gazdar, AF; Girard, L; He, B; Jablons, DM; Li, Y; Liu, C; Lo, Y; Mikami, I; Minna, JD; Newton, RC; Peyton, M; Reguart, N; Scherle, PA; Vaddi, K; Yang, G; Yao, W; Zhou, BB1

Other Studies

2 other study(ies) available for gefitinib and incb3619

ArticleYear
SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes.
    Journal of medicinal chemistry, 2015, Aug-13, Volume: 58, Issue:15

    Topics: ADAM Proteins; ADAM17 Protein; Animals; Cell Line; CHO Cells; Cricetinae; Cricetulus; Humans; In Vitro Techniques; Molecular Probes; Structure-Activity Relationship; Substrate Specificity

2015
Targeting ADAM-mediated ligand cleavage to inhibit HER3 and EGFR pathways in non-small cell lung cancer.
    Cancer cell, 2006, Volume: 10, Issue:1

    Topics: ADAM Proteins; ADAM17 Protein; Animals; Apoptosis; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; ErbB Receptors; Female; Gefitinib; Gene Expression; Humans; Ligands; Mice; Mice, Inbred BALB C; Mice, Nude; Models, Biological; Paclitaxel; Piperidines; Protease Inhibitors; Protein Kinase Inhibitors; Quinazolines; Receptor, ErbB-3; Signal Transduction; Spiro Compounds; Xenograft Model Antitumor Assays

2006