Page last updated: 2024-09-03

gefitinib and gsk343

gefitinib has been researched along with gsk343 in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(gsk343)
Trials
(gsk343)
Recent Studies (post-2010) (gsk343)
5,2315662,91943043

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)gsk343 (IC50)
Polycomb protein EEDHomo sapiens (human)0.122
Histone-binding protein RBBP4Homo sapiens (human)0.122
Polycomb protein SUZ12Homo sapiens (human)0.122
Histone-lysine N-methyltransferase EZH2Homo sapiens (human)1.0255
Histone-binding protein RBBP7Homo sapiens (human)0.004
Zinc finger protein AEBP2Homo sapiens (human)0.24
Histone-lysine N-methyltransferase EZH1Homo sapiens (human)0.24

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Chen, C; Chen, J; Gong, H; Li, W; Li, Y; Liu, C; Liu, H; Liu, M; Shi, R; Yuan, Y; Zhang, H; Zhang, Z1

Other Studies

1 other study(ies) available for gefitinib and gsk343

ArticleYear
EZH2 inhibitors reverse resistance to gefitinib in primary EGFR wild-type lung cancer cells.
    BMC cancer, 2020, Dec-04, Volume: 20, Issue:1

    Topics: Adenosine; Adult; Aged; Animals; Apoptosis; Carcinoma, Non-Small-Cell Lung; Cell Cycle; Cell Line, Tumor; Cell Movement; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Drug Synergism; Enhancer of Zeste Homolog 2 Protein; Female; Gefitinib; Gene Expression Regulation, Neoplastic; Genes, erbB-1; Humans; Indazoles; Lung Neoplasms; Mice; Mice, Inbred BALB C; Mice, Nude; Middle Aged; Neoplasm Invasiveness; Neoplasm Proteins; Protein Kinase Inhibitors; Pyridones; RNA Interference; RNA, Neoplasm; RNA, Small Interfering; Signal Transduction

2020