Page last updated: 2024-09-03

gefitinib and fosbretabulin

gefitinib has been researched along with fosbretabulin in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(fosbretabulin)
Trials
(fosbretabulin)
Recent Studies (post-2010) (fosbretabulin)
5,2315662,9194970320

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)fosbretabulin (IC50)
Tubulin polymerization-promoting proteinHomo sapiens (human)1.016
Tubulin alpha-1A chainSus scrofa (pig)1.82
Tubulin beta chainSus scrofa (pig)1.9428
Tubulin beta-4A chainHomo sapiens (human)1.663
Tubulin beta chainHomo sapiens (human)1.663
ATP-dependent translocase ABCB1Homo sapiens (human)0.009
Tubulin alpha-3C chainHomo sapiens (human)1.663
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)1.08
Delta-type opioid receptorMus musculus (house mouse)1.005
Delta-type opioid receptorRattus norvegicus (Norway rat)0.81
Mu-type opioid receptorMus musculus (house mouse)1.2
Tubulin alpha-1B chainHomo sapiens (human)1.663
Tubulin alpha-4A chainHomo sapiens (human)1.663
Tubulin beta-4B chainHomo sapiens (human)1.663
Vesicular acetylcholine transporterTetronarce californica (Pacific electric ray)1.8
Tubulin beta-3 chainHomo sapiens (human)1.5801
Tubulin beta-2A chainHomo sapiens (human)1.663
Beta-tubulin Leishmania donovani1.95
Tubulin beta-8 chainHomo sapiens (human)1.663
Tubulin beta-2B chainBos taurus (cattle)1.4484
Tubulin alpha-3E chainHomo sapiens (human)1.663
Tubulin alpha-1A chainHomo sapiens (human)1.663
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)1.4928
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)1.4037
Tubulin alpha-1C chainHomo sapiens (human)1.663
Tubulin beta-6 chainHomo sapiens (human)1.663
Tubulin beta-2B chainHomo sapiens (human)1.663
Tubulin beta-1 chainHomo sapiens (human)1.6366

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, L; He, L; Liu, Y; Ma, L; Nie, C; Pu, Y; Shao, M; Wang, F; Wu, W; Wu, Y; Yang, Z; Yu, K1

Other Studies

1 other study(ies) available for gefitinib and fosbretabulin

ArticleYear
Synthesis and biological evaluation of diarylthiazole derivatives as antimitotic and antivascular agents with potent antitumor activity.
    Bioorganic & medicinal chemistry, 2015, Jul-01, Volume: 23, Issue:13

    Topics: Angiogenesis Inhibitors; Animals; Antimitotic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Line, Tumor; Cell Movement; Colchicine; Colonic Neoplasms; Drug Resistance, Neoplasm; Female; G2 Phase Cell Cycle Checkpoints; Gene Expression; Human Umbilical Vein Endothelial Cells; Humans; Mice; Mice, Inbred BALB C; Protein Binding; Stilbenes; Structure-Activity Relationship; Thiazoles; Tubulin Modulators; Xenograft Model Antitumor Assays

2015