Page last updated: 2024-09-03

gefitinib and cvt 313

gefitinib has been researched along with cvt 313 in 2 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(cvt 313)
Trials
(cvt 313)
Recent Studies (post-2010) (cvt 313)
5,2315662,91919011

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)cvt 313 (IC50)
Cyclin-T1Homo sapiens (human)2.3
Cyclin-dependent kinase 1Homo sapiens (human)3.7
G2/mitotic-specific cyclin-B1Homo sapiens (human)3.7
Cyclin-A2Homo sapiens (human)0.22
G1/S-specific cyclin-E1Homo sapiens (human)0.176
Cyclin-dependent kinase 2Homo sapiens (human)0.198
Cyclin-dependent kinase 7Homo sapiens (human)9.2
Cyclin-dependent kinase 9Homo sapiens (human)2.3
Cyclin-HHomo sapiens (human)9.2
CDK-activating kinase assembly factor MAT1Homo sapiens (human)9.2
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.419
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.419

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Dai, L; Hu, ZD; Li, XL; Sun, YX; Tao, YF; Wang, AM; Wang, SP; Wu, Q; Yang, AL; Zhang, J1

Other Studies

2 other study(ies) available for gefitinib and cvt 313

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
A network pharmacology approach to investigate the anticancer mechanism of cinobufagin against hepatocellular carcinoma via downregulation of EGFR-CDK2 signaling.
    Toxicology and applied pharmacology, 2021, 11-15, Volume: 431

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Bufanolides; Carcinoma, Hepatocellular; Cell Proliferation; Cyclin-Dependent Kinase 2; Down-Regulation; Drug Synergism; ErbB Receptors; Gefitinib; Gene Expression Regulation, Neoplastic; Gene Regulatory Networks; Hep G2 Cells; Humans; Liver Neoplasms; M Phase Cell Cycle Checkpoints; Network Pharmacology; Protein Interaction Maps; Protein Kinase Inhibitors; Purines; Signal Transduction

2021