Page last updated: 2024-09-03

gefitinib and chalcone

gefitinib has been researched along with chalcone in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(chalcone)
Trials
(chalcone)
Recent Studies (post-2010) (chalcone)
5,2315662,9192,015221,086

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)chalcone (IC50)
perilipin-5Homo sapiens (human)4.245
perilipin-1Homo sapiens (human)4.194
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)4.2195
Amine oxidase [flavin-containing] AHomo sapiens (human)1.41
Amine oxidase [flavin-containing] BHomo sapiens (human)1.41
Sortase AStreptococcus mutans5

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jeong, JH; Kwon, TK; Oh, YJ; Seo, YH1

Other Studies

1 other study(ies) available for gefitinib and chalcone

ArticleYear
Chalcone-templated Hsp90 inhibitors and their effects on gefitinib resistance in non-small cell lung cancer (NSCLC).
    Archives of pharmacal research, 2017, Volume: 40, Issue:1

    Topics: Antineoplastic Agents; Carcinoma, Non-Small-Cell Lung; Cell Survival; Chalcone; Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Gefitinib; HSP90 Heat-Shock Proteins; Humans; Lung Neoplasms; Molecular Docking Simulation; Protein Structure, Secondary; Quinazolines

2017