Page last updated: 2024-09-03

gefitinib and ceritinib

gefitinib has been researched along with ceritinib in 5 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(ceritinib)
Trials
(ceritinib)
Recent Studies (post-2010) (ceritinib)
5,2315662,91932935322

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)ceritinib (IC50)
Tyrosine-protein kinase JAK2Homo sapiens (human)1.385
Rho-associated protein kinase 2Homo sapiens (human)1.27
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)3.7
Tyrosine-protein kinase ABL1Homo sapiens (human)1.25
Epidermal growth factor receptorHomo sapiens (human)0.7757
High affinity nerve growth factor receptorHomo sapiens (human)2.727
Insulin receptorHomo sapiens (human)0.1525
Tyrosine-protein kinase LckHomo sapiens (human)0.616
NucleophosminHomo sapiens (human)0.026
Tyrosine-protein kinase LynHomo sapiens (human)1.573
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)1.352
Insulin-like growth factor 1 receptorHomo sapiens (human)0.209
Hepatocyte growth factor receptorHomo sapiens (human)1.5933
Cytochrome P450 3A4Homo sapiens (human)3.36
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)0.2697
Tyrosine-protein kinase FgrHomo sapiens (human)1.947
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 22.86
Mast/stem cell growth factor receptor KitHomo sapiens (human)2.0675
Cyclin-dependent kinase 4Homo sapiens (human)4.72
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)1.694
Platelet-derived growth factor receptor alphaHomo sapiens (human)1.14
Fibroblast growth factor receptor 2Homo sapiens (human)0.26
Fibroblast growth factor receptor 4Homo sapiens (human)0.95
Fibroblast growth factor receptor 3Homo sapiens (human)0.43
Tyrosine-protein kinase JAK1Homo sapiens (human)3.73
Cyclin-dependent kinase 2Homo sapiens (human)3.97
Vascular endothelial growth factor receptor 2Homo sapiens (human)4.21
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)1.0965
Transcription factor ETV6Homo sapiens (human)3.25
Tyrosine-protein kinase ZAP-70Homo sapiens (human)9.7
Tyrosine-protein kinase SYKHomo sapiens (human)3.05
Tyrosine-protein kinase JAK3Homo sapiens (human)7.92
Tyrosine-protein kinase BTKHomo sapiens (human)3.36
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.25
BDNF/NT-3 growth factors receptorHomo sapiens (human)1.829
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)0.023
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)2.24
Echinoderm microtubule-associated protein-like 4Homo sapiens (human)0.5935
ALK tyrosine kinase receptorHomo sapiens (human)0.1102

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (60.00)24.3611
2020's2 (40.00)2.80

Authors

AuthorsStudies
Aiche, S; Bassermann, F; Becker, W; Canevari, G; Casale, E; Depaolini, SR; Ehrlich, HC; Felder, ER; Feuchtinger, A; Garz, AK; Gohlke, BO; Götze, K; Greif, PA; Hahne, H; Heinzlmeir, S; Helm, D; Huenges, J; Jeremias, I; Kayser, G; Klaeger, S; Koch, H; Koenig, PA; Kramer, K; Kuster, B; Médard, G; Meng, C; Petzoldt, S; Polzer, H; Preissner, R; Qiao, H; Reinecke, M; Reiter, K; Rueckert, L; Ruland, J; Ruprecht, B; Schlegl, J; Schmidt, T; Schneider, S; Schoof, M; Spiekermann, K; Tõnisson, N; Vick, B; Vooder, T; Walch, A; Wilhelm, M; Wu, Z; Zecha, J; Zolg, DP1
Ding, K; Lu, X; Smaill, JB1
Cho, HJ; Chung, DH; Jeon, YK; Keam, B; Kim, DW; Kim, TM; Koh, J; Lee, DS; Lee, SH; Won, JK1
Garber, K1
Fujita, A; Hatsuyama, T; Inotsume, N; Mukai, Y; Sato, H; Toda, T; Wakamoto, A; Yoshida, T1

Reviews

1 review(s) available for gefitinib and ceritinib

ArticleYear
Medicinal Chemistry Strategies for the Development of Kinase Inhibitors Targeting Point Mutations.
    Journal of medicinal chemistry, 2020, 10-08, Volume: 63, Issue:19

    Topics: Chemistry, Pharmaceutical; Humans; Point Mutation; Protein Kinase Inhibitors

2020

Other Studies

4 other study(ies) available for gefitinib and ceritinib

ArticleYear
The target landscape of clinical kinase drugs.
    Science (New York, N.Y.), 2017, 12-01, Volume: 358, Issue:6367

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Cytokines; Drug Discovery; fms-Like Tyrosine Kinase 3; Humans; Leukemia, Myeloid, Acute; Lung Neoplasms; Mice; Molecular Targeted Therapy; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proteomics; Xenograft Model Antitumor Assays

2017
Concomitant ALK translocation and EGFR mutation in lung cancer: a comparison of direct sequencing and sensitive assays and the impact on responsiveness to tyrosine kinase inhibitor.
    Annals of oncology : official journal of the European Society for Medical Oncology, 2015, Volume: 26, Issue:2

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anaplastic Lymphoma Kinase; Antineoplastic Agents; Carcinoma, Non-Small-Cell Lung; Crizotinib; DNA Mutational Analysis; Female; Gefitinib; Genes, erbB-1; High-Throughput Nucleotide Sequencing; Humans; Immunohistochemistry; In Situ Hybridization, Fluorescence; Lung Neoplasms; Male; Middle Aged; Mutation; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Pyrimidines; Quinazolines; Real-Time Polymerase Chain Reaction; Receptor Protein-Tyrosine Kinases; Sensitivity and Specificity; Sulfones; Translocation, Genetic

2015
Oncologists push beyond new lung cancer genomic testing guidelines.
    Journal of the National Cancer Institute, 2015, Volume: 107, Issue:2

    Topics: Anaplastic Lymphoma Kinase; Antineoplastic Agents; Crizotinib; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; Genetic Testing; Genomics; Humans; Lung Neoplasms; Medical Oncology; Molecular Targeted Therapy; Mutation; Practice Guidelines as Topic; Precision Medicine; Pyrazoles; Pyridines; Pyrimidines; Quinazolines; Receptor Protein-Tyrosine Kinases; Societies, Medical; Sulfones; Translocation, Genetic

2015
An Liquid Chromatography-Tandem Mass Spectrometry Method for the Simultaneous Determination of Afatinib, Alectinib, Ceritinib, Crizotinib, Dacomitinib, Erlotinib, Gefitinib, and Osimertinib in Human Serum.
    Therapeutic drug monitoring, 2021, 12-01, Volume: 43, Issue:6

    Topics: Acrylamides; Afatinib; Aniline Compounds; Carbazoles; Chromatography, Liquid; Crizotinib; Erlotinib Hydrochloride; Gefitinib; Humans; Lung Neoplasms; Piperidines; Protein Kinase Inhibitors; Pyrimidines; Quinazolinones; Sulfones; Tandem Mass Spectrometry

2021