Page last updated: 2024-09-03

gefitinib and cc-292

gefitinib has been researched along with cc-292 in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(cc-292)
Trials
(cc-292)
Recent Studies (post-2010) (cc-292)
5,2315662,91933532

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)cc-292 (IC50)
Tyrosine-protein kinase JAK2Homo sapiens (human)0.5337
Epidermal growth factor receptorHomo sapiens (human)0.442
Tyrosine-protein kinase LynHomo sapiens (human)4.4
Tyrosine-protein kinase TecHomo sapiens (human)0.0062
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)2.665
Tyrosine-protein kinase JAK3Homo sapiens (human)0.4626
Tyrosine-protein kinase BTKHomo sapiens (human)0.1163
Early activation antigen CD69Homo sapiens (human)3.1
Sigma intracellular receptor 2Rattus norvegicus (Norway rat)0.5337

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Chen, L; Li, Y; Liu, K; Ma, T; Ma, X; Sun, H; Sun, X; Wang, C; Zheng, X; Zhu, Y1

Other Studies

1 other study(ies) available for gefitinib and cc-292

ArticleYear
Synthesis and biological activity of thieno[3,2-d]pyrimidines as potent JAK3 inhibitors for the treatment of idiopathic pulmonary fibrosis.
    Bioorganic & medicinal chemistry, 2020, 01-15, Volume: 28, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Disease Models, Animal; Dose-Response Relationship, Drug; Epithelial Cells; Female; Humans; Idiopathic Pulmonary Fibrosis; Janus Kinase 3; Mice; Mice, Inbred C57BL; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship

2020