Page last updated: 2024-09-03

gefitinib and bms345541

gefitinib has been researched along with bms345541 in 3 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(bms345541)
Trials
(bms345541)
Recent Studies (post-2010) (bms345541)
5,2315662,91998063

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)bms345541 (IC50)
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)1
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)4.54
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)3.1

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Knight, ZA; Shokat, KM1
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP1

Reviews

1 review(s) available for gefitinib and bms345541

ArticleYear
Features of selective kinase inhibitors.
    Chemistry & biology, 2005, Volume: 12, Issue:6

    Topics: Animals; Drug Evaluation, Preclinical; Humans; Phosphoric Monoester Hydrolases; Protein Kinase Inhibitors; Substrate Specificity

2005

Other Studies

2 other study(ies) available for gefitinib and bms345541

ArticleYear
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011
Comprehensive analysis of kinase inhibitor selectivity.
    Nature biotechnology, 2011, Oct-30, Volume: 29, Issue:11

    Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity

2011