Page last updated: 2024-09-03

gefitinib and bms 708163

gefitinib has been researched along with bms 708163 in 1 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(bms 708163)
Trials
(bms 708163)
Recent Studies (post-2010) (bms 708163)
5,2315662,91946543

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)bms 708163 (IC50)
Presenilin-1Homo sapiens (human)0.0006
Presenilin-2Homo sapiens (human)0.0006
Gamma-secretase subunit APH-1BHomo sapiens (human)0.0006
NicastrinHomo sapiens (human)0.0006
Gamma-secretase subunit APH-1AHomo sapiens (human)0.0006
Gamma-secretase subunit PEN-2Homo sapiens (human)0.0006

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
He, C; He, J; Wei, S; Xie, M1

Other Studies

1 other study(ies) available for gefitinib and bms 708163

ArticleYear
γ Secretase inhibitor BMS-708163 reverses resistance to EGFR inhibitor via the PI3K/Akt pathway in lung cancer.
    Journal of cellular biochemistry, 2015, Volume: 116, Issue:6

    Topics: Amyloid Precursor Protein Secretases; Animals; Apoptosis; Cell Line, Tumor; Cell Survival; ErbB Receptors; Female; Gefitinib; Immunohistochemistry; Lung Neoplasms; Mice; Mice, Inbred BALB C; Oxadiazoles; Phosphatidylinositol 3-Kinases; Proto-Oncogene Proteins c-akt; Quinazolines; Sulfonamides

2015