Page last updated: 2024-09-03

gefitinib and antimycin a

gefitinib has been researched along with antimycin a in 3 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(antimycin a)
Trials
(antimycin a)
Recent Studies (post-2010) (antimycin a)
5,2315662,91937020

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)antimycin a (IC50)
Mitochondrial succinate dehydrogenase subunit C Zymoseptoria tritici0.002
Succinate dehydrogenase [ubiquinone] iron-sulfur subunit, mitochondrialZymoseptoria tritici0.002
Mitogen-activated protein kinase 1Homo sapiens (human)2.116

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Abou Samra, A; Ariffin, A; Awang, K; Bignon, J; Daressy, F; Desrat, S; Fourneau, C; Gapil Tiamas, S; Hoong Leong, K; Litaudon, M; Roussi, F; Steinmetz, V1

Other Studies

3 other study(ies) available for gefitinib and antimycin a

ArticleYear
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Pro-apoptotic carboxamide analogues of natural fislatifolic acid targeting Mcl-1 and Bcl-2.
    Bioorganic & medicinal chemistry letters, 2020, 04-01, Volume: 30, Issue:7

    Topics: Amides; Antineoplastic Agents; Apoptosis; bcl-X Protein; Cell Line, Tumor; Cyclohexanecarboxylic Acids; Drug Screening Assays, Antitumor; Humans; Myeloid Cell Leukemia Sequence 1 Protein; Small Molecule Libraries; Stereoisomerism

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