Page last updated: 2024-09-03

gefitinib and 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin

gefitinib has been researched along with 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin in 2 studies

Compound Research Comparison

Studies
(gefitinib)
Trials
(gefitinib)
Recent Studies (post-2010)
(gefitinib)
Studies
(17-(dimethylaminoethylamino)-17-demethoxygeldanamycin)
Trials
(17-(dimethylaminoethylamino)-17-demethoxygeldanamycin)
Recent Studies (post-2010) (17-(dimethylaminoethylamino)-17-demethoxygeldanamycin)
5,2315662,9192559168

Protein Interaction Comparison

ProteinTaxonomygefitinib (IC50)17-(dimethylaminoethylamino)-17-demethoxygeldanamycin (IC50)
Lysine-specific demethylase 6BHomo sapiens (human)0.4
Lysine-specific demethylase 4BHomo sapiens (human)0.7
Heat shock protein HSP 90-alphaHomo sapiens (human)0.1699
Heat shock protein HSP 90-betaHomo sapiens (human)0.2724
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0036
Lysine-specific demethylase 5AHomo sapiens (human)0.13
Hypoxia-inducible factor 1-alphaHomo sapiens (human)0.043
Endothelial PAS domain-containing protein 1Homo sapiens (human)0.0335
Lysine-specific demethylase 4CHomo sapiens (human)0.7

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ando, M; Dote, H; Jida, M; Kawasaki, K; Kiura, K; Kobayashi, N; Kubo, T; Miyoshi, S; Ogino, A; Otani, H; Soh, J; Toyooka, S; Ueno, T; Yamamoto, H1
Akashi, M; Chin, TM; Doan, NB; Koeffler, HP; Mori, S; Said, JW; Sudo, M1

Other Studies

2 other study(ies) available for gefitinib and 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin

ArticleYear
The anti-proliferative effect of heat shock protein 90 inhibitor, 17-DMAG, on non-small-cell lung cancers being resistant to EGFR tyrosine kinase inhibitor.
    Lung cancer (Amsterdam, Netherlands), 2012, Volume: 75, Issue:2

    Topics: Animals; Antineoplastic Agents; Apoptosis; Benzoquinones; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Drug Resistance, Neoplasm; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; HSP90 Heat-Shock Proteins; Humans; Lactams, Macrocyclic; Lung Neoplasms; Mice; Mutation; Quinazolines; Xenograft Model Antitumor Assays

2012
Inhibiting proliferation of gefitinib-resistant, non-small cell lung cancer.
    Cancer chemotherapy and pharmacology, 2013, Volume: 71, Issue:5

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzoquinones; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cell Proliferation; Drug Resistance, Neoplasm; Drug Synergism; ErbB Receptors; Gefitinib; Humans; Hydroxamic Acids; Lactams, Macrocyclic; Lung Neoplasms; Mice; Mice, Nude; Mutation; Protein Kinase Inhibitors; PTEN Phosphohydrolase; Quinazolines; Sulfonamides; Xenograft Model Antitumor Assays

2013