gbr 12935 and piperidines

gbr 12935 has been researched along with piperidines in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's2 (33.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ross, SB1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
Allard, P; Norlén, M1
Beardsley, PM; Cook, CD; Davis, MC; Dutta, AK; Fei, XS; Reith, ME1
Chen, N; Dutta, AK; Maiti, S; Reith, ME; Zhen, J1
Gigante, E; Good, CH; Hoffman, AF; Lupica, CR; Morales, M; Root, DH; Zhang, S1

Other Studies

6 other study(ies) available for gbr 12935 and piperidines

ArticleYear
Heterogeneous binding of sigma radioligands in the rat brain and liver: possible relationship to subforms of cytochrome P-450.
    Pharmacology & toxicology, 1991, Volume: 68, Issue:4

    Topics: Animals; Brain; Cytochrome P-450 Enzyme System; Guanidines; Haloperidol; Kinetics; Ligands; Liver; Male; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Subcellular Fractions

1991
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
[3H]GBR 12935 binding in platelets: a possible association with cytochrome P-450IID6?
    European journal of pharmacology, 1997, Aug-06, Volume: 332, Issue:2

    Topics: Antipsychotic Agents; Blood Platelets; Culture Techniques; Cytochrome P-450 Enzyme System; Dopamine Antagonists; Enzyme Inhibitors; Flupenthixol; Humans; Ligands; Lobeline; Piperazines; Piperidines; Quinidine

1997
Expansion of structure-activity studies of piperidine analogues of 1-[2-(diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine (GBR 12935) compounds by altering substitutions in the N-benzyl moiety and behavioral pharmacology of selected molecules.
    Journal of medicinal chemistry, 2002, Jan-31, Volume: 45, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Piperidines; Radioligand Assay; Rats; Serotonin; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Symporters

2002
Interaction between a hydroxypiperidine analogue of 4-(2-benzhydryloxy-ethyl)-1-(4-fluorobenzyl)piperidine and Aspartate 68 in the human dopamine transporter.
    European journal of pharmacology, 2004, Dec-03, Volume: 506, Issue:1

    Topics: Animals; Aspartic Acid; Benzhydryl Compounds; Binding Sites; Binding, Competitive; Biological Transport; Cell Line; Cell Membrane; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Humans; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Mutation; Nerve Tissue Proteins; Norepinephrine; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Serotonin; Stereoisomerism; Synaptosomes; Tritium

2004
Norepinephrine activates dopamine D4 receptors in the rat lateral habenula.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, Feb-25, Volume: 35, Issue:8

    Topics: Animals; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopaminergic Neurons; Habenula; Isoxazoles; Male; Norepinephrine; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D4; RNA, Messenger; Ventral Tegmental Area; Vesicular Monoamine Transport Proteins

2015