gamma-aminobutyric acid and spiperone

gamma-aminobutyric acid has been researched along with spiperone in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199028 (73.68)18.7374
1990's6 (15.79)18.2507
2000's2 (5.26)29.6817
2010's2 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Enna, SJ; Möhler, H; Okada, T1
Bird, ED; Enna, SJ; Reisine, TD; Spokes, E; Yamamura, HI1
Fung, YK; Lau, YS1
Colmers, WF; Pan, ZZ; Williams, JT1
Khorram, O; McCann, SM; Mizunuma, H1
Cross, AJ; Crow, TJ; Ferrier, IN; Johnson, JA; Johnstone, EC; Owen, F; Owens, DG; Poulter, M1
Kalaria, RN; Prince, AK1
Cassel, G; Persson, SA; Sellström, A1
Arbilla, S; Bartholini, G; Fage, D; Langer, SZ; Oblin, A; Scatton, B; Zivkovic, B1
Kaufman, WR; Lindsay, PJ1
Arbilla, S; Bartholini, G; Claustre, Y; Dedek, J; Dennis, T; Langer, SZ; Lloyd, KG; Scatton, B; Zivkovic, B1
Altar, CA; Heikkila, RE; Manzino, L; Marien, MR1
Jones, DL1
Bunn, SJ; Hanley, MR; Wilkin, GP1
Flohé, L; Günzler, WA; Hennies, HH1
Oka, M; Shimizu, M; Yamada, K; Yoshida, K1
Hruska, RE; Silbergeld, EK1
Cheney, DL; Costa, E; Gandolfi, O; Hong, JS1
Cross, A; Rossor, M1
Govoni, S; Memo, M; Saiani, L; Spano, PF; Trabucchi, M1
Enna, SJ; Ferkany, JW; Strong, R1
Biggio, G; Concas, A; Corda, MG; Corongiu, FP; Guarneri, P; Rossetti, Z1
Jones, DL; Mogenson, GJ1
Gardner, CR; Huot-Olivier, S; Klein, J; Mallorga, P; Palfreyman, MG1
Silbergeld, EK1
Cohen, G; Dembiec-Cohen, D; Hwang, E; Mytilineou, C; Van Woert, M1
Dakshinamurti, K; Paulose, CS1
Enna, SJ; Ferkany, JW1
Pecins-Thompson, M; Peris, J1
Kanazawa, I; Kimura, M; Murata, M1
Blier, P; De Montigny, C; Lista, A1
Blier, P; de Montigny, C; Mongeau, R; Weiss, M1
Araujo, DM; Cherry, SR; Kornblum, HI; Tatsukawa, KJ; Toyokuni, T1
Chesneau, D; de la Riva, C; Fabre-Nys, C; Hinton, MR; Kendrick, KM; Locatelli, A; Ohkura, S1

Reviews

1 review(s) available for gamma-aminobutyric acid and spiperone

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

37 other study(ies) available for gamma-aminobutyric acid and spiperone

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Benzodiasepine and neurotransmitter receptor binding in rat brain after chronic administration of diazepam or phenobarbital.
    Brain research, 1978, Nov-10, Volume: 156, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Dopamine; gamma-Aminobutyric Acid; Neurotransmitter Agents; Phenobarbital; Quinuclidines; Rats; Receptors, Dopamine; Receptors, Drug; Receptors, Neurotransmitter; Spiperone

1978
Pre- and postsynaptic neurochemical alterations in Alzheimer's disease.
    Brain research, 1978, Dec-29, Volume: 159, Issue:2

    Topics: Aged; Alzheimer Disease; Caudate Nucleus; Choline O-Acetyltransferase; Dementia; Frontal Lobe; gamma-Aminobutyric Acid; Hippocampus; Humans; Middle Aged; Putamen; Quinuclidines; Receptors, Neurotransmitter; Spiperone; Synapses

1978
Chronic effects of nicotine on mesolimbic dopaminergic system in rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Dextroamphetamine; Dopamine; Dopamine Antagonists; gamma-Aminobutyric Acid; Injections; Limbic System; Male; Methyltyrosines; Motor Activity; Nicotine; Nucleus Accumbens; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Nicotinic; Spiperone; Tyrosine 3-Monooxygenase

1992
5-HT-mediated synaptic potentials in the dorsal raphe nucleus: interactions with excitatory amino acid and GABA neurotransmission.
    Journal of neurophysiology, 1989, Volume: 62, Issue:2

    Topics: Animals; Electric Stimulation; Fluoxetine; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neurons; Pons; Raphe Nuclei; Rats; Serotonin; Spiperone; Synapses

1989
Purification of a non-dopaminergic and non-GABAergic prolactin release-inhibiting factor (PIF) in sheep stalk-median eminence.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1985, Volume: 178, Issue:1

    Topics: Animals; Cells, Cultured; Chromatography, Gel; Dopamine; Epinephrine; Estradiol; gamma-Aminobutyric Acid; Median Eminence; Norepinephrine; Pituitary Gland, Anterior; Prolactin; Prolactin Release-Inhibiting Factors; Rats; Sheep; Spiperone

1985
Chemical and structural changes in the brain in patients with movement disorder.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Acetylcholine; Antipsychotic Agents; Brain; Choline O-Acetyltransferase; Dopamine; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Homovanillic Acid; Humans; Movement Disorders; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Schizophrenia; Spiperone

1985
Decreased neurotransmitter receptor binding in striatum and cortex from adult hypothyroid rats.
    Brain research, 1986, Feb-05, Volume: 364, Issue:2

    Topics: Animals; Choline O-Acetyltransferase; Corpus Striatum; Dioxanes; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypothyroidism; Muscimol; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Spiperone; Tyrosine 3-Monooxygenase; Visual Cortex

1986
Acute cyanide intoxication and central transmitter systems.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1985, Volume: 5, Issue:6 Pt 2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids; Animals; Apomorphine; Brain; Cyanides; Cyclic GMP; Dopamine; gamma-Aminobutyric Acid; Homovanillic Acid; Levodopa; Male; Neurotransmitter Agents; Norepinephrine; Rats; Rats, Inbred Strains; Spiperone

1985
Influence of GABA mimetics and lithium on biochemical manifestations of striatal dopamine target cell hypersensitivity.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Haloperidol; Kinetics; Lithium; Rats; Receptors, Dopamine; Spiperone; Synapses; Synaptic Transmission

1985
Potentiation of salivary fluid secretion in ixodid ticks: a new receptor system for gamma-aminobutyric acid.
    Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:8

    Topics: Animals; Bicuculline; Dopamine; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Muscimol; Picrotoxin; Receptors, GABA-A; Saliva; Spiperone; Sulpiride; Ticks

1986
Fengabine, a novel antidepressant GABAergic agent. II. Effect on cerebral noradrenergic, serotonergic and GABAergic transmission in the rat.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Animals; Antidepressive Agents; Brain; Chlorophenols; Clonidine; Dihydroalprenolol; gamma-Aminobutyric Acid; Imipramine; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Spiperone; Synaptic Transmission

1987
1-Methyl-4-phenylpyridine (MPP+): regional dopamine neuron uptake, toxicity, and novel rotational behavior following dopamine receptor proliferation.
    European journal of pharmacology, 1986, Nov-19, Volume: 131, Issue:2-3

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Autoradiography; Basal Ganglia; Brain; Dopamine; gamma-Aminobutyric Acid; Injections; Male; Neurons; Pyridinium Compounds; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1986
Cardiovascular and drinking responses elicited by central administration of angiotensin II: differential effects of GABA injected into the ventral tegmental area and spiperone injected into the nucleus accumbens.
    Brain research bulletin, 1986, Volume: 17, Issue:2

    Topics: Angiotensin II; Animals; Blood Pressure; Brain; Drinking Behavior; gamma-Aminobutyric Acid; Heart Rate; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Septal Nuclei; Spiperone; Tegmentum Mesencephali

1986
Autoradiographic localization of peripheral benzodiazepine, dihydroalprenolol and arginine vasopressin binding sites in the pituitaries of control, stalk transected and Brattleboro rats.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Alprenolol; Animals; Arginine Vasopressin; Autoradiography; Benzodiazepines; Benzodiazepinones; Binding Sites; Dihydroalprenolol; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Intermediate Filament Proteins; Male; Pituitary Gland; Rats; Rats, Brattleboro; Rats, Inbred Strains; Spiperone

1986
Influence of supidimide on brain neurotransmitter systems of rats and mice.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:11

    Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Aminobutyrate Transaminase; Adenylyl Cyclases; Animals; Binding, Competitive; Brain; Brain Chemistry; Catechol O-Methyltransferase; Dopamine; Electroshock; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Mice; Monoamine Oxidase; Neurotransmitter Agents; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, GABA-A; Serotonin; Species Specificity; Spiperone; Thalidomide; Tryptophan; Tyrosine 3-Monooxygenase

1984
Avoidance enhancement and discriminative response control by anxiolytics with drugs acting on the GABA system.
    Japanese journal of pharmacology, 1980, Volume: 30, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Avoidance Learning; Discrimination Learning; Drug Synergism; gamma-Aminobutyric Acid; Male; Methyltyrosines; Mice; Picrotoxin; Rats; Semicarbazides; Spiperone

1980
Inhibition of neurotransmitter receptor binding by ergot derivatives.
    Journal of neuroscience research, 1981, Volume: 6, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Bromocriptine; Dioxanes; Ergolines; Ergot Alkaloids; gamma-Aminobutyric Acid; Lysergic Acid Diethylamide; Male; Metergoline; Organ Specificity; Quinuclidinyl Benzilate; Rats; Receptors, Neurotransmitter; Serotonin; Spiperone; Structure-Activity Relationship; Synapses

1981
On the neurotoxicity of chlordecone: a role for gamma-aminobutyric acid and serotonin.
    Brain research, 1984, Jun-11, Volume: 303, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Brain; Chlordecone; gamma-Aminobutyric Acid; Insecticides; Ketanserin; Male; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Spiperone

1984
Dopamine D-1 and D-2 receptors in Huntington's disease.
    European journal of pharmacology, 1983, Mar-25, Volume: 88, Issue:2-3

    Topics: Aged; Brain; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Kinetics; Male; Middle Aged; Putamen; Receptors, Dopamine; Spiperone; Substantia Nigra; Thioxanthenes

1983
Impairment of brain neurotransmitter receptors in aged rats.
    Mechanisms of ageing and development, 1980, Volume: 12, Issue:1

    Topics: Aging; Animals; Brain; Corpus Striatum; gamma-Aminobutyric Acid; Male; Olfactory Bulb; Pituitary Gland; Rats; Receptors, Cell Surface; Receptors, Dopamine; Spiperone

1980
Drug-induced alterations in neurotransmitter receptor binding and function.
    Advances in biochemical psychopharmacology, 1980, Volume: 21

    Topics: 4-Aminobutyrate Transaminase; Animals; Behavior, Animal; Brain; Corpus Striatum; Female; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Rats; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, Dopamine; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Neurotransmitter; Spiperone; Synaptic Membranes

1980
Methyl mercury enhances [3H]diazepam binding in different areas of the rat brain.
    Brain research, 1981, Dec-14, Volume: 229, Issue:1

    Topics: Animals; Brain; Diazepam; gamma-Aminobutyric Acid; Male; Methylmercury Compounds; Muscimol; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Retina; Spiperone

1981
Central injections of spiperone and GABA: attenuation of angiotensin II stimulated thirst.
    Canadian journal of physiology and pharmacology, 1982, Volume: 60, Issue:5

    Topics: Angiotensin II; Animals; Butyrophenones; gamma-Aminobutyric Acid; Globus Pallidus; Male; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Spiperone; Tegmentum Mesencephali; Thirst

1982
Chronic elevation of brain GABA by gamma-vinyl GABA treatment does not alter the sensitivity of GABAergic or dopaminergic receptors in rat CNS.
    Psychopharmacology, 1983, Volume: 79, Issue:2-3

    Topics: Adenylyl Cyclases; Aminocaproates; Animals; Brain Chemistry; Diazepam; gamma-Aminobutyric Acid; Male; Motor Activity; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Spiperone; Vigabatrin

1983
Indirectly acting neurotoxins.
    Acta psychiatrica Scandinavica. Supplementum, 1983, Volume: 303

    Topics: Aminolevulinic Acid; Animals; Brain; Dopamine; Estradiol; Female; gamma-Aminobutyric Acid; Lead Poisoning; Male; Porphyrias; Porphyrins; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Dopamine; Receptors, GABA-A; Seizures; Spiperone; Synapses; Synaptic Transmission

1983
Explant cultures of dog substantia nigra and striatum: a model for the study of nigro-striatal dopamine neurons.
    Journal of neural transmission. Supplementum, 1983, Volume: 19

    Topics: Animals; Autoradiography; Cell Differentiation; Corpus Striatum; Culture Techniques; Dogs; Dopamine; gamma-Aminobutyric Acid; Homovanillic Acid; Microscopy, Fluorescence; Neural Pathways; Neurons; Receptors, Dopamine; Spiperone; Substantia Nigra; Synaptic Transmission

1983
Consequences of brain monoamine changes in the pyridoxine-deficient young rat.
    Progress in clinical and biological research, 1984, Volume: 144A

    Topics: Animals; Brain; Dopamine; gamma-Aminobutyric Acid; Kinetics; Male; Pyridoxal Phosphate; Rats; Rats, Inbred Strains; Serotonin; Spiperone; Tissue Distribution; Vitamin B 6 Deficiency

1984
Interaction between GABA agonists and the cholinergic muscarinic system in rat corpus striatum.
    Life sciences, 1980, Jul-14, Volume: 27, Issue:2

    Topics: Animals; Atropine; Choline; Corpus Striatum; gamma-Aminobutyric Acid; Kinetics; Male; Parasympathetic Nervous System; Rats; Receptors, Dopamine; Spiperone

1980
Behavioral and neurochemical changes caused by repeated ethanol and cocaine administration.
    Psychopharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Autoradiography; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Convulsants; Dopamine; Ethanol; gamma-Aminobutyric Acid; Limbic System; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Substantia Nigra

1993
Roles of dopamine and its receptors in generation of choreic movements.
    Advances in neurology, 1993, Volume: 60

    Topics: Afferent Pathways; Animals; Brain Mapping; Cerebral Cortex; Choline O-Acetyltransferase; Chorea; Corpus Striatum; Disease Models, Animal; Dopamine; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kainic Acid; Levodopa; Macaca; Neurons; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Substantia Nigra; Synapses; Tyrosine 3-Monooxygenase

1993
Differential properties of pre- and postsynaptic 5-hydroxytryptamine1A receptors in the dorsal raphe and hippocampus: I. Effect of spiperone.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Drug Antagonism; gamma-Aminobutyric Acid; Hippocampus; Male; Methiothepin; Neurons; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Synapses

1993
Effect of acute, short- and long-term milnacipran administration on rat locus coeruleus noradrenergic and dorsal raphe serotonergic neurons.
    Neuropharmacology, 1998, Volume: 37, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Agonists; Adrenergic Uptake Inhibitors; Animals; Biological Transport; Brimonidine Tartrate; Clonidine; Cyclopropanes; Desipramine; Drug Administration Schedule; gamma-Aminobutyric Acid; Hippocampus; Hypothalamus; Injections, Subcutaneous; Kinetics; Locus Coeruleus; Lysergic Acid Diethylamide; Male; Mesencephalon; Milnacipran; Neurons; Norepinephrine; Quinoxalines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Spiperone; Time Factors

1998
Deficits in striatal dopamine D(2) receptors and energy metabolism detected by in vivo microPET imaging in a rat model of Huntington's disease.
    Experimental neurology, 2000, Volume: 166, Issue:2

    Topics: Animals; Autoradiography; Benzazepines; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Energy Metabolism; Female; Fluorodeoxyglucose F18; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Huntington Disease; In Situ Hybridization; Nerve Degeneration; Neurotoxins; Quinolinic Acid; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Substantia Nigra; Tomography, Emission-Computed; Tritium

2000
Biphasic role of dopamine on female sexual behaviour via D2 receptors in the mediobasal hypothalamus.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Aspartic Acid; Citrulline; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Estradiol; Extracellular Space; Female; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Goats; Hypothalamus, Middle; Luteinizing Hormone; Microdialysis; Norepinephrine; Ovariectomy; Pimozide; Prolactin; Quinpirole; Receptors, Dopamine D2; Serotonin; Sexual Behavior, Animal; Spiperone; Taurine; Time Factors

2003