gallopamil and veratridine

gallopamil has been researched along with veratridine in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199017 (58.62)18.7374
1990's6 (20.69)18.2507
2000's2 (6.90)29.6817
2010's4 (13.79)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E1
Ahnert, G; Glossmann, H; Habermann, E1
Bartfai, T; Breakefield, XO; Greengard, P; Study, RE1
Rosenberger, LB; Triggle, DJ1
Catterall, WA; Galper, JB2
Ferrante, J; Rutledge, A; Triggle, DJ1
Kuramoto, K; Morita, Y; Sorimachi, M; Yamagami, K1
Ikeda, K; Koyano, H; Sato, M; Yoshizaki, K1
Furukawa, T; Katsuragi, T; Usune, S1
Payza, K; Russell, JT1
Nishimura, S; Sorimachi, M; Yada, T; Yamagami, K1
Liles, WC; Nathanson, NM1
Bourguignon, JP; Debougnoux, G; Franchimont, P; Gerard, A; Rose, J1
Dinerstein, RJ; Miller, RJ; Perney, TM1
Drouva, SV; Epelbaum, J; Hery, M; Kordon, C; Laplante, E; Tapia-Arancibia, L1
Barraco, R; Moron, M; Wu, PH1
Erlichman, J; Fleckman, A; Fleischer, N; Schubart, UK1
Conn, PM; Rogers, DC; Seay, SG1
Dannies, PS; Scammell, JG1
Corcoran, JJ; Kirshner, N1
Corcoran, JJ; Kilpatrick, DL; Kirshner, N; Slepetis, RJ1
Pezzementi, L; Schmidt, J1
Brenci, S; Indiveri, F; Lotti, G; Musso, NR1

Other Studies

29 other study(ies) available for gallopamil and veratridine

ArticleYear
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship

2008
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
    Bioorganic & medicinal chemistry, 2016, Apr-15, Volume: 24, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine

2016
Investigations on the mechanism of cyclic guanosine monophosphate increase due to depolarizing agents as studied with sea anemone toxin II in mouse cerebellar slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 307, Issue:2

    Topics: Adenosine Deaminase; Animals; Calcium; Cerebellum; Cnidarian Venoms; Cyclic GMP; Gallopamil; In Vitro Techniques; Mice; Neuromuscular Depolarizing Agents; Peptides; Potassium; Sea Anemones; Tetrodotoxin; Veratridine; Xanthines

1979
Voltage-sensitive calcium channels regulate guanosine 3',5'-cyclic monophosphate levels in neuroblastoma cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1978, Volume: 75, Issue:12

    Topics: Carbachol; Cell Line; Cobalt; Cyclic AMP; Cyclic GMP; Gallopamil; Ion Channels; Membrane Potentials; Neurons; Potassium; Receptors, Muscarinic; Veratridine

1978
The mechanism of action of ionophore A 23187 on guinea pig intestinal smooth muscle.
    Canadian journal of physiology and pharmacology, 1979, Volume: 57, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Calcimycin; Calcium; Calcium Radioisotopes; Dioxolanes; Gallopamil; Guinea Pigs; In Vitro Techniques; Intestines; Muscle Contraction; Muscle, Smooth; Nifedipine; Tetrodotoxin; Veratridine

1979
Inhibition of sodium channels by D600.
    Molecular pharmacology, 1979, Volume: 15, Issue:1

    Topics: Binding, Competitive; Calcium; Cells, Cultured; Gallopamil; Ion Channels; Myocardium; Neoplasms, Experimental; Neuroblastoma; Sodium; Verapamil; Veratridine

1979
Developmental changes in the sensitivity of embryonic heart cells to tetrodotoxin and D600.
    Developmental biology, 1978, Volume: 65, Issue:1

    Topics: Age Factors; Animals; Biological Transport; Chick Embryo; Culture Techniques; Electric Conductivity; Gallopamil; Heart; Myocardial Contraction; Sodium; Tetrodotoxin; Verapamil; Veratridine

1978
The effects of chronic depolarization on L-type 1,4-dihydropyridine-sensitive, voltage-dependent Ca2+ channels in chick neural retina and rat cardiac cells.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:7

    Topics: Animals; Calcimycin; Calcium Channels; Cells, Cultured; Chick Embryo; Dihydropyridines; Down-Regulation; Gallopamil; Heart; In Vitro Techniques; Kinetics; Myocardium; Neuromuscular Depolarizing Agents; Neurons; Potassium; Rats; Retina; Veratridine

1991
GABA inhibits the rise in cytosolic free calcium concentration in depolarized immature cerebellar Purkinje cells.
    Neuroscience letters, 1991, Jan-28, Volume: 122, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aging; Animals; Calcium; Cerebellum; Cytosol; Gallopamil; gamma-Aminobutyric Acid; Kinetics; Purkinje Cells; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Veratridine

1991
Response of cytosolic calcium to anoxia and cyanide in cultured glomus cells of newborn rabbit carotid body.
    Brain research, 1991, Jun-14, Volume: 551, Issue:1-2

    Topics: Animals; Animals, Newborn; Calcium; Carotid Body; Cells, Cultured; Cyanides; Cytosol; Gallopamil; Hypoxia; Rabbits; Tetrodotoxin; Veratridine

1991
Inhibition by ouabain and veratridine of acetylcholine-evoked phasic contraction in the guinea-pig taenia coli.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:6

    Topics: Acetylcholine; Amiloride; Animals; Calcium; Colon; Dose-Response Relationship, Drug; Fluorometry; Fura-2; Gallopamil; Guinea Pigs; Muscle Contraction; Muscle, Smooth; Ouabain; Potassium; Sodium; Veratridine

1991
Activation and inactivation of oxytocin and vasopressin release from isolated nerve endings (neurosecretosomes) of the rat neurohypophysis.
    Journal of neurochemistry, 1991, Volume: 57, Issue:2

    Topics: Animals; Calcium; Calcium Channel Blockers; Gallopamil; Ionomycin; Kinetics; Male; Membrane Potentials; Nerve Endings; Oxytocin; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains; Vasopressins; Veratridine

1991
Spontaneous and secretagogue-induced changes in cytosolic free Ca concentration measured by microfluorimetry with fura-2 on single bovine adrenal chromaffin cells.
    The Japanese journal of physiology, 1989, Volume: 39, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Adrenal Medulla; Animals; Benzofurans; Calcium; Cattle; Cells, Cultured; Cytophotometry; Cytosol; Fluorescent Dyes; Fura-2; Gallopamil; In Vitro Techniques; Meglumine; Nicotine; Tetrodotoxin; Veratridine

1989
Regulation of muscarinic acetylcholine receptor number in cultured neuronal cells by chronic membrane depolarization.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Line; Cobalt; Cyclic GMP; Gallopamil; Membrane Potentials; Mice; Neurons; Quinuclidinyl Benzilate; Receptors, Muscarinic; Tetrodotoxin; Veratridine

1987
Pulsatile release of gonadotropin-releasing hormone (GnRH) from the rat hypothalamus in vitro: calcium and glucose dependency and inhibition by superactive GnRH analogs.
    Endocrinology, 1987, Volume: 121, Issue:3

    Topics: Animals; Buserelin; Calcium; Egtazic Acid; Gallopamil; Glucose; Gonadotropin-Releasing Hormone; Hypothalamus; Male; Periodicity; Rats; Rats, Inbred Strains; Triptorelin Pamoate; Veratridine

1987
Depolarization-induced increases in intracellular free calcium detected in single cultured neuronal cells.
    Neuroscience letters, 1984, Oct-12, Volume: 51, Issue:2

    Topics: Calcium; Cell Line; Cobalt; Gallopamil; Ion Channels; Ionophores; Membrane Potentials; Neurons; Nicotinic Acids; Nimodipine; Potassium; Veratridine

1984
Ionic channels involved in the LHRH and SRIF release from rat mediobasal hypothalamus.
    Neuroendocrinology, 1981, Volume: 32, Issue:3

    Topics: Animals; Calcium; Cell Membrane; Gallopamil; Gonadotropin-Releasing Hormone; Hypothalamus; In Vitro Techniques; Ion Channels; Magnesium; Male; Potassium; Rats; Sodium; Somatostatin; Veratridine

1981
Organic calcium channel blockers enhance [3H]purine release from rat brain cortical synaptosomes.
    Neurochemical research, 1984, Volume: 9, Issue:8

    Topics: Adenosine; Animals; Calcium Channel Blockers; Cerebral Cortex; Diltiazem; Egtazic Acid; Gallopamil; Glutamates; Glutamic Acid; Male; Mitochondria; Nifedipine; Potassium; Purines; Rats; Rats, Inbred Strains; Synaptosomes; Veratridine

1984
Effect of trifluoperazine, D600, and phenytoin on depolarization- and thyrotropin-releasing hormone-induced thyrotropin release from rat pituitary tissue.
    Endocrinology, 1981, Volume: 108, Issue:6

    Topics: Animals; Calcium; Gallopamil; Ion Channels; Male; Membrane Potentials; Phenytoin; Pituitary Gland, Anterior; Potassium; Rats; Sodium; Thyrotropin; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil; Veratridine

1981
Structure-function relationship of calcium ion channel antagonists at the pituitary gonadotrope.
    Endocrinology, 1983, Volume: 113, Issue:5

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Female; Gallopamil; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Pituitary Gland; Rats; Structure-Activity Relationship; Verapamil; Veratridine

1983
Veratridine and ouabain stimulate calcium-dependent prolactin release.
    Endocrinology, 1983, Volume: 113, Issue:4

    Topics: Animals; Bromocriptine; Calcium; Cells, Cultured; Gallopamil; Male; Ouabain; Pituitary Gland, Anterior; Prolactin; Rats; Sodium; Tetrodotoxin; Verapamil; Veratridine; Veratrine

1983
Inhibition of calcium uptake, sodium uptake, and catecholamine secretion by methoxyverapamil (D600) in primary cultures of adrenal medulla cells.
    Journal of neurochemistry, 1983, Volume: 40, Issue:4

    Topics: Adrenal Medulla; Animals; Biological Transport, Active; Calcium; Catecholamines; Cattle; Cells, Cultured; Gallopamil; Kinetics; Nicotine; Sodium; Tetrodotoxin; Verapamil; Veratridine

1983
Calcium uptake and catecholamine secretion by cultured bovine adrenal medulla cells.
    Journal of neurochemistry, 1982, Volume: 38, Issue:2

    Topics: Adrenal Medulla; Animals; Calcium; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Dose-Response Relationship, Drug; Gallopamil; Nicotine; Potassium; Time Factors; Tubocurarine; Veratridine

1982
Ryanodine alters the rate of acetylcholine receptor synthesis in chick skeletal muscle cell cultures.
    The Journal of biological chemistry, 1981, Dec-25, Volume: 256, Issue:24

    Topics: Acetylcholinesterase; Alkaloids; Animals; Cell Membrane; Cells, Cultured; Chick Embryo; Dantrolene; Gallopamil; Kinetics; Muscles; Receptors, Cholinergic; Ryanodine; Veratridine

1981
Acetylcholine-induced, calcium-dependent norepinephrine outflow from peripheral human lymphocytes.
    Journal of neuroimmunology, 1998, Jul-01, Volume: 87, Issue:1-2

    Topics: Acetylcholine; Adult; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Female; Gallopamil; Humans; Ionomycin; Levodopa; Lymphocytes; Male; Norepinephrine; Tyrosine; Veratridine

1998