gallopamil and colforsin

gallopamil has been researched along with colforsin in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19909 (47.37)18.7374
1990's9 (47.37)18.2507
2000's0 (0.00)29.6817
2010's1 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Alibhai, KN; Huizinga, JD; Richardson, D1
Dolphin, AC1
Efrat, S; Fleischer, N; Surana, M1
Höllt, V; Kley, N; Loeffler, JP; Pittius, CW1
Rorsman, P1
Afar, R; Geertsen, S; Quik, M; Trifaró, JM1
Auguet, M; Braquet, P; Clostre, F; Delaflotte, S; Pirotzky, E1
Critchlow, LM; Hoskins, DD; Vijayaraghavan, S1
Dave, JR; Eiden, LE; Eskay, RL; Lozovsky, D; Waschek, JA1
Henquin, JC; Meissner, HP1
Dannies, PS; Delbeke, D; Scammell, JG1
Huizinga, JD; Liu, LW1
Alekseev, AE; Kokoz, YM; Korystova, AF; Mavlyutova, DA1
Bernhardt, SJ; Lindemann, B; Naim, M; Zehavi, U1
Fleischer, N; Leiser, M1
Sjöholm, A1
Laychock, SG; Lee, B1

Other Studies

19 other study(ies) available for gallopamil and colforsin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
On the pharmacological and physiological role of glibenclamide-sensitive potassium channels in colonic smooth muscle.
    Pharmacology & toxicology, 1992, Volume: 71, Issue:5

    Topics: Animals; Benzopyrans; Carbachol; Colforsin; Colon; Cromakalim; Dogs; Drug Interactions; Electric Stimulation; Female; Gallopamil; Glyburide; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Stereoisomerism

1992
Ca2+ channel currents in rat sensory neurones: interaction between guanine nucleotides, cyclic AMP and Ca2+ channel ligands.
    The Journal of physiology, 1991, Volume: 432

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Drug Interactions; Gallopamil; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Neurons, Afferent; Nicotinic Acids; Oxadiazoles; Phosphorylation; Rats

1991
Glucose induces insulin gene transcription in a murine pancreatic beta-cell line.
    The Journal of biological chemistry, 1991, Jun-15, Volume: 266, Issue:17

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Line; Cell Nucleus; Colforsin; Cyclic AMP; Gallopamil; Genes; Glucose; Insulin; Insulinoma; Kinetics; Mice; Mice, Transgenic; Pancreatic Neoplasms; Promoter Regions, Genetic; Rats; Transcription, Genetic; Uridine Triphosphate

1991
Involvement of ion channels in the induction of proenkephalin A gene expression by nicotine and cAMP in bovine chromaffin cells.
    The Journal of biological chemistry, 1987, Mar-25, Volume: 262, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Enkephalins; Gallopamil; Gene Expression Regulation; Ion Channels; Nicotine; Nifedipine; Protein Precursors; RNA, Messenger; Sodium; Tubocurarine; Verapamil

1987
Two types of Ca2+ currents with different sensitivities to organic Ca2+ channel antagonists in guinea pig pancreatic alpha 2 cells.
    The Journal of general physiology, 1988, Volume: 91, Issue:2

    Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Cobalt; Colforsin; Electrophysiology; Gallopamil; Guinea Pigs; Ion Channels; Islets of Langerhans; Membrane Potentials; Nifedipine; Tetrodotoxin

1988
Regulation of alpha-bungarotoxin sites in chromaffin cells in culture by nicotinic receptor ligands, K+, and cAMP.
    Molecular pharmacology, 1988, Volume: 34, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenylyl Cyclases; Adrenal Medulla; alpha7 Nicotinic Acetylcholine Receptor; Biological Transport; Bucladesine; Bungarotoxins; Carbachol; Cells, Cultured; Colforsin; Enzyme Activation; Gallopamil; Nicotine; Norepinephrine; Potassium; Receptors, Cholinergic; Receptors, Nicotinic; Tubocurarine

1988
Effects of atrial natriuretic factor (ANF) on phenylephrine-triggered intra- and extracellular calcium dependent contraction in rat aorta.
    Journal of autonomic pharmacology, 1989, Volume: 9, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Atrial Natriuretic Factor; Calcium; Colforsin; Cyclic AMP; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains

1989
Evidence for a role for cellular alkalinization in the cyclic adenosine 3',5'-monophosphate-mediated initiation of motility in bovine caput spermatozoa.
    Biology of reproduction, 1985, Volume: 32, Issue:3

    Topics: Animals; Bicarbonates; Cattle; Colforsin; Cyclic AMP; Dipyridamole; Diterpenes; Epididymis; Gallopamil; Hydrogen-Ion Concentration; Ionophores; Male; Sperm Motility; Spermatozoa; Theophylline

1985
Calcium-independent and calcium-dependent mechanisms regulate corticotropin-releasing factor-stimulated proopiomelanocortin peptide secretion and messenger ribonucleic acid production.
    Endocrinology, 1987, Volume: 120, Issue:1

    Topics: Animals; Barium; Calcium; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Gallopamil; Gene Expression Regulation; Male; Pituitary Gland, Anterior; Pro-Opiomelanocortin; Prolactin; Rats; RNA, Messenger

1987
The ionic, electrical, and secretory effects of endogenous cyclic adenosine monophosphate in mouse pancreatic B cells: studies with forskolin.
    Endocrinology, 1984, Volume: 115, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Cobalt; Colforsin; Cyclic AMP; Diterpenes; Dose-Response Relationship, Drug; Electrophysiology; Female; Gallopamil; Glucose; Insulin; Islets of Langerhans; Membrane Potentials; Mice; Rubidium

1984
Difference in calcium requirements for forskolin-induced release of prolactin from normal pituitary cells and GH4C1 cells in culture.
    Endocrinology, 1984, Volume: 114, Issue:4

    Topics: Animals; Antihypertensive Agents; Calcium; Cell Line; Cells, Cultured; Colforsin; Cyclic AMP; Diterpenes; Gallopamil; Kinetics; Male; Pituitary Gland, Anterior; Pituitary Neoplasms; Potassium; Rats; Rats, Inbred Strains

1984
Canine colonic circular muscle generates action potentials without the pacemaker component.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Barium; Calcium Channels; Colforsin; Colon; Dogs; Electric Stimulation; Electrophysiology; Female; Gallopamil; In Vitro Techniques; Male; Microelectrodes; Muscle, Smooth; Neuromuscular Depolarizing Agents; Potassium; Potassium Channels

1994
Potential-dependent Ca2+ currents in isolated heart cells of hibernators.
    Biochemistry and molecular biology international, 1994, Volume: 33, Issue:2

    Topics: Animals; Calcium; Calcium Channels; Cells, Cultured; Colforsin; Electric Conductivity; Electrophysiology; Gallopamil; Heart; Hibernation; Isoproterenol; Membrane Potentials; Myocardium; Nifedipine; Patch-Clamp Techniques; Sciuridae

1994
Changes in IP3 and cytosolic Ca2+ in response to sugars and non-sugar sweeteners in transduction of sweet taste in the rat.
    The Journal of physiology, 1996, Jan-15, Volume: 490 ( Pt 2)

    Topics: Amiloride; Animals; Calcium; Carbohydrates; Colforsin; Cyclic AMP; Fluorescent Dyes; Fura-2; Gallopamil; Image Processing, Computer-Assisted; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Metals; Microscopy, Fluorescence; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Saccharin; Signal Transduction; Sucrose; Sweetening Agents; Taste Buds

1996
cAMP-dependent phosphorylation of the cardiac-type alpha 1 subunit of the voltage-dependent Ca2+ channel in a murine pancreatic beta-cell line.
    Diabetes, 1996, Volume: 45, Issue:10

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium Channels; Calcium Channels, L-Type; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophoresis, Polyacrylamide Gel; Gallopamil; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Macromolecular Substances; Mice; Myocardium; Phosphoproteins; Phosphorylation

1996
Glucose stimulates islet beta-cell mitogenesis through GTP-binding proteins and by protein kinase C-dependent mechanisms.
    Diabetes, 1997, Volume: 46, Issue:7

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Atrial Natriuretic Factor; Calcium Channel Blockers; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; DNA; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gallopamil; Glucose; GTP-Binding Proteins; Insulin; Insulin Secretion; Ionomycin; Ionophores; Islets of Langerhans; Pertussis Toxin; Pregnancy; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Thionucleotides; Virulence Factors, Bordetella

1997
Atrial natriuretic peptide and cyclic nucleotides affect glucose-induced Ca2+ responses in single pancreatic islet beta-cells: correlation with (Ca[2+] + Mg2+)-ATPase activity.
    Diabetes, 1997, Volume: 46, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atrial Natriuretic Factor; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gallopamil; Glucose; Islets of Langerhans; Male; Nucleotides, Cyclic; Rats; Rats, Sprague-Dawley; Thapsigargin

1997