gallamine triethiodide and tacrine

gallamine triethiodide has been researched along with tacrine in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's2 (22.22)18.2507
2000's4 (44.44)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Ellis, J; Seidenberg, M1
Cross, AJ; Green, AR; Hunter, AJ; Jones, JA; Murray, TK1
Aldunate, R; Inestrosa, NC; Muñoz, FJ1
Ellis, J; Huang, XP1
Cieslik, JS; Elsinghorst, PW; Gütschow, M; Mohr, K; Tränkle, C1
Christian, L; Gütschow, M; Inhester, T; Petzold, S; Pietsch, M1
Agnusdei, M; Belinskaya, T; Borriello, M; Brindisi, M; Butini, S; Campiani, G; Catalanotti, B; Fattorusso, C; Fiorini, I; Gemma, S; Nacci, V; Novellino, E; Panico, A; Persico, M; Ros, S; Saxena, A1

Other Studies

9 other study(ies) available for gallamine triethiodide and tacrine

ArticleYear
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Two allosteric modulators interact at a common site on cardiac muscarinic receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Gallamine Triethiodide; Gallic Acid; In Vitro Techniques; Myocardium; Obidoxime Chloride; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Tacrine

1992
The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Aminoacridines; Animals; Behavior, Animal; Brain Chemistry; Cholinesterase Inhibitors; Gallamine Triethiodide; In Vitro Techniques; Male; Mice; Myocardium; N-Methylscopolamine; Nicotine; Oxotremorine; Parasympathetic Nervous System; Physostigmine; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Tacrine

1989
Peripheral binding site is involved in the neurotrophic activity of acetylcholinesterase.
    Neuroreport, 1999, Nov-26, Volume: 10, Issue:17

    Topics: Acetylcholinesterase; Animals; Binding Sites; Cell Division; Cells, Cultured; Cholinesterase Inhibitors; DNA; Dose-Response Relationship, Drug; Edrophonium; Formazans; Gallamine Triethiodide; Nerve Growth Factors; Neurites; Neurons; PC12 Cells; Propidium; Protein Structure, Tertiary; Rats; Spinal Cord; Tacrine; Tetrazolium Salts

1999
Mutational disruption of a conserved disulfide bond in muscarinic acetylcholine receptors attenuates positive homotropic cooperativity between multiple allosteric sites and has subtype-dependent effects on the affinities of muscarinic allosteric ligands.
    Molecular pharmacology, 2007, Volume: 71, Issue:3

    Topics: Allosteric Site; Amino Acid Sequence; Base Sequence; Disulfides; Gallamine Triethiodide; Isoindoles; Molecular Sequence Data; Mutagenesis, Site-Directed; N-Methylscopolamine; Phthalimides; Receptors, Muscarinic; Structure-Activity Relationship; Tacrine

2007
First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor.
    Journal of medicinal chemistry, 2007, Nov-15, Volume: 50, Issue:23

    Topics: Acetylcholinesterase; Allosteric Regulation; Animals; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Drug Design; Gallamine Triethiodide; Humans; In Vitro Techniques; Ligands; Models, Molecular; Myocardium; Radioligand Assay; Receptor, Muscarinic M2; Structure-Activity Relationship; Swine; Tacrine

2007
Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile.
    The FEBS journal, 2009, Volume: 276, Issue:8

    Topics: Acetonitriles; Acetylcholinesterase; Acetylthiocholine; Animals; Cholinesterase Inhibitors; Electrophorus; Gallamine Triethiodide; Hydrolysis; Kinetics; Tacrine

2009
Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Computational Biology; Crystallography, X-Ray; Drug Design; Humans; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Tacrine

2008