gallamine triethiodide has been researched along with tacrine in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (11.11) | 18.7374 |
1990's | 2 (22.22) | 18.2507 |
2000's | 4 (44.44) | 29.6817 |
2010's | 2 (22.22) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ | 1 |
Ekins, S; Williams, AJ; Xu, JJ | 1 |
Ellis, J; Seidenberg, M | 1 |
Cross, AJ; Green, AR; Hunter, AJ; Jones, JA; Murray, TK | 1 |
Aldunate, R; Inestrosa, NC; Muñoz, FJ | 1 |
Ellis, J; Huang, XP | 1 |
Cieslik, JS; Elsinghorst, PW; Gütschow, M; Mohr, K; Tränkle, C | 1 |
Christian, L; Gütschow, M; Inhester, T; Petzold, S; Pietsch, M | 1 |
Agnusdei, M; Belinskaya, T; Borriello, M; Brindisi, M; Butini, S; Campiani, G; Catalanotti, B; Fattorusso, C; Fiorini, I; Gemma, S; Nacci, V; Novellino, E; Panico, A; Persico, M; Ros, S; Saxena, A | 1 |
9 other study(ies) available for gallamine triethiodide and tacrine
Article | Year |
---|---|
Developing structure-activity relationships for the prediction of hepatotoxicity.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes | 2010 |
A predictive ligand-based Bayesian model for human drug-induced liver injury.
Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands | 2010 |
Two allosteric modulators interact at a common site on cardiac muscarinic receptors.
Topics: Allosteric Regulation; Animals; Binding Sites; Gallamine Triethiodide; Gallic Acid; In Vitro Techniques; Myocardium; Obidoxime Chloride; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Tacrine | 1992 |
The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro.
Topics: Aminoacridines; Animals; Behavior, Animal; Brain Chemistry; Cholinesterase Inhibitors; Gallamine Triethiodide; In Vitro Techniques; Male; Mice; Myocardium; N-Methylscopolamine; Nicotine; Oxotremorine; Parasympathetic Nervous System; Physostigmine; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Tacrine | 1989 |
Peripheral binding site is involved in the neurotrophic activity of acetylcholinesterase.
Topics: Acetylcholinesterase; Animals; Binding Sites; Cell Division; Cells, Cultured; Cholinesterase Inhibitors; DNA; Dose-Response Relationship, Drug; Edrophonium; Formazans; Gallamine Triethiodide; Nerve Growth Factors; Neurites; Neurons; PC12 Cells; Propidium; Protein Structure, Tertiary; Rats; Spinal Cord; Tacrine; Tetrazolium Salts | 1999 |
Mutational disruption of a conserved disulfide bond in muscarinic acetylcholine receptors attenuates positive homotropic cooperativity between multiple allosteric sites and has subtype-dependent effects on the affinities of muscarinic allosteric ligands.
Topics: Allosteric Site; Amino Acid Sequence; Base Sequence; Disulfides; Gallamine Triethiodide; Isoindoles; Molecular Sequence Data; Mutagenesis, Site-Directed; N-Methylscopolamine; Phthalimides; Receptors, Muscarinic; Structure-Activity Relationship; Tacrine | 2007 |
First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor.
Topics: Acetylcholinesterase; Allosteric Regulation; Animals; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Drug Design; Gallamine Triethiodide; Humans; In Vitro Techniques; Ligands; Models, Molecular; Myocardium; Radioligand Assay; Receptor, Muscarinic M2; Structure-Activity Relationship; Swine; Tacrine | 2007 |
Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile.
Topics: Acetonitriles; Acetylcholinesterase; Acetylthiocholine; Animals; Cholinesterase Inhibitors; Electrophorus; Gallamine Triethiodide; Hydrolysis; Kinetics; Tacrine | 2009 |
Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.
Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Computational Biology; Crystallography, X-Ray; Drug Design; Humans; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Tacrine | 2008 |