gallamine triethiodide and oxotremorine

gallamine triethiodide has been researched along with oxotremorine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199011 (50.00)18.7374
1990's8 (36.36)18.2507
2000's2 (9.09)29.6817
2010's1 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bernhardt, G; Gmeiner, P; Hübner, H; Keller, M; Pegoli, A; She, X; Wifling, D1
Biggs, DF; Yang, ZJ1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Aas, P1
Boselli, C; Kenakin, T1
Cross, AJ; Green, AR; Hunter, AJ; Jones, JA; Murray, TK1
Delen, FM; Ehlert, FJ; Friedman, DJ; Self, DW; Yun, SH1
Chaudhry, IA; Duncalf, D; Foldes, FF; Goldiner, PL; Harsing, LG; Kobayashi, O; Nagashima, H; Vizi, ES1
Limas, C; Limas, CJ1
Choo, LK; Mitchelson, F1
Ehlert, FJ1
Constanti, A; Williams, SH1
Mulder, AH; Schoffelmeer, AN; Van Vliet, BJ; Wardeh, G1
Ehlert, FJ; Jenden, DJ1
Dóda, M; Gellén, B; György, L1
De Neef, P; Domenach, V; Vandermeers, A; Vandermeers-Piret, MC; Waelbroeck, M1
Cheng, JT; Hung, YC; Lin, SN; Tong, YC1
Christopoulos, A; Mitchelson, F1
Dement, WC; Mignot, E; Nishino, S; Reid, MS; Siegel, JM; Tafti, M1
Fukaya, M; Fukudome, Y; Kano, M; Manabe, T; Matsui, M; Ohno-Shosaku, T; Omori, Y; Taketo, MM; Tsubokawa, H; Watanabe, M1
Antony, J; Grossmüller, M; Holzgrabe, U; Mohr, K; Tränkle, C1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1

Other Studies

22 other study(ies) available for gallamine triethiodide and oxotremorine

ArticleYear
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M
    Journal of medicinal chemistry, 2017, 04-27, Volume: 60, Issue:8

    Topics: Benzodiazepinones; Binding Sites; Molecular Dynamics Simulation; Muscarinic Antagonists; Radioisotopes; Receptor, Muscarinic M2

2017
Muscarinic receptors and parasympathetic neurotransmission in guinea-pig trachea.
    European journal of pharmacology, 1991, Feb-14, Volume: 193, Issue:3

    Topics: Animals; Arecoline; Bethanidine; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Muscarinic Antagonists; Oxotremorine; Parasympathetic Nervous System; Pilocarpine; Pirenzepine; Receptors, Muscarinic; Synaptic Transmission; Trachea

1991
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Prejunctional control of cholinergic nerves in airway smooth muscle exerted by muscarinic, purinergic and glutamergic receptors.
    Progress in brain research, 1990, Volume: 84

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aspartic Acid; Bronchi; Diamines; Gallamine Triethiodide; Glutamates; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxotremorine; Parasympatholytics; Rats; Rats, Inbred Strains; Receptors, Glutamate; Receptors, Muscarinic; Receptors, Neurotransmitter; Receptors, Purinergic; Trachea

1990
Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: Allosteric Regulation; Animals; Atropine; Binding Sites; Carbachol; Dose-Response Relationship, Drug; Gallamine Triethiodide; In Vitro Techniques; Male; Muscarine; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine; Trachea

1989
The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Aminoacridines; Animals; Behavior, Animal; Brain Chemistry; Cholinesterase Inhibitors; Gallamine Triethiodide; In Vitro Techniques; Male; Mice; Myocardium; N-Methylscopolamine; Nicotine; Oxotremorine; Parasympathetic Nervous System; Physostigmine; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Tacrine

1989
Coupling of subtypes of the muscarinic receptor to adenylate cyclase in the corpus striatum and heart.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Gallamine Triethiodide; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Pirenzepine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives

1989
Direct evidence that pancuronium and gallamine enhance the release of norepinephrine from the atrial sympathetic nerve by inhibiting prejunctional muscarinic receptors.
    Journal of the autonomic nervous system, 1987, Volume: 18, Issue:1

    Topics: Adrenergic Fibers; Animals; Atropine; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; Male; Norepinephrine; Oxotremorine; Pancuronium; Receptors, Muscarinic; Tubocurarine; Vecuronium Bromide

1987
Carbachol induces desensitization of cardiac beta-adrenergic receptors through muscarinic M1 receptors.
    Biochemical and biophysical research communications, 1985, Apr-30, Volume: 128, Issue:2

    Topics: Animals; Carbachol; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Gallamine Triethiodide; Heart; Myocardium; Oxotremorine; Propanolamines; Protein Kinase C; Protein Kinases; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Muscarinic; Time Factors; Tissue Distribution

1985
Displacement of [3H]oxotremorine-M binding by muscarinic antagonists in guinea-pig atrial and ileal membrane homogenates.
    European journal of pharmacology, 1988, Jul-07, Volume: 151, Issue:2

    Topics: Animals; Atropine; Binding, Competitive; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Oxotremorine; Parasympatholytics; Piperidines

1988
Gallamine allosterically antagonizes muscarinic receptor-mediated inhibition of adenylate cyclase activity in the rat myocardium.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Algorithms; Animals; Dose-Response Relationship, Drug; Gallamine Triethiodide; Heart; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1988
A quantitative study of the effects of some muscarinic antagonists on the guinea-pig olfactory cortex slice.
    British journal of pharmacology, 1988, Volume: 93, Issue:4

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Drug Interactions; Evoked Potentials; Gallamine Triethiodide; Guinea Pigs; In Vitro Techniques; Oxotremorine; Parasympathomimetics; Pirenzepine

1988
Muscarine receptor-mediated modulation of [3H]dopamine and [14C]acetylcholine release from rat neostriatal slices: selective antagonism by gallamine but not pirenzepine.
    European journal of pharmacology, 1986, Sep-09, Volume: 128, Issue:3

    Topics: Acetylcholine; Animals; Corpus Striatum; Dopamine; Gallamine Triethiodide; In Vitro Techniques; Male; Oxotremorine; Parasympatholytics; Pirenzepine; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1986
The binding of a 2-chloroethylamine derivative of oxotremorine (BM 123) to muscarinic receptors in the rat cerebral cortex.
    Molecular pharmacology, 1985, Volume: 28, Issue:2

    Topics: Alkylation; Animals; Atropine; Benzodiazepinones; Binding Sites; Binding, Competitive; Cerebral Cortex; Gallamine Triethiodide; Kinetics; N-Methylscopolamine; Oxotremorine; Pirenzepine; Pyrrolidinones; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Structure-Activity Relationship; Thiosulfates

1985
Influence of the surgical isolation of the hypothalamus on oxotremorine-induced rage reaction and sympathetic response in the cat.
    Acta physiologica Academiae Scientiarum Hungaricae, 1972, Volume: 42, Issue:2

    Topics: Anger; Animals; Arecoline; Behavior, Animal; Cats; Female; Gallamine Triethiodide; Hypothalamus; Male; Muscle Contraction; Nictitating Membrane; Oxotremorine; Pentylenetetrazole

1972
Binding of the labelled muscarinic toxin 125I-MT1 to rat brain muscarinic M1 receptors.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Alkaloids; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Elapid Venoms; Furans; Gallamine Triethiodide; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Naphthalenes; Oxotremorine; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Protein Binding; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Synaptic Membranes; Tubocurarine

1996
Pharmacological characterization of the muscarinic receptor subtypes responsible for the contractile response in the rat urinary bladder.
    Journal of autonomic pharmacology, 1997, Volume: 17, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Analysis of Variance; Animals; Bethanechol; Diamines; Dose-Response Relationship, Drug; Female; Gallamine Triethiodide; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nicotinic Antagonists; Oxotremorine; Parasympatholytics; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Structure-Activity Relationship; Urinary Bladder

1997
Application of an allosteric ternary complex model to the technique of pharmacological resultant analysis.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:8

    Topics: Animals; Binding, Competitive; Gallamine Triethiodide; Kinetics; Mathematical Computing; Models, Biological; Muscarinic Agonists; Muscarinic Antagonists; Nicotinic Antagonists; Oxotremorine; Pharmacology; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine; Trachea

1997
Neuropharmacological characterization of basal forebrain cholinergic stimulated cataplexy in narcoleptic canines.
    Experimental neurology, 1998, Volume: 151, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Animals; Atropine; Behavior, Animal; Carbachol; Cataplexy; Cholinergic Fibers; Dogs; Feeding Behavior; Female; GABA Agonists; Gallamine Triethiodide; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Muscimol; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Oxotremorine; Piperidines; Pirenzepine; Prosencephalon

1998
Two distinct classes of muscarinic action on hippocampal inhibitory synapses: M2-mediated direct suppression and M1/M3-mediated indirect suppression through endocannabinoid signalling.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: Animals; Animals, Newborn; Benzoxazines; Blotting, Western; Brain; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Carrier Proteins; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Endocannabinoids; GABA Plasma Membrane Transport Proteins; Gallamine Triethiodide; Heterozygote; Hippocampus; Immunohistochemistry; In Vitro Techniques; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Knockout; Morpholines; Muscarinic Agonists; Naphthalenes; Neural Inhibition; Nicotinic Antagonists; Oxotremorine; Patch-Clamp Techniques; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Signal Transduction; Synapses

2004
Allosteric site in M2 acetylcholine receptors: evidence for a major conformational change upon binding of an orthosteric agonist instead of an antagonist.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:4

    Topics: Allosteric Regulation; Allosteric Site; Animals; Binding, Competitive; Gallamine Triethiodide; In Vitro Techniques; Isoindoles; Muscarinic Agonists; Muscarinic Antagonists; Myocardium; N-Methylscopolamine; Obidoxime Chloride; Oxotremorine; Phthalimides; Protein Conformation; Pyridinium Compounds; Receptor, Muscarinic M2; Swine

2006
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998