gallamine triethiodide and afdx 116

gallamine triethiodide has been researched along with afdx 116 in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19906 (33.33)18.7374
1990's10 (55.56)18.2507
2000's2 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kimura, T; Satoh, S; Shimamura, T1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Birdsall, NJ; Eveleigh, P; Hulme, EC; Pedder, EK; Poyner, D1
Bast, A; Doelman, CJ; Nagtegaal, JE; Rodrigues de Miranda, JF; Sprong, RC1
Ashe, JH; Olito, AC; Yarosh, CA1
Michel, AD; Whiting, RL2
Elzinga, CR; Meurs, H; Roffel, AF; Zaagsma, J2
Gilbert, MJ; Newberry, NR1
Delen, FM; Ehlert, FJ; Friedman, DJ; Self, DW; Yun, SH1
Brown, DA; Marrion, NV; Marsh, SJ; Smart, TG1
Kunysz, EL; Michel, AD; Whiting, RL1
Hamstra, JJ; Roffel, AF; Santing, RE; ten Berge, RE; Zaagsma, J1
Bargas, J; Galarraga, E; Hernández-Echeagaray, E1
Fitzgerald, RS; Shirahata, M; Wang, HY1
Christopoulos, A; Lanzafame, A; Mitchelson, F1
Kovacs, I; Roeske, WR; Varga, EV; Waite, SL; Yamamura, HI1

Other Studies

18 other study(ies) available for gallamine triethiodide and afdx 116

ArticleYear
Effects of pirenzepine, AF-DX 116 and gallamine on the release of catecholamines from the dog adrenal gland in response to splanchnic nerve stimulation: interaction of M1 and M2 receptors with nicotinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Adrenal Glands; Animals; Catecholamines; Dogs; Electric Stimulation; Female; Gallamine Triethiodide; Hexamethonium; Hexamethonium Compounds; Male; Parasympatholytics; Pirenzepine; Receptors, Muscarinic; Receptors, Nicotinic; Splanchnic Nerves

1991
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Modulation of the structure-binding relationships of antagonists for muscarinic acetylcholine receptor subtypes.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Animals; Centrifugation; Cerebral Cortex; Cholic Acids; Digitonin; Gallamine Triethiodide; Heart; In Vitro Techniques; Lacrimal Apparatus; Membranes; Muscarinic Antagonists; Myocardium; Parasympatholytics; Piperidines; Pirenzepine; Rats; Structure-Activity Relationship

1991
Prejunctional muscarinic receptors on cholinergic nerves in guinea pig airways are of the M2 subtype.
    European journal of pharmacology, 1991, Jan-25, Volume: 193, Issue:1

    Topics: Animals; Diamines; Electric Stimulation; Gallamine Triethiodide; Guinea Pigs; In Vitro Techniques; Male; Parasympathetic Nervous System; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1991
Differential effects of the muscarinic M2 antagonists, AF-DX 116 and gallamine, on single neurons of rabbit sympathetic ganglia.
    Neuropharmacology, 1990, Volume: 29, Issue:8

    Topics: Action Potentials; Animals; Electrophysiology; Gallamine Triethiodide; Ganglia, Sympathetic; Membrane Potentials; Membranes; Methacholine Compounds; Neurons; Parasympatholytics; Pirenzepine; Rabbits

1990
The binding of [3H]4-diphenylacetoxy-N-methylpiperidine methiodide to longitudinal ileal smooth muscle muscarinic receptors.
    European journal of pharmacology, 1990, Feb-06, Volume: 176, Issue:2

    Topics: Animals; Binding, Competitive; Diamines; Gallamine Triethiodide; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Piperidines; Pirenzepine; Receptors, Muscarinic

1990
Allosteric interactions of three muscarine antagonists at bovine tracheal smooth muscle and cardiac M2 receptors.
    European journal of pharmacology, 1989, Mar-07, Volume: 172, Issue:1

    Topics: Animals; Cattle; Dexetimide; Diamines; Gallamine Triethiodide; Heart; In Vitro Techniques; Membrane Proteins; Muscle, Smooth; Parasympatholytics; Pirenzepine; Receptors, Muscarinic; Trachea

1989
Biphasic dose-response curve to muscarine on the rat superior cervical ganglion.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Animals; Dose-Response Relationship, Drug; Gallamine Triethiodide; Ganglia, Spinal; In Vitro Techniques; Muscarine; Pertussis Toxin; Pirenzepine; Rats; Virulence Factors, Bordetella

1989
Coupling of subtypes of the muscarinic receptor to adenylate cyclase in the corpus striatum and heart.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Gallamine Triethiodide; Male; Myocardium; N-Methylscopolamine; Oxotremorine; Pirenzepine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; RNA, Messenger; Scopolamine Derivatives

1989
Muscarinic suppression of the M-current in the rat sympathetic ganglion is mediated by receptors of the M1-subtype.
    British journal of pharmacology, 1989, Volume: 98, Issue:2

    Topics: Animals; Calcium; Gallamine Triethiodide; Ganglia, Spinal; Ganglia, Sympathetic; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Piperidines; Pirenzepine; Potassium Channels; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives

1989
Functional and direct binding studies using subtype selective muscarinic receptor antagonists.
    British journal of pharmacology, 1988, Volume: 93, Issue:3

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; Dicyclomine; Diphenylacetic Acids; Gallamine Triethiodide; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Myocardium; Phenethylamines; Phenylacetates; Pirenzepine; Receptors, Muscarinic

1988
Direct binding studies on ileal and cardiac muscarinic receptors.
    British journal of pharmacology, 1987, Volume: 92, Issue:4

    Topics: Animals; Gallamine Triethiodide; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Membranes; Muscle, Smooth; Myocardium; N-Methylscopolamine; Pirenzepine; Receptors, Muscarinic; Scopolamine Derivatives

1987
No evidence for a role of muscarinic M2 receptors in functional antagonism in bovine trachea.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Animals; Bronchoconstrictor Agents; Cattle; Dose-Response Relationship, Drug; Gallamine Triethiodide; Histamine; In Vitro Techniques; Isoproterenol; Methacholine Chloride; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Trachea

1995
Dysfunction of muscarinic M2 receptors after the early allergic reaction: possible contribution to bronchial hyperresponsiveness in allergic guinea-pigs.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Inhalation; Allergens; Animals; Asthma; Benzodiazepinones; Bronchial Hyperreactivity; Diamines; Disease Models, Animal; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart; Histamine; Hypersensitivity; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea

1995
3-Alpha-chloro-imperialine, a potent blocker of cholinergic presynaptic modulation of glutamatergic afferents in the rat neostriatum.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 4-Aminopyridine; Afferent Pathways; Animals; Atropine; Bicuculline; Carbachol; Cevanes; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; Gallamine Triethiodide; Muscarine; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Neurons; Pirenzepine; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Muscarinic; Synapses

1998
Acetylcholine is released from in vitro cat carotid bodies during hypoxic stimulation.
    Advances in experimental medicine and biology, 2000, Volume: 475

    Topics: Acetylcholine; Animals; Atropine; Carotid Body; Cats; Gallamine Triethiodide; Hypoxia; In Vitro Techniques; Mecamylamine; Parasympatholytics; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic

2000
The allosteric interaction of otenzepad (AF-DX 116) at muscarinic M2 receptors in guinea pig atria.
    European journal of pharmacology, 2001, Mar-30, Volume: 416, Issue:3

    Topics: Acetylcholine; Allosteric Regulation; Animals; Atropine; Carbachol; Cardiotonic Agents; Dexetimide; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart Atria; In Vitro Techniques; Kinetics; Male; Muscarinic Antagonists; N-Methylscopolamine; Nicotinic Antagonists; Parasympatholytics; Phthalimides; Pirenzepine; Quaternary Ammonium Compounds; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic

2001
Pharmacological comparison of the cloned human and rat M2 muscarinic receptor genes expressed in the murine fibroblast (B82) cell line.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Amino Acid Sequence; Animals; Carbachol; Cloning, Molecular; Cyclic AMP; Humans; Mice; Molecular Sequence Data; Muscarinic Agonists; Muscarinic Antagonists; Phosphatidylinositols; Radioligand Assay; Rats; Receptors, Muscarinic; Sequence Alignment; Sequence Homology, Amino Acid; Signal Transduction; Species Specificity

1998