Page last updated: 2024-09-04

gadolinium dtpa and mocetinostat

gadolinium dtpa has been researched along with mocetinostat in 13 studies

Compound Research Comparison

Studies
(gadolinium dtpa)
Trials
(gadolinium dtpa)
Recent Studies (post-2010)
(gadolinium dtpa)
Studies
(mocetinostat)
Trials
(mocetinostat)
Recent Studies (post-2010) (mocetinostat)
12,6546644,05121,7353908,606

Protein Interaction Comparison

ProteinTaxonomygadolinium dtpa (IC50)mocetinostat (IC50)
Histone deacetylase 3Homo sapiens (human)0.7851
Nuclear receptor corepressor 1Homo sapiens (human)0.022
Cytochrome P450 3A4Homo sapiens (human)0.57
Cytochrome P450 2D6Homo sapiens (human)0.102
Cytochrome P450 2C19Homo sapiens (human)0.102
Histone deacetylase 4Homo sapiens (human)0.5717
Histone deacetylase 1Homo sapiens (human)0.3433
Histone deacetylase 7Homo sapiens (human)0.6725
Histone deacetylase 2Homo sapiens (human)0.3537
Histone deacetylase 11 Homo sapiens (human)0.6386
Histone deacetylase 8Homo sapiens (human)0.6725
Histone deacetylase 6Homo sapiens (human)0.5717
Histone deacetylase 5Homo sapiens (human)0.6725
Nuclear receptor corepressor 2Homo sapiens (human)0.045

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (38.46)29.6817
2010's6 (46.15)24.3611
2020's2 (15.38)2.80

Authors

AuthorsStudies
Bogdanov, AA; Chen, JW; Querol, M1
Aikawa, E; Breckwoldt, MO; Chen, JW; Moskowitz, MA; Qiu, S; Rodriguez, E; Stangenberg, L; Weissleder, R1
Bogdanov, AA; DeLeo, MJ; Ford, JC; Gounis, MJ; Hong, B; Wakhloo, AK1
Bogdanov, A; Chen, JW; Chen, Y; Hamilton, AM; Hegele, RA; Querol, M; Reynolds, F; Rodriguez, E; Rogers, KA; Ronald, JA; Rutt, BK; Weissleder, R1
Mahmood, U1
Aikawa, E; Breckwoldt, MO; Chen, JW; Iwamoto, Y; Nahrendorf, M; Panizzi, P; Rodriguez, E; Su, HS; Weissleder, R1
Bogdanov, AA; Chueh, JY; Gounis, MJ; Kühn, AL; van der Bom, IM; Wakhloo, AK; Zheng, S1
Ali, M; Bure, L; Chen, JW; Hsieh, KL; Iwamoto, Y; Jacobs, AH; Li, D; Pulli, B; Schob, S; Wojtkiewicz, GR1
Bryan, RN1
Ali, M; Bure, L; Chen, JW; Choi, Y; Corey, KE; Guimaraes, AR; Iwamoto, Y; Masia, R; Pulli, B; Wang, C; Wojtkiewicz, G; Zeller, MW1
Bogdanov, AA; Caravan, P; Gounis, MJ; Hoang, DM; Leporati, A; Mazzanti, ML; Rodríguez-Rodríguez, A; Wadghiri, YZ; Wakhloo, AK; Weaver, JP1
Chen, JW; Cheng, D; Jalali Motlagh, N; Kuellenberg, EG; Schmidt, SP; Stocker, R; Wang, C; Wojtkiewicz, GR1
Cao, W; Chen, K; Lei, J; Li, Y; Liu, X; Liu, Y; Tan, B; Xia, Q; Xia, Z; Xiao, B; Zhong, L; Zhu, C; Zhu, J1

Other Studies

13 other study(ies) available for gadolinium dtpa and mocetinostat

ArticleYear
A paramagnetic contrast agent with myeloperoxidase-sensing properties.
    Organic & biomolecular chemistry, 2006, May-21, Volume: 4, Issue:10

    Topics: Contrast Media; Gadolinium; Gadolinium DTPA; Hydrogen Peroxide; Ligands; Magnetic Resonance Imaging; Peroxidase

2006
Tracking the inflammatory response in stroke in vivo by sensing the enzyme myeloperoxidase.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Nov-25, Volume: 105, Issue:47

    Topics: Animals; Disease Models, Animal; Gadolinium DTPA; Inflammation; Magnetic Resonance Imaging; Mice; Mice, Inbred C57BL; Peroxidase; Stroke

2008
Carotid artery brain aneurysm model: in vivo molecular enzyme-specific MR imaging of active inflammation in a pilot study.
    Radiology, 2009, Volume: 252, Issue:3

    Topics: Aneurysm; Angiography, Digital Subtraction; Animals; Carotid Artery Diseases; Carotid Artery, Common; Cerebral Angiography; Contrast Media; Disease Models, Animal; Feasibility Studies; Gadolinium DTPA; Image Enhancement; Inflammation; Magnetic Resonance Imaging; Peroxidase; Pilot Projects; Rabbits

2009
Enzyme-sensitive magnetic resonance imaging targeting myeloperoxidase identifies active inflammation in experimental rabbit atherosclerotic plaques.
    Circulation, 2009, Aug-18, Volume: 120, Issue:7

    Topics: Animals; Aorta, Thoracic; Atherosclerosis; Disease Models, Animal; Gadolinium DTPA; Hypercholesterolemia; Inflammation; Macrophages; Magnetic Resonance Imaging; Male; Peroxidase; Rabbits; Regression Analysis

2009
Science to practice: can an enzyme-sensitive MR contrast agent be used to image inflammation in aneurysms?
    Radiology, 2009, Volume: 252, Issue:3

    Topics: Animals; Carotid Artery Diseases; Carotid Artery, Common; Cerebral Angiography; Contrast Media; Dilatation, Pathologic; Disease Models, Animal; Gadolinium DTPA; Image Enhancement; Inflammation; Intracranial Aneurysm; Magnetic Resonance Imaging; Peroxidase; Rabbits

2009
Vasculitis: molecular imaging by targeting the inflammatory enzyme myeloperoxidase.
    Radiology, 2012, Volume: 262, Issue:1

    Topics: Animals; Aorta; Cell Movement; Chromatography, High Pressure Liquid; Contrast Media; Gadolinium DTPA; Immunohistochemistry; Mice; Molecular Imaging; Mucocutaneous Lymph Node Syndrome; Peroxidase; Random Allocation; Statistics, Nonparametric

2012
MR imaging of myeloperoxidase activity in a model of the inflamed aneurysm wall.
    AJNR. American journal of neuroradiology, 2015, Volume: 36, Issue:1

    Topics: Animals; Disease Models, Animal; Gadolinium DTPA; Image Enhancement; Intracranial Aneurysm; Magnetic Resonance Angiography; Male; Motion; Neuroimaging; Peroxidase; Phantoms, Imaging; Rabbits; Radiography; Signal-To-Noise Ratio

2015
Multiple sclerosis: myeloperoxidase immunoradiology improves detection of acute and chronic disease in experimental model.
    Radiology, 2015, Volume: 275, Issue:2

    Topics: Acute Disease; Animals; Chronic Disease; Contrast Media; Disease Models, Animal; Encephalomyelitis, Autoimmune, Experimental; Female; Gadolinium DTPA; Mice; Multiple Sclerosis; Peroxidase; Radionuclide Imaging

2015
Science to practice: myeloperoxidase immunoradiology improves detection of acute and chronic experimental multiple sclerosis.
    Radiology, 2015, Volume: 275, Issue:2

    Topics: Animals; Contrast Media; Female; Gadolinium DTPA; Multiple Sclerosis; Peroxidase; Radionuclide Imaging

2015
Molecular MR Imaging of Myeloperoxidase Distinguishes Steatosis from Steatohepatitis in Nonalcoholic Fatty Liver Disease.
    Radiology, 2017, Volume: 284, Issue:2

    Topics: Adult; Animals; Biopsy; Contrast Media; Diagnosis, Differential; Disease Models, Animal; Fatty Liver; Female; Gadolinium DTPA; Humans; Immunoenzyme Techniques; Magnetic Resonance Imaging; Mice; Middle Aged; Molecular Imaging; Non-alcoholic Fatty Liver Disease; Oxidative Stress; Peroxidase

2017
High-resolution Imaging of Myeloperoxidase Activity Sensors in Human Cerebrovascular Disease.
    Scientific reports, 2018, 05-16, Volume: 8, Issue:1

    Topics: Adolescent; Adult; Aged; Biosensing Techniques; Cerebrovascular Disorders; Contrast Media; Female; Gadolinium DTPA; Humans; Image Processing, Computer-Assisted; Magnetic Resonance Imaging; Male; Middle Aged; Peroxidase; Phantoms, Imaging; Prospective Studies; Young Adult

2018
Highly Efficient Activatable MRI Probe to Sense Myeloperoxidase Activity.
    Journal of medicinal chemistry, 2021, 05-13, Volume: 64, Issue:9

    Topics: Animals; Atherosclerosis; Binding Sites; Calcium; Catalytic Domain; Cell Survival; Contrast Media; Disease Models, Animal; Drug Design; Female; Gadolinium DTPA; Half-Life; Magnetic Resonance Imaging; Mice; Mice, Inbred BALB C; Peroxidase; RAW 264.7 Cells; Signal-To-Noise Ratio; Tissue Distribution; Zinc

2021
An activatable Mn(II) MRI probe for detecting peroxidase activity in vitro and in vivo.
    Journal of inorganic biochemistry, 2022, Volume: 236

    Topics: Animals; Contrast Media; Edetic Acid; Gadolinium DTPA; Horseradish Peroxidase; Hydrogen Peroxide; Magnetic Resonance Imaging; Manganese; Mice; Peroxidase; Phenols; Protons; Tyrosine; Uric Acid; Water

2022