Page last updated: 2024-09-04

fusidic acid and tauro-24,25-dihydrofusidate

fusidic acid has been researched along with tauro-24,25-dihydrofusidate in 22 studies

Compound Research Comparison

Studies
(fusidic acid)
Trials
(fusidic acid)
Recent Studies (post-2010)
(fusidic acid)
Studies
(tauro-24,25-dihydrofusidate)
Trials
(tauro-24,25-dihydrofusidate)
Recent Studies (post-2010) (tauro-24,25-dihydrofusidate)
1,7421173442210

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19904 (18.18)18.7374
1990's17 (77.27)18.2507
2000's1 (4.55)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Mitra, AK; Shao, Z1
Illum, L; Richardson, JL; Thomas, NW1
Bantle, S; Beglinger, C; Drewe, J; Kissel, T; Rummelt, A1
Lee, WA; Narog, BA; Patapoff, TW; Wang, YJ1
Breimer, DD; de Boer, AG; Heijligers-Feijen, CD; van Hoogdalem, EJ; Verhoef, JC1
Borden, L; Ennis, RD; Lee, WA1
Baldwin, PA; Grimm, CJ; Klingbeil, CK; Longenecker, JP1
Hermens, WA; Hooymans, PM; Merkus, FW; Verhoef, JC1
Deurloo, MJ; Hermens, WA; Merkus, FW; Romeyn, SG; Verhoef, JC1
Breimer, DD; de Boer, AG; Heijligers-Feijen, CD; Mathôt, RA; van Bree, JB; van Hoogdalem, EJ; Verhoef, JC; Wackwitz, AT1
Merkle, HP; Raehs, SC; Sandow, J; Wirth, K1
Carey, MC; Dubovi, EJ; Flier, JS; Longenecker, JP; Moses, AC; Silver, RD1
Blom-Roosemalen, MC; Breimer, DD; de Boer, AG; Hurni, MA; Nagelkerke, JF; Noach, AB1
Hosoya, K; Kubo, H; Morimoto, Y; Natsume, H; Sugibayashi, K2
Bengtsson, P; Ennis, RD; Lee, WA; Longenecker, JP1
Albertsson-Wikland, K; Diczfalusy, M; Flyg, C; Hedin, L; Olsson, B; Petersson, AS; Rosberg, S1
Chung, YB; Han, K; Lee, MJ; Moon, DC; Park, JS; Robinson, JR1
Adriaens, E; Mertens, J; Remon, JP; Voorspoels, J1
Cullander, C; Marttin, E; Merkus, FW; Nagelkerke, JF; Romeijn, SG; Verhoef, JC1
Akutsu, T; Hosoya, K; Kubo, H; Morimoto, Y; Natsume, H; Sugibayashi, K1
Agu, RU; Augustijns, P; Jorissen, M; Kinget, R; Verbeke, N; Willems, T1

Trials

1 trial(s) available for fusidic acid and tauro-24,25-dihydrofusidate

ArticleYear
Tolerability and absorption enhancement of intranasally administered octreotide by sodium taurodihydrofusidate in healthy subjects.
    Pharmaceutical research, 1992, Volume: 9, Issue:1

    Topics: Administration, Intranasal; Adult; Biological Availability; Double-Blind Method; Drug Evaluation; Drug Interactions; Female; Fusidic Acid; Humans; Lasers; Male; Octreotide; Reference Values; Scattering, Radiation

1992

Other Studies

21 other study(ies) available for fusidic acid and tauro-24,25-dihydrofusidate

ArticleYear
Nasal membrane and intracellular protein and enzyme release by bile salts and bile salt-fatty acid mixed micelles: correlation with facilitated drug transport.
    Pharmaceutical research, 1992, Volume: 9, Issue:9

    Topics: 5'-Nucleotidase; Acyclovir; Animals; Bile Acids and Salts; Fatty Acids; Fusidic Acid; Glycocholic Acid; L-Lactate Dehydrogenase; Linoleic Acid; Linoleic Acids; Male; Membrane Proteins; Nasal Mucosa; Rats; Rats, Sprague-Dawley; Taurocholic Acid

1992
Vaginal absorption of insulin in the rat: effect of penetration enhancers on insulin uptake and mucosal histology.
    Pharmaceutical research, 1992, Volume: 9, Issue:7

    Topics: Absorption; Adjuvants, Pharmaceutic; Administration, Intravaginal; Animals; Blood Glucose; Buffers; Epithelial Cells; Epithelium; Female; Fusidic Acid; Insulin; Lysophospholipids; Rats; Rats, Wistar; Vagina

1992
Intranasal bioavailability of insulin powder formulations: effect of permeation enhancer-to-protein ratio.
    Journal of pharmaceutical sciences, 1991, Volume: 80, Issue:8

    Topics: Absorption; Adjuvants, Pharmaceutic; Administration, Intranasal; Aerosols; Animals; Biological Availability; Female; Fusidic Acid; Insulin; Nasal Mucosa; Permeability; Powders; Proteins; Solutions

1991
Absorption enhancement of rectally infused insulin by sodium tauro-24,25-dihydrofusidate (STDHF) in rats.
    Pharmaceutical research, 1990, Volume: 7, Issue:2

    Topics: Administration, Rectal; Animals; Biological Availability; Blood Glucose; Edetic Acid; Fusidic Acid; Infusions, Intravenous; Insulin; Intestinal Absorption; Male; Rats; Rats, Inbred Strains; Stimulation, Chemical

1990
The effects of permeation enhancers on the surface morphology of the rat nasal mucosa: a scanning electron microscopy study.
    Pharmaceutical research, 1990, Volume: 7, Issue:5

    Topics: Animals; Bile Acids and Salts; Buffers; Cell Membrane Permeability; Dose-Response Relationship, Drug; Fusidic Acid; Male; Microscopy, Electron, Scanning; Nasal Mucosa; Phosphates; Polyethylene Glycols; Rats; Rats, Inbred Strains; Surface-Active Agents; Time Factors

1990
The effect of sodium tauro-24,25-dihydrofusidate on the nasal absorption of human growth hormone in three animal models.
    Pharmaceutical research, 1990, Volume: 7, Issue:5

    Topics: Absorption; Animals; Biological Availability; Dose-Response Relationship, Drug; Fusidic Acid; Growth Hormone; Humans; Male; Nasal Mucosa; Rabbits; Rats; Rats, Inbred Strains; Sheep; Structure-Activity Relationship; Surface-Active Agents

1990
Effects of absorption enhancers on human nasal tissue ciliary movement in vitro.
    Pharmaceutical research, 1990, Volume: 7, Issue:2

    Topics: Absorption; Adenoids; Adjuvants, Pharmaceutic; Chemical Phenomena; Chemistry, Physical; Fusidic Acid; Humans; In Vitro Techniques; Insulin; Micelles; Mucociliary Clearance; Nasal Mucosa

1990
Absorption enhancement of intranasally administered insulin by sodium taurodihydrofusidate (STDHF) in rabbits and rats.
    Pharmaceutical research, 1989, Volume: 6, Issue:10

    Topics: Administration, Intranasal; Animals; Biological Availability; Blood Glucose; Excipients; Fusidic Acid; Injections, Intravenous; Insulin; Male; Rabbits; Rats; Rats, Inbred Strains

1989
Rectal absorption enhancement of cefoxitin and desglycinamide arginine vasopressin by sodium tauro-24,25-dihydrofusidate in conscious rats.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Animals; Arginine Vasopressin; Biological Availability; Cefoxitin; Fusidic Acid; Intestinal Absorption; Male; Rats; Rats, Inbred Strains; Rectum; Stimulation, Chemical

1989
The adjuvant effect of bacitracin on nasal absorption of gonadorelin and buserelin in rats.
    Pharmaceutical research, 1988, Volume: 5, Issue:11

    Topics: Absorption; Adjuvants, Pharmaceutic; Animals; Bacitracin; Buserelin; Dose-Response Relationship, Drug; Female; Fusidic Acid; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Male; Nasal Mucosa; Ovulation; Rats; Rats, Inbred Strains; Rosaniline Dyes

1988
Effects of sodium taurodihydrofusidate on nasal absorption of insulin in sheep.
    Journal of pharmaceutical sciences, 1987, Volume: 76, Issue:5

    Topics: Absorption; Animals; Biological Availability; Female; Fusidic Acid; Hemolysis; Injections, Intravenous; Insulin; Nasal Mucosa; Rabbits; Sheep

1987
Permeability enhancement in Caco-2 cell monolayers by sodium salicylate and sodium taurodihydrofusidate: assessment of effect-reversibility and imaging of transepithelial transport routes by confocal laser scanning microscopy.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Adjuvants, Pharmaceutic; Biological Transport; Cell Membrane; Cell Membrane Permeability; Colonic Neoplasms; Dextrans; Electrophysiology; Epithelium; Fluorescein; Fluorescein-5-isothiocyanate; Fluoresceins; Fusidic Acid; Humans; Intestinal Absorption; Lasers; Lipid Metabolism; Microscopy; Sodium Salicylate; Trypan Blue; Tumor Cells, Cultured

1993
Evaluation of enhancers to increase nasal absorption using Ussing chamber technique.
    Biological & pharmaceutical bulletin, 1994, Volume: 17, Issue:2

    Topics: Absorption; Adjuvants, Pharmaceutic; Animals; Deoxycholic Acid; Dextrans; Fluorescein-5-isothiocyanate; Fusidic Acid; Lysophosphatidylcholines; Male; Nasal Mucosa; Phospholipids; Polidocanol; Polyethylene Glycols; Proteins; Rabbits; Sodium Dodecyl Sulfate

1994
The bioavailability of intranasal salmon calcitonin in healthy volunteers with and without a permeation enhancer.
    Pharmaceutical research, 1994, Volume: 11, Issue:5

    Topics: Adjuvants, Pharmaceutic; Administration, Intranasal; Adult; Biological Availability; Calcitonin; Female; Fusidic Acid; Humans; Male; Radioimmunoassay

1994
Intranasal administration of human growth hormone (hGH) in combination with a membrane permeation enhancer in patients with GH deficiency: a pharmacokinetic study.
    The Journal of clinical endocrinology and metabolism, 1993, Volume: 76, Issue:4

    Topics: Administration, Intranasal; Adolescent; Adult; Dose-Response Relationship, Drug; Drug Combinations; Female; Fusidic Acid; Growth Hormone; Humans; Injections, Subcutaneous; Male; Nasal Mucosa; Radioimmunoassay

1993
Identification of enzymatic degradation products of luteinizing hormone releasing hormone (LHRH)/[D-Ala6] LHRH in rabbit mucosal homogenates.
    Pharmaceutical research, 1995, Volume: 12, Issue:10

    Topics: Amino Acid Sequence; Animals; Edetic Acid; Female; Fusidic Acid; Gonadotropin-Releasing Hormone; Hydrolysis; In Vitro Techniques; Molecular Sequence Data; Mucous Membrane; Rabbits

1995
Effect of absorption enhancers on ciliated epithelium: a novel in vivo toxicity screening method using rotifers.
    Pharmaceutical research, 1997, Volume: 14, Issue:4

    Topics: 2-Hydroxypropyl-beta-cyclodextrin; Animals; beta-Cyclodextrins; Cilia; Cyclodextrins; Deoxycholic Acid; Epithelium; Fusidic Acid; Microscopy, Electron, Scanning; Phosphatidylcholines; Rotifera

1997
Confocal laser scanning microscopic visualization of the transport of dextrans after nasal administration to rats: effects of absorption enhancers.
    Pharmaceutical research, 1997, Volume: 14, Issue:5

    Topics: Absorption; Adjuvants, Pharmaceutic; Administration, Intranasal; Animals; Biological Transport, Active; Dextrans; Epithelium; Fixatives; Fluorescein-5-isothiocyanate; Fusidic Acid; Male; Microscopy, Confocal; Molecular Weight; Nasal Mucosa; Rats; Rats, Wistar; Stimulation, Chemical

1997
Effect of sodium taurodihydrofusidate on nasal drug delivery: differences in its concentration and penetrant molecular weight.
    Archives of pharmacal research, 1994, Volume: 17, Issue:2

    Topics: Adjuvants, Pharmaceutic; Administration, Intranasal; Animals; Anti-Asthmatic Agents; Cromolyn Sodium; Dextrans; Fluorescein-5-isothiocyanate; Fusidic Acid; In Vitro Techniques; Male; Molecular Weight; Nasal Mucosa; Rabbits

1994
Evaluation of bile acids and fusidate derivative as nasal absorption enhancers using an electrophysiological technique.
    Biological & pharmaceutical bulletin, 1999, Volume: 22, Issue:10

    Topics: Absorption; Administration, Inhalation; Animals; Bile Acids and Salts; Biological Transport; Dextrans; Dose-Response Relationship, Drug; Electric Impedance; Electrophysiology; Evaluation Studies as Topic; Fusidic Acid; In Vitro Techniques; Male; Membrane Potentials; Nasal Mucosa; Rabbits; Time Factors

1999
In-vitro nasal drug delivery studies: comparison of derivatised, fibrillar and polymerised collagen matrix-based human nasal primary culture systems for nasal drug delivery studies.
    The Journal of pharmacy and pharmacology, 2001, Volume: 53, Issue:11

    Topics: Administration, Intranasal; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Cilia; Collagen; Drug Delivery Systems; Fluorescein; Fusidic Acid; Humans; L-Lactate Dehydrogenase; Malate Dehydrogenase; Microscopy, Electron, Scanning; Nasal Mucosa

2001