furosemide and enalaprilat anhydrous

furosemide has been researched along with enalaprilat anhydrous in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19903 (13.04)18.7374
1990's9 (39.13)18.2507
2000's3 (13.04)29.6817
2010's8 (34.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ax, F; Bonham, NM; Hallberg, A; Karlén, A; Lennernäs, H; Winiwarter, S1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Avdeef, A; Tam, KY1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bellman, K; Knegtel, RM; Settimo, L1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Andersson, G; Held, P; Sigurdsson, A; Swedberg, K1
Anderson, GH; Hellwig, B; Kopecky, RT; McAfee, JG; Patchin, D; Roskopf, M; Thomas, FD1
Ayers, C; Davidson, R; DiPette, D; Fisher, M; Guthrie, G; Rucinska, E; Rutledge, J; Schwartz, S1
Denton, DA; Di Nicolantonio, R; McKinley, MJ; Weisinger, RS1
de Jong, PE; de Zeeuw, D; Donker, AJ; Navis, GJ; van der Hem, GK1
Connelly, JF; Zigmont, EA1
Berdeaux, A; Giudicelli, JF; Richard, V1
Berdeaux, A; Ghaleh, B; Giudicelli, JF; Richard, V1
Ferraro, T; May, C; Tarjan, E; Weisinger, RS1
Blossom, G; Czako, PF; Glover, JL; Juleff, R; Long, GW; Misra, DC1
Bak, M; Christensen, S; Petersen, JS; Poulsen, LB; Shalmi, M1
Kutina, AV; Natochin, IuV; Shakhmatova, EI1

Reviews

1 review(s) available for furosemide and enalaprilat anhydrous

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

2 trial(s) available for furosemide and enalaprilat anhydrous

ArticleYear
Enalaprilat in acute myocardial infarction: tolerability and effects on the renin-angiotensin system.
    International journal of cardiology, 1991, Volume: 33, Issue:1

    Topics: Aged; Blood Pressure; Enalaprilat; Female; Furosemide; Humans; Infusions, Intravenous; Injections, Intravenous; Male; Metoprolol; Middle Aged; Myocardial Infarction; Nitroglycerin; Renin-Angiotensin System; Thrombolytic Therapy

1991
Effect of intravenous enalaprilat in moderate and severe systemic hypertension.
    The American journal of cardiology, 1988, Nov-15, Volume: 62, Issue:16

    Topics: Antihypertensive Agents; Double-Blind Method; Enalapril; Enalaprilat; Female; Furosemide; Humans; Hypertension; Infusions, Intravenous; Male; Middle Aged; Multicenter Studies as Topic; Placebos; Random Allocation

1988

Other Studies

20 other study(ies) available for furosemide and enalaprilat anhydrous

ArticleYear
Correlation of human jejunal permeability (in vivo) of drugs with experimentally and theoretically derived parameters. A multivariate data analysis approach.
    Journal of medicinal chemistry, 1998, Dec-03, Volume: 41, Issue:25

    Topics: Humans; Intestinal Absorption; Jejunum; Models, Biological; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Structure-Activity Relationship

1998
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
    Journal of medicinal chemistry, 2010, May-13, Volume: 53, Issue:9

    Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Enalaprilat-enhanced renography in a rat model of renovascular hypertension.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1990, Volume: 31, Issue:4

    Topics: Animals; Enalaprilat; Furosemide; Hypertension, Renovascular; Kidney; Male; Organotechnetium Compounds; Pentetic Acid; Radioisotope Renography; Rats; Rats, Inbred Strains; Succimer; Technetium Tc 99m Dimercaptosuccinic Acid; Technetium Tc 99m Pentetate; Time Factors

1990
The effect of captopril or enalaprilic acid on the Na appetite of Na-deplete rats.
    Clinical and experimental pharmacology & physiology, 1988, Volume: 15, Issue:1

    Topics: Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Appetite; Captopril; Drinking; Enalaprilat; Food Deprivation; Furosemide; Male; Rats; Rats, Inbred Strains; Sodium; Sodium, Dietary; Water Deprivation

1988
Blood pressure response to enalaprilic acid in essential hypertension: dose-response and effect of pre-treatment with furosemide.
    European journal of clinical pharmacology, 1985, Volume: 29, Issue:1

    Topics: Adult; Aged; Aldosterone; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Dose-Response Relationship, Drug; Enalapril; Enalaprilat; Female; Furosemide; Heart Rate; Humans; Hypertension; Male; Middle Aged; Renin

1985
Intravenous antihypertensive agents for patients unable to take oral medications.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 1995, Jul-15, Volume: 52, Issue:14

    Topics: Adrenergic beta-Antagonists; Antihypertensive Agents; Calcium Channel Blockers; Enalaprilat; Furosemide; Humans; Hydralazine; Hypertension; Injections, Intravenous; Labetalol; Methyldopa; Nitroglycerin; Nitroprusside; Vasodilator Agents

1995
Systemic and coronary effects of the angiotensin II receptor antagonist EXP3174 in dogs.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:1

    Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Coronary Circulation; Dogs; Enalaprilat; Female; Furosemide; Hemodynamics; Imidazoles; Losartan; Male; Renin-Angiotensin System; Tetrazoles

1993
Comparison of the effects of EXP3174, an angiotensin II antagonist and enalaprilat on myocardial infarct size in anaesthetized dogs.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: Anesthesia; Angiotensin I; Angiotensin II; Animals; Antihypertensive Agents; Blood Pressure; Coronary Circulation; Disease Models, Animal; Dogs; Enalaprilat; Female; Furosemide; Heart Rate; Imidazoles; Injections, Intravenous; Losartan; Male; Myocardial Infarction; Myocardial Ischemia; Myocardial Reperfusion Injury; Renin-Angiotensin System; Tetrazoles

1993
Converting enzyme inhibition in rabbits: effects on sodium and water intake/excretion and blood pressure.
    Physiology & behavior, 1993, Volume: 53, Issue:2

    Topics: Animals; Blood Pressure; Enalaprilat; Female; Furosemide; Male; Natriuresis; Rabbits; Sodium Chloride; Thirst; Water-Electrolyte Balance

1993
Protective effects of enalaprilat against postischemic renal failure.
    The Journal of surgical research, 1993, Volume: 54, Issue:3

    Topics: Analysis of Variance; Animals; Blood Urea Nitrogen; Creatinine; Dogs; Enalaprilat; Furosemide; Ischemia; Kidney; Mannitol; Renal Insufficiency; Time Factors

1993
Effects of angiotensin-converting enzyme inhibition on renal adaptations to acute furosemide administration in conscious rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:1

    Topics: Absorption; Adaptation, Physiological; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Body Fluids; Consciousness; Drug Interactions; Enalaprilat; Female; Furosemide; Heart Rate; Kidney; Kidney Tubules; Peptidyl-Dipeptidase A; Potassium; Rats; Rats, Wistar; Renal Circulation; Sodium; Solutions; Time Factors; Water

1993
[Influence of the angiotensin converting enzyme inhibition on the functional proteinuria in rats].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2009, Volume: 95, Issue:10

    Topics: Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Diuresis; Diuretics; Dose-Response Relationship, Drug; Enalaprilat; Female; Furosemide; Glomerular Filtration Rate; Kidney; Peptidyl-Dipeptidase A; Potassium; Proteinuria; Rats; Rats, Wistar; Vasotocin; Water

2009