Page last updated: 2024-09-03

furamidine and db 820

furamidine has been researched along with db 820 in 8 studies

Compound Research Comparison

Studies
(furamidine)
Trials
(furamidine)
Recent Studies (post-2010)
(furamidine)
Studies
(db 820)
Trials
(db 820)
Recent Studies (post-2010) (db 820)
108132801

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (75.00)29.6817
2010's2 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boykin, DW; Brun, R; Easterbrook, JD; Ismail, MA; Tanious, FA; Wilson, WD1
Anbazhagan, M; Boykin, DW; Bridges, AS; Brun, R; Francesconi, I; Hall, JE; Hu, Q; Ismail, MA; Kumar, A; Mathis, AM; Saulter, J; Tanious, FA; Tidwell, RR; Wenzler, T; Wilson, WD1
Arafa, RK; Boykin, DW; Brun, R; Ismail, MA; Tanious, FA; Wenzler, T; Wilson, WD1
Boykin, DW; Brun, R; Hall, JE; Ismail, MA; Tidwell, RR; Wenzler, T1
Arafa, RK; Boykin, DW; Brun, R; Hu, L; Ismail, MA; Munde, M; Patel, A; Wenzler, T; Wilson, WD1
Anbazhagan, M; Boykin, DW; Brun, R; Gillingwater, K; Kumar, A; Tidwell, RR1
Boykin, DW; Branowska, D; Brun, R; Farahat, AA; Kumar, A; Liu, Y; Wenzler, T; Wilson, WD1
Bondada, L; Boykin, DW; Brun, R; Hu, L; Munde, M; Patel, A; Wang, MZ; Wenzler, T; Wilson, WD; Yang, S1

Other Studies

8 other study(ies) available for furamidine and db 820

ArticleYear
Synthesis and antiprotozoal activity of aza-analogues of furamidine.
    Journal of medicinal chemistry, 2003, Oct-23, Volume: 46, Issue:22

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Aza Compounds; Benzamidines; Mice; Plasmodium falciparum; Prodrugs; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2003
Diphenyl furans and aza analogs: effects of structural modification on in vitro activity, DNA binding, and accumulation and distribution in trypanosomes.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:8

    Topics: Animals; Benzamidines; DNA, Protozoan; Dose-Response Relationship, Drug; Furans; Inhibitory Concentration 50; Organelles; Parasitic Sensitivity Tests; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense

2007
Synthesis and antiprotozoal activity of novel bis-benzamidino imidazo[1,2-a]pyridines and 5,6,7,8-tetrahydro-imidazo[1,2-a]pyridines.
    Bioorganic & medicinal chemistry, 2008, Jan-15, Volume: 16, Issue:2

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Combinatorial Chemistry Techniques; Disease Models, Animal; Inhibitory Concentration 50; Mice; Molecular Structure; Plasmodium falciparum; Prodrugs; Pyridines; Trypanosoma brucei rhodesiense

2008
New treatment option for second-stage African sleeping sickness: in vitro and in vivo efficacy of aza analogs of DB289.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:10

    Topics: Animals; Benzamidines; Central Nervous System; Female; Furans; Mice; Molecular Structure; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei gambiense; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2009
Synthesis and activity of azaterphenyl diamidines against Trypanosoma brucei rhodesiense and Plasmodium falciparum.
    Bioorganic & medicinal chemistry, 2009, Sep-15, Volume: 17, Issue:18

    Topics: Animals; Antiprotozoal Agents; Inhibitory Concentration 50; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2009
In vivo investigations of selected diamidine compounds against Trypanosoma evansi using a mouse model.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:12

    Topics: Animals; Disease Models, Animal; Female; Mice; Parasitic Sensitivity Tests; Pentamidine; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2009
Synthesis and antiprotozoal activity of 2,5-bis[amidinoaryl]thiazoles.
    Bioorganic & medicinal chemistry, 2010, May-15, Volume: 18, Issue:10

    Topics: Administration, Oral; Animals; Antimalarials; Antiprotozoal Agents; Disease Models, Animal; DNA, Protozoan; Drug Stability; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Rats; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2010
Synthesis and antiprotozoal activity of dicationic 2,6-diphenylpyrazines and aza-analogues.
    Bioorganic & medicinal chemistry, 2013, Nov-01, Volume: 21, Issue:21

    Topics: Animals; Antiprotozoal Agents; Aza Compounds; Cations; Cell Line; Cell Survival; Disease Models, Animal; Mice; Myoblasts; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Poly dA-dT; Prodrugs; Pyrazines; Rats; Structure-Activity Relationship; Transition Temperature; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2013