Page last updated: 2024-08-26

fulvestrant and estrone

fulvestrant has been researched along with estrone in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (33.33)18.2507
2000's5 (33.33)29.6817
2010's4 (26.67)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Bellavance, E; Luu-The, V; Poirier, D1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Potter, BV; Purohit, A; Reed, MJ; Roberts, CJ; Williams, GJ1
Newton, CJ1
Biberger, C; von Angerer, E1
Bélanger, A; Candas, B; Gauthier, S; Labrie, C; Labrie, F; Li, X; Martel, C; Mérand, Y; Provencher, L1
Gorodeski, GI1
Robinson, JA; Spelsberg, TC; Turner, RT; Waters, KM1
Dubey, RK; Gillespie, DG; Imthurn, B; Jackson, EK; Keller, PJ; Zacharia, LC1
Atkin, SL; Bilko, D; Newton, CJ; Pappa, S1
Ansell, PJ; Ganjam, VK; Harada, N; Honda, S; Lubahn, DB; Newton, LG; Philips, BJ; Rottinghaus, GE; Welshons, WV1
De Felici, M; Farini, D; La Sala, G1
Coombes, RC; Januszewski, A; Palmieri, C; Stanway, S1
Dias, NJ; Selcer, KW1
Bazgier, V; Berka, K; Holcakova, J; Hrstka, R; Kolarova, T; Kudova, E; Kvasnica, M; Oklestkova, J; Rarova, L; Strnad, M; Tichy, V; Vonka, P1

Reviews

2 review(s) available for fulvestrant and estrone

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Irosustat: a first-generation steroid sulfatase inhibitor in breast cancer.
    Expert review of anticancer therapy, 2011, Volume: 11, Issue:2

    Topics: Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Clinical Trials, Phase II as Topic; Dehydroepiandrosterone Sulfate; Estradiol; Estrone; Female; Fulvestrant; Humans; Neoplasms, Hormone-Dependent; Steryl-Sulfatase; Sulfonic Acids; Tamoxifen

2011

Other Studies

13 other study(ies) available for fulvestrant and estrone

ArticleYear
Potent and selective steroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 7, an enzyme that catalyzes the reduction of the key hormones estrone and dihydrotestosterone.
    Journal of medicinal chemistry, 2009, Dec-10, Volume: 52, Issue:23

    Topics: 17-Hydroxysteroid Dehydrogenases; Androstane-3,17-diol; Androstanes; Biocatalysis; Cell Line; Dihydrotestosterone; Enzyme Inhibitors; Estradiol; Estrone; Humans; Inhibitory Concentration 50; Oxidation-Reduction; Substrate Specificity

2009
In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate.
    International journal of cancer, 1995, Sep-27, Volume: 63, Issue:1

    Topics: Animals; Arylsulfatases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estradiol; Estrone; Female; Fulvestrant; Liver; Mammary Neoplasms, Experimental; Rats; Rats, Wistar; Steryl-Sulfatase; Sulfatases; Tamoxifen; Time Factors

1995
Estrogen receptor blockade by the pure antiestrogen, ZM 182780, induces death of pituitary tumour cells.
    The Journal of steroid biochemistry and molecular biology, 1995, Volume: 55, Issue:3-4

    Topics: Animals; Cell Death; Culture Media; Culture Media, Conditioned; DNA Damage; Dose-Response Relationship, Drug; Estradiol; Estriol; Estrogen Antagonists; Estrone; Fulvestrant; Hydroxytestosterones; Luciferases; Pituitary Neoplasms; Prolactin; Rats; Receptors, Estrogen; Steroids; Time Factors; Tumor Cells, Cultured

1995
2-Phenylindoles with sulfur containing side chains. Estrogen receptor affinity, antiestrogenic potency, and antitumor activity.
    The Journal of steroid biochemistry and molecular biology, 1996, Volume: 58, Issue:1

    Topics: Animals; Antineoplastic Agents, Hormonal; Breast Neoplasms; Cattle; Cell Division; Estradiol; Estrogen Antagonists; Estrone; Female; Fulvestrant; HeLa Cells; Humans; Indoles; Mammary Neoplasms, Experimental; Mice; Organ Size; Receptors, Estrogen; Sulfur; Tamoxifen; Transcriptional Activation; Tumor Cells, Cultured; Uterus; Vitellogenins

1996
Comparison of the effects of the new orally active antiestrogen EM-800 with ICI 182 780 and toremifene on estrogen-sensitive parameters in the ovariectomized mouse.
    Endocrinology, 1998, Volume: 139, Issue:5

    Topics: Animals; Benzopyrans; Estradiol; Estrogen Antagonists; Estrogens; Estrone; Female; Fulvestrant; Mice; Mice, Inbred BALB C; Organ Size; Ovariectomy; Propionates; Receptors, Estrogen; Toremifene; Uterus; Vagina

1998
Estrogen increases the permeability of the cultured human cervical epithelium by modulating cell deformability.
    The American journal of physiology, 1998, Volume: 275, Issue:3

    Topics: Actins; Cell Line; Cell Membrane Permeability; Cells, Cultured; Cervix Uteri; Chlorides; Diethylstilbestrol; Egtazic Acid; Epithelial Cells; Estradiol; Estriol; Estrogen Antagonists; Estrogens; Estrone; Female; Fulvestrant; Humans; Kinetics; Progesterone; Sodium; Tamoxifen

1998
Direct action of naturally occurring estrogen metabolites on human osteoblastic cells.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2000, Volume: 15, Issue:3

    Topics: Alkaline Phosphatase; Bone Matrix; Cell Differentiation; Cell Line; Enzyme Induction; Estradiol; Estrogen Receptor alpha; Estrogens; Fulvestrant; Humans; Hydroxyestrones; Osteoblasts; Osteocalcin; Receptors, Estrogen; Recombinant Fusion Proteins; RNA, Messenger

2000
Clinically used estrogens differentially inhibit human aortic smooth muscle cell growth and mitogen-activated protein kinase activity.
    Arteriosclerosis, thrombosis, and vascular biology, 2000, Volume: 20, Issue:4

    Topics: Aorta; Becaplermin; Cell Division; Cells, Cultured; DNA; Enzyme Inhibitors; Estradiol; Estriol; Estrogen Antagonists; Estrogens; Estrone; Female; Fulvestrant; Humans; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis

2000
Dexamethasone blocks antioestrogen- and oxidant-induced death of pituitary tumour cells.
    The Journal of endocrinology, 2001, Volume: 169, Issue:2

    Topics: Adenosine Triphosphate; Cell Death; Dexamethasone; Estradiol; Estrogen Receptor Modulators; Estrone; Flow Cytometry; Flutamide; Fulvestrant; Glucocorticoids; Glyceraldehyde-3-Phosphate Dehydrogenases; Gonanes; Humans; Hydrogen Peroxide; Microscopy, Fluorescence; Mifepristone; Pituitary Neoplasms; Reactive Oxygen Species; Receptor Cross-Talk; Receptors, Cell Surface; Transfection; Tumor Cells, Cultured

2001
Estrogen receptor-independent catechol estrogen binding activity: protein binding studies in wild-type, Estrogen receptor-alpha KO, and aromatase KO mice tissues.
    Biochemistry, 2004, Jun-01, Volume: 43, Issue:21

    Topics: Animals; Aromatase; Binding, Competitive; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Estrogens, Catechol; Female; Fulvestrant; Hydroxyestrones; Kidney; Liver; Male; Mice; Mice, Knockout; Ovary; Proteins; Receptors, Estrogen; Substrate Specificity; Tissue Distribution; Uterus

2004
Estrogenic in vitro assay on mouse embryonic Leydig cells.
    The International journal of developmental biology, 2010, Volume: 54, Issue:4

    Topics: Animals; Biological Assay; Cell Differentiation; Cells, Cultured; Estradiol; Estrogen Antagonists; Estrogen Receptor alpha; Estrogens; Estrone; Female; Fulvestrant; Genes, Reporter; Humans; Leydig Cells; Luciferases; Male; Mice; Phytoestrogens; Response Elements; Testis; Transcription Factor AP-1; Transfection

2010
Steroid sulfatase mediated growth Sof human MG-63 pre-osteoblastic cells.
    Steroids, 2014, Volume: 88

    Topics: Cell Line; Cell Proliferation; Enzyme Inhibitors; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogen Receptor Modulators; Estrone; Fulvestrant; Gene Expression Regulation, Enzymologic; Humans; Osteoblasts; RNA, Messenger; Steryl-Sulfatase

2014
Small change - big consequence: The impact of C15-C16 double bond in a D‑ring of estrone on estrogen receptor activity.
    The Journal of steroid biochemistry and molecular biology, 2023, Volume: 233

    Topics: Breast Neoplasms; Cell Line, Tumor; Estradiol; Estrogen Receptor alpha; Estrone; Female; Fulvestrant; Humans; Molecular Docking Simulation; Receptors, Estrogen; Tamoxifen

2023