Page last updated: 2024-09-02

fr 139317 and verapamil

fr 139317 has been researched along with verapamil in 1 studies

Study Comparison

Studies
(fr 139317)
Trials
(fr 139317)
Recent Studies (post-2010)
(fr 139317)
Studies
(verapamil)
Trials
(verapamil)
Recent Studies (post-2010)
(verapamil)
219081762115272067

Protein Interaction Comparison

ProteinTaxonomyfr 139317 (IC50)verapamil (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)6.8
Multidrug resistance-associated protein 4Homo sapiens (human)133
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.2
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
Bile salt export pumpHomo sapiens (human)131.5
ATP-dependent translocase ABCB1Mus musculus (house mouse)2
ATP-dependent translocase ABCB1Homo sapiens (human)18.7117
Cytochrome P450 3A4Homo sapiens (human)16.6238
Alpha-2A adrenergic receptorHomo sapiens (human)0.579
Cytochrome P450 2C9 Homo sapiens (human)22
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.02
ATP-dependent translocase ABCB1Mus musculus (house mouse)64.3333
Catechol O-methyltransferaseHomo sapiens (human)0.2
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)8
Histamine H2 receptorHomo sapiens (human)2.59
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.442
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.02
Sodium-dependent serotonin transporterHomo sapiens (human)0.24
Multidrug resistance-associated protein 1 Homo sapiens (human)5.598
D(3) dopamine receptorHomo sapiens (human)0.186
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.165
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)6.8
Cytochrome P450 2J2Homo sapiens (human)22
D(2) dopamine receptorRattus norvegicus (Norway rat)200
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.2
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.3945
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.2
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)24.1417
Sodium channel protein type 5 subunit alphaHomo sapiens (human)41.5
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)192.0001
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)232

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kendall, DA; O'Sullivan, SE; Randall, MD1

Other Studies

1 other study(ies) available for fr 139317 and verapamil

ArticleYear
The effects of Delta9-tetrahydrocannabinol in rat mesenteric vasculature, and its interactions with the endocannabinoid anandamide.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Apamin; Arachidonic Acids; Azepines; Barium Compounds; Biological Factors; Calcium; Cannabinoid Receptor Modulators; Capsaicin; Charybdotoxin; Chlorides; Cyclohexanols; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Endocannabinoids; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Vasodilation; Verapamil

2005