fr 139317 has been researched along with phosphoramidon in 6 studies
| Studies (fr 139317) | Trials (fr 139317) | Recent Studies (post-2010) (fr 139317) | Studies (phosphoramidon) | Trials (phosphoramidon) | Recent Studies (post-2010) (phosphoramidon) |
|---|---|---|---|---|---|
| 219 | 0 | 8 | 781 | 12 | 33 |
| 219 | 0 | 8 | 781 | 12 | 33 |
| 219 | 0 | 8 | 781 | 12 | 33 |
| 219 | 0 | 8 | 781 | 12 | 33 |
| 219 | 0 | 8 | 781 | 12 | 33 |
| 219 | 0 | 8 | 781 | 12 | 33 |
| Protein | Taxonomy | fr 139317 (IC50) | phosphoramidon (IC50) |
|---|---|---|---|
| Thermolysin | Bacillus thermoproteolyticus | 0.033 | |
| Neprilysin | Rattus norvegicus (Norway rat) | 0.0578 | |
| Neprilysin | Oryctolagus cuniculus (rabbit) | 0.0028 | |
| Neprilysin | Homo sapiens (human) | 0.0405 | |
| Angiotensin-converting enzyme | Homo sapiens (human) | 0.615 | |
| Endothelin-converting enzyme 1 | Homo sapiens (human) | 1.0695 | |
| P2Y purinoceptor 12 | Homo sapiens (human) | 0.017 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 4 (66.67) | 18.2507 |
| 2000's | 1 (16.67) | 29.6817 |
| 2010's | 1 (16.67) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Aghai, Z; Bax, WA; Saxena, PR; van Tricht, CL; Wassenaar, C | 1 |
| Albert, U; Edvinsson, L; Ekelund, U; Mellander, S | 1 |
| Chilian, WM; DeFily, DV; Nishikawa, Y | 1 |
| Bellissant, E; Durand-Castel, X; Goineau, S; Guillo, P; Pape, D | 1 |
| Fukushima, Y; Hisa, H; Kimura, T; Kuwakubo, F; Matsumoto, T; Matsumura, Y; Nagayama, T; Satoh, S; Suzuki-Kusaba, M; Yoshida, M | 1 |
| Clark, JC; Davenport, AP; Fryer, TD; Johnström, P; Maguire, JJ; Pickard, JD; Richards, HK | 1 |
6 other study(ies) available for fr 139317 and phosphoramidon
| Article | Year |
|---|---|
Different endothelin receptors involved in endothelin-1- and sarafotoxin S6B-induced contractions of the human isolated coronary artery.
Topics: Adolescent; Adult; Azepines; Child; Child, Preschool; Coronary Vessels; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Endothelium, Vascular; Female; Glycopeptides; Humans; In Vitro Techniques; Indoles; Infant; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Peptides, Cyclic; Protease Inhibitors; Protein Precursors; Receptors, Endothelin; Vasoconstrictor Agents; Viper Venoms | 1994 |
In-vivo effects of endothelin-1 and ETA receptor blockade on arterial, venous and capillary functions in skeletal muscle.
Topics: Animals; Arteries; Azepines; Blood Pressure; Capillaries; Cats; Endothelin Receptor Antagonists; Endothelins; Glycopeptides; Hyperemia; Indoles; Muscle Tonus; Muscles; Neprilysin; Regional Blood Flow; Sympathectomy; Vascular Resistance; Vasoconstriction; Vasodilation; Veins | 1993 |
Endothelin antagonists block alpha1-adrenergic constriction of coronary arterioles.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Arterioles; Azepines; Coronary Vessels; Dogs; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Glycopeptides; Hemodynamics; Indoles; Phenylephrine; Propranolol; Receptor, Endothelin A; Vasoconstriction | 1999 |
Endothelin, but not angiotensin II, contributes to the hypoxic contractile response of large isolated pulmonary arteries in the rat.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Azepines; Bosentan; Calcium; Calcium Channel Blockers; Endothelin Receptor Antagonists; Endothelins; Endothelium, Vascular; Extracellular Space; Glycopeptides; Hypoxia; In Vitro Techniques; Indoles; Lisinopril; Losartan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Pulmonary Artery; Rats; Rats, Wistar; Sulfonamides | 1999 |
Role of endogenous endothelins in catecholamine secretion in the rat adrenal gland.
Topics: Adrenal Glands; Animals; Azepines; Catecholamines; Dose-Response Relationship, Drug; Electric Stimulation; Endothelin-1; Endothelins; Epinephrine; Glycopeptides; In Vitro Techniques; Indoles; Male; Norepinephrine; Oligopeptides; Piperidines; Rats; Rats, Wistar | 2000 |
Positron emission tomography of [18F]-big endothelin-1 reveals renal excretion but tissue-specific conversion to [18F]-endothelin-1 in lung and liver.
Topics: Animals; Aspartic Acid Endopeptidases; Autoradiography; Azepines; Endothelin A Receptor Antagonists; Endothelin-1; Endothelin-Converting Enzymes; Enzyme Activation; Fluorine Radioisotopes; Glycopeptides; Half-Life; Indoles; Infusions, Intravenous; Kidney; Lung; Male; Metalloendopeptidases; Molecular Imaging; Molecular Probe Techniques; Positron-Emission Tomography; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Tissue Distribution; Whole Body Imaging | 2010 |