Page last updated: 2024-09-02

fr 139317 and 1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-

fr 139317 has been researched along with 1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)- in 7 studies

Study Comparison

Studies
(fr 139317)
Trials
(fr 139317)
Recent Studies (post-2010)
(fr 139317)
Studies
(1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-)
Trials
(1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-)
Recent Studies (post-2010)
(1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-)
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Protein Interaction Comparison

ProteinTaxonomyfr 139317 (IC50)1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)- (IC50)

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (57.14)18.2507
2000's3 (42.86)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
D'Amico, M; Di Filippo, C; Rossi, F1
Docherty, C; MacLean, MR1
D'Amico, M; Di Filippo, C; Esposito, F; Filippelli, A; Rossi, F1
D'Amico, M; Di Filippo, C; Filippelli, A; Rossi, F1
D'Amico, M; Di Filippo, C; Filippelli, A; Piegari, E; Rinaldi, B; Rossi, F1
Berrino, L; D'Amico, M; Di Filippo, C; Giugliano, D; Marfella, R; Rossi, F1
Goto, K1

Reviews

1 review(s) available for fr 139317 and 1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-

ArticleYear
[Discovery of endothelin and its significance].
    Nihon rinsho. Japanese journal of clinical medicine, 2004, Volume: 62 Suppl 9

    Topics: Amino Acid Sequence; Animals; Azepines; Cardiovascular Diseases; Drug Design; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Humans; Indans; Indoles; Molecular Sequence Data; Peptides, Cyclic; Pyrimidines; Receptors, Endothelin; Sulfonamides; Vasoconstriction

2004

Other Studies

6 other study(ies) available for fr 139317 and 1h-indene-2-carboxylic acid, 1-(1,3-benzodioxol-5-yl)-3-(2- (carboxymethoxy)-4-methoxyphenyl)-2,3-dihydro-5-propoxy-, (1s,2r,3s)-

ArticleYear
Depressor responses to endothelin-1 into the superior colliculus of rats: predominant role of endothelin ET(B) receptors.
    European journal of pharmacology, 1998, Apr-17, Volume: 347, Issue:1

    Topics: Animals; Autoradiography; Azepines; Blood Pressure; Endothelin Receptor Antagonists; Endothelin-1; Heart Rate; Indans; Indoles; Male; Microinjections; Oligopeptides; Piperidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Superior Colliculi

1998
Development of endothelin receptors in perinatal rabbit pulmonary resistance arteries.
    British journal of pharmacology, 1998, Volume: 124, Issue:6

    Topics: Acetylcholine; Animals; Azepines; Endothelin-1; In Vitro Techniques; Indans; Indoles; Norepinephrine; Oligopeptides; Piperidines; Potassium Chloride; Pulmonary Artery; Rabbits; Receptors, Endothelin; Serotonin; Vascular Resistance; Viper Venoms

1998
Injection of endothelin-1 into the raphe obscurus of rats induces depressor responses predominantly through endothelin ET(A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:6

    Topics: Animals; Autoradiography; Azepines; Blood Pressure; Depression, Chemical; Endothelin Receptor Antagonists; Endothelin-1; Indans; Indoles; Male; Microinjections; Oligopeptides; Piperidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin

1999
Endothelin receptor antagonists reduce the pressor effects of angiotensin II into the periaqueductal gray area of rats.
    Life sciences, 1999, Volume: 65, Issue:9

    Topics: Angiotensin II; Animals; Azepines; Blood Pressure; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelin-1; Indans; Indoles; Male; Oligopeptides; Periaqueductal Gray; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin

1999
Local administration of ETA (but not ETB) blockers into the PAG area of the brain decreases blood pressure of DOCA-salt rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:2

    Topics: Analysis of Variance; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Desoxycorticosterone; Electrophoresis, Agar Gel; Endothelin Receptor Antagonists; Endothelin-1; Glyceraldehyde-3-Phosphate Dehydrogenases; Heart Rate; Hypertension; Indans; Indoles; Male; Oligopeptides; Periaqueductal Gray; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2002
Endothelin-1 receptor antagonists reduce cardiac electrical instability induced by high glucose in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:3

    Topics: Animals; Azepines; Dose-Response Relationship, Drug; Electrocardiography; Endothelin Receptor Antagonists; Glucose; Heart; Heart Conduction System; In Vitro Techniques; Indans; Indoles; Long QT Syndrome; Male; Oligopeptides; Piperidines; Rats; Receptor, Endothelin A; Receptors, Endothelin

2002