fr 120480 has been researched along with cholecystokinin in 10 studies
Studies (fr 120480) | Trials (fr 120480) | Recent Studies (post-2010) (fr 120480) | Studies (cholecystokinin) | Trials (cholecystokinin) | Recent Studies (post-2010) (cholecystokinin) |
---|---|---|---|---|---|
32 | 0 | 8 | 10,914 | 466 | 1,074 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 7 (70.00) | 18.2507 |
2000's | 3 (30.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Itoh, H; Kinoshita, T; Matsuo, T; Satoh, Y; Sogabe, H; Tada, T; Takaya, T; Yoshida, K | 1 |
Fukuyama, S; Kihara, N; Koda, S; Morokoshi, N; Nakashima, K; Yasuda, T | 1 |
Funakoshi, A; Miyasaka, K | 1 |
Otsuki, M; Tachibana, I | 1 |
Deguchi, S; Nakashima, K; Shimatani, K; Tada, T; Yasuda, T | 1 |
Hara, H; Kasai, T; Narakino, H; Nishi, T | 1 |
Biernat, M; Guilloteau, P; Le Huërou-Luron, I; Sosak-Swiderska, B; Sysa, P; Zabielski, R | 1 |
Bernard, C; Biernat, M; Chayvialle, JA; Guilloteau, P; Morisset, J; Podgurniak, P; Romé, V; Zabielski, R | 1 |
An, YP; Cui, H; Cui, ZJ; Xiao, R | 1 |
Cui, ZJ; Xiao, R | 1 |
10 other study(ies) available for fr 120480 and cholecystokinin
Article | Year |
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Studies on a novel, potent and orally effective cholecystokinin A antagonist, FK-480. Synthesis and structure-activity relationships of FK-480 and related compounds.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Cholecystokinin; Drug Evaluation; Drug Stability; Gastric Emptying; In Vitro Techniques; Indoles; Mice; Pancreas; Prodrugs; Rats; Sincalide; Structure-Activity Relationship | 1994 |
Mechanism of optical isomerization of (S)-N-[1-(2-fluorophenyl)-3,4,6,7- tetrahydro-4-oxopyrrolo[3,2,1-jk] [1,4]-benzodiazepine-3-yl]-1H- indole-2-carboxamide (FK480) in soft capsules containing polyethylene glycol 400 and glycerol.
Topics: Benzodiazepinones; Capsules; Cholecystokinin; Formates; Glycerol; Indoles; Isomerism; Polyethylene Glycols | 1994 |
Effect of a new cholecystokinin antagonist (FK 480) on gene expression of cholecystokinin and secretin in rat intestine.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Gene Expression; Indoles; Intestinal Mucosa; Male; Rats; Rats, Wistar; RNA, Messenger; Secretin | 1994 |
Effects of a new benzodiazepine derivative cholecystokinin receptor antagonist FK480 on pancreatic exocrine secretion in anesthetized rats.
Topics: Administration, Oral; Animals; Benzodiazepinones; Ceruletide; Cholecystokinin; Dose-Response Relationship, Drug; Indoles; Injections, Intravenous; Male; Pancreas; Proteins; Rats; Rats, Wistar; Receptors, Cholecystokinin | 1994 |
Solvent dependence of optical rotation of (S)-N-[1-(2-fluorophenyl)- 3,4,6,7-tetrahydro-4-oxo-pyrrolo[3,2,1-jk][1,4]benzodiazepine-3-yl]- 1H-indole-2-carboxamide.
Topics: Benzodiazepinones; Cholecystokinin; Circular Dichroism; Crystallography; Indoles; Magnetic Resonance Spectroscopy; Optical Rotation; Solvents; X-Ray Diffraction | 1993 |
CK-independent increases in pancreatic secretion induced by dietary protein in chronic BPJ-diverted rats.
Topics: Animals; Atropine; Benzodiazepinones; Bile; Cholecystokinin; Devazepide; Diet; Hormone Antagonists; Indoles; Male; Pancreas; Pancreatic Juice; Proteins; Rats; Rats, Sprague-Dawley | 1996 |
Small intestinal and pancreatic microstructures are modified by an intraduodenal CCK-A receptor antagonist administration in neonatal calves.
Topics: Animals; Animals, Newborn; Benzodiazepinones; Cattle; Cholecystokinin; Duodenum; Hormone Antagonists; Indoles; Intestine, Small; Pancreas; Pancreatic Juice; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Vacuoles | 1999 |
Bovine pancreatic secretion in the first week of life: potential involvement of intestinal CCK receptors.
Topics: Animals; Animals, Newborn; Benzodiazepinones; Cattle; Cholecystokinin; Colostrum; Indoles; Intestinal Mucosa; Milk; Pancreas; Pancreatic Polypeptide; Peptide Fragments; Postprandial Period; Rats; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Time Factors | 2002 |
Selective activation by photodynamic action of cholecystokinin receptor in the freshly isolated rat pancreatic acini.
Topics: Amylases; Animals; Atropine; Benzodiazepinones; Bethanechol; Calcium; Cholecystokinin; Indoles; Light; Organometallic Compounds; Pancreas; Photochemotherapy; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Receptors, Muscarinic | 2003 |
Mutual dependence of VIP/PACAP and CCK receptor signaling for a physiological role in duck exocrine pancreatic secretion.
Topics: Amylases; Animals; Benzodiazepinones; Calcium; Cholecystokinin; Colforsin; Ducks; Gastrins; In Vitro Techniques; Indoles; Intracellular Membranes; Neuropeptides; Oscillometry; Osmolar Concentration; Pancreas; Pituitary Adenylate Cyclase-Activating Polypeptide; Protein Kinase C; Receptors, Cholecystokinin; Signal Transduction; Vasoactive Intestinal Peptide | 2004 |