fpl 64176 has been researched along with pyrroles in 75 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 20 (26.67) | 18.2507 |
2000's | 35 (46.67) | 29.6817 |
2010's | 18 (24.00) | 24.3611 |
2020's | 2 (2.67) | 2.80 |
Authors | Studies |
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Kunze, DL; Rampe, D | 1 |
Dage, RC; Rampe, D | 1 |
Lacerda, AE; Rampe, D | 1 |
Rampe, D; Triggle, DJ; Zheng, W | 1 |
Cheung, CW; Gigg, M; Hartley, SA; Jones, LM; Usowicz, MM | 1 |
Anderson, B; Dage, RC; Li, T; Rampe, D; Rapien-Pryor, V | 1 |
Baxter, AJ; Dixon, J; Ince, F; Manners, CN; Teague, SJ | 1 |
Dooley, DJ; Feuerstein, TJ; Ginap, T | 1 |
Bergamaschi, A; Malgaroli, A; Scheller, RH; Ting, AE; Tsien, RW; Villa, A; Wendland, B | 1 |
Györke, S; Palade, P; Yasui, K | 1 |
Adams, ME; Mori, Y; Sather, WA; Tanabe, T; Tsien, RW; Zhang, JF | 1 |
Glossmann, H; Grabner, M; Hering, S; Striessnig, J; Wang, Z | 1 |
Bading, H; Chawla, S; Hardingham, GE; Johnson, CM | 1 |
Crumling, MA; Meriney, SD; White, MG | 1 |
Fuhlendorff, J; Gromada, J; Madsen, P; Springborg, J; Varming, AR | 1 |
Handrock, R; Haverich, A; Herzig, S; Hirt, S; Mittmann, C; Schröder, F | 1 |
Chen, Y; Cheng, H; Deng, LH; Lakatta, EG; Sham, JS; Song, LS; Stern, MD | 1 |
Barczak, A; Konradi, C; Leveque, JC; Lewis, SE; Macías, W; Rajadhyaksha, A | 1 |
Handrock, R; Herzig, S; Hofmann, F; Lauven, M; Müller, A | 1 |
Drew, T; Jinnah, HA; Kim, BS; Rothstein, JD; Visser, JE; Yitta, S | 1 |
Bers, DM; Zhou, Z | 1 |
Brownstone, RM; Carlin, KP; Jiang, Z | 1 |
Brownstone, RM; Carlin, KP; Jiang, Z; Jones, KE; Jordan, LM | 1 |
Drew, T; Hess, EJ; Ho, T; Jinnah, HA; Rothstein, JD; Sepkuty, JP; Yitta, S | 1 |
Fan, JS; Palade, P; Yuan, Y | 1 |
Coyne, MD; Gwathmey, JK; Kim, CS | 1 |
Plummer, MR; Schjott, JM | 1 |
Bers, DM; Katoh, H; Schlotthauer, K | 1 |
Janczewski, AM; Lakatta, EG; Stern, MD | 1 |
Barczak, A; Carlson, R; Konradi, C; Macías, W; Rajadhyaksha, A | 1 |
Fan, J; Palade, P; Yuan, Y | 1 |
Barrett, CF; Liu, L; Rittenhouse, AR | 1 |
Altier, C; Bourinet, E; Nargeot, J; Spaetgens, RL; Zamponi, GW | 1 |
Albillos, A; Alonso, MT; Alvarez, J; Cuchillo-Ibáñez, I; G García, A; García-Sancho, J; Montero, M; Olivares, R | 1 |
Cano-Abad, MF; Gabilan, NH; García, AG; López, MG; Villarroya, M | 1 |
Altschuld, RA; Cheng, Y; Dumitrescu, C; Efimov, IR; Narayan, P | 1 |
Fan, JS; Palade, P | 1 |
Frank, AJ; Kelly, JE; Lokuta, AJ; Reddy, ST; Wasserstrom, JA; Wasserstrom, LA | 1 |
Barrett, CF; Gonzalez, PK; Liu, L; Rittenhouse, AR | 1 |
Adachi-Akahane, S; Ichijo, H; Nagao, T; Yamaguchi, S; Yoshioka, K; Zhorov, BS | 1 |
Carlson, RR; Dudman, JT; Konradi, C; Macías, W | 1 |
Bowden, SE; Cloues, RK; Marrion, NV; Shepherd, D; Tavalin, SJ | 1 |
Chawla, S; Huang, CL | 1 |
Bean, BP; McDonough, SI; Mori, Y | 1 |
Feller, MB; Muir-Robinson, G; Torborg, C; Wang, CT | 1 |
Hormuzdi, S; Lewen, A; Misgeld, U; Monyer, H; Titz, S | 1 |
Baker, SP; Bellvé, KD; Carmichael, J; De Crescenzo, V; Fogarty, KE; Lai, FA; Lemos, JR; Lifshitz, LM; Tuft, RA; Walsh, JV; Zhuge, R; Zissimopoulos, S | 1 |
Hong, Z; Isenberg, B; Keirstead, SA; Lee, EH; Reyes, M; Ross, JJ; Tranquillo, RT; Verfaillie, CM; Weir, EK; Willenbring, B; Zeng, L | 1 |
Chen, X; Dore, J; Liu, Y | 1 |
Allen, DD; Gaasch, JA; Geldenhuys, WJ; Lockman, PR; Van der Schyf, CJ | 1 |
Binder, MD; Moritz, AT; Newkirk, G; Powers, RK | 1 |
Grenett, HE; Huang, J; Ku, DD; Urthaler, F; Wolkowicz, PE; Wu, HC | 1 |
Ghais, NS; Grace, AA; Huang, CL; Zhang, Y | 1 |
Adermark, L; Lovinger, DM; Talani, G | 1 |
Banik, NL; Del Re, AM; Ray, SK; Sribnick, EA; Woodward, JJ | 1 |
Amobi, N; Guillebaud, J; Smith, IC | 1 |
Fraser, JA; Grace, AA; Huang, CL; Killeen, MJ; Schwiening, C; Zhang, Y | 1 |
Amobi, N; Guillebaud, J; Smith, CH | 1 |
Atlas, D; Hagalili, Y; Marom, M; Sebag, A; Tzvier, L | 1 |
Cui, JH; Kim, WM; Yoon, MH | 1 |
Cao, C; Khurana, S; Lin, H; Pallone, TL; Zhang, Z | 1 |
Aureliano, M; Gutierrez-Merino, C; Marques-da-Silva, D; Samhan-Arias, AK; Tiago, T | 1 |
Cheetham, CC; Dang, MT; Li, Y; Lovinger, DM; Lu, J; Vo, V; Yokoi, F | 1 |
Amobi, NI; Guillebaud, J; Smith, IC | 1 |
Cao, X; Fang, YY; Gao, TM; Hou, FQ; Hu, HH; Li, SJ; Wang, P; Yan, HC; Zhu, XH | 1 |
Allen, DD; Geldenhuys, WJ; Jones-Higgins, MR; Lockman, JA; Patrick, JD; Van der Schyf, CJ | 1 |
Arranz-Tagarro, JA; Calvo-Gallardo, E; de Pascual, R; Fernández-Morales, JC; Gandía, L; García, AG; Olivares, R; Padín, JF; Vestring, S | 1 |
Alkam, T; Chebolu, S; Darmani, NA; Vaezi, M; Zhong, W | 1 |
Amberg, GC; Clay, CM; Dang, AK; Magee, C; Murtazina, DA; Navratil, AM | 1 |
Eugen, T; Philipp, K; Stanislav, B; Steffen, H | 1 |
Colbran, RJ; Pasek, JG; Wang, X | 1 |
Ke, L; Liao, Q; Nian, W; Ouyang, W; Wang, X; Zhang, R; Zhang, Z | 1 |
Chan, JD; McCusker, P | 1 |
Okada, H; Yasuda, K; Yoshida, A | 1 |
Horita, M; Takadera, T; Uema, S | 1 |
1 review(s) available for fpl 64176 and pyrroles
Article | Year |
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Direct Estimation of CaV1.2 Gating Parameters: Quantification of Voltage Sensor - Pore Transductions and their Modulation by FLP 64176.
Topics: Calcium Channel Agonists; Calcium Channels, L-Type; HEK293 Cells; Humans; Ion Channel Gating; Pyrroles | 2015 |
74 other study(ies) available for fpl 64176 and pyrroles
Article | Year |
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Characterization of the effects of a new Ca2+ channel activator, FPL 64176, in GH3 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Cells, Cultured; Electric Conductivity; In Vitro Techniques; Ion Channel Gating; Pituitary Gland, Anterior; Pyrroles; Rats | 1992 |
Functional interactions between two Ca2+ channel activators, (S)-Bay K 8644 and FPL 64176, in smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Drug Interactions; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Muscle, Smooth, Vascular; Pyrroles; Rats | 1992 |
A new site for the activation of cardiac calcium channels defined by the nondihydropyridine FPL 64176.
Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Dihydropyridines; Electrophysiology; Heart; Heart Ventricles; Isradipine; Myocardium; Potassium; Pyrroles; Rats; Ventricular Function | 1991 |
Pharmacological, radioligand binding, and electrophysiological characteristics of FPL 64176, a novel nondihydropyridine Ca2+ channel activator, in cardiac and vascular preparations.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Isradipine; Male; Myocardium; Potassium; Pyrroles; Radioligand Assay; Rats; Vasoconstriction; Verapamil | 1991 |
Allosteric interactions at L-type calcium channels between FPL 64176 and the enantiomers of the dihydropyridine Bay K 8644.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Allosteric Regulation; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Guinea Pigs; In Vitro Techniques; Ion Channel Gating; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Pyrroles; Stereoisomerism | 1995 |
Comparison of the in vitro and in vivo cardiovascular effects of two structurally distinct Ca++ channel activators, BAY K 8644 and FPL 64176.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Blood Pressure; Calcium Channels; Guinea Pigs; Heart; In Vitro Techniques; Male; Myocardial Contraction; Pyrroles; Rats | 1993 |
Discovery and synthesis of methyl 2,5-dimethyl-4-[2- (phenylmethyl)benzoyl]-1H-pyrrole-3-carboxylate (FPL 64176) and analogues: the first examples of a new class of calcium channel activator.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Guinea Pigs; Myocardial Contraction; Pyrroles; Rats; Stereoisomerism; Structure-Activity Relationship | 1993 |
The non-dihydropyridine L-type voltage-sensitive calcium channel activator FPL 64176 enhances K(+)-evoked efflux of [3H]norepinephrine from rat neocortical slices.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium Channels; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; In Vitro Techniques; Isradipine; Kinetics; Male; Norepinephrine; Potassium; Pyrroles; Rats; Rats, Sprague-Dawley; Tritium | 1993 |
Presynaptic component of long-term potentiation visualized at individual hippocampal synapses.
Topics: Amino Acid Sequence; Animals; Calcium-Binding Proteins; Cells, Cultured; Glutamic Acid; Hippocampus; Long-Term Potentiation; Membrane Glycoproteins; Molecular Sequence Data; Nerve Tissue Proteins; Neurons; Patch-Clamp Techniques; Potassium; Presynaptic Terminals; Pyrroles; Rats; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Synaptic Vesicles; Synaptotagmins | 1995 |
Negative control mechanism with features of adaptation controls Ca2+ release in cardiac myocytes.
Topics: Animals; Calcium; Calcium Channel Agonists; Cells, Cultured; Heart; Homeostasis; Kinetics; Membrane Potentials; Myocardium; Pyrroles; Rats; Rats, Sprague-Dawley; Ryanodine; Time Factors | 1994 |
Distinctive biophysical and pharmacological properties of class A (BI) calcium channel alpha 1 subunits.
Topics: Animals; Biophysical Phenomena; Biophysics; Cadmium; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Electrophysiology; Kinetics; Mollusk Venoms; omega-Conotoxins; Peptides; Pyrroles; Spider Venoms | 1993 |
Transfer of 1,4-dihydropyridine sensitivity from L-type to class A (BI) calcium channels.
Topics: Amino Acid Sequence; Animals; Binding Sites; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Carps; Dihydropyridines; Ion Channel Gating; Isradipine; Molecular Sequence Data; omega-Agatoxin IVA; omega-Conotoxins; Peptide Fragments; Peptides; Protein Structure, Tertiary; Pyrroles; Rabbits; Recombinant Fusion Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Spider Venoms | 1996 |
Distinct functions of nuclear and cytoplasmic calcium in the control of gene expression.
Topics: Animals; Calcium; Calcium Channel Agonists; Cell Line; Cell Nucleus; Chelating Agents; Cyclic AMP Response Element-Binding Protein; Cytoplasm; DNA-Binding Proteins; Egtazic Acid; Gene Expression Regulation; Genes, fos; Humans; Mice; Nuclear Proteins; Potassium Chloride; Pyrroles; Second Messenger Systems; Serum Response Factor; Transcription Factors; Transcription, Genetic | 1997 |
Developmental changes in calcium current pharmacology and somatostatin inhibition in chick parasympathetic neurons.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Ciliary Body; Ganglia, Parasympathetic; Hormone Antagonists; Neurons; Nitrendipine; omega-Conotoxin GVIA; Patch-Clamp Techniques; Peptides; Pyrroles; Somatostatin; Synapses | 1997 |
Increase in [Ca2+]i and subsequent insulin release from beta TC3-cells with the L-type Ca(2+)-channel activator, FPL 64176.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Antigens, Polyomavirus Transforming; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Glyburide; Insulin; Insulin Secretion; Insulinoma; Kinetics; Mice; Mice, Transgenic; Pancreatic Neoplasms; Promoter Regions, Genetic; Pyrroles; Simian virus 40; Tumor Cells, Cultured | 1997 |
Single-channel properties of L-type calcium channels from failing human ventricle.
Topics: Adult; Aged; Calcium; Calcium Channel Agonists; Calcium Channels; Female; Heart; Heart Failure; Heart Ventricles; Humans; Ion Channel Gating; Male; Middle Aged; Patch-Clamp Techniques; Pyrroles | 1998 |
Termination of Ca2+ release by a local inactivation of ryanodine receptors in cardiac myocytes.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Electrophysiology; Male; Myocardium; Pyrroles; Rats; Rats, Wistar; Ryanodine Receptor Calcium Release Channel | 1998 |
L-Type Ca(2+) channels are essential for glutamate-mediated CREB phosphorylation and c-fos gene expression in striatal neurons.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; Gene Expression Regulation; Glutamic Acid; Magnesium; Neurons; Phosphorylation; Proto-Oncogene Proteins c-fos; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sodium | 1999 |
Interaction of three structurally distinct Ca2+ channel activators with single L-type Ca2+ channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Azocines; Calcium Channel Agonists; Calcium Channels; CHO Cells; Cricetinae; Electrophysiology; Pyrroles | 1999 |
Calcium channel activation and self-biting in mice.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aggression; Animals; Behavior, Animal; Bites and Stings; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; Diltiazem; Ion Channel Gating; Mice; Mice, Inbred C57BL; Nifedipine; Nimodipine; Nitrendipine; Pyrroles; Self-Injurious Behavior | 1999 |
Ca2+ influx via the L-type Ca2+ channel during tail current and above current reversal potential in ferret ventricular myocytes.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Electric Conductivity; Electrophysiology; Heart Ventricles; Myocardium; Pyrroles | 2000 |
Characterization of calcium currents in functionally mature mouse spinal motoneurons.
Topics: Animals; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, P-Type; Calcium Channels, Q-Type; Calcium Channels, T-Type; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred BALB C; Motor Neurons; Nifedipine; Patch-Clamp Techniques; Pyrroles; Spinal Cord | 2000 |
Dendritic L-type calcium currents in mouse spinal motoneurons: implications for bistability.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cats; Computer Simulation; Dendrites; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred BALB C; Models, Neurological; Motor Neurons; Nifedipine; Patch-Clamp Techniques; Pyrroles; Spinal Cord | 2000 |
Calcium channel agonists and dystonia in the mouse.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain Mapping; Calcium Channel Agonists; Calcium Channels; Dose-Response Relationship, Drug; Dystonia; Electroencephalography; Electromyography; Locomotion; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Neurologic Examination; Pyrroles | 2000 |
Kinetic effects of FPL 64176 on L-type Ca2+ channels in cardiac myocytes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Heart Ventricles; Kinetics; Male; Myocardium; Pyrroles; Rats; Rats, Sprague-Dawley; Ventricular Function | 2000 |
Voltage-dependent calcium channels in ventricular cells of rainbow trout: effect of temperature changes in vitro.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adaptation, Physiological; Animals; Barium; Body Temperature; Cadmium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cardiotonic Agents; Cold Temperature; Colforsin; Heart Ventricles; In Vitro Techniques; Ion Channel Gating; Isoproterenol; Membrane Potentials; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Nifedipine; Oncorhynchus mykiss; Patch-Clamp Techniques; Pyrroles; Tetrodotoxin | 2000 |
Sustained activation of hippocampal Lp-type voltage-gated calcium channels by tetanic stimulation.
Topics: Action Potentials; Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Cells, Cultured; Electric Stimulation; Embryo, Mammalian; Hippocampus; Long-Term Potentiation; Patch-Clamp Techniques; Pyramidal Cells; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate | 2000 |
Transmission of information from cardiac dihydropyridine receptor to ryanodine receptor: evidence from BayK 8644 effects on resting Ca(2+) sparks.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cells, Cultured; Ferrets; Heart; Heart Ventricles; Ion Channel Gating; Membrane Potentials; Microscopy, Confocal; Myocardium; Nifedipine; Pyrroles; Receptor Cross-Talk; Ryanodine Receptor Calcium Release Channel | 2000 |
Voltage-independent changes in L-type Ca(2+) current uncoupled from SR Ca(2+) release in cardiac myocytes.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Chelating Agents; Egtazic Acid; Electric Conductivity; Electrophysiology; Heart Ventricles; Myocardium; Pyrroles; Rats; Sarcoplasmic Reticulum | 2000 |
Potassium chloride depolarization mediates CREB phosphorylation in striatal neurons in an NMDA receptor-dependent manner.
Topics: Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium-Calmodulin-Dependent Protein Kinase Type 1; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Corpus Striatum; Cyclic AMP Response Element-Binding Protein; DNA-Binding Proteins; Excitatory Amino Acid Antagonists; Fetus; Gene Expression Regulation; Hippocampus; Membrane Potentials; Neurons; Nuclear Proteins; Phosphorylation; Potassium Chloride; Pyrroles; Rats; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Serum Response Factor | 2001 |
FPL-64176 modifies pore properties of L-type Ca(2+) channels.
Topics: Animals; Cadmium; Calcium Channel Agonists; Calcium Channels, L-Type; Cobalt; Electric Conductivity; Heart Ventricles; Male; Myocardium; Permeability; Pyrroles; Rats; Rats, Sprague-Dawley | 2001 |
Arachidonic acid reversibly enhances N-type calcium current at an extracellular site.
Topics: Animals; Animals, Newborn; Arachidonic Acid; Calcium Channel Agonists; Cell Membrane; Cells, Cultured; Guanosine Diphosphate; Kinetics; Membrane Potentials; Neurons; omega-Conotoxin GVIA; Pyrroles; Rats; Rats, Sprague-Dawley; Serum Albumin, Bovine; Superior Cervical Ganglion; Tetrodotoxin; Thionucleotides | 2001 |
Multiple structural elements contribute to voltage-dependent facilitation of neuronal alpha 1C (CaV1.2) L-type calcium channels.
Topics: Animals; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, R-Type; Cation Transport Proteins; Humans; Ion Channel Gating; Membrane Potentials; Neurons; Oocytes; Patch-Clamp Techniques; Pyrroles; Structure-Activity Relationship; Xenopus | 2001 |
Control of secretion by mitochondria depends on the size of the local [Ca2+] after chromaffin cell stimulation.
Topics: Adrenal Medulla; Aequorin; Animals; Caffeine; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Cattle; Cell Membrane; Cells, Cultured; Chromaffin Cells; Fura-2; Membrane Potentials; Mitochondria; Nisoldipine; omega-Conotoxin GVIA; omega-Conotoxins; Potassium; Pyrroles; Ryanodine Receptor Calcium Release Channel | 2001 |
Calcium entry through L-type calcium channels causes mitochondrial disruption and chromaffin cell death.
Topics: Adrenal Medulla; Animals; Apoptosis; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cattle; Chromaffin Cells; Cytochrome c Group; Cytoprotection; Free Radicals; Mitochondria; Necrosis; Nimodipine; Pyrroles | 2001 |
Phase I and phase II of short-term mechanical restitution in perfused rat left ventricles.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Benzylamines; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Enzyme Inhibitors; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Perfusion; Pyrroles; Rats; Rats, Sprague-Dawley; Ryanodine; Sarcolemma; Sarcoplasmic Reticulum; Sulfonamides; Systole; Thapsigargin; Time Factors; Vasodilation; Ventricular Function, Left | 2002 |
Effects of FPL 64176 on Ca transients in voltage-clamped rat ventricular myocytes.
Topics: Action Potentials; Animals; Calcium; Calcium Channel Agonists; Heart Ventricles; Male; Myocardium; Patch-Clamp Techniques; Pyrroles; Rats; Rats, Sprague-Dawley | 2002 |
Activation of cardiac ryanodine receptors by the calcium channel agonist FPL-64176.
Topics: Animals; Calcium; Calcium Channel Agonists; Cats; Dogs; Dose-Response Relationship, Drug; Heart Ventricles; Humans; Ion Channel Gating; Microsomes; Muscle, Skeletal; Myocardium; Pyrroles; Ryanodine Receptor Calcium Release Channel | 2002 |
The calcium channel ligand FPL 64176 enhances L-type but inhibits N-type neuronal calcium currents.
Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, N-Type; Membrane Potentials; Neural Inhibition; Neurons; PC12 Cells; Pyrroles; Rats | 2003 |
Key roles of Phe1112 and Ser1115 in the pore-forming IIIS5-S6 linker of L-type Ca2+ channel alpha1C subunit (CaV 1.2) in binding of dihydropyridines and action of Ca2+ channel agonists.
Topics: Alanine; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; Isradipine; Phenylalanine; Point Mutation; Protein Subunits; Pyrroles; Rats; Repetitive Sequences, Nucleic Acid; Serine | 2003 |
Striatal proenkephalin gene induction: coordinated regulation by cyclic AMP and calcium pathways.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antihypertensive Agents; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Carcinogens; Cells, Cultured; Colforsin; Corpus Striatum; Cyclic AMP; Drug Interactions; Embryo, Mammalian; Enkephalins; Enzyme Inhibitors; Gene Expression Regulation, Developmental; Humans; Isoquinolines; Neurons; Nifedipine; Protein Precursors; Pyrroles; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate; Transcriptional Activation; Transfection | 2003 |
Modulation of single channels underlying hippocampal L-type current enhancement by agonists depends on the permeant ion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Electric Conductivity; Hippocampus; In Vitro Techniques; Permeability; Pyrroles; Rats; Rats, Sprague-Dawley; Time Factors | 2004 |
FPL-64176 alters both charge movement and Ca2+ release properties in amphibian muscle fibres.
Topics: Animals; Calcium Channel Agonists; Calcium Signaling; In Vitro Techniques; Membrane Potentials; Muscle Fibers, Skeletal; Pyrroles; Rana temporaria; Ryanodine Receptor Calcium Release Channel | 2004 |
FPL 64176 modification of Ca(V)1.2 L-type calcium channels: dissociation of effects on ionic current and gating current.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Biophysics; Calcium Channel Agonists; Calcium Channels; Cell Line; Cesium; Cricetinae; Electrophysiology; Ion Channel Gating; Ions; Kinetics; Membrane Potentials; Models, Theoretical; Plasmids; Potassium Channels; Pyrroles; Rabbits; Time Factors; Transfection | 2005 |
L-type calcium channel agonist induces correlated depolarizations in mice lacking the beta2 subunit nAChRs.
Topics: Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Electrophysiology; Mice; Mice, Transgenic; Patch-Clamp Techniques; Pyrroles; Receptors, Nicotinic; Retinal Ganglion Cells; Synaptic Transmission | 2004 |
Intracellular acidification in neurons induced by ammonium depends on KCC2 function.
Topics: Animals; Bumetanide; Calcium; Calcium Channel Agonists; Cells, Cultured; Diagnostic Imaging; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Female; Furosemide; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Hippocampus; Hydrogen-Ion Concentration; Immunohistochemistry; Intracellular Space; K Cl- Cotransporters; Mesencephalon; Neuroglia; Neurons; Potassium Chloride; Pregnancy; Pyrroles; Quaternary Ammonium Compounds; Rats; Rats, Wistar; Sodium Potassium Chloride Symporter Inhibitors; Symporters; Time Factors; Transfection | 2006 |
Dihydropyridine receptors and type 1 ryanodine receptors constitute the molecular machinery for voltage-induced Ca2+ release in nerve terminals.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Membrane; Electric Stimulation; Electrophysiology; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Mice; Nerve Endings; Neurons; Nifedipine; Pyrroles; Ryanodine Receptor Calcium Release Channel | 2006 |
Cytokine-induced differentiation of multipotent adult progenitor cells into functional smooth muscle cells.
Topics: Animals; Animals, Newborn; Becaplermin; Calcium Channel Agonists; Calcium Channels, L-Type; Cell Differentiation; Cells, Cultured; Cytokines; Fibrin; Flow Cytometry; Gene Expression; Humans; Mice; Mice, Inbred C57BL; Multipotent Stem Cells; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Pyrroles; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Swine; Transcription Factors; Transforming Growth Factor beta | 2006 |
Calcium influx through L-type channels generates protein kinase M to induce burst firing of dopamine cells in the rat ventral tegmental area.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Calpain; Dopamine; Female; Glutamine; Protein Kinase C; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Ventral Tegmental Area | 2007 |
Voltage-gated calcium channels provide an alternate route for iron uptake in neuronal cell cultures.
Topics: Animals; Blotting, Western; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Cells, Cultured; Data Interpretation, Statistical; Electrophysiology; Ion Channel Gating; Iron; Neurons; Nimodipine; PC12 Cells; Phenotype; Pyrroles; Rats | 2007 |
Facilitation of somatic calcium channels can evoke prolonged tail currents in rat hypoglossal motoneurons.
Topics: Animals; Animals, Newborn; Brain Stem; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cell Nucleus; Dose-Response Relationship, Radiation; Electric Conductivity; Electric Stimulation; Female; Hypoglossal Nerve; In Vitro Techniques; Male; Membrane Potentials; Motor Neurons; Patch-Clamp Techniques; Pyrroles; Rats; Rats, Sprague-Dawley | 2007 |
A pharmacological model for calcium overload-induced tachycardia in isolated rat left atria.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzazepines; Boron Compounds; Calcium; Calcium Channel Agonists; Cardiotonic Agents; Cyclic Nucleotide-Gated Cation Channels; Heart Atria; In Vitro Techniques; Male; Ouabain; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; RNA, Messenger; Ryanodine; Tachycardia | 2007 |
Arrhythmogenic actions of the Ca2+ channel agonist FPL-64716 in Langendorff-perfused murine hearts.
Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Diltiazem; Disease Models, Animal; Electric Stimulation; Heart; Homeostasis; Indoles; Mice; Mice, Inbred Strains; Myocytes, Cardiac; Nifedipine; Pyrroles; Sarcoplasmic Reticulum; Tachycardia, Ventricular | 2009 |
Endocannabinoid-dependent plasticity at GABAergic and glutamatergic synapses in the striatum is regulated by synaptic activity.
Topics: Action Potentials; Animals; Arachidonic Acids; Calcium Channel Agonists; Calcium Channels, L-Type; Cannabinoid Receptor Modulators; Endocannabinoids; Female; gamma-Aminobutyric Acid; Glutamic Acid; Male; Neostriatum; Neuronal Plasticity; Neurons; Organ Culture Techniques; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Synapses; Synaptic Transmission | 2009 |
Estrogen attenuates glutamate-induced cell death by inhibiting Ca2+ influx through L-type voltage-gated Ca2+ channels.
Topics: Animals; Apoptosis; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Calpain; Caspase 3; Cell Line; Cell Physiological Phenomena; Electric Capacitance; Estradiol; Estrogens; Glutamic Acid; Intracellular Space; Membrane Potentials; Mice; Neurons; Neuroprotective Agents; Pyrroles; Rats | 2009 |
Contractile actions of L-type Ca2+ agonists in human vas deferens and effects of structurally different Ca2+ antagonists.
Topics: Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Humans; In Vitro Techniques; Male; Muscle Contraction; Phenothiazines; Potassium; Pyrroles; Vas Deferens | 2010 |
Acute atrial arrhythmogenesis in murine hearts following enhanced extracellular Ca(2+) entry depends on intracellular Ca(2+) stores.
Topics: Aniline Compounds; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Caffeine; Calcium; Calcium Channels, L-Type; Calcium Signaling; Heart; Heart Atria; Mice; Myocytes, Cardiac; Nifedipine; Pyrroles; Xanthenes | 2010 |
Comparative effects of T-type and L-type Ca(2+)-antagonists against noradrenaline-induced contractions of human vas deferens.
Topics: Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Flunarizine; Humans; Male; Mibefradil; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Pyrroles; Vas Deferens | 2010 |
Conformational changes induced in voltage-gated calcium channel Cav1.2 by BayK 8644 or FPL64176 modify the kinetics of secretion independently of Ca2+ influx.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Electrochemical Techniques; Lanthanum; Membrane Potentials; Mutation; Protein Conformation; Protein Subunits; Pyrroles; Rats | 2010 |
Role of PKG-L-type calcium channels in the antinociceptive effect of intrathecal sildenafil.
Topics: Animals; Calcium Channel Agonists; Calcium Channels, L-Type; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Male; Pain; Pain Measurement; Piperazines; Protein Kinase Inhibitors; Purines; Pyrroles; Rats; Rats, Sprague-Dawley; Sildenafil Citrate; Sulfones | 2010 |
Voltage-gated divalent currents in descending vasa recta pericytes.
Topics: Animals; Barium; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Kidney Medulla; Mibefradil; Models, Animal; Nickel; Nifedipine; omega-Agatoxin IVA; Patch-Clamp Techniques; Pericytes; Pyrroles; Rats | 2010 |
Early disruption of the actin cytoskeleton in cultured cerebellar granule neurons exposed to 3-morpholinosydnonimine-oxidative stress is linked to alterations of the cytosolic calcium concentration.
Topics: Actin Cytoskeleton; Animals; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Cells, Cultured; Cerebellum; Molsidomine; Neurons; Nifedipine; Oxidative Stress; Peroxynitrous Acid; Pyrroles; Rats; Rats, Wistar | 2011 |
An anticholinergic reverses motor control and corticostriatal LTD deficits in Dyt1 ΔGAG knock-in mice.
Topics: Animals; Calcium Channel Agonists; Corpus Striatum; Disease Models, Animal; Dystonia Musculorum Deformans; Gene Knock-In Techniques; Humans; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Mice; Mice, Transgenic; Molecular Chaperones; Muscarinic Antagonists; Pyrroles; Receptors, Dopamine D2; Trihexyphenidyl | 2012 |
Perspective on the role of P2X-purinoceptor activation in human vas deferens contractility.
Topics: 4-Aminopyridine; Adenosine Triphosphate; Amides; Apamin; Calcium Channel Agonists; Calcium Channels, L-Type; Humans; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle Contraction; Norepinephrine; Peptides; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Purinergic P2X Receptor Agonists; Pyridines; Pyrophosphatases; Pyrroles; Receptors, Purinergic P2X; rho-Associated Kinases; Suramin; Vas Deferens | 2012 |
An L-type calcium channel agonist, bay K8644, extends the window of intervention against ischemic neuronal injury.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain Ischemia; Butadienes; Calcium Channels, L-Type; Extracellular Signal-Regulated MAP Kinases; Maze Learning; Memory; Neurons; Neuroprotective Agents; Nitriles; Phosphorylation; Pyrroles; Rats; Rats, Sprague-Dawley; Rats, Wistar | 2013 |
NGP1-01, a multi-targeted polycyclic cage amine, attenuates brain endothelial cell death in iron overload conditions.
Topics: Amines; Animals; Apoptosis; Arabidopsis Proteins; Blood-Brain Barrier; Bridged-Ring Compounds; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Carrier Proteins; Cell Survival; Endothelial Cells; Iron Overload; Nerve Degeneration; Neuroprotective Agents; Pyrroles; Rats; Receptors, N-Methyl-D-Aspartate; Transcription Factors | 2012 |
Plasmalemmal sodium-calcium exchanger shapes the calcium and exocytotic signals of chromaffin cells at physiological temperature.
Topics: Animals; Bromides; Caffeine; Calcium Channel Blockers; Calcium Signaling; Catecholamines; Cattle; Cell Membrane; Cells, Cultured; Chromaffin Cells; Exocytosis; Histamine; Kinetics; Membrane Potentials; Nifedipine; Patch-Clamp Techniques; Potassium; Potassium Compounds; Pyrroles; Sodium-Calcium Exchanger; Temperature | 2013 |
Broad-spectrum antiemetic potential of the L-type calcium channel antagonist nifedipine and evidence for its additive antiemetic interaction with the 5-HT(3) receptor antagonist palonosetron in the least shrew (Cryptotis parva).
Topics: Animals; Antiemetics; Calcium Channel Blockers; Calcium Channels, L-Type; Drug Synergism; Female; Isoquinolines; Male; Nifedipine; Palonosetron; Pyrroles; Quinuclidines; Receptors, Serotonin, 5-HT3; Serotonin 5-HT3 Receptor Antagonists; Shrews; Vomiting | 2014 |
GnRH evokes localized subplasmalemmal calcium signaling in gonadotropes.
Topics: Animals; Calcium Signaling; Cell Line; Electrophysiology; Gonadotrophs; Gonadotropin-Releasing Hormone; Mice; Microscopy, Fluorescence; Nicardipine; Pyrroles | 2014 |
Differential CaMKII regulation by voltage-gated calcium channels in the striatum.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Chelating Agents; Corpus Striatum; Egtazic Acid; Enzyme Inhibitors; Gene Expression Regulation; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Pyrroles; Receptors, Glutamate; Signal Transduction; Spider Venoms | 2015 |
Effect of fluoride exposure on mRNA expression of cav1.2 and calcium signal pathway apoptosis regulators in PC12 cells.
Topics: Animals; Apoptosis; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Fluorides; Fluorosis, Dental; Nifedipine; PC12 Cells; Pyrroles; Rats; RNA, Messenger; Signal Transduction | 2017 |
Anti-schistosomal action of the calcium channel agonist FPL-64176.
Topics: Animals; Biotinylation; Calcium Channel Agonists; Calcium Signaling; Female; Helminth Proteins; Male; Mice; Microscopy, Electron, Transmission; Pyrroles; Real-Time Polymerase Chain Reaction; Schistosoma mansoni; Schistosomiasis mansoni | 2019 |
Conflicting Nongenomic Effects of Progesterone in the Myometrium of Pregnant Rats.
Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels, L-Type; Female; Hormone Antagonists; Mifepristone; Myometrium; Nifedipine; Organ Culture Techniques; Oxytocin; Potassium Chloride; Pregnancy; Progesterone; Pyrroles; Rats, Wistar; Uterine Contraction; Verapamil | 2021 |
Protective effects of calcium ions via L-type calcium channels and NMDA receptors on prostaglandin E
Topics: Animals; Apoptosis; Calcium; Calcium Channel Agonists; Calcium Channels, L-Type; Calcium Signaling; Carbazoles; Cells, Cultured; Cerebral Cortex; Dinoprostone; Enzyme Inhibitors; Ions; N-Methylaspartate; Neurons; Protective Agents; Protein Kinase C; Pyrroles; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate | 2021 |