Page last updated: 2024-09-04

fpl 52757 and metergoline

fpl 52757 has been researched along with metergoline in 1 studies

Compound Research Comparison

Studies
(fpl 52757)
Trials
(fpl 52757)
Recent Studies (post-2010)
(fpl 52757)
Studies
(metergoline)
Trials
(metergoline)
Recent Studies (post-2010) (metergoline)
6216563744

Protein Interaction Comparison

ProteinTaxonomyfpl 52757 (IC50)metergoline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.0007
Bile salt export pumpHomo sapiens (human)10
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)0.366
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0041
Alpha-2A adrenergic receptorHomo sapiens (human)0.058
Cytochrome P450 2D6Homo sapiens (human)0.2
D(2) dopamine receptorHomo sapiens (human)0.063
Alpha-2B adrenergic receptorHomo sapiens (human)0.016
Alpha-2C adrenergic receptorHomo sapiens (human)0.189
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0062
Substance-K receptorHomo sapiens (human)4.071
D(1A) dopamine receptorHomo sapiens (human)0.074
AcetylcholinesteraseHomo sapiens (human)1.344
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.366
Histamine H2 receptorHomo sapiens (human)0.975
Alpha-1D adrenergic receptorHomo sapiens (human)0.136
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0007
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0062
Sodium-dependent serotonin transporterHomo sapiens (human)0.59
Histamine H1 receptorHomo sapiens (human)4.133
D(3) dopamine receptorHomo sapiens (human)0.0077
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 6Homo sapiens (human)0.028
Sodium-dependent dopamine transporter Homo sapiens (human)0.063

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1

Other Studies

1 other study(ies) available for fpl 52757 and metergoline

ArticleYear
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012