Compounds > formestane

Page last updated: 2024-08-21

formestane and ketoconazole

formestane has been researched along with ketoconazole in 11 studies

Research

Studies (11)

Timeframe	Studies, this research(%)	All Research%
pre-1990	2 (18.18)	18.7374
1990's	4 (36.36)	18.2507
2000's	2 (18.18)	29.6817
2010's	3 (27.27)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Cole, PA; Robinson, CH	1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J	1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J	1
Majetich, G; Shimkus, JM	1
Ayub, M; Levell, MJ	2
Armstrong, DT; Glasier, MA; Khalil, MW; Lang, T; Morley, P	1
Bhatnagar, AS; King, EJ; Purba, HS; Richert, P	1
Moslemi, S; Seralini, GE	1
Aceves-Ramos, A; Gaona, B; Romano, MC; Valdez, RA; Willms, K	1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL	1

Reviews

2 review(s) available for formestane and ketoconazole

Article	Year
Mechanism and inhibition of cytochrome P-450 aromatase. Journal of medicinal chemistry, 1990, Volume: 33, Issue:11 Topics: Affinity Labels; Aromatase; Aromatase Inhibitors; Binding, Competitive; Humans; Molecular Structure; Photochemistry	1990
The taiwaniaquinoids: a review. Journal of natural products, 2010, Feb-26, Volume: 73, Issue:2 Topics: Biological Products; Cupressaceae; Diterpenes; Molecular Structure	2010

Other Studies

9 other study(ies) available for formestane and ketoconazole

Article	Year
Chemical genetics reveals a complex functional ground state of neural stem cells. Nature chemical biology, 2007, Volume: 3, Issue:5 Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells	2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum. Nature chemical biology, 2009, Volume: 5, Issue:10 Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection	2009
The inhibition of human prostatic aromatase activity by imidazole drugs including ketoconazole and 4-hydroxyandrostenedione. Biochemical pharmacology, 1990, Oct-01, Volume: 40, Issue:7 Topics: Androstenedione; Aromatase Inhibitors; Estradiol; Estrone; Humans; Imidazoles; Ketoconazole; Male; Prostate; Structure-Activity Relationship	1990
Formation of 4-oestrene-3,17-dione (19-norandrostenedione) by porcine granulosa cells in vitro is inhibited by the aromatase inhibitor 4-hydroxyandrostenedione and the cytochrome P-450 inhibitors aminoglutethimide phosphate and ketoconazole. The Journal of endocrinology, 1989, Volume: 120, Issue:2 Topics: Aminoglutethimide; Androstenedione; Animals; Cells, Cultured; Female; Granulosa Cells; Ketoconazole; Swine	1989
Structure-activity relationships of the inhibition of human placental aromatase by imidazole drugs including ketoconazole. Journal of steroid biochemistry, 1988, Volume: 31, Issue:1 Topics: Aminoglutethimide; Androstenedione; Aromatase Inhibitors; Humans; Imidazoles; Ketoconazole; Microsomes; Placenta; Structure-Activity Relationship	1988
Effect of aromatase inhibitors on estrogen 2-hydroxylase in rat liver. The Journal of steroid biochemistry and molecular biology, 1994, Volume: 48, Issue:2-3 Topics: Aminoglutethimide; Androstenedione; Animals; Aromatase Inhibitors; Binding, Competitive; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Estradiol; Estrone; Fadrozole; Female; Ketoconazole; Microsomes, Liver; Rats; Rats, Sprague-Dawley; Steroid Hydroxylases; Substrate Specificity	1994
Inhibition and inactivation of equine aromatase by steroidal and non-steroidal compounds. A comparison with human aromatase inhibition. Journal of enzyme inhibition, 1997, Volume: 12, Issue:4 Topics: Androstenedione; Animals; Aromatase Inhibitors; Enzyme Activation; Fadrozole; Horses; Humans; Imidazoles; Ketoconazole; Male; Miconazole; Substrate Specificity	1997
Steroid synthesis by Taenia crassiceps WFU cysticerci is regulated by enzyme inhibitors. General and comparative endocrinology, 2013, Jul-01, Volume: 188 Topics: Androstenedione; Animals; Chromatography, Thin Layer; Danazol; Desoxycorticosterone; Enzyme Inhibitors; Estradiol; Ketoconazole; Steroids; Taenia	2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics. PloS one, 2016, Volume: 11, Issue:10 Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat	2016