flutamide has been researched along with metribolone in 24 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (4.17) | 18.7374 |
1990's | 14 (58.33) | 18.2507 |
2000's | 8 (33.33) | 29.6817 |
2010's | 1 (4.17) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
de Launoit, Y; Dufour, M; Labrie, F; Simard, J; Veilleux, R | 1 |
Bellward, GD; Pak, RC; Sunahara, GI | 1 |
Bravo, AI; Calandra, RS; Capurro, MI; Donaldson, M; Luthy, IA; Mordoh, J; Morvillo, V; Quintans, C | 1 |
D'Eramo, G; Di Silverio, F; Felli, MP; Frati, L; Gulino, A; Lubrano, C; Maroder, M; Ravenna, L; Sciarra, F; Vacca, A | 1 |
Govindan, MV; Koutsilieris, M; Pagé, N; Warriar, N | 1 |
Berrevoets, CA; Mulder, E; Veldscholte, J | 1 |
Fanger, GR; Henderson, LP; Maue, RA; Tabb, JS; Wilson, EM | 1 |
Burnstein, KL; Cameron, DJ; Dai, JL; Maiorino, CA | 1 |
Jimenez, J; Luizzi, MF; Sonnenschein, C; Soto, AM; Szelei, J | 1 |
Bartsch, G; Cronauer, MV; Culig, Z; Hittmair, A; Hobisch, A; Klocker, H; Radmayr, C; Zhang, J | 1 |
Judd, J; Kremer, M; Oursler, MJ; Pascoe, D; Pederson, L; Riggs, BL; Spelsberg, TC | 1 |
Bisht, D; Chakraborti, PK; Rana, S | 1 |
Funder, JW; Li, H; Liu, JP; Zhu, X | 1 |
Fan, Z; Mendelsohn, J; Ye, D | 1 |
Caplan, AJ; Cheetham, ME; Fliss, AE; Melville, MW; Rao, J | 1 |
Lumbroso, S; Moras, D; Nicolas, JC; Poujol, N; Sultan, C; Tahiri, B; Wurtz, JM | 1 |
Jones, GR; Lyng, FM; Rommerts, FF | 1 |
Appa Rao, KB; Gui, Y; Lessey, BA; Lovely, LP | 1 |
Gao, AC; Hou, M; Lee, SO; Lou, W; Onate, SA | 1 |
Lemaire, G; Mauvais, P; Michel, S; Rahmani, R; Terouanne, B | 1 |
Farla, P; Hersmus, R; Houtsmuller, AB; Trapman, J | 1 |
Chang, CY; Elbi, C; Hager, GL; Hendarwanto, A; Klokk, TI; Kurys, P; Nagaich, AK; Saatcioglu, F; Slagsvold, T | 1 |
Bowles, HJ; Burchiel, SW; Dennis, MK; Edwards, BS; MacKenzie, DA; Prossnitz, ER; Sklar, LA; Thompson, TA | 1 |
Dits, NF; Erkens-Schulze, S; Jenster, G; Marques, RB; van Ijcken, WF; van Weerden, WM | 1 |
24 other study(ies) available for flutamide and metribolone
Article | Year |
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Characteristics of the biphasic action of androgens and of the potent antiproliferative effects of the new pure antiestrogen EM-139 on cell cycle kinetic parameters in LNCaP human prostatic cancer cells.
Topics: Androgens; Androstane-3,17-diol; Binding, Competitive; Cell Cycle; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Antagonism; Estradiol; Estrogen Antagonists; Estrone; Flow Cytometry; Flutamide; Humans; In Vitro Techniques; Male; Metribolone; Piperidines; Prostatic Neoplasms; Raloxifene Hydrochloride; Tamoxifen; Testosterone; Time Factors; Tumor Cells, Cultured | 1991 |
Effect of flutamide on hepatic cytosolic methyltrienolone (R1881) binding kinetics and testosterone responsive hepatic drug and steroid metabolism in the adult male rat.
Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Androgen-Binding Protein; Anilides; Animals; Aryl Hydrocarbon Hydroxylases; Benzopyrene Hydroxylase; Body Weight; Castration; Cytosol; Estrenes; Female; Flutamide; Kinetics; Liver; Male; Metribolone; Organ Size; Rats; Receptors, Androgen; Sex Factors; Testosterone | 1987 |
Atypical androgen receptor in the human melanoma cell line IIB-MEL-J.
Topics: Androgen Antagonists; Animals; Antibodies, Monoclonal; Antineoplastic Agents, Hormonal; Binding, Competitive; Cell Division; Dihydrotestosterone; Estradiol; Flutamide; Humans; Hydrocortisone; Immunohistochemistry; Male; Melanoma; Metribolone; Mice; Mice, Nude; Progesterone; Receptors, Androgen; Testosterone; Tumor Cells, Cultured | 1995 |
Androgenic and antiandrogenic control on epidermal growth factor, epidermal growth factor receptor, and androgen receptor expression in human prostate cancer cell line LNCaP.
Topics: Androgen Antagonists; Blotting, Northern; Down-Regulation; Epidermal Growth Factor; ErbB Receptors; Flutamide; Gene Expression; Humans; Male; Metribolone; Prostatic Neoplasms; Protein Binding; Radioimmunoassay; Receptors, Androgen; RNA, Messenger; Time Factors; Tumor Cells, Cultured | 1995 |
Interaction of antiandrogen-androgen receptor complexes with DNA and transcription activation.
Topics: Androgen Antagonists; Animals; Binding, Competitive; Blotting, Western; Cell Line; Chloramphenicol O-Acetyltransferase; Chlorocebus aethiops; Cyproterone Acetate; Dihydrotestosterone; DNA; Flutamide; Gene Expression Regulation; Humans; Imidazoles; Imidazolidines; Kidney; Kinetics; Mammary Tumor Virus, Mouse; Metribolone; Receptors, Androgen; Recombinant Proteins; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection | 1993 |
Effects of antiandrogens on transformation and transcription activation of wild-type and mutated (LNCaP) androgen receptors.
Topics: Adenocarcinoma; Alanine; Amino Acid Sequence; Androgen Antagonists; Anilides; Animals; Blotting, Western; Cell Line; Cell Nucleus; Chloramphenicol O-Acetyltransferase; Cyproterone Acetate; Dose-Response Relationship, Drug; Flutamide; Humans; Male; Metribolone; Mutagenesis, Site-Directed; Nitriles; Point Mutation; Prostatic Neoplasms; Receptors, Androgen; Recombinant Proteins; Threonine; Tosyl Compounds; Transcription, Genetic; Transfection; Transformation, Genetic; Tumor Cells, Cultured | 1993 |
Suppression of sodium channel function in differentiating C2 muscle cells stably overexpressing rat androgen receptors.
Topics: Acetylcholine; Androgen Antagonists; Animals; Bungarotoxins; Cell Differentiation; Cell Line; Dihydrotestosterone; Flutamide; Gene Expression; Metribolone; Mice; Muscles; Rats; Receptors, Androgen; Receptors, Cholinergic; Sodium Channels; Transfection | 1994 |
Androgen and glucocorticoid regulation of androgen receptor cDNA expression.
Topics: Cell Line; Cyproterone Acetate; Cytomegalovirus; DNA, Complementary; Dose-Response Relationship, Drug; Down-Regulation; Flutamide; Gene Expression; Glucocorticoids; Humans; Metribolone; Promoter Regions, Genetic; Protein Biosynthesis; Receptors, Androgen; Receptors, Glucocorticoid; RNA, Messenger; Testosterone Congeners; Time Factors; Transfection; Tumor Cells, Cultured | 1995 |
Androgen-induced inhibition of proliferation in human breast cancer MCF7 cells transfected with androgen receptor.
Topics: Androgen Antagonists; Androgens; Anilides; Blotting, Western; Breast Neoplasms; Cell Cycle; Cell Division; Dihydrotestosterone; Dose-Response Relationship, Drug; Female; Flutamide; Humans; In Vitro Techniques; Metribolone; Nandrolone; Nitriles; Receptors, Androgen; Testosterone; Testosterone Congeners; Tosyl Compounds; Transfection; Tumor Cells, Cultured | 1997 |
Synergistic activation of androgen receptor by androgen and luteinizing hormone-releasing hormone in prostatic carcinoma cells.
Topics: Androgen Antagonists; Anilides; Bucladesine; Cell Line; Chloramphenicol O-Acetyltransferase; Cyclic AMP; Flutamide; Genes, Reporter; Gonadotropin-Releasing Hormone; Humans; Kinetics; Male; Metribolone; Nitriles; Prostate-Specific Antigen; Prostatic Neoplasms; Receptors, Androgen; Recombinant Fusion Proteins; Testosterone Congeners; Tosyl Compounds; Transcriptional Activation; Transfection; Tumor Cells, Cultured | 1997 |
Androgens regulate bone resorption activity of isolated osteoclasts in vitro.
Topics: Acid Phosphatase; Androgen Antagonists; Androgens; Animals; Bone Resorption; Cathepsin B; Chickens; Dihydrotestosterone; Flutamide; Genes, Reporter; Humans; Isoenzymes; Metribolone; Mice; Osteoclasts; Receptors, Androgen; Regulatory Sequences, Nucleic Acid; Tartrate-Resistant Acid Phosphatase; Transfection; Transforming Growth Factor beta | 1999 |
Synergistic activation of yeast-expressed rat androgen receptor by modulators of protein kinase-A.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 8-Bromo Cyclic Adenosine Monophosphate; Androgens; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyproterone; Dihydrotestosterone; Enzyme Inhibitors; Flutamide; Gene Expression Regulation; Genes, Reporter; Metribolone; Okadaic Acid; Rats; Receptors, Androgen; Regulatory Sequences, Nucleic Acid; RNA, Messenger; Saccharomyces cerevisiae; Signal Transduction; Transcriptional Activation; Transformation, Genetic | 1999 |
Androgen stimulates mitogen-activated protein kinase in human breast cancer cells.
Topics: Androgen Antagonists; Breast Neoplasms; Calcium-Calmodulin-Dependent Protein Kinases; DNA Replication; Dose-Response Relationship, Drug; Enzyme Activation; Female; Flutamide; Humans; Metribolone; Testosterone Congeners; Tumor Cells, Cultured | 1999 |
Androgen and epidermal growth factor down-regulate cyclin-dependent kinase inhibitor p27Kip1 and costimulate proliferation of MDA PCa 2a and MDA PCa 2b prostate cancer cells.
Topics: Androgen Antagonists; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Cell Cycle Proteins; Cell Division; Cyclin-Dependent Kinase Inhibitor p27; Cyclin-Dependent Kinases; Cycloheximide; Dihydrotestosterone; Down-Regulation; Drug Synergism; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Flutamide; Humans; Male; Metribolone; Microtubule-Associated Proteins; Prostatic Neoplasms; Protein Synthesis Inhibitors; Receptors, Androgen; Testosterone Congeners; Trastuzumab; Tumor Cells, Cultured; Tumor Suppressor Proteins | 1999 |
Domain requirements of DnaJ-like (Hsp40) molecular chaperones in the activation of a steroid hormone receptor.
Topics: Binding Sites; Binding, Competitive; Flutamide; Gene Deletion; Genetic Complementation Test; Heat-Shock Proteins; HSP40 Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Humans; Metribolone; Molecular Chaperones; Mutation; Phenotype; Protein Binding; Protein Structure, Tertiary; Radioligand Assay; Receptors, Androgen; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Suppression, Genetic; Tritium; Zinc Fingers | 1999 |
Specific recognition of androgens by their nuclear receptor. A structure-function study.
Topics: Amino Acid Sequence; Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Anilides; Binding Sites; Computer Simulation; Cyproterone Acetate; Dose-Response Relationship, Drug; Flutamide; Humans; Ligands; Metribolone; Models, Molecular; Molecular Sequence Data; Nitriles; Progesterone; Promegestone; Receptors, Androgen; Sequence Alignment; Tosyl Compounds; Transcriptional Activation | 2000 |
Rapid androgen actions on calcium signaling in rat sertoli cells and two human prostatic cell lines: similar biphasic responses between 1 picomolar and 100 nanomolar concentrations.
Topics: Androgen Antagonists; Androgens; Animals; Calcium Signaling; Cell Line; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Gap Junctions; Humans; Kinetics; Male; Metribolone; Prostate; Prostatic Neoplasms; Rats; Rats, Wistar; Sertoli Cells; Testosterone; Tumor Cells, Cultured | 2000 |
Characterization of androgen receptors in a well-differentiated endometrial adenocarcinoma cell line (Ishikawa).
Topics: Adenocarcinoma; Alkaline Phosphatase; Androgens; Cell Differentiation; Cell Nucleus; Diethylstilbestrol; Dihydrotestosterone; Endometrial Neoplasms; Endometrium; Estradiol; Estrogen Receptor Modulators; Estrogens; Female; Flutamide; Fulvestrant; Humans; Metribolone; Progesterone; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; Tumor Cells, Cultured | 2000 |
Interleukin-4 enhances prostate-specific antigen expression by activation of the androgen receptor and Akt pathway.
Topics: Androgen Antagonists; Cell Nucleus; Chromones; Colonic Neoplasms; Enzyme Inhibitors; Flutamide; Gene Expression; Humans; Interleukin-4; Male; Metribolone; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Prostate-Specific Antigen; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Receptors, Androgen; Response Elements; RNA, Messenger; Signal Transduction; Testosterone Congeners; Tumor Cells, Cultured | 2003 |
Effect of organochlorine pesticides on human androgen receptor activation in vitro.
Topics: Androgen Antagonists; Binding, Competitive; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Flutamide; Humans; Inhibitory Concentration 50; Insecticides; Male; Metribolone; Receptors, Androgen; Testosterone Congeners | 2004 |
Antiandrogens prevent stable DNA-binding of the androgen receptor.
Topics: Androgen Antagonists; Androgen Receptor Antagonists; Androgens; Anilides; Blotting, Western; Carcinoma, Hepatocellular; Cell Line, Tumor; Cells, Cultured; Computer Simulation; DNA; DNA-Binding Proteins; DNA, Neoplasm; Flutamide; Green Fluorescent Proteins; Humans; Liver Neoplasms; Male; Metribolone; Nitriles; Prostatic Neoplasms; Receptors, Androgen; Recombinant Fusion Proteins; Tosyl Compounds | 2005 |
Ligand-specific dynamics of the androgen receptor at its response element in living cells.
Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Anilides; Animals; Cell Line, Tumor; Chromatin Assembly and Disassembly; Cyproterone Acetate; Dihydrotestosterone; Female; Fluorescence Recovery After Photobleaching; Flutamide; Genes, Reporter; Green Fluorescent Proteins; In Situ Hybridization, Fluorescence; Ligands; Luciferases; Mammary Neoplasms, Animal; Mammary Tumor Virus, Mouse; Metribolone; Mice; Microscopy, Video; Mifepristone; Models, Biological; Nitriles; Plasmids; Promoter Regions, Genetic; Receptors, Androgen; Response Elements; Testosterone; Tosyl Compounds; Transcription, Genetic | 2007 |
A multifunctional androgen receptor screening assay using the high-throughput Hypercyt flow cytometry system.
Topics: Androgen Receptor Antagonists; Androgens; Cell Line, Tumor; Drug Evaluation, Preclinical; Flow Cytometry; Flutamide; Humans; Male; Metribolone; Receptors, Androgen; Transcriptional Activation; Transfection | 2008 |
Modulation of androgen receptor signaling in hormonal therapy-resistant prostate cancer cell lines.
Topics: Androgen Antagonists; Antineoplastic Agents, Hormonal; Base Sequence; Cell Line, Tumor; DNA Primers; Drug Resistance, Neoplasm; Flutamide; Gene Expression Profiling; Humans; Male; Metribolone; Oligonucleotide Array Sequence Analysis; Prostatic Neoplasms; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction | 2011 |