flutamide and cyproterone

flutamide has been researched along with cyproterone in 109 studies

Research

Studies (109)

TimeframeStudies, this research(%)All Research%
pre-199073 (66.97)18.7374
1990's24 (22.02)18.2507
2000's9 (8.26)29.6817
2010's2 (1.83)24.3611
2020's1 (0.92)2.80

Authors

AuthorsStudies
Ackerman, JH; Bell, MR; Christiansen, RG; D'Ambra, TE; Herrmann, JL; Kullnig, RK; Mallamo, JP; Opalka, CJ; Snyder, BW; Winneker, RC1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY1
Neri, RO1
Chisholm, GD; Ghanadian, R; Smith, CB; Williams, G1
Bruchovsky, N; Callaway, T; Comeau, T; Lakey, WH; Lieskovsky, G; Rennie, P; Shnitka, T; Wilkin, P1
Takayasu, S2
Datta, JK; Kumari, GL; Roy, S1
Munshi, SR; Nagendranath, N; Raman, G; Sheth, AR1
Liao, S; Tymoczko, JL1
Hillier, SG; Knazek, RA; Ross, GT1
Cuthbertson, TL; Li, JJ; Li, SA1
Bardin, CW; Brown, TR; Greene, FE1
Gidari, AS; Lane, SE; Levere, RD1
Schmidt, JD1
Chung, LW; Ferland-Raymond, G1
Harman, SM; Louvet, JP; Ross, GT; Schrieber, JR1
Neri, RO; Peets, EA1
Coffey, DS; Sufrin, G1
Beato, M; Bock, K; Filmer, A; Hackenberg, R; Hawighorst, T; Schulz, KD; Slater, EP1
Ameye, F; Baert, L; Oyen, R; Van De Voorde, W; Van Poppel, H1
Schmeller, N1
Imai, K; Kawashima, K; Nakata, S; Shimizu, N; Suzuki, T; Takahashi, O; Watanabe, K; Yamanaka, H1
Radoś, N; Tarle, M1
Cantabrana, B; Garcia Valencia, V; Gutierrez, M; Hidalgo, A; Sanchez, M1
el Etreby, MF; Habenicht, UF; Neumann, F1
Schulze, H; Senge, T1
D'Eramo, G; Di Silverio, F; Sciarra, F1
Schröder, FH2
Concolino, G; Di Silverio, F; Sciarra, F; Toscano, V1
Arbusow, V; Bojar, H; Fittler, F; Klobeck, HG; Schulz, P; Wolf, D1
Cusan, L; Labrie, C; Labrie, F; Lapointe, S; Plante, M1
Concolino, G; Conti, C; Di Silverio, F; Lubrano, C; Petrangeli, E; Sciarra, F; Toscano, V1
Labrie, F; Lapointe, S; Plante, M1
Le Guellec, R; Léger, JG; Tenniswood, MP1
Namer, M1
Baylink, DJ; Farley, JR; Kasperk, CH; Linkhart, TA; Turner, RT; Wergedal, JE1
Shaw, CJ; Snyder, BW; Wagner, MM; Winneker, RC1
Waxman, J1
Milsted, RA1
Ganten, D; Ganten, U; Schröder, G; Stock, G; Witt, M; Zimmermann, F1
Gupta, G; Setty, BS; Srivastava, A1
Mowszowicz, I1
Furr, BJ2
Daricello, G; Pavone, C; Pavone-Macaluso, M; Romano, C; Serretta, V1
Combettes, C; Durand-Seme, V; Leveque, JL; Querleux, B; Saint-Leger, D1
Gangnerau, MN; Picon, R1
Dias, JA; Swift, TA1
Abel, P; Cox, J; Farah, N; Fleming, J; Hewitt, G; O'Donoghue, EP; Sandow, J; Sikora, K; Waxman, J; Williams, G1
Sathyanesan, AG; Shrivastava, VK1
Sogani, PC; Whitmore, WF1
Soloway, MS1
Haider, S; Rai, U1
Alexandre, C; Balthazart, J2
Cunningham, GR; Kong, AY; Shao, TC1
Gutiérrez Cecchini, B; Hidalgo Balsera, A; Manso Rodríguez, G; Sala Blanco, J1
Fair, WR; Sogani, PC1
Ayub, M; Levell, MJ1
Dupront, A; Meyer, BH; Pottier, J; Tremblay, D1
el Etreby, MF; Habenicht, UF; Louton, T; Nishino, Y; Schröder, HG1
el Etreby, MF; Habenicht, UF; Neumann, F; Schröder, H1
Bruchovsky, N; Fletcher, T; Foekens, JA; Goldenberg, SL; Lawson, D; Rennie, PS1
Donn, F; Tamm, J; Volkwein, U1
Clos, V; Esteve, A; Jane, F; Salva, P1
Bouffioux, C1
Alioth, H; Müller, J; Senn, E1
Tokarz, RR1
Boublil, JL; Cavaglione, G; Kather, R; Namer, M1
Neumann, F1
Labrie, F; Poyet, P1
Wilson, FE1
Datta, JK; Roy, S1
Bullock, LP; Ventura, SM1
Jacobi, GH; Wenderoth, UK1
Hano, R; Knuth, UA; Nieschlag, E1
Ahmed, K; Davis, AT; Wilson, MJ1
Das, RP; Kumari, GL; Roy, S1
Rees, J; Shuster, S1
Lax, ER; Schriefers, H1
Panse, GT1
Baumann, P; Lax, ER; Schriefers, H1
Peluso, JJ; Steger, RW; Stude, D1
King, RJ; Yates, J1
Pandha, H; Waxman, J1
Hagen, R; Hoppe, F; Romalo, G; Schwab, B; Schweikert, HU1
Antoniou, G; Giannikos, L; Grigoriou, O; Karakitsos, P; Konidaris, S; Papadias, C1
Cutler, GB; Merke, DP1
Denis, L; Mahler, C; Verhelst, J1
De Markowsky, EE; Malgor, LA; Valsecia, M; Vergés, E1
Hirai, S; Matsubara, S1
Bisht, D; Chakraborti, PK; Rana, S1
Durmuşoğlu, F; Erenus, M; Gürbüz, O; Yücelten, D1
Benten, WP; Guo, Z; Lieberherr, M; Stamm, O; Wrehlke, C; Wunderlich, F1
Collette, L; de Reijke, TM; Schröder, FH; Whelan, P1
Man, RY; Quan, A; Teoh, H1
Leung, SW; Man, RY; Quan, A; Teoh, H1
Drapier-Faure, E; Faure, M1
Corradi, LS; Góes, RM; Leite Vilamaior, PS; Oliveira, SM; Taboga, SR1
Aguilera Tubet, C; Ballestero Diego, R; Roca Edreira, A; Villanueva Peña, A; Zubillaga Guerrero, S1
Delvoye, N; Gannon, PO; Lapointe, R; Mes-Masson, AM; Poisson, AO; Saad, F1
Alves, A; Gouveia, TIA; Mota, IH; Santos, MSF; Silva, AMT1

Reviews

19 review(s) available for flutamide and cyproterone

ArticleYear
Antiandrogens.
    Advances in sex hormone research, 1976, Volume: 2

    Topics: Acne Vulgaris; Androgen Antagonists; Animals; Biological Assay; Comb and Wattles; Cyproterone; Female; Fertility; Flutamide; Genitalia, Male; Hirsutism; Male; Phthalimides; Progesterone; Prostatic Hyperplasia; Prostatic Neoplasms; Sebaceous Glands; Sebum; Sex Differentiation; Sexual Behavior, Animal; Sexual Dysfunction, Physiological; Steroids

1976
Androgen receptors and the molecular basis for the action of antiadrogens in the ventral prostate.
    Journal of reproduction and fertility. Supplement, 1976, Issue:24 suppl

    Topics: Androgen Antagonists; Animals; Carrier Proteins; Contraceptive Agents, Male; Cyproterone; Cytosol; Dihydrotestosterone; Flutamide; Genes; Male; Molecular Conformation; Prostate; Protein Binding; Rats; Receptors, Androgen; Receptors, Steroid; RNA; Transcription, Genetic

1976
Chemotherapy of prostatic cancer.
    The Urologic clinics of North America, 1975, Volume: 2, Issue:1

    Topics: Aged; Alkylating Agents; Antibiotics, Antineoplastic; Antimetabolites; Antineoplastic Agents; Bromocriptine; Cyproterone; Depression, Chemical; Diethylstilbestrol; Drug Therapy, Combination; Estramustine; Fluorouracil; Flutamide; Health Facilities; Hematologic Diseases; Humans; Kinetics; Male; Mitosis; Nitrogen Mustard Compounds; Prostatic Neoplasms

1975
Cancer of the prostate. Mechanisms of action of antiandrogens.
    Acta urologica Belgica, 1991, Volume: 59, Issue:4

    Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Gonadotropin-Releasing Hormone; Humans; Luteinizing Hormone; Male; Prostatic Neoplasms; Rats; Testosterone

1991
Antiandrogenic substances in the management of prostatic cancer.
    Recent results in cancer research. Fortschritte der Krebsforschung. Progres dans les recherches sur le cancer, 1990, Volume: 118

    Topics: Androgen Antagonists; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Prostatic Neoplasms

1990
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
    Progress in clinical and biological research, 1990, Volume: 359

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds

1990
Clinical applications of antiandrogens.
    Journal of steroid biochemistry, 1988, Volume: 31, Issue:4B

    Topics: Androgen Antagonists; Breast Neoplasms; Cyproterone; Cyproterone Acetate; Female; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Hyperplasia; Prostatic Neoplasms; Puberty, Precocious; Skin Diseases; Spironolactone

1988
Initiation of LHRH monotherapy for prostate cancer.
    Progress in clinical and biological research, 1989, Volume: 303

    Topics: Androgen Antagonists; Antineoplastic Agents; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Flutamide; Gonadotropin-Releasing Hormone; Humans; Male; Prostatic Neoplasms

1989
[Antiandrogens. Mechanisms and paradoxical effects].
    Annales d'endocrinologie, 1989, Volume: 50, Issue:3

    Topics: 5-alpha Reductase Inhibitors; Androgen Antagonists; Androgens; Anilides; Cimetidine; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Nitriles; Spironolactone; Tosyl Compounds

1989
Androgen blockade and suppression for prostate carcinoma.
    Lancet (London, England), 1989, Oct-28, Volume: 2, Issue:8670

    Topics: Androgen Antagonists; Cyproterone; Drug Administration Schedule; Drug Therapy, Combination; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms

1989
Flutamide and other antiandrogens in the treatment of advanced prostatic carcinoma.
    Cancer treatment and research, 1988, Volume: 39

    Topics: Androgen Antagonists; Androgens; Anilides; Antineoplastic Agents; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Megestrol; Megestrol Acetate; Prostatic Neoplasms

1988
Treatment of advanced prostatic cancer.
    The Urologic clinics of North America, 1987, Volume: 14, Issue:2

    Topics: Adrenalectomy; Aminoglutethimide; Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Clinical Trials as Topic; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Estrogens; Flutamide; Glucocorticoids; Humans; Ketoconazole; Male; Megestrol; Megestrol Acetate; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms; Spironolactone; Time Factors

1987
Advantages and disadvantages of pure antiandrogens and of antiandrogens of the cyproterone acetate-type in the treatment of prostatic cancer.
    Progress in clinical and biological research, 1988, Volume: 260

    Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Female; Flutamide; Glucuronidase; Gonadotropin-Releasing Hormone; Guinea Pigs; Kidney; Male; Mice; Prostatic Neoplasms; Rats; Sex Differentiation; Time Factors

1988
[LHRH agonists combined with antiandrogens in the treatment of metastasizing prostatic carcinoma].
    Schweizerische Rundschau fur Medizin Praxis = Revue suisse de medecine Praxis, 1985, Nov-26, Volume: 74, Issue:48

    Topics: Androgen Antagonists; Animals; Buserelin; Cyproterone; Cyproterone Acetate; Dogs; Drug Therapy, Combination; Flutamide; Humans; Male; Neoplasm Metastasis; Orchiectomy; Prostatic Neoplasms; Rats; Receptors, Cell Surface; Receptors, LHRH

1985
New forms and future perspectives in endocrine treatment of prostatic carcinoma.
    Progress in clinical and biological research, 1984, Volume: 153

    Topics: Aminoglutethimide; Androgen Antagonists; Cyproterone; Cyproterone Acetate; Estrogen Antagonists; Flutamide; Hormones; Humans; Male; Pituitary Hormone-Releasing Hormones; Prolactin; Prostatic Neoplasms

1984
Clinical pharmacokinetics of the antiandrogens and their efficacy in prostate cancer.
    Clinical pharmacokinetics, 1998, Volume: 34, Issue:5

    Topics: Androgen Antagonists; Anilides; Antineoplastic Agents, Hormonal; Clinical Trials as Topic; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Tosyl Compounds

1998
Maximum androgen blockade in advanced prostate cancer: an overview of the randomised trials. Prostate Cancer Trialists' Collaborative Group.
    Lancet (London, England), 2000, Apr-29, Volume: 355, Issue:9214

    Topics: Aged; Androgen Antagonists; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Orchiectomy; Prostatic Neoplasms; Randomized Controlled Trials as Topic; Survival Analysis

2000
[What is the role of hormonal treatments in acne?].
    Annales de dermatologie et de venereologie, 2001, Volume: 128 Supp 1

    Topics: Acne Vulgaris; Androgen Antagonists; Cyproterone; Estrogens; Flutamide; Glucocorticoids; Hormone Antagonists; Humans; Mineralocorticoid Receptor Antagonists; Nandrolone; Patient Selection; Progestins; Spironolactone; Treatment Outcome

2001
First-line treatment of metastatic prostate cancer. Androgen suppression for symptomatic disease.
    Prescrire international, 2013, Volume: 22, Issue:135

    Topics: Androgen Antagonists; Antineoplastic Agents, Hormonal; Bone Neoplasms; Cyproterone; Estrogens; Flutamide; Goserelin; Humans; Male; Neoplasms, Hormone-Dependent; Orchiectomy; Practice Guidelines as Topic; Prostatic Neoplasms; Time Factors; Treatment Outcome

2013

Trials

13 trial(s) available for flutamide and cyproterone

ArticleYear
Advanced prostatic cancer: clinical and hormonal response to flutamide in patients pretreated with LHRH analogue and cyproterone acetate.
    European urology, 1990, Volume: 18, Issue:1

    Topics: Aged; Androgen Antagonists; Anilides; Buserelin; Clinical Trials as Topic; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Goserelin; Humans; Male; Middle Aged; Prostatic Neoplasms; Random Allocation

1990
Antiandrogens: clinical applications.
    The Journal of steroid biochemistry and molecular biology, 1990, Nov-20, Volume: 37, Issue:3

    Topics: Acne Vulgaris; Adult; Androgen Antagonists; Cyproterone; Cyproterone Acetate; Dermatitis, Seborrheic; Female; Flutamide; Hirsutism; Humans; Male; Prostatic Neoplasms; Spironolactone

1990
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
    Progress in clinical and biological research, 1990, Volume: 359

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds

1990
Effects of two different medical treatments on dihydrotestosterone content and androgen receptors in human benign prostatic hyperplasia.
    Journal of steroid biochemistry, 1988, Volume: 30, Issue:1-6

    Topics: Androgen Antagonists; Anilides; Cell Nucleus; Cyproterone; Cyproterone Acetate; Cytosol; Dihydrotestosterone; Flutamide; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Androgen; Tamoxifen

1988
Short-term anti-androgen therapy and very long-acting depot gonadotrophin-releasing hormone agonist for prostatic cancer.
    Progress in clinical and biological research, 1989, Volume: 303

    Topics: Aged; Aged, 80 and over; Androgen Antagonists; Buserelin; Clinical Trials as Topic; Cyproterone; Cyproterone Acetate; Delayed-Action Preparations; Flutamide; Humans; Male; Middle Aged; Prostatic Neoplasms; Random Allocation

1989
The clinical and endocrine assessment of three different antiandrogen regimens combined with a very long-acting gonadotrophin-releasing hormone analogue.
    American journal of clinical oncology, 1988, Volume: 11 Suppl 2

    Topics: Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Buserelin; Cyproterone; Cyproterone Acetate; Delayed-Action Preparations; Flutamide; Humans; Male; Middle Aged; Neoplasm Metastasis; Neoplasms, Hormone-Dependent; Phosphoric Monoester Hydrolases; Prostatic Neoplasms; Random Allocation; Testosterone

1988
Treatment of advanced prostatic cancer.
    The Urologic clinics of North America, 1987, Volume: 14, Issue:2

    Topics: Adrenalectomy; Aminoglutethimide; Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Clinical Trials as Topic; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Estrogens; Flutamide; Glucocorticoids; Humans; Ketoconazole; Male; Megestrol; Megestrol Acetate; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms; Spironolactone; Time Factors

1987
The effect of short term treatment with cyproterone acetate or flutamide on the metabolism of 5 alpha-dihydrotestosterone in human testicular tissue.
    Journal of steroid biochemistry, 1988, Volume: 31, Issue:2

    Topics: Aged; Aged, 80 and over; Anilides; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Male; Middle Aged; Testis

1988
Total androgen blockade in advanced prostatic cancer. Critical review and personal experience.
    European urology, 1988, Volume: 15, Issue:3-4

    Topics: Androgen Antagonists; Buserelin; Cyproterone; Cyproterone Acetate; Flutamide; Goserelin; Humans; Male; Multicenter Studies as Topic; Orchiectomy; Prostatic Neoplasms; Time Factors

1988
Effect of flutamide or cyproterone acetate on pituitary and testicular hormones in normal men.
    The Journal of clinical endocrinology and metabolism, 1984, Volume: 59, Issue:5

    Topics: Adult; Anilides; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Estradiol; Flutamide; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; Humans; Luteinizing Hormone; Male; Pituitary Function Tests; Pituitary Hormones; Prolactin; Testicular Hormones; Testosterone

1984
Comparison of flutamide and cyproterone acetate in the treatment of hirsutism: a randomized controlled trial.
    Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology, 1996, Volume: 10, Issue:2

    Topics: Adolescent; Adult; Androgen Antagonists; Cyproterone; Female; Flutamide; Hirsutism; Hormones; Humans; Prospective Studies

1996
Recurrence rate of hirsutism after 3 different antiandrogen therapies.
    Journal of the American Academy of Dermatology, 1999, Volume: 41, Issue:1

    Topics: Androgen Antagonists; Contraceptives, Oral; Cyproterone; Female; Flutamide; Hirsutism; Humans; Luteinizing Hormone; Recurrence; Spironolactone; Testosterone

1999
Prostate cancer treated by anti-androgens: is sexual function preserved? EORTC Genitourinary Group. European Organization for Research and Treatment of Cancer.
    British journal of cancer, 2000, Volume: 82, Issue:2

    Topics: Aged; Androgen Antagonists; Cyproterone; Erectile Dysfunction; Flutamide; Humans; Male; Middle Aged; Prospective Studies; Prostatic Neoplasms; Quality of Life; Sexuality

2000

Other Studies

79 other study(ies) available for flutamide and cyproterone

ArticleYear
Antiandrogenic steroidal sulfonylpyrazoles.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:8

    Topics: Androgen Antagonists; Animals; Male; Molecular Structure; Orchiectomy; Organ Size; Pregnanes; Prostate; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Androgen; Structure-Activity Relationship; Testosterone; X-Ray Diffraction

1990
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
    Chemical research in toxicology, 2012, Oct-15, Volume: 25, Issue:10

    Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding

2012
The effect of antiandrogens and stilboestrol on the cytosol receptor in rat prostate.
    British journal of urology, 1977, Volume: 49, Issue:7

    Topics: Androgen Antagonists; Animals; Chlormadinone Acetate; Cyproterone; Cytosol; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Male; Nandrolone; Prostate; Rats; Receptors, Androgen; Receptors, Steroid

1977
Androgen receptors in benign and malignant prostatic tissue.
    Transactions of the American Association of Genito-Urinary Surgeons, 1979, Volume: 71

    Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Androgen Antagonists; Animals; Cyproterone; Dihydrotestosterone; Estrenes; Flutamide; Humans; Male; Prostatic Hyperplasia; Prostatic Neoplasms; Rats; Receptors, Androgen; Receptors, Steroid

1979
Effect of antiandrogens on the binding of androgen to cytosol and nuclei of hamster sebaceous glands.
    Archives of dermatological research, 1979, Feb-23, Volume: 264, Issue:1

    Topics: Androgen Antagonists; Androstanes; Androstanols; Animals; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Dihydrotestosterone; Estrenes; Flutamide; In Vitro Techniques; Male; Prostate; Receptors, Androgen; Receptors, Steroid; Sebaceous Glands; Seminal Vesicles; Steroids, Heterocyclic; Testosterone

1979
Evidence for a role of androgens in the growth and maturation of ovarian follicles in rats.
    Hormone research, 1978, Volume: 9, Issue:2

    Topics: Androgens; Animals; Corpus Luteum; Cyproterone; Diestrus; Estradiol; Estrus; Female; Flutamide; Ovarian Follicle; Ovary; Pregnancy; Rats

1978
Testicular phosphatase activity in rats treated with cyproterone acetate & flutamide.
    Indian journal of experimental biology, 1977, Volume: 15, Issue:9

    Topics: Acid Phosphatase; Alkaline Phosphatase; Anilides; Animals; Cyproterone; Flutamide; Male; Rats; Testis

1977
Androgen binding to cytosol and nuclei of hamster sebaceous glands.
    Journal of steroid biochemistry, 1978, Volume: 9, Issue:2

    Topics: Androgens; Animals; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Dihydrotestosterone; Estradiol; Flutamide; Male; Progesterone; Receptors, Androgen; Sebaceous Glands

1978
Androgenic stimulation of progesterone production by granulosa cells from preantral ovarian follicles: further in vitro studies using replicate cell cultures.
    Endocrinology, 1977, Volume: 100, Issue:6

    Topics: Animals; Cells, Cultured; Cyproterone; Diethylstilbestrol; Female; Flutamide; Granulosa Cells; Ovarian Follicle; Ovary; Progesterone; Rats; Testosterone

1977
Specific androgen binding in the kidney and estrogen-dependent renal carcinoma of the Syrian hamster.
    Endocrinology, 1977, Volume: 101, Issue:4

    Topics: Androgens; Animals; Castration; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Diethylstilbestrol; Dihydrotestosterone; Estrogens; Flutamide; Kidney; Kidney Neoplasms; Liver; Male; Progesterone; Receptors, Androgen; Receptors, Steroid

1977
Androgen receptor dependent and independent activities of testosterone on hepatic microsomal drug metabolism.
    Endocrinology, 1976, Volume: 99, Issue:5

    Topics: Animals; Castration; Cyproterone; Cytochrome P-450 Enzyme System; Ethylmorphine-N-Demethylase; Female; Flutamide; Liver; Male; Mice; Mice, Inbred BALB C; Microsomes, Liver; Organ Size; Quinone Reductases; Rats; Receptors, Androgen; Receptors, Steroid; Testosterone

1976
Induction of delta-aminolevulinic acid synthetase by flutamide, a non-steroidal antiandrogen.
    Biochimica et biophysica acta, 1976, Nov-18, Volume: 451, Issue:1

    Topics: 5-Aminolevulinate Synthetase; Aminoisobutyric Acids; Anilides; Animals; Anti-Bacterial Agents; Cells, Cultured; Chick Embryo; Cyproterone; Enzyme Induction; Flutamide; Mitochondria, Liver

1976
Differences among rat sex accessory glands in their neonatal androgen dependency.
    Endocrinology, 1975, Volume: 97, Issue:1

    Topics: Age Factors; Androstanes; Animals; Animals, Newborn; Castration; Cyproterone; DNA; Flutamide; Ketosteroids; Male; Prostate; Protein Biosynthesis; Rats; RNA; Seminal Vesicles; Steroids, Heterocyclic; Testis; Testosterone; Thymidine; Tritium

1975
Evidence of a role of adrogens in follicular maturation.
    Endocrinology, 1975, Volume: 97, Issue:2

    Topics: Androgens; Androstenedione; Animals; Chorionic Gonadotropin; Cyproterone; Diethylstilbestrol; Dihydrotestosterone; Estradiol; Female; Flutamide; Humans; Hydrocortisone; Hydroxyprogesterones; Hypophysectomy; Organ Size; Ovarian Follicle; Ovary; Pituitary Gland; Progesterone; Rats; Testosterone

1975
Biological aspects of antiandrogens.
    Journal of steroid biochemistry, 1975, Volume: 6, Issue:6

    Topics: Androgen Antagonists; Anilides; Animals; Castration; Cyproterone; DNA; Dose-Response Relationship, Drug; Flutamide; Male; Organ Size; Organ Specificity; Prostate; Rats; Seminal Vesicles; Testis; Testosterone

1975
Flutamide. Mechanism of action of a new nonsteroidal antiandrogen.
    Investigative urology, 1976, Volume: 13, Issue:6

    Topics: Anilides; Animals; Castration; Chemical Phenomena; Chemistry; Cyproterone; DNA; Flutamide; Genitalia, Male; Male; Prostate; Rats; Seminal Vesicles; Testosterone

1976
Regulation of androgen receptor mRNA and protein level by steroid hormones in human mammary cancer cells.
    The Journal of steroid biochemistry and molecular biology, 1992, Volume: 43, Issue:7

    Topics: Blotting, Northern; Breast Neoplasms; Cyproterone; Dihydrotestosterone; Estradiol; Flutamide; Gene Expression Regulation, Neoplastic; Hormones; Humans; Immunohistochemistry; Progesterone Congeners; Radioligand Assay; Receptors, Androgen; RNA, Messenger; Steroids; Tumor Cells, Cultured

1992
Neo-adjuvant hormonotherapy does not facilitate radical prostatectomy.
    Acta urologica Belgica, 1992, Volume: 60, Issue:3

    Topics: Aged; Antineoplastic Combined Chemotherapy Protocols; Blood Loss, Surgical; Chemotherapy, Adjuvant; Cyproterone; Estramustine; Flutamide; Humans; Male; Middle Aged; Prostatectomy; Prostatic Neoplasms

1992
[A 79-year-old man with metastatic prostate cancer, treated with Zoladex, flutamide, calcitonin and Ostac, suffers from frequent troublesome sweating with palpitation and angina pectoris, especially at night. Is there a therapy?].
    Der Internist, 1992, Volume: 33, Issue:4

    Topics: Aged; Androgen Antagonists; Angina Pectoris; Buserelin; Calcitonin; Cyproterone; Cyproterone Acetate; Flutamide; Goserelin; Humans; Hyperhidrosis; Male; Prostatic Neoplasms

1992
[A study of the androgenic activity of anti-androgen].
    Nihon Naibunpi Gakkai zasshi, 1990, Jun-20, Volume: 66, Issue:6

    Topics: Androgen Antagonists; Aniline Compounds; Animals; Arginase; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Estradiol; Flutamide; Male; Medroxyprogesterone; Organ Size; Ornithine Decarboxylase; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen; Seminal Vesicles

1990
Investigation on serum neurone-specific enolase in prostate cancer diagnosis and monitoring: comparative study of a multiple tumor marker assay.
    The Prostate, 1991, Volume: 19, Issue:1

    Topics: Acid Phosphatase; Antigens, Neoplasm; Antineoplastic Agents; APUD Cells; Biomarkers, Tumor; Carcinoembryonic Antigen; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Estramustine; Flutamide; Humans; Male; Orchiectomy; Phosphopyruvate Hydratase; Prostate-Specific Antigen; Prostatic Neoplasms

1991
Effects of steroidal and non-steroidal antiandrogens on the left atrium of the rat in vitro.
    General pharmacology, 1991, Volume: 22, Issue:6

    Topics: Androgen Antagonists; Animals; Calcium; Chlormadinone Acetate; Cimetidine; Cyproterone; Electric Stimulation; Female; Flutamide; Heart; Heart Atria; In Vitro Techniques; Male; Medroxyprogesterone; Myocardial Contraction; Rats; Rats, Inbred Strains; Spironolactone; Steroids; Stimulation, Chemical

1991
Influence of different types of antiandrogens on luteinizing hormone-releasing hormone analogue-induced testosterone surge in patients with metastatic carcinoma of the prostate.
    The Journal of urology, 1990, Volume: 144, Issue:4

    Topics: Acid Phosphatase; Aged; Androgen Antagonists; Buserelin; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Goserelin; Humans; Luteinizing Hormone; Male; Premedication; Prostatic Neoplasms; Testosterone; Time Factors

1990
The synthetic androgen mibolerone induces transient suppression of the transformed phenotype in an androgen responsive human prostatic carcinoma cell line.
    Andrologia, 1990, Volume: 22 Suppl 1

    Topics: Androgen Antagonists; Androgens; Cell Division; Cell Transformation, Neoplastic; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Male; Nandrolone; Prostatic Neoplasms; Receptors, Androgen; RNA, Messenger; Tumor Cells, Cultured

1990
Analysis of the androgenic activity of synthetic "progestins" currently used for the treatment of prostate cancer.
    Journal of steroid biochemistry, 1987, Volume: 28, Issue:4

    Topics: Adrenal Glands; Animals; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Male; Medroxyprogesterone; Medroxyprogesterone Acetate; Megestrol; Megestrol Acetate; Organ Size; Ornithine Decarboxylase; Progesterone Congeners; Prostate; Prostatic Neoplasms; Rats; Rats, Inbred Strains; Spironolactone

1987
Stimulatory effect of synthetic progestins currently used for the treatment of prostate cancer on growth of the androgen-sensitive Shionogi tumor in mice.
    Journal of steroid biochemistry, 1988, Volume: 31, Issue:1

    Topics: Androgens; Animals; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Female; Flutamide; Male; Mammary Neoplasms, Experimental; Medroxyprogesterone; Medroxyprogesterone Acetate; Megestrol; Megestrol Acetate; Mice; Progesterone Congeners; Prostatic Neoplasms

1988
Treatment with antiandrogens induces an androgen-repressed gene in the rat ventral prostate.
    The Prostate, 1988, Volume: 13, Issue:2

    Topics: Androgen Antagonists; Androgens; Animals; Blotting, Northern; Body Weight; Cell Survival; Cell-Free System; Cyproterone; Cyproterone Acetate; Flutamide; Gene Expression Regulation; Male; Orchiectomy; Organ Size; Prostate; Protein Biosynthesis; Rats; Rats, Inbred Strains; RNA

1988
Androgens directly stimulate proliferation of bone cells in vitro.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Alkaline Phosphatase; Androgens; Animals; Binding, Competitive; Cell Count; Cell Differentiation; Cell Division; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; DNA; Dose-Response Relationship, Drug; Fluoxymesterone; Flutamide; Humans; Methenolone; Mice; Osteoblasts; Testosterone; Tumor Cells, Cultured

1989
Antiandrogens do not reverse androgen-induced inhibition of sex hormone-binding globulin levels in adult female rhesus monkeys.
    Endocrinology, 1989, Volume: 125, Issue:2

    Topics: Androgen Antagonists; Androgens; Animals; Biomarkers; Cyproterone; Cyproterone Acetate; Female; Flutamide; Macaca; Macaca mulatta; Methyltestosterone; Ovariectomy; Pregnanes; Pyrazoles; Sex Hormone-Binding Globulin

1989
Sexual dimorphism of blood pressure in spontaneously hypertensive rats: effects of anti-androgen treatment.
    Journal of hypertension, 1989, Volume: 7, Issue:9

    Topics: Androgen Antagonists; Anilides; Animals; Animals, Newborn; Blood Pressure; Cyproterone; Cyproterone Acetate; Female; Flutamide; Male; Orchiectomy; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Sex Characteristics; Species Specificity; Testosterone

1989
Effect of antiandrogens on some key enzymes of glycolysis in epididymis and ventral prostate of rat.
    Indian journal of experimental biology, 1989, Volume: 27, Issue:4

    Topics: Androgen Antagonists; Animals; Body Weight; Cyproterone; Cyproterone Acetate; Enzymes; Epididymis; Estradiol; Flutamide; Glycolysis; Male; Nandrolone; Organ Size; Prostate; Rats

1989
"Casodex" (ICI 176,334)--a new, pure, peripherally-selective anti-androgen: preclinical studies.
    Hormone research, 1989, Volume: 32 Suppl 1

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Rats; Tosyl Compounds

1989
[Antiandrogens in monotherapy or combined therapy for treatment of advanced cancer of the prostate].
    Archivos espanoles de urologia, 1989, Volume: 42 Suppl 2

    Topics: Aged; Aged, 80 and over; Androgen Antagonists; Anilides; Antineoplastic Agents; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Flutamide; Follow-Up Studies; Humans; Imidazoles; Imidazolidines; Male; Middle Aged; Neoplasm Staging; Nitriles; Orchiectomy; Prostatic Neoplasms; Tosyl Compounds

1989
Imaging the hamster flank organ by an ultrasonic technique: a new approach to animal tests.
    The British journal of dermatology, 1989, Volume: 121, Issue:6

    Topics: Animals; Cricetinae; Cyproterone; Female; Flutamide; Male; Mesocricetus; Orchiectomy; Sebaceous Glands; Skin; Spironolactone; Testosterone; Ultrasonography

1989
Onset of steroidogenesis and differentiation of functional LH receptors in rat fetal testicular cultures.
    Archives of andrology, 1987, Volume: 18, Issue:3

    Topics: Aminoglutethimide; Animals; Binding, Competitive; Bucladesine; Cyproterone; Cyproterone Acetate; Dehydroepiandrosterone; Flutamide; Gestational Age; Luteinizing Hormone; Male; Organ Culture Techniques; Progesterone; Rats; Rats, Inbred Strains; Receptors, LH; Testis; Testosterone

1987
Testosterone suppression of ornithine decarboxylase activity in rat Sertoli cells.
    Endocrinology, 1988, Volume: 123, Issue:2

    Topics: Animals; Bucladesine; Cells, Cultured; Cyclic AMP; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Enzyme Induction; Estradiol; Flutamide; Follicle Stimulating Hormone; Male; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Sertoli Cells; Testosterone

1988
Combined treatment with flutamide and surgical or medical (LHRH agonist) castration in metastatic prostatic cancer.
    Lancet (London, England), 1986, Jan-04, Volume: 1, Issue:8471

    Topics: Anilides; Combined Modality Therapy; Cyproterone; Flutamide; Gonadotropin-Releasing Hormone; Humans; Male; Megestrol; Neoplasm Metastasis; Orchiectomy; Prostatic Neoplasms; Receptors, Cell Surface; Receptors, LHRH

1986
Effect of antiandrogens on the hypothalamic gamma-aminobutyric acid (GABA) and glutamate contents of the Indian palm squirrel (Funambulus pennanti, Wroughton).
    Experimental and clinical endocrinology, 1986, Volume: 87, Issue:3

    Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Female; Flutamide; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hypothalamus; Organ Size; Sciuridae

1986
Treatment of prostatic cancer. Newer forms of androgen deprivation.
    Postgraduate medicine, 1986, Volume: 80, Issue:1

    Topics: Androgen Antagonists; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Megestrol; Megestrol Acetate; Neoplasm Metastasis; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms

1986
Effects of cyproterone acetate and flutamide on the testis and epididymis of the Indian wall lizard, Hemidactylus flaviviridis (Ruppell).
    General and comparative endocrinology, 1986, Volume: 64, Issue:3

    Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Epididymis; Epithelial Cells; Flutamide; Leydig Cells; Lizards; Male; Organ Size; Spermatogenesis; Spermatozoa; Testis

1986
Inhibition of testosterone metabolism in the brain and cloacal gland of the quail by specific inhibitors and antihormones.
    The Journal of endocrinology, 1987, Volume: 112, Issue:2

    Topics: Androgen Antagonists; Androstanes; Androstatrienes; Animals; Azasteroids; Cloaca; Coturnix; Cyproterone; Cyproterone Acetate; Estrogen Antagonists; Flutamide; Hypothalamus; Male; Nitromifene; Quail; Tamoxifen; Testosterone

1987
Acid phosphatase activity: a marker of androgen action in prostate explant cultures.
    The Prostate, 1987, Volume: 10, Issue:1

    Topics: Acid Phosphatase; Animals; Cells, Cultured; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Estradiol; Flutamide; Hydrocortisone; Male; Prostate; Rats; Rats, Inbred Strains

1987
Effects of metabolism inhibitors, antiestrogens and antiandrogens on the androgen and estrogen induced sexual behavior in Japanese quail.
    Physiology & behavior, 1986, Volume: 38, Issue:4

    Topics: Androgens; Androstatrienes; Animals; Coturnix; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Estrogens; Flutamide; Male; Orchiectomy; Quail; Sexual Behavior, Animal; Tamoxifen; Testosterone

1986
[Effects of cyproterone acetate and flutamide on blood calcium and bone structure].
    Archivos espanoles de urologia, 1986, Volume: 39, Issue:8

    Topics: Androgen Antagonists; Anilides; Animals; Bone and Bones; Calcium; Cyproterone; Cyproterone Acetate; Flutamide; Male; Rats; Rats, Inbred Strains

1986
Inhibition of rat testicular 17 alpha-hydroxylase and 17,20-lyase activities by anti-androgens (flutamide, hydroxyflutamide, RU23908, cyproterone acetate) in vitro.
    Journal of steroid biochemistry, 1987, Volume: 28, Issue:1

    Topics: Aldehyde-Lyases; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Cytochrome P-450 Enzyme System; Flutamide; Imidazoles; Imidazolidines; Kinetics; Male; Microsomes; Rats; Rats, Inbred Strains; Steroid 17-alpha-Hydroxylase; Steroid Hydroxylases; Testis

1987
The kinetics of antiandrogens in humans.
    Progress in clinical and biological research, 1987, Volume: 243A

    Topics: Androgen Antagonists; Anilides; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Neoplasms

1987
Effect of cyproterone acetate in comparison to flutamide and megestrol acetate on the ventral prostate, seminal vesicle, and adrenal glands of adult male rats.
    The Prostate, 1987, Volume: 11, Issue:4

    Topics: Adrenal Glands; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Organ Size; Prostate; Rats; Rats, Inbred Strains; Seminal Vesicles

1987
ICI 176,334: a novel non-steroidal, peripherally-selective antiandrogen.
    Progress in clinical and biological research, 1988, Volume: 260

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostate; Radioligand Assay; Rats; Receptors, Androgen; Seminal Vesicles; Testosterone; Tosyl Compounds

1988
Relative effectiveness of alternative androgen withdrawal therapies in initiating regression of rat prostate.
    The Journal of urology, 1988, Volume: 139, Issue:6

    Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Gonadotropin-Releasing Hormone; Imidazoles; Imidazolidines; Leuprolide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen

1988
Microsomal effects of cyproterone acetate and flutamide in rat testis.
    General pharmacology, 1988, Volume: 19, Issue:3

    Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Cytochrome b Group; Cytochrome P-450 Enzyme System; Cytochromes b5; Flutamide; In Vitro Techniques; Luteinizing Hormone; Male; Microsomes; NADPH-Ferrihemoprotein Reductase; Rats; Rats, Inbred Strains; Testis; Testosterone

1988
Effects of the antiandrogens cyproterone acetate and flutamide on male reproductive behavior in a lizard (Anolis sagrei).
    Hormones and behavior, 1987, Volume: 21, Issue:1

    Topics: Aggression; Anilides; Animals; Cyproterone; Dihydrotestosterone; Female; Flutamide; Lizards; Male; Organ Size; Sexual Behavior, Animal; Social Dominance; Testis; Testosterone

1987
[Cancer of the prostate: new hormone therapies].
    Bulletin du cancer, 1986, Volume: 73, Issue:1

    Topics: Androgen Antagonists; Cyproterone; Flutamide; Humans; Ketoconazole; Male; Medroxyprogesterone; Megestrol; Neoplasms, Hormone-Dependent; Progestins; Prostatic Neoplasms; Tamoxifen

1986
Principles of endocrine manipulation in the treatment of prostatic cancer.
    Progress in clinical and biological research, 1985, Volume: 185A

    Topics: Androgen Antagonists; Animals; Castration; Cyproterone; Estrogens; Flutamide; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Male; Neoplasms, Hormone-Dependent; Progestins; Prostatic Neoplasms; Rats; Testosterone

1985
Comparison of the antiandrogenic/androgenic activities of flutamide, cyproterone acetate and megestrol acetate.
    Molecular and cellular endocrinology, 1985, Volume: 42, Issue:3

    Topics: Adrenal Glands; Anilides; Animals; Cyproterone; Dihydrotestosterone; Flutamide; Follicle Stimulating Hormone; Luteinizing Hormone; Male; Megestrol; Orchiectomy; Organ Size; Prostate; Rats; Rats, Inbred Strains

1985
An androgen-independent mechanism maintains photorefractoriness in male tree sparrows (Spizella arborea).
    The Journal of endocrinology, 1985, Volume: 107, Issue:1

    Topics: Animals; Birds; Castration; Cyproterone; Flutamide; Light; Luteinizing Hormone; Male; Radioimmunoassay; Testosterone

1985
Effect of anti-androgens on the morphological & biochemical changes induced by testosterone in rat uterus.
    Indian journal of experimental biology, 1980, Volume: 18, Issue:5

    Topics: Anilides; Animals; Cyproterone; Female; Flutamide; Glycogen; Proteins; Rats; RNA; Sialic Acids; Testosterone; Uterus

1980
Stimulation of ribonucleic acid polymerase activity in mouse kidney.
    Endocrinology, 1983, Volume: 112, Issue:2

    Topics: Animals; Cyproterone; Cyproterone Acetate; DNA-Directed RNA Polymerases; Female; Flutamide; Kidney; Medroxyprogesterone; Mice; Mice, Inbred C57BL; Progesterone; Receptors, Androgen; Receptors, Steroid; RNA Polymerase I; RNA Polymerase II; Testosterone

1983
Effects of antiandrogens (cyproterone acetate and flutamide) on the activity of nuclear protein phosphokinases and phosphatases of rat ventral prostate.
    Molecular pharmacology, 1980, Volume: 17, Issue:2

    Topics: Alkaline Phosphatase; Anilides; Animals; Castration; Cell Nucleus; Chromatin; Cyproterone; Flutamide; Male; Phosphoric Monoester Hydrolases; Prostate; Protein Kinases; Rats; Testosterone

1980
Effect of 17-hydroxy progesterone caproate, flutamide & cyproterone acetate on genital organs & fertility of male rats--a comparative study.
    Indian journal of experimental biology, 1980, Volume: 18, Issue:11

    Topics: 17 alpha-Hydroxyprogesterone Caproate; Anilides; Animals; Contraceptive Agents, Male; Cyproterone; Cyproterone Acetate; Fertility; Flutamide; Genitalia, Male; Hydroxyprogesterones; Male; Organ Specificity; Progesterone Congeners; Rats

1980
Pubertal induction of sweat gland activity.
    Clinical science (London, England : 1979), 1981, Volume: 60, Issue:6

    Topics: Acne Vulgaris; Adult; Child; Cyproterone; Cyproterone Acetate; Female; Flutamide; Humans; Male; Middle Aged; Puberty; Sex Factors; Sweat Glands; Sweating; Testosterone

1981
Sex-specific action of antiandrogens on androgen induced changes in hepatic microsomal 3 beta-hydroxysteroid dehydrogenase and 5 alpha-reductase activity in the rat.
    Acta endocrinologica, 1981, Volume: 98, Issue:2

    Topics: 3-Hydroxysteroid Dehydrogenases; 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Androgen Antagonists; Anilides; Animals; Castration; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Female; Flutamide; Male; Microsomes, Liver; Organ Size; Oxidoreductases; Rats; Sex Factors

1981
Effects of antiandrogens on glycogen metabolism of spermatozoa from caput epididymidis.
    Indian journal of experimental biology, 1981, Volume: 19, Issue:9

    Topics: Anilides; Animals; Contraceptive Agents, Male; Cyproterone; Cyproterone Acetate; Flutamide; Glycogen; Male; Mice; Spermatozoa

1981
Antiandrogenic effects of oestradiol on enzyme activities of hepatic steroid metabolism.
    Experimental and clinical endocrinology, 1983, Volume: 82, Issue:2

    Topics: 3-alpha-Hydroxysteroid Dehydrogenase (B-Specific); 3-Hydroxysteroid Dehydrogenases; 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Animals; Castration; Cyproterone; Dihydrotestosterone; Estradiol; Female; Flutamide; Male; Microsomes, Liver; Oxidoreductases; Rats; Rats, Inbred Strains

1983
Role of androgens in hCG-induced ovulation in PMSG-primed immature rats.
    Acta endocrinologica, 1980, Volume: 93, Issue:4

    Topics: 3-Hydroxysteroid Dehydrogenases; Androgens; Anilides; Animals; Chorionic Gonadotropin; Cyproterone; Estradiol; Female; Flutamide; Gonadotropins, Equine; Ovarian Follicle; Ovulation; Progesterone; Rats

1980
Antiandrogen effects on androgen-responsive mammary tumour cells in culture.
    Journal of steroid biochemistry, 1981, Volume: 14, Issue:9

    Topics: Anilides; Animals; Cell Division; Cells, Cultured; Cyproterone; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Mammary Neoplasms, Experimental; Mice; Receptors, Androgen; Testosterone

1981
Anti-androgens in treatment of prostate cancer.
    Lancet (London, England), 1995, Oct-14, Volume: 346, Issue:8981

    Topics: Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Meta-Analysis as Topic; Prostatic Neoplasms

1995
Juvenile nasopharyngeal fibroma: androgen receptors and their significance for tumor growth.
    The Laryngoscope, 1994, Volume: 104, Issue:9

    Topics: Cell Division; Child; Cholestenone 5 alpha-Reductase; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Fibroblasts; Fibroma; Flutamide; Humans; Male; Nasopharyngeal Neoplasms; Oxidoreductases; Receptors, Androgen; Scrotum; Skin; Testosterone; Tritium; Tumor Cells, Cultured

1994
New approaches to the treatment of congenital adrenal hyperplasia.
    JAMA, 1997, Apr-02, Volume: 277, Issue:13

    Topics: Adrenal Hyperplasia, Congenital; Age Determination by Skeleton; Androgen Antagonists; Child; Cyproterone; Drug Therapy, Combination; Female; Fludrocortisone; Flutamide; Growth; Humans; Hydrocortisone; Mineralocorticoid Receptor Antagonists; Spironolactone; Testolactone

1997
Blockade of the in vitro effects of testosterone and erythropoietin on Cfu-E and Bfu-E proliferation by pretreatment of the donor rats with cyproterone and flutamide.
    Acta physiologica, pharmacologica et therapeutica latinoamericana : organo de la Asociacion Latinoamericana de Ciencias Fisiologicas y [de] la Asociacion Latinoamericana de Farmacologia, 1998, Volume: 48, Issue:2

    Topics: Androgen Antagonists; Animals; Bone Marrow Cells; Cells, Cultured; Cyproterone; Erythroid Precursor Cells; Erythropoiesis; Erythropoietin; Flutamide; Male; Premedication; Rats; Testosterone

1998
Influence of anti-androgens on the anterior horn cells of rat spinal cord: morphometric and in-situ hybridization studies.
    Journal of the neurological sciences, 1998, Nov-26, Volume: 161, Issue:1

    Topics: Androgen Antagonists; Animals; Anterior Horn Cells; Cell Count; Cell Size; Choline O-Acetyltransferase; Cyproterone; Flutamide; In Situ Hybridization; Male; Rats; Rats, Wistar; RNA, Messenger

1998
Synergistic activation of yeast-expressed rat androgen receptor by modulators of protein kinase-A.
    Journal of molecular biology, 1999, Feb-26, Volume: 286, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 8-Bromo Cyclic Adenosine Monophosphate; Androgens; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyproterone; Dihydrotestosterone; Enzyme Inhibitors; Flutamide; Gene Expression Regulation; Genes, Reporter; Metribolone; Okadaic Acid; Rats; Receptors, Androgen; Regulatory Sequences, Nucleic Acid; RNA, Messenger; Saccharomyces cerevisiae; Signal Transduction; Transcriptional Activation; Transformation, Genetic

1999
Testosterone signaling through internalizable surface receptors in androgen receptor-free macrophages.
    Molecular biology of the cell, 1999, Volume: 10, Issue:10

    Topics: Androgen Antagonists; Animals; Calcium; Cell Line; Cyproterone; Endocytosis; Estradiol; Estrenes; Flow Cytometry; Flutamide; Macrophages; Mice; Mice, Knockout; Microscopy, Confocal; Pertussis Toxin; Pyrrolidinones; Receptors, Androgen; Receptors, Cell Surface; Serum Albumin, Bovine; Signal Transduction; Testosterone; Type C Phospholipases; Virulence Factors, Bordetella

1999
Acute impairment of relaxation by low levels of testosterone in porcine coronary arteries.
    Cardiovascular research, 2000, Volume: 45, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Analysis of Variance; Androgen Receptor Antagonists; Animals; Bradykinin; Calcimycin; Coronary Vessels; Cromakalim; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Flutamide; Ionophores; Male; Nitroprusside; Swine; Testosterone; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2000
Differential effects of 17beta-estradiol and testosterone on the contractile responses of porcine coronary arteries.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Androgen Antagonists; Androgen Receptor Antagonists; Animals; Coronary Vessels; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelin-1; Estradiol; Estrogen Antagonists; Female; Flutamide; Fulvestrant; In Vitro Techniques; Isotonic Solutions; Male; Potassium Chloride; Receptors, Estrogen; Serotonin; Swine; Tamoxifen; Testosterone; Vasoconstriction

2000
Cellular and extracellular behavior in the gerbil (Meriones unguiculatus) ventral prostate following different types of castration and the consequences of testosterone replacement.
    Cell biology international, 2007, Volume: 31, Issue:3

    Topics: Acid Phosphatase; Androgen Antagonists; Animals; Cyproterone; Disease Models, Animal; Endoplasmic Reticulum, Rough; Endothelium; Flutamide; Gerbillinae; Immunohistochemistry; Male; Microscopy, Electron, Transmission; Orchiectomy; Organ Size; Prostate; Prostatic Hyperplasia; Protein Tyrosine Phosphatases; Receptors, Androgen; Testosterone

2007
[Mediastinal lymph nodes during the course of a metastatic prostate cancer].
    Actas urologicas espanolas, 2007, Volume: 31, Issue:6

    Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Antineoplastic Combined Chemotherapy Protocols; Bone Neoplasms; Cyproterone; Diphosphonates; Estramustine; Fatal Outcome; Flutamide; Humans; Imidazoles; Ketoconazole; Lung Neoplasms; Lymphatic Metastasis; Male; Mediastinum; Neoplasms, Hormone-Dependent; Prostatic Neoplasms; Radionuclide Imaging; Skin Neoplasms; Triptorelin Pamoate; Zoledronic Acid

2007
Characterization of the intra-prostatic immune cell infiltration in androgen-deprived prostate cancer patients.
    Journal of immunological methods, 2009, Aug-31, Volume: 348, Issue:1-2

    Topics: Androgen Antagonists; Androgens; Antineoplastic Agents, Hormonal; Cyproterone; Flutamide; Humans; Killer Cells, Natural; Leuprolide; Lymphocytes, Tumor-Infiltrating; Macrophages; Male; Neoplasm Recurrence, Local; Prostatic Neoplasms; T-Lymphocytes

2009
Are cytostatic drugs in surface waters a potential threat?
    The Science of the total environment, 2022, Dec-20, Volume: 853

    Topics: Child; Chlorambucil; Cyclophosphamide; Cyproterone; Cytostatic Agents; Drinking Water; Environmental Monitoring; Etoposide; Flutamide; Humans; Mycophenolic Acid; Pharmaceutical Preparations; Rivers; Tamoxifen; Water Pollutants, Chemical

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