flutamide has been researched along with cyproterone in 109 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 73 (66.97) | 18.7374 |
1990's | 24 (22.02) | 18.2507 |
2000's | 9 (8.26) | 29.6817 |
2010's | 2 (1.83) | 24.3611 |
2020's | 1 (0.92) | 2.80 |
Authors | Studies |
---|---|
Ackerman, JH; Bell, MR; Christiansen, RG; D'Ambra, TE; Herrmann, JL; Kullnig, RK; Mallamo, JP; Opalka, CJ; Snyder, BW; Winneker, RC | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY | 1 |
Neri, RO | 1 |
Chisholm, GD; Ghanadian, R; Smith, CB; Williams, G | 1 |
Bruchovsky, N; Callaway, T; Comeau, T; Lakey, WH; Lieskovsky, G; Rennie, P; Shnitka, T; Wilkin, P | 1 |
Takayasu, S | 2 |
Datta, JK; Kumari, GL; Roy, S | 1 |
Munshi, SR; Nagendranath, N; Raman, G; Sheth, AR | 1 |
Liao, S; Tymoczko, JL | 1 |
Hillier, SG; Knazek, RA; Ross, GT | 1 |
Cuthbertson, TL; Li, JJ; Li, SA | 1 |
Bardin, CW; Brown, TR; Greene, FE | 1 |
Gidari, AS; Lane, SE; Levere, RD | 1 |
Schmidt, JD | 1 |
Chung, LW; Ferland-Raymond, G | 1 |
Harman, SM; Louvet, JP; Ross, GT; Schrieber, JR | 1 |
Neri, RO; Peets, EA | 1 |
Coffey, DS; Sufrin, G | 1 |
Beato, M; Bock, K; Filmer, A; Hackenberg, R; Hawighorst, T; Schulz, KD; Slater, EP | 1 |
Ameye, F; Baert, L; Oyen, R; Van De Voorde, W; Van Poppel, H | 1 |
Schmeller, N | 1 |
Imai, K; Kawashima, K; Nakata, S; Shimizu, N; Suzuki, T; Takahashi, O; Watanabe, K; Yamanaka, H | 1 |
Radoś, N; Tarle, M | 1 |
Cantabrana, B; Garcia Valencia, V; Gutierrez, M; Hidalgo, A; Sanchez, M | 1 |
el Etreby, MF; Habenicht, UF; Neumann, F | 1 |
Schulze, H; Senge, T | 1 |
D'Eramo, G; Di Silverio, F; Sciarra, F | 1 |
Schröder, FH | 2 |
Concolino, G; Di Silverio, F; Sciarra, F; Toscano, V | 1 |
Arbusow, V; Bojar, H; Fittler, F; Klobeck, HG; Schulz, P; Wolf, D | 1 |
Cusan, L; Labrie, C; Labrie, F; Lapointe, S; Plante, M | 1 |
Concolino, G; Conti, C; Di Silverio, F; Lubrano, C; Petrangeli, E; Sciarra, F; Toscano, V | 1 |
Labrie, F; Lapointe, S; Plante, M | 1 |
Le Guellec, R; Léger, JG; Tenniswood, MP | 1 |
Namer, M | 1 |
Baylink, DJ; Farley, JR; Kasperk, CH; Linkhart, TA; Turner, RT; Wergedal, JE | 1 |
Shaw, CJ; Snyder, BW; Wagner, MM; Winneker, RC | 1 |
Waxman, J | 1 |
Milsted, RA | 1 |
Ganten, D; Ganten, U; Schröder, G; Stock, G; Witt, M; Zimmermann, F | 1 |
Gupta, G; Setty, BS; Srivastava, A | 1 |
Mowszowicz, I | 1 |
Furr, BJ | 2 |
Daricello, G; Pavone, C; Pavone-Macaluso, M; Romano, C; Serretta, V | 1 |
Combettes, C; Durand-Seme, V; Leveque, JL; Querleux, B; Saint-Leger, D | 1 |
Gangnerau, MN; Picon, R | 1 |
Dias, JA; Swift, TA | 1 |
Abel, P; Cox, J; Farah, N; Fleming, J; Hewitt, G; O'Donoghue, EP; Sandow, J; Sikora, K; Waxman, J; Williams, G | 1 |
Sathyanesan, AG; Shrivastava, VK | 1 |
Sogani, PC; Whitmore, WF | 1 |
Soloway, MS | 1 |
Haider, S; Rai, U | 1 |
Alexandre, C; Balthazart, J | 2 |
Cunningham, GR; Kong, AY; Shao, TC | 1 |
Gutiérrez Cecchini, B; Hidalgo Balsera, A; Manso Rodríguez, G; Sala Blanco, J | 1 |
Fair, WR; Sogani, PC | 1 |
Ayub, M; Levell, MJ | 1 |
Dupront, A; Meyer, BH; Pottier, J; Tremblay, D | 1 |
el Etreby, MF; Habenicht, UF; Louton, T; Nishino, Y; Schröder, HG | 1 |
el Etreby, MF; Habenicht, UF; Neumann, F; Schröder, H | 1 |
Bruchovsky, N; Fletcher, T; Foekens, JA; Goldenberg, SL; Lawson, D; Rennie, PS | 1 |
Donn, F; Tamm, J; Volkwein, U | 1 |
Clos, V; Esteve, A; Jane, F; Salva, P | 1 |
Bouffioux, C | 1 |
Alioth, H; Müller, J; Senn, E | 1 |
Tokarz, RR | 1 |
Boublil, JL; Cavaglione, G; Kather, R; Namer, M | 1 |
Neumann, F | 1 |
Labrie, F; Poyet, P | 1 |
Wilson, FE | 1 |
Datta, JK; Roy, S | 1 |
Bullock, LP; Ventura, SM | 1 |
Jacobi, GH; Wenderoth, UK | 1 |
Hano, R; Knuth, UA; Nieschlag, E | 1 |
Ahmed, K; Davis, AT; Wilson, MJ | 1 |
Das, RP; Kumari, GL; Roy, S | 1 |
Rees, J; Shuster, S | 1 |
Lax, ER; Schriefers, H | 1 |
Panse, GT | 1 |
Baumann, P; Lax, ER; Schriefers, H | 1 |
Peluso, JJ; Steger, RW; Stude, D | 1 |
King, RJ; Yates, J | 1 |
Pandha, H; Waxman, J | 1 |
Hagen, R; Hoppe, F; Romalo, G; Schwab, B; Schweikert, HU | 1 |
Antoniou, G; Giannikos, L; Grigoriou, O; Karakitsos, P; Konidaris, S; Papadias, C | 1 |
Cutler, GB; Merke, DP | 1 |
Denis, L; Mahler, C; Verhelst, J | 1 |
De Markowsky, EE; Malgor, LA; Valsecia, M; Vergés, E | 1 |
Hirai, S; Matsubara, S | 1 |
Bisht, D; Chakraborti, PK; Rana, S | 1 |
Durmuşoğlu, F; Erenus, M; Gürbüz, O; Yücelten, D | 1 |
Benten, WP; Guo, Z; Lieberherr, M; Stamm, O; Wrehlke, C; Wunderlich, F | 1 |
Collette, L; de Reijke, TM; Schröder, FH; Whelan, P | 1 |
Man, RY; Quan, A; Teoh, H | 1 |
Leung, SW; Man, RY; Quan, A; Teoh, H | 1 |
Drapier-Faure, E; Faure, M | 1 |
Corradi, LS; Góes, RM; Leite Vilamaior, PS; Oliveira, SM; Taboga, SR | 1 |
Aguilera Tubet, C; Ballestero Diego, R; Roca Edreira, A; Villanueva Peña, A; Zubillaga Guerrero, S | 1 |
Delvoye, N; Gannon, PO; Lapointe, R; Mes-Masson, AM; Poisson, AO; Saad, F | 1 |
Alves, A; Gouveia, TIA; Mota, IH; Santos, MSF; Silva, AMT | 1 |
19 review(s) available for flutamide and cyproterone
Article | Year |
---|---|
Antiandrogens.
Topics: Acne Vulgaris; Androgen Antagonists; Animals; Biological Assay; Comb and Wattles; Cyproterone; Female; Fertility; Flutamide; Genitalia, Male; Hirsutism; Male; Phthalimides; Progesterone; Prostatic Hyperplasia; Prostatic Neoplasms; Sebaceous Glands; Sebum; Sex Differentiation; Sexual Behavior, Animal; Sexual Dysfunction, Physiological; Steroids | 1976 |
Androgen receptors and the molecular basis for the action of antiadrogens in the ventral prostate.
Topics: Androgen Antagonists; Animals; Carrier Proteins; Contraceptive Agents, Male; Cyproterone; Cytosol; Dihydrotestosterone; Flutamide; Genes; Male; Molecular Conformation; Prostate; Protein Binding; Rats; Receptors, Androgen; Receptors, Steroid; RNA; Transcription, Genetic | 1976 |
Chemotherapy of prostatic cancer.
Topics: Aged; Alkylating Agents; Antibiotics, Antineoplastic; Antimetabolites; Antineoplastic Agents; Bromocriptine; Cyproterone; Depression, Chemical; Diethylstilbestrol; Drug Therapy, Combination; Estramustine; Fluorouracil; Flutamide; Health Facilities; Hematologic Diseases; Humans; Kinetics; Male; Mitosis; Nitrogen Mustard Compounds; Prostatic Neoplasms | 1975 |
Cancer of the prostate. Mechanisms of action of antiandrogens.
Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Gonadotropin-Releasing Hormone; Humans; Luteinizing Hormone; Male; Prostatic Neoplasms; Rats; Testosterone | 1991 |
Antiandrogenic substances in the management of prostatic cancer.
Topics: Androgen Antagonists; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Prostatic Neoplasms | 1990 |
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds | 1990 |
Clinical applications of antiandrogens.
Topics: Androgen Antagonists; Breast Neoplasms; Cyproterone; Cyproterone Acetate; Female; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Hyperplasia; Prostatic Neoplasms; Puberty, Precocious; Skin Diseases; Spironolactone | 1988 |
Initiation of LHRH monotherapy for prostate cancer.
Topics: Androgen Antagonists; Antineoplastic Agents; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Flutamide; Gonadotropin-Releasing Hormone; Humans; Male; Prostatic Neoplasms | 1989 |
[Antiandrogens. Mechanisms and paradoxical effects].
Topics: 5-alpha Reductase Inhibitors; Androgen Antagonists; Androgens; Anilides; Cimetidine; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Nitriles; Spironolactone; Tosyl Compounds | 1989 |
Androgen blockade and suppression for prostate carcinoma.
Topics: Androgen Antagonists; Cyproterone; Drug Administration Schedule; Drug Therapy, Combination; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms | 1989 |
Flutamide and other antiandrogens in the treatment of advanced prostatic carcinoma.
Topics: Androgen Antagonists; Androgens; Anilides; Antineoplastic Agents; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Megestrol; Megestrol Acetate; Prostatic Neoplasms | 1988 |
Treatment of advanced prostatic cancer.
Topics: Adrenalectomy; Aminoglutethimide; Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Clinical Trials as Topic; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Estrogens; Flutamide; Glucocorticoids; Humans; Ketoconazole; Male; Megestrol; Megestrol Acetate; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms; Spironolactone; Time Factors | 1987 |
Advantages and disadvantages of pure antiandrogens and of antiandrogens of the cyproterone acetate-type in the treatment of prostatic cancer.
Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Female; Flutamide; Glucuronidase; Gonadotropin-Releasing Hormone; Guinea Pigs; Kidney; Male; Mice; Prostatic Neoplasms; Rats; Sex Differentiation; Time Factors | 1988 |
[LHRH agonists combined with antiandrogens in the treatment of metastasizing prostatic carcinoma].
Topics: Androgen Antagonists; Animals; Buserelin; Cyproterone; Cyproterone Acetate; Dogs; Drug Therapy, Combination; Flutamide; Humans; Male; Neoplasm Metastasis; Orchiectomy; Prostatic Neoplasms; Rats; Receptors, Cell Surface; Receptors, LHRH | 1985 |
New forms and future perspectives in endocrine treatment of prostatic carcinoma.
Topics: Aminoglutethimide; Androgen Antagonists; Cyproterone; Cyproterone Acetate; Estrogen Antagonists; Flutamide; Hormones; Humans; Male; Pituitary Hormone-Releasing Hormones; Prolactin; Prostatic Neoplasms | 1984 |
Clinical pharmacokinetics of the antiandrogens and their efficacy in prostate cancer.
Topics: Androgen Antagonists; Anilides; Antineoplastic Agents, Hormonal; Clinical Trials as Topic; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Tosyl Compounds | 1998 |
Maximum androgen blockade in advanced prostate cancer: an overview of the randomised trials. Prostate Cancer Trialists' Collaborative Group.
Topics: Aged; Androgen Antagonists; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Orchiectomy; Prostatic Neoplasms; Randomized Controlled Trials as Topic; Survival Analysis | 2000 |
[What is the role of hormonal treatments in acne?].
Topics: Acne Vulgaris; Androgen Antagonists; Cyproterone; Estrogens; Flutamide; Glucocorticoids; Hormone Antagonists; Humans; Mineralocorticoid Receptor Antagonists; Nandrolone; Patient Selection; Progestins; Spironolactone; Treatment Outcome | 2001 |
First-line treatment of metastatic prostate cancer. Androgen suppression for symptomatic disease.
Topics: Androgen Antagonists; Antineoplastic Agents, Hormonal; Bone Neoplasms; Cyproterone; Estrogens; Flutamide; Goserelin; Humans; Male; Neoplasms, Hormone-Dependent; Orchiectomy; Practice Guidelines as Topic; Prostatic Neoplasms; Time Factors; Treatment Outcome | 2013 |
13 trial(s) available for flutamide and cyproterone
Article | Year |
---|---|
Advanced prostatic cancer: clinical and hormonal response to flutamide in patients pretreated with LHRH analogue and cyproterone acetate.
Topics: Aged; Androgen Antagonists; Anilides; Buserelin; Clinical Trials as Topic; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Goserelin; Humans; Male; Middle Aged; Prostatic Neoplasms; Random Allocation | 1990 |
Antiandrogens: clinical applications.
Topics: Acne Vulgaris; Adult; Androgen Antagonists; Cyproterone; Cyproterone Acetate; Dermatitis, Seborrheic; Female; Flutamide; Hirsutism; Humans; Male; Prostatic Neoplasms; Spironolactone | 1990 |
Pure antiandrogens as monotherapy in prospective studies of prostatic carcinoma.
Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Nitriles; Prospective Studies; Prostatic Neoplasms; Tosyl Compounds | 1990 |
Effects of two different medical treatments on dihydrotestosterone content and androgen receptors in human benign prostatic hyperplasia.
Topics: Androgen Antagonists; Anilides; Cell Nucleus; Cyproterone; Cyproterone Acetate; Cytosol; Dihydrotestosterone; Flutamide; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Androgen; Tamoxifen | 1988 |
Short-term anti-androgen therapy and very long-acting depot gonadotrophin-releasing hormone agonist for prostatic cancer.
Topics: Aged; Aged, 80 and over; Androgen Antagonists; Buserelin; Clinical Trials as Topic; Cyproterone; Cyproterone Acetate; Delayed-Action Preparations; Flutamide; Humans; Male; Middle Aged; Prostatic Neoplasms; Random Allocation | 1989 |
The clinical and endocrine assessment of three different antiandrogen regimens combined with a very long-acting gonadotrophin-releasing hormone analogue.
Topics: Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Buserelin; Cyproterone; Cyproterone Acetate; Delayed-Action Preparations; Flutamide; Humans; Male; Middle Aged; Neoplasm Metastasis; Neoplasms, Hormone-Dependent; Phosphoric Monoester Hydrolases; Prostatic Neoplasms; Random Allocation; Testosterone | 1988 |
Treatment of advanced prostatic cancer.
Topics: Adrenalectomy; Aminoglutethimide; Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Clinical Trials as Topic; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Estrogens; Flutamide; Glucocorticoids; Humans; Ketoconazole; Male; Megestrol; Megestrol Acetate; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms; Spironolactone; Time Factors | 1987 |
The effect of short term treatment with cyproterone acetate or flutamide on the metabolism of 5 alpha-dihydrotestosterone in human testicular tissue.
Topics: Aged; Aged, 80 and over; Anilides; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Male; Middle Aged; Testis | 1988 |
Total androgen blockade in advanced prostatic cancer. Critical review and personal experience.
Topics: Androgen Antagonists; Buserelin; Cyproterone; Cyproterone Acetate; Flutamide; Goserelin; Humans; Male; Multicenter Studies as Topic; Orchiectomy; Prostatic Neoplasms; Time Factors | 1988 |
Effect of flutamide or cyproterone acetate on pituitary and testicular hormones in normal men.
Topics: Adult; Anilides; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Estradiol; Flutamide; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; Humans; Luteinizing Hormone; Male; Pituitary Function Tests; Pituitary Hormones; Prolactin; Testicular Hormones; Testosterone | 1984 |
Comparison of flutamide and cyproterone acetate in the treatment of hirsutism: a randomized controlled trial.
Topics: Adolescent; Adult; Androgen Antagonists; Cyproterone; Female; Flutamide; Hirsutism; Hormones; Humans; Prospective Studies | 1996 |
Recurrence rate of hirsutism after 3 different antiandrogen therapies.
Topics: Androgen Antagonists; Contraceptives, Oral; Cyproterone; Female; Flutamide; Hirsutism; Humans; Luteinizing Hormone; Recurrence; Spironolactone; Testosterone | 1999 |
Prostate cancer treated by anti-androgens: is sexual function preserved? EORTC Genitourinary Group. European Organization for Research and Treatment of Cancer.
Topics: Aged; Androgen Antagonists; Cyproterone; Erectile Dysfunction; Flutamide; Humans; Male; Middle Aged; Prospective Studies; Prostatic Neoplasms; Quality of Life; Sexuality | 2000 |
79 other study(ies) available for flutamide and cyproterone
Article | Year |
---|---|
Antiandrogenic steroidal sulfonylpyrazoles.
Topics: Androgen Antagonists; Animals; Male; Molecular Structure; Orchiectomy; Organ Size; Pregnanes; Prostate; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Androgen; Structure-Activity Relationship; Testosterone; X-Ray Diffraction | 1990 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding | 2012 |
The effect of antiandrogens and stilboestrol on the cytosol receptor in rat prostate.
Topics: Androgen Antagonists; Animals; Chlormadinone Acetate; Cyproterone; Cytosol; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Male; Nandrolone; Prostate; Rats; Receptors, Androgen; Receptors, Steroid | 1977 |
Androgen receptors in benign and malignant prostatic tissue.
Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Androgen Antagonists; Animals; Cyproterone; Dihydrotestosterone; Estrenes; Flutamide; Humans; Male; Prostatic Hyperplasia; Prostatic Neoplasms; Rats; Receptors, Androgen; Receptors, Steroid | 1979 |
Effect of antiandrogens on the binding of androgen to cytosol and nuclei of hamster sebaceous glands.
Topics: Androgen Antagonists; Androstanes; Androstanols; Animals; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Dihydrotestosterone; Estrenes; Flutamide; In Vitro Techniques; Male; Prostate; Receptors, Androgen; Receptors, Steroid; Sebaceous Glands; Seminal Vesicles; Steroids, Heterocyclic; Testosterone | 1979 |
Evidence for a role of androgens in the growth and maturation of ovarian follicles in rats.
Topics: Androgens; Animals; Corpus Luteum; Cyproterone; Diestrus; Estradiol; Estrus; Female; Flutamide; Ovarian Follicle; Ovary; Pregnancy; Rats | 1978 |
Testicular phosphatase activity in rats treated with cyproterone acetate & flutamide.
Topics: Acid Phosphatase; Alkaline Phosphatase; Anilides; Animals; Cyproterone; Flutamide; Male; Rats; Testis | 1977 |
Androgen binding to cytosol and nuclei of hamster sebaceous glands.
Topics: Androgens; Animals; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Dihydrotestosterone; Estradiol; Flutamide; Male; Progesterone; Receptors, Androgen; Sebaceous Glands | 1978 |
Androgenic stimulation of progesterone production by granulosa cells from preantral ovarian follicles: further in vitro studies using replicate cell cultures.
Topics: Animals; Cells, Cultured; Cyproterone; Diethylstilbestrol; Female; Flutamide; Granulosa Cells; Ovarian Follicle; Ovary; Progesterone; Rats; Testosterone | 1977 |
Specific androgen binding in the kidney and estrogen-dependent renal carcinoma of the Syrian hamster.
Topics: Androgens; Animals; Castration; Cell Nucleus; Cricetinae; Cyproterone; Cytosol; Diethylstilbestrol; Dihydrotestosterone; Estrogens; Flutamide; Kidney; Kidney Neoplasms; Liver; Male; Progesterone; Receptors, Androgen; Receptors, Steroid | 1977 |
Androgen receptor dependent and independent activities of testosterone on hepatic microsomal drug metabolism.
Topics: Animals; Castration; Cyproterone; Cytochrome P-450 Enzyme System; Ethylmorphine-N-Demethylase; Female; Flutamide; Liver; Male; Mice; Mice, Inbred BALB C; Microsomes, Liver; Organ Size; Quinone Reductases; Rats; Receptors, Androgen; Receptors, Steroid; Testosterone | 1976 |
Induction of delta-aminolevulinic acid synthetase by flutamide, a non-steroidal antiandrogen.
Topics: 5-Aminolevulinate Synthetase; Aminoisobutyric Acids; Anilides; Animals; Anti-Bacterial Agents; Cells, Cultured; Chick Embryo; Cyproterone; Enzyme Induction; Flutamide; Mitochondria, Liver | 1976 |
Differences among rat sex accessory glands in their neonatal androgen dependency.
Topics: Age Factors; Androstanes; Animals; Animals, Newborn; Castration; Cyproterone; DNA; Flutamide; Ketosteroids; Male; Prostate; Protein Biosynthesis; Rats; RNA; Seminal Vesicles; Steroids, Heterocyclic; Testis; Testosterone; Thymidine; Tritium | 1975 |
Evidence of a role of adrogens in follicular maturation.
Topics: Androgens; Androstenedione; Animals; Chorionic Gonadotropin; Cyproterone; Diethylstilbestrol; Dihydrotestosterone; Estradiol; Female; Flutamide; Humans; Hydrocortisone; Hydroxyprogesterones; Hypophysectomy; Organ Size; Ovarian Follicle; Ovary; Pituitary Gland; Progesterone; Rats; Testosterone | 1975 |
Biological aspects of antiandrogens.
Topics: Androgen Antagonists; Anilides; Animals; Castration; Cyproterone; DNA; Dose-Response Relationship, Drug; Flutamide; Male; Organ Size; Organ Specificity; Prostate; Rats; Seminal Vesicles; Testis; Testosterone | 1975 |
Flutamide. Mechanism of action of a new nonsteroidal antiandrogen.
Topics: Anilides; Animals; Castration; Chemical Phenomena; Chemistry; Cyproterone; DNA; Flutamide; Genitalia, Male; Male; Prostate; Rats; Seminal Vesicles; Testosterone | 1976 |
Regulation of androgen receptor mRNA and protein level by steroid hormones in human mammary cancer cells.
Topics: Blotting, Northern; Breast Neoplasms; Cyproterone; Dihydrotestosterone; Estradiol; Flutamide; Gene Expression Regulation, Neoplastic; Hormones; Humans; Immunohistochemistry; Progesterone Congeners; Radioligand Assay; Receptors, Androgen; RNA, Messenger; Steroids; Tumor Cells, Cultured | 1992 |
Neo-adjuvant hormonotherapy does not facilitate radical prostatectomy.
Topics: Aged; Antineoplastic Combined Chemotherapy Protocols; Blood Loss, Surgical; Chemotherapy, Adjuvant; Cyproterone; Estramustine; Flutamide; Humans; Male; Middle Aged; Prostatectomy; Prostatic Neoplasms | 1992 |
[A 79-year-old man with metastatic prostate cancer, treated with Zoladex, flutamide, calcitonin and Ostac, suffers from frequent troublesome sweating with palpitation and angina pectoris, especially at night. Is there a therapy?].
Topics: Aged; Androgen Antagonists; Angina Pectoris; Buserelin; Calcitonin; Cyproterone; Cyproterone Acetate; Flutamide; Goserelin; Humans; Hyperhidrosis; Male; Prostatic Neoplasms | 1992 |
[A study of the androgenic activity of anti-androgen].
Topics: Androgen Antagonists; Aniline Compounds; Animals; Arginase; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Estradiol; Flutamide; Male; Medroxyprogesterone; Organ Size; Ornithine Decarboxylase; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen; Seminal Vesicles | 1990 |
Investigation on serum neurone-specific enolase in prostate cancer diagnosis and monitoring: comparative study of a multiple tumor marker assay.
Topics: Acid Phosphatase; Antigens, Neoplasm; Antineoplastic Agents; APUD Cells; Biomarkers, Tumor; Carcinoembryonic Antigen; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Estramustine; Flutamide; Humans; Male; Orchiectomy; Phosphopyruvate Hydratase; Prostate-Specific Antigen; Prostatic Neoplasms | 1991 |
Effects of steroidal and non-steroidal antiandrogens on the left atrium of the rat in vitro.
Topics: Androgen Antagonists; Animals; Calcium; Chlormadinone Acetate; Cimetidine; Cyproterone; Electric Stimulation; Female; Flutamide; Heart; Heart Atria; In Vitro Techniques; Male; Medroxyprogesterone; Myocardial Contraction; Rats; Rats, Inbred Strains; Spironolactone; Steroids; Stimulation, Chemical | 1991 |
Influence of different types of antiandrogens on luteinizing hormone-releasing hormone analogue-induced testosterone surge in patients with metastatic carcinoma of the prostate.
Topics: Acid Phosphatase; Aged; Androgen Antagonists; Buserelin; Cyproterone; Cyproterone Acetate; Drug Therapy, Combination; Flutamide; Goserelin; Humans; Luteinizing Hormone; Male; Premedication; Prostatic Neoplasms; Testosterone; Time Factors | 1990 |
The synthetic androgen mibolerone induces transient suppression of the transformed phenotype in an androgen responsive human prostatic carcinoma cell line.
Topics: Androgen Antagonists; Androgens; Cell Division; Cell Transformation, Neoplastic; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Humans; Male; Nandrolone; Prostatic Neoplasms; Receptors, Androgen; RNA, Messenger; Tumor Cells, Cultured | 1990 |
Analysis of the androgenic activity of synthetic "progestins" currently used for the treatment of prostate cancer.
Topics: Adrenal Glands; Animals; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Flutamide; Male; Medroxyprogesterone; Medroxyprogesterone Acetate; Megestrol; Megestrol Acetate; Organ Size; Ornithine Decarboxylase; Progesterone Congeners; Prostate; Prostatic Neoplasms; Rats; Rats, Inbred Strains; Spironolactone | 1987 |
Stimulatory effect of synthetic progestins currently used for the treatment of prostate cancer on growth of the androgen-sensitive Shionogi tumor in mice.
Topics: Androgens; Animals; Chlormadinone Acetate; Cyproterone; Cyproterone Acetate; Female; Flutamide; Male; Mammary Neoplasms, Experimental; Medroxyprogesterone; Medroxyprogesterone Acetate; Megestrol; Megestrol Acetate; Mice; Progesterone Congeners; Prostatic Neoplasms | 1988 |
Treatment with antiandrogens induces an androgen-repressed gene in the rat ventral prostate.
Topics: Androgen Antagonists; Androgens; Animals; Blotting, Northern; Body Weight; Cell Survival; Cell-Free System; Cyproterone; Cyproterone Acetate; Flutamide; Gene Expression Regulation; Male; Orchiectomy; Organ Size; Prostate; Protein Biosynthesis; Rats; Rats, Inbred Strains; RNA | 1988 |
Androgens directly stimulate proliferation of bone cells in vitro.
Topics: Alkaline Phosphatase; Androgens; Animals; Binding, Competitive; Cell Count; Cell Differentiation; Cell Division; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; DNA; Dose-Response Relationship, Drug; Fluoxymesterone; Flutamide; Humans; Methenolone; Mice; Osteoblasts; Testosterone; Tumor Cells, Cultured | 1989 |
Antiandrogens do not reverse androgen-induced inhibition of sex hormone-binding globulin levels in adult female rhesus monkeys.
Topics: Androgen Antagonists; Androgens; Animals; Biomarkers; Cyproterone; Cyproterone Acetate; Female; Flutamide; Macaca; Macaca mulatta; Methyltestosterone; Ovariectomy; Pregnanes; Pyrazoles; Sex Hormone-Binding Globulin | 1989 |
Sexual dimorphism of blood pressure in spontaneously hypertensive rats: effects of anti-androgen treatment.
Topics: Androgen Antagonists; Anilides; Animals; Animals, Newborn; Blood Pressure; Cyproterone; Cyproterone Acetate; Female; Flutamide; Male; Orchiectomy; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Sex Characteristics; Species Specificity; Testosterone | 1989 |
Effect of antiandrogens on some key enzymes of glycolysis in epididymis and ventral prostate of rat.
Topics: Androgen Antagonists; Animals; Body Weight; Cyproterone; Cyproterone Acetate; Enzymes; Epididymis; Estradiol; Flutamide; Glycolysis; Male; Nandrolone; Organ Size; Prostate; Rats | 1989 |
"Casodex" (ICI 176,334)--a new, pure, peripherally-selective anti-androgen: preclinical studies.
Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostatic Neoplasms; Rats; Tosyl Compounds | 1989 |
[Antiandrogens in monotherapy or combined therapy for treatment of advanced cancer of the prostate].
Topics: Aged; Aged, 80 and over; Androgen Antagonists; Anilides; Antineoplastic Agents; Combined Modality Therapy; Cyproterone; Cyproterone Acetate; Flutamide; Follow-Up Studies; Humans; Imidazoles; Imidazolidines; Male; Middle Aged; Neoplasm Staging; Nitriles; Orchiectomy; Prostatic Neoplasms; Tosyl Compounds | 1989 |
Imaging the hamster flank organ by an ultrasonic technique: a new approach to animal tests.
Topics: Animals; Cricetinae; Cyproterone; Female; Flutamide; Male; Mesocricetus; Orchiectomy; Sebaceous Glands; Skin; Spironolactone; Testosterone; Ultrasonography | 1989 |
Onset of steroidogenesis and differentiation of functional LH receptors in rat fetal testicular cultures.
Topics: Aminoglutethimide; Animals; Binding, Competitive; Bucladesine; Cyproterone; Cyproterone Acetate; Dehydroepiandrosterone; Flutamide; Gestational Age; Luteinizing Hormone; Male; Organ Culture Techniques; Progesterone; Rats; Rats, Inbred Strains; Receptors, LH; Testis; Testosterone | 1987 |
Testosterone suppression of ornithine decarboxylase activity in rat Sertoli cells.
Topics: Animals; Bucladesine; Cells, Cultured; Cyclic AMP; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Enzyme Induction; Estradiol; Flutamide; Follicle Stimulating Hormone; Male; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Sertoli Cells; Testosterone | 1988 |
Combined treatment with flutamide and surgical or medical (LHRH agonist) castration in metastatic prostatic cancer.
Topics: Anilides; Combined Modality Therapy; Cyproterone; Flutamide; Gonadotropin-Releasing Hormone; Humans; Male; Megestrol; Neoplasm Metastasis; Orchiectomy; Prostatic Neoplasms; Receptors, Cell Surface; Receptors, LHRH | 1986 |
Effect of antiandrogens on the hypothalamic gamma-aminobutyric acid (GABA) and glutamate contents of the Indian palm squirrel (Funambulus pennanti, Wroughton).
Topics: Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Female; Flutamide; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hypothalamus; Organ Size; Sciuridae | 1986 |
Treatment of prostatic cancer. Newer forms of androgen deprivation.
Topics: Androgen Antagonists; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Male; Megestrol; Megestrol Acetate; Neoplasm Metastasis; Orchiectomy; Pituitary Hormone-Releasing Hormones; Prostatic Neoplasms | 1986 |
Effects of cyproterone acetate and flutamide on the testis and epididymis of the Indian wall lizard, Hemidactylus flaviviridis (Ruppell).
Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Epididymis; Epithelial Cells; Flutamide; Leydig Cells; Lizards; Male; Organ Size; Spermatogenesis; Spermatozoa; Testis | 1986 |
Inhibition of testosterone metabolism in the brain and cloacal gland of the quail by specific inhibitors and antihormones.
Topics: Androgen Antagonists; Androstanes; Androstatrienes; Animals; Azasteroids; Cloaca; Coturnix; Cyproterone; Cyproterone Acetate; Estrogen Antagonists; Flutamide; Hypothalamus; Male; Nitromifene; Quail; Tamoxifen; Testosterone | 1987 |
Acid phosphatase activity: a marker of androgen action in prostate explant cultures.
Topics: Acid Phosphatase; Animals; Cells, Cultured; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Estradiol; Flutamide; Hydrocortisone; Male; Prostate; Rats; Rats, Inbred Strains | 1987 |
Effects of metabolism inhibitors, antiestrogens and antiandrogens on the androgen and estrogen induced sexual behavior in Japanese quail.
Topics: Androgens; Androstatrienes; Animals; Coturnix; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Estrogens; Flutamide; Male; Orchiectomy; Quail; Sexual Behavior, Animal; Tamoxifen; Testosterone | 1986 |
[Effects of cyproterone acetate and flutamide on blood calcium and bone structure].
Topics: Androgen Antagonists; Anilides; Animals; Bone and Bones; Calcium; Cyproterone; Cyproterone Acetate; Flutamide; Male; Rats; Rats, Inbred Strains | 1986 |
Inhibition of rat testicular 17 alpha-hydroxylase and 17,20-lyase activities by anti-androgens (flutamide, hydroxyflutamide, RU23908, cyproterone acetate) in vitro.
Topics: Aldehyde-Lyases; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Cytochrome P-450 Enzyme System; Flutamide; Imidazoles; Imidazolidines; Kinetics; Male; Microsomes; Rats; Rats, Inbred Strains; Steroid 17-alpha-Hydroxylase; Steroid Hydroxylases; Testis | 1987 |
The kinetics of antiandrogens in humans.
Topics: Androgen Antagonists; Anilides; Cyproterone; Cyproterone Acetate; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Prostatic Neoplasms | 1987 |
Effect of cyproterone acetate in comparison to flutamide and megestrol acetate on the ventral prostate, seminal vesicle, and adrenal glands of adult male rats.
Topics: Adrenal Glands; Androgen Antagonists; Animals; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Organ Size; Prostate; Rats; Rats, Inbred Strains; Seminal Vesicles | 1987 |
ICI 176,334: a novel non-steroidal, peripherally-selective antiandrogen.
Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Dogs; Flutamide; Imidazoles; Imidazolidines; Male; Nitriles; Prostate; Radioligand Assay; Rats; Receptors, Androgen; Seminal Vesicles; Testosterone; Tosyl Compounds | 1988 |
Relative effectiveness of alternative androgen withdrawal therapies in initiating regression of rat prostate.
Topics: Anilides; Animals; Cyproterone; Cyproterone Acetate; Diethylstilbestrol; Dihydrotestosterone; Flutamide; Gonadotropin-Releasing Hormone; Imidazoles; Imidazolidines; Leuprolide; Male; Megestrol; Megestrol Acetate; Orchiectomy; Prostate; Rats; Rats, Inbred Strains; Receptors, Androgen | 1988 |
Microsomal effects of cyproterone acetate and flutamide in rat testis.
Topics: Androgen Antagonists; Anilides; Animals; Cyproterone; Cyproterone Acetate; Cytochrome b Group; Cytochrome P-450 Enzyme System; Cytochromes b5; Flutamide; In Vitro Techniques; Luteinizing Hormone; Male; Microsomes; NADPH-Ferrihemoprotein Reductase; Rats; Rats, Inbred Strains; Testis; Testosterone | 1988 |
Effects of the antiandrogens cyproterone acetate and flutamide on male reproductive behavior in a lizard (Anolis sagrei).
Topics: Aggression; Anilides; Animals; Cyproterone; Dihydrotestosterone; Female; Flutamide; Lizards; Male; Organ Size; Sexual Behavior, Animal; Social Dominance; Testis; Testosterone | 1987 |
[Cancer of the prostate: new hormone therapies].
Topics: Androgen Antagonists; Cyproterone; Flutamide; Humans; Ketoconazole; Male; Medroxyprogesterone; Megestrol; Neoplasms, Hormone-Dependent; Progestins; Prostatic Neoplasms; Tamoxifen | 1986 |
Principles of endocrine manipulation in the treatment of prostatic cancer.
Topics: Androgen Antagonists; Animals; Castration; Cyproterone; Estrogens; Flutamide; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Male; Neoplasms, Hormone-Dependent; Progestins; Prostatic Neoplasms; Rats; Testosterone | 1985 |
Comparison of the antiandrogenic/androgenic activities of flutamide, cyproterone acetate and megestrol acetate.
Topics: Adrenal Glands; Anilides; Animals; Cyproterone; Dihydrotestosterone; Flutamide; Follicle Stimulating Hormone; Luteinizing Hormone; Male; Megestrol; Orchiectomy; Organ Size; Prostate; Rats; Rats, Inbred Strains | 1985 |
An androgen-independent mechanism maintains photorefractoriness in male tree sparrows (Spizella arborea).
Topics: Animals; Birds; Castration; Cyproterone; Flutamide; Light; Luteinizing Hormone; Male; Radioimmunoassay; Testosterone | 1985 |
Effect of anti-androgens on the morphological & biochemical changes induced by testosterone in rat uterus.
Topics: Anilides; Animals; Cyproterone; Female; Flutamide; Glycogen; Proteins; Rats; RNA; Sialic Acids; Testosterone; Uterus | 1980 |
Stimulation of ribonucleic acid polymerase activity in mouse kidney.
Topics: Animals; Cyproterone; Cyproterone Acetate; DNA-Directed RNA Polymerases; Female; Flutamide; Kidney; Medroxyprogesterone; Mice; Mice, Inbred C57BL; Progesterone; Receptors, Androgen; Receptors, Steroid; RNA Polymerase I; RNA Polymerase II; Testosterone | 1983 |
Effects of antiandrogens (cyproterone acetate and flutamide) on the activity of nuclear protein phosphokinases and phosphatases of rat ventral prostate.
Topics: Alkaline Phosphatase; Anilides; Animals; Castration; Cell Nucleus; Chromatin; Cyproterone; Flutamide; Male; Phosphoric Monoester Hydrolases; Prostate; Protein Kinases; Rats; Testosterone | 1980 |
Effect of 17-hydroxy progesterone caproate, flutamide & cyproterone acetate on genital organs & fertility of male rats--a comparative study.
Topics: 17 alpha-Hydroxyprogesterone Caproate; Anilides; Animals; Contraceptive Agents, Male; Cyproterone; Cyproterone Acetate; Fertility; Flutamide; Genitalia, Male; Hydroxyprogesterones; Male; Organ Specificity; Progesterone Congeners; Rats | 1980 |
Pubertal induction of sweat gland activity.
Topics: Acne Vulgaris; Adult; Child; Cyproterone; Cyproterone Acetate; Female; Flutamide; Humans; Male; Middle Aged; Puberty; Sex Factors; Sweat Glands; Sweating; Testosterone | 1981 |
Sex-specific action of antiandrogens on androgen induced changes in hepatic microsomal 3 beta-hydroxysteroid dehydrogenase and 5 alpha-reductase activity in the rat.
Topics: 3-Hydroxysteroid Dehydrogenases; 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Androgen Antagonists; Anilides; Animals; Castration; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Female; Flutamide; Male; Microsomes, Liver; Organ Size; Oxidoreductases; Rats; Sex Factors | 1981 |
Effects of antiandrogens on glycogen metabolism of spermatozoa from caput epididymidis.
Topics: Anilides; Animals; Contraceptive Agents, Male; Cyproterone; Cyproterone Acetate; Flutamide; Glycogen; Male; Mice; Spermatozoa | 1981 |
Antiandrogenic effects of oestradiol on enzyme activities of hepatic steroid metabolism.
Topics: 3-alpha-Hydroxysteroid Dehydrogenase (B-Specific); 3-Hydroxysteroid Dehydrogenases; 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Animals; Castration; Cyproterone; Dihydrotestosterone; Estradiol; Female; Flutamide; Male; Microsomes, Liver; Oxidoreductases; Rats; Rats, Inbred Strains | 1983 |
Role of androgens in hCG-induced ovulation in PMSG-primed immature rats.
Topics: 3-Hydroxysteroid Dehydrogenases; Androgens; Anilides; Animals; Chorionic Gonadotropin; Cyproterone; Estradiol; Female; Flutamide; Gonadotropins, Equine; Ovarian Follicle; Ovulation; Progesterone; Rats | 1980 |
Antiandrogen effects on androgen-responsive mammary tumour cells in culture.
Topics: Anilides; Animals; Cell Division; Cells, Cultured; Cyproterone; Dihydrotestosterone; Dose-Response Relationship, Drug; Flutamide; Mammary Neoplasms, Experimental; Mice; Receptors, Androgen; Testosterone | 1981 |
Anti-androgens in treatment of prostate cancer.
Topics: Androgen Antagonists; Antineoplastic Combined Chemotherapy Protocols; Cyproterone; Flutamide; Humans; Imidazoles; Imidazolidines; Male; Meta-Analysis as Topic; Prostatic Neoplasms | 1995 |
Juvenile nasopharyngeal fibroma: androgen receptors and their significance for tumor growth.
Topics: Cell Division; Child; Cholestenone 5 alpha-Reductase; Cyproterone; Cyproterone Acetate; Dihydrotestosterone; Fibroblasts; Fibroma; Flutamide; Humans; Male; Nasopharyngeal Neoplasms; Oxidoreductases; Receptors, Androgen; Scrotum; Skin; Testosterone; Tritium; Tumor Cells, Cultured | 1994 |
New approaches to the treatment of congenital adrenal hyperplasia.
Topics: Adrenal Hyperplasia, Congenital; Age Determination by Skeleton; Androgen Antagonists; Child; Cyproterone; Drug Therapy, Combination; Female; Fludrocortisone; Flutamide; Growth; Humans; Hydrocortisone; Mineralocorticoid Receptor Antagonists; Spironolactone; Testolactone | 1997 |
Blockade of the in vitro effects of testosterone and erythropoietin on Cfu-E and Bfu-E proliferation by pretreatment of the donor rats with cyproterone and flutamide.
Topics: Androgen Antagonists; Animals; Bone Marrow Cells; Cells, Cultured; Cyproterone; Erythroid Precursor Cells; Erythropoiesis; Erythropoietin; Flutamide; Male; Premedication; Rats; Testosterone | 1998 |
Influence of anti-androgens on the anterior horn cells of rat spinal cord: morphometric and in-situ hybridization studies.
Topics: Androgen Antagonists; Animals; Anterior Horn Cells; Cell Count; Cell Size; Choline O-Acetyltransferase; Cyproterone; Flutamide; In Situ Hybridization; Male; Rats; Rats, Wistar; RNA, Messenger | 1998 |
Synergistic activation of yeast-expressed rat androgen receptor by modulators of protein kinase-A.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 8-Bromo Cyclic Adenosine Monophosphate; Androgens; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyproterone; Dihydrotestosterone; Enzyme Inhibitors; Flutamide; Gene Expression Regulation; Genes, Reporter; Metribolone; Okadaic Acid; Rats; Receptors, Androgen; Regulatory Sequences, Nucleic Acid; RNA, Messenger; Saccharomyces cerevisiae; Signal Transduction; Transcriptional Activation; Transformation, Genetic | 1999 |
Testosterone signaling through internalizable surface receptors in androgen receptor-free macrophages.
Topics: Androgen Antagonists; Animals; Calcium; Cell Line; Cyproterone; Endocytosis; Estradiol; Estrenes; Flow Cytometry; Flutamide; Macrophages; Mice; Mice, Knockout; Microscopy, Confocal; Pertussis Toxin; Pyrrolidinones; Receptors, Androgen; Receptors, Cell Surface; Serum Albumin, Bovine; Signal Transduction; Testosterone; Type C Phospholipases; Virulence Factors, Bordetella | 1999 |
Acute impairment of relaxation by low levels of testosterone in porcine coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Analysis of Variance; Androgen Receptor Antagonists; Animals; Bradykinin; Calcimycin; Coronary Vessels; Cromakalim; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Flutamide; Ionophores; Male; Nitroprusside; Swine; Testosterone; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2000 |
Differential effects of 17beta-estradiol and testosterone on the contractile responses of porcine coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Androgen Antagonists; Androgen Receptor Antagonists; Animals; Coronary Vessels; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelin-1; Estradiol; Estrogen Antagonists; Female; Flutamide; Fulvestrant; In Vitro Techniques; Isotonic Solutions; Male; Potassium Chloride; Receptors, Estrogen; Serotonin; Swine; Tamoxifen; Testosterone; Vasoconstriction | 2000 |
Cellular and extracellular behavior in the gerbil (Meriones unguiculatus) ventral prostate following different types of castration and the consequences of testosterone replacement.
Topics: Acid Phosphatase; Androgen Antagonists; Animals; Cyproterone; Disease Models, Animal; Endoplasmic Reticulum, Rough; Endothelium; Flutamide; Gerbillinae; Immunohistochemistry; Male; Microscopy, Electron, Transmission; Orchiectomy; Organ Size; Prostate; Prostatic Hyperplasia; Protein Tyrosine Phosphatases; Receptors, Androgen; Testosterone | 2007 |
[Mediastinal lymph nodes during the course of a metastatic prostate cancer].
Topics: Adenocarcinoma; Androgen Antagonists; Androgens; Antineoplastic Combined Chemotherapy Protocols; Bone Neoplasms; Cyproterone; Diphosphonates; Estramustine; Fatal Outcome; Flutamide; Humans; Imidazoles; Ketoconazole; Lung Neoplasms; Lymphatic Metastasis; Male; Mediastinum; Neoplasms, Hormone-Dependent; Prostatic Neoplasms; Radionuclide Imaging; Skin Neoplasms; Triptorelin Pamoate; Zoledronic Acid | 2007 |
Characterization of the intra-prostatic immune cell infiltration in androgen-deprived prostate cancer patients.
Topics: Androgen Antagonists; Androgens; Antineoplastic Agents, Hormonal; Cyproterone; Flutamide; Humans; Killer Cells, Natural; Leuprolide; Lymphocytes, Tumor-Infiltrating; Macrophages; Male; Neoplasm Recurrence, Local; Prostatic Neoplasms; T-Lymphocytes | 2009 |
Are cytostatic drugs in surface waters a potential threat?
Topics: Child; Chlorambucil; Cyclophosphamide; Cyproterone; Cytostatic Agents; Drinking Water; Environmental Monitoring; Etoposide; Flutamide; Humans; Mycophenolic Acid; Pharmaceutical Preparations; Rivers; Tamoxifen; Water Pollutants, Chemical | 2022 |