flutamide and cycloheximide

flutamide has been researched along with cycloheximide in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.56)18.7374
1990's5 (27.78)18.2507
2000's8 (44.44)29.6817
2010's4 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Mora, G; Muldoon, TG; Steinsapir, J1
Bardin, CW; Jänne, OA; Kontula, KK; Seppänen, PJ; van Duyne, P1
Cantabrana, B; Gutierrez, M; Hidalgo, A; Sánchez Aparicio, JA1
Varriale, B1
Galosy, S; Gudmundsson, GO; Newcomer, B; Sridaran, R; Talamantes, F; Thordarson, G1
Fan, Z; Mendelsohn, J; Ye, D1
Man, RY; Quan, A; Teoh, H1
Leung, SW; Man, RY; Quan, A; Teoh, H1
Lou, YR; Nazarova, N; Pennanen, P; Qiao, S; Tuohimaa, P1
Lou, YR; Nazarova, N; Talonpoika, R; Tuohimaa, P1
Hareramadas, B; Rai, U1
Brogley, M; Chinnaiyan, A; Dhanasekaran, S; Hofer, MD; Kuefer, R; Lapensee, EW; O'Mahony, OA; Pienta, KJ; Rehman, H; Robins, DM; Rubin, MA; Steinkamp, MP1
Díaz, M; Gómez, T; González-Montelongo, MC; Marín, R; Marrero-Alonso, J1
Centurión, D; Cobos-Puc, LE; González-Hernández, A; Maassenvandenbrink, A; Muñoz-Islas, E; Ramírez-Rosas, MB; Sánchez-López, A; Villalón, CM1
Kai, L; Levenson, AS1
Avellar, MC; Callera, GE; Camargo, LL; Carvalho, MH; Chignalia, AZ; Fortes, ZB; Laurindo, FR; Lopes, LR; Montezano, AC; Schuldt, EZ; Tostes, RC; Touyz, RM1

Other Studies

18 other study(ies) available for flutamide and cycloheximide

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Effects of steroidal and non-steroidal antiandrogens on the androgen binding properties of the rat ventral prostate androgen receptor.
    Biochimica et biophysica acta, 1991, Aug-13, Volume: 1094, Issue:1

    Topics: Androgen Antagonists; Animals; Cycloheximide; Flutamide; Imidazoles; Imidazolidines; Kinetics; Male; Prostate; Rats; Receptors, Androgen

1991
Effect of a nonsteroidal antiandrogen, flutamide, on androgen receptor dynamics and ornithine decarboxylase gene expression in mouse kidney.
    Endocrinology, 1985, Volume: 116, Issue:1

    Topics: Anilides; Animals; Cell Nucleus; Cycloheximide; Female; Flutamide; Gene Expression Regulation; Kidney; Male; Mice; Nucleic Acid Hybridization; Ornithine Decarboxylase; Rats; Rats, Inbred Strains; Receptors, Androgen; Receptors, Steroid; RNA, Messenger; Testosterone

1985
Effects of androgens on isolated rat uterus.
    Life sciences, 1993, Volume: 53, Issue:3

    Topics: Animals; Cycloheximide; Cyproterone Acetate; Dactinomycin; Dihydrotestosterone; Drug Interactions; Female; Flutamide; In Vitro Techniques; Muscle Contraction; Rats; Rats, Wistar; Uterus

1993
Autoinduction of androgen receptor mRNA in primary cultures of hamster (Mesocricetus auratus) harderian gland cells.
    General and comparative endocrinology, 1996, Volume: 102, Issue:3

    Topics: Actins; Androgen Antagonists; Animals; Autoradiography; Blotting, Northern; Cells, Cultured; Cricetinae; Cycloheximide; DNA, Complementary; Dose-Response Relationship, Drug; Flutamide; Gene Expression Regulation; Harderian Gland; Male; Mesocricetus; Phosphorus Radioisotopes; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Androgen; Reference Standards; RNA, Messenger; Testosterone; Time Factors

1996
Interaction of mouse placental lactogens and androgens in regulating progesterone release in cultured mouse luteal cells.
    Endocrinology, 1997, Volume: 138, Issue:8

    Topics: Androgen Receptor Antagonists; Androgens; Androstenedione; Animals; Aromatase Inhibitors; Cattle; Cells, Cultured; Cycloheximide; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Fadrozole; Female; Flutamide; Luteal Cells; Mice; Placental Lactogen; Pregnancy; Progesterone; Prolactin; Protein Synthesis Inhibitors; Rabbits; Testosterone

1997
Androgen and epidermal growth factor down-regulate cyclin-dependent kinase inhibitor p27Kip1 and costimulate proliferation of MDA PCa 2a and MDA PCa 2b prostate cancer cells.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 1999, Volume: 5, Issue:8

    Topics: Androgen Antagonists; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Cell Cycle Proteins; Cell Division; Cyclin-Dependent Kinase Inhibitor p27; Cyclin-Dependent Kinases; Cycloheximide; Dihydrotestosterone; Down-Regulation; Drug Synergism; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Flutamide; Humans; Male; Metribolone; Microtubule-Associated Proteins; Prostatic Neoplasms; Protein Synthesis Inhibitors; Receptors, Androgen; Testosterone Congeners; Trastuzumab; Tumor Cells, Cultured; Tumor Suppressor Proteins

1999
Acute impairment of relaxation by low levels of testosterone in porcine coronary arteries.
    Cardiovascular research, 2000, Volume: 45, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Analysis of Variance; Androgen Receptor Antagonists; Animals; Bradykinin; Calcimycin; Coronary Vessels; Cromakalim; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Flutamide; Ionophores; Male; Nitroprusside; Swine; Testosterone; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2000
Differential effects of 17beta-estradiol and testosterone on the contractile responses of porcine coronary arteries.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Androgen Antagonists; Androgen Receptor Antagonists; Animals; Coronary Vessels; Cycloheximide; Cyproterone; Dactinomycin; Dose-Response Relationship, Drug; Endothelin-1; Estradiol; Estrogen Antagonists; Female; Flutamide; Fulvestrant; In Vitro Techniques; Isotonic Solutions; Male; Potassium Chloride; Receptors, Estrogen; Serotonin; Swine; Tamoxifen; Testosterone; Vasoconstriction

2000
Inhibition of fatty acid synthase expression by 1alpha,25-dihydroxyvitamin D3 in prostate cancer cells.
    The Journal of steroid biochemistry and molecular biology, 2003, Volume: 85, Issue:1

    Topics: Androgen Antagonists; Anilides; Calcitriol; Cerulenin; Cycloheximide; Down-Regulation; Enzyme Inhibitors; Fatty Acid Synthases; Flutamide; Gene Expression Regulation, Neoplastic; Humans; Male; Nitriles; Oligonucleotide Array Sequence Analysis; Prostatic Neoplasms; Protein Synthesis Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tosyl Compounds; Tumor Cells, Cultured

2003
5alpha-dihydrotestosterone inhibits 1alpha,25-dihydroxyvitamin D3-induced expression of CYP24 in human prostate cancer cells.
    The Prostate, 2005, May-15, Volume: 63, Issue:3

    Topics: Androgen Receptor Antagonists; Androgens; Anilides; Calcitriol; Cycloheximide; Cytochrome P-450 Enzyme System; Dihydrotestosterone; Drug Interactions; Flutamide; Gene Expression Regulation, Enzymologic; Humans; Male; Nitriles; Prostatic Neoplasms; Protein Synthesis Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Steroid Hydroxylases; Tosyl Compounds; Tumor Cells, Cultured; Vitamin D3 24-Hydroxylase

2005
Mechanism of androgen-induced thymic atrophy in the wall lizard, Hemidactylus flaviviridis: an in vitro study.
    General and comparative endocrinology, 2005, Volume: 144, Issue:1

    Topics: Androgen Antagonists; Androgens; Animals; Apoptosis; Caspases; Cell Proliferation; Cycloheximide; Dactinomycin; Dihydrotestosterone; Flutamide; In Vitro Techniques; Lizards; Male; Protein Synthesis Inhibitors; Thymus Gland

2005
Treatment-dependent androgen receptor mutations in prostate cancer exploit multiple mechanisms to evade therapy.
    Cancer research, 2009, May-15, Volume: 69, Issue:10

    Topics: Amino Acid Substitution; Anilides; Antineoplastic Agents; Autopsy; Cycloheximide; DNA Primers; Flutamide; Humans; Lymphatic Metastasis; Male; Mutation; Nitriles; Prostatic Neoplasms; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; RNA, Neoplasm; Tosyl Compounds

2009
Androgens induce nongenomic stimulation of colonic contractile activity through induction of calcium sensitization and phosphorylation of LC20 and CPI-17.
    Molecular endocrinology (Baltimore, Md.), 2010, Volume: 24, Issue:5

    Topics: Amides; Androgens; Animals; Benzophenanthridines; Blotting, Western; Calcium; Colon; Cycloheximide; Dactinomycin; Dihydrotestosterone; Enzyme Inhibitors; Finasteride; Flutamide; In Vitro Techniques; Male; Mice; Models, Biological; Models, Theoretical; Muscle Contraction; Muscle, Smooth; Phosphorylation; Protein Kinase C; Pyridines; Receptors, Androgen; rho-Associated Kinases; Signal Transduction; Testosterone

2010
Pharmacological evidence that Ca²+ channels and, to a lesser extent, K+ channels mediate the relaxation of testosterone in the canine basilar artery.
    Steroids, 2011, Volume: 76, Issue:4

    Topics: 4-Aminopyridine; Adenine; Aminoglutethimide; Androgen Receptor Antagonists; Animals; Aromatase Inhibitors; Barium Compounds; Basilar Artery; Calcium Channel Blockers; Calcium Channels; Chlorides; Cycloheximide; Dactinomycin; Dogs; Enzyme Inhibitors; Flutamide; In Vitro Techniques; Male; Nifedipine; Nucleic Acid Synthesis Inhibitors; Oxadiazoles; Potassium Channel Blockers; Potassium Channels; Protein Synthesis Inhibitors; Quinoxalines; Testosterone; Vasodilation; Vasodilator Agents

2011
Combination of resveratrol and antiandrogen flutamide has synergistic effect on androgen receptor inhibition in prostate cancer cells.
    Anticancer research, 2011, Volume: 31, Issue:10

    Topics: Androgen Antagonists; Caspase 3; Cell Line, Tumor; Cell Proliferation; Cycloheximide; Dihydrotestosterone; Down-Regulation; Drug Synergism; Flutamide; Gene Expression Regulation, Neoplastic; Humans; Male; Prostate-Specific Antigen; Prostatic Neoplasms; Proteasome Endopeptidase Complex; Protein Processing, Post-Translational; Receptors, Androgen; Resveratrol; RNA, Messenger; Stilbenes; Transcriptional Activation

2011
Testosterone induces vascular smooth muscle cell migration by NADPH oxidase and c-Src-dependent pathways.
    Hypertension (Dallas, Tex. : 1979), 2012, Volume: 59, Issue:6

    Topics: Androgen Antagonists; Androgens; Animals; Cell Movement; Cells, Cultured; Cycloheximide; Dactinomycin; Flutamide; Immunoblotting; Male; Muscle, Smooth, Vascular; NADH, NADPH Oxidoreductases; NADPH Oxidase 1; NADPH Oxidase 4; NADPH Oxidases; Protein Synthesis Inhibitors; Proto-Oncogene Proteins pp60(c-src); Pyrimidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Reactive Oxygen Species; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Testosterone

2012