fluphenazine and sk&f 7172-a2

fluphenazine has been researched along with sk&f 7172-a2 in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19905 (31.25)18.7374
1990's9 (56.25)18.2507
2000's1 (6.25)29.6817
2010's1 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chesselet, MF; Weiss-Wunder, LT1
Chesselet, MF; Weiss, LT1
Thermos, K; Weiss, B; Winkler, JD2
Wreggett, KA1
Cross, J; Glazer, L; Hait, WN; Kaiser, C; Kennedy, KA1
Qin, ZH; Wang, Y; Weiss, B; Zhang, SP; Zhou, LW1
Aloyo, VJ; Chen, JF; Qin, ZH; Weiss, B1
Qin, ZH; Weiss, B1
Qin, ZH; Weiss, B; Zhou, LW1
Chen, JF; Weiss, B1
Qin, ZH; Weiss, B; Zhang, SP1
Ekokoski, E; Törnquist, K1
Davidkova, G; Morabito, M; Weiss, B; Zhang, SP; Zhou, LW1
Hwang, MK; Kim, SH; Min, YK1
Chai, Y; Lin, YF1

Other Studies

16 other study(ies) available for fluphenazine and sk&f 7172-a2

ArticleYear
Acute and repeated administration of fluphenazine-N-mustard alters levels of tyrosine hydroxylase mRNA in subsets of mesencephalic dopaminergic neurons.
    Neuroscience, 1992, Volume: 49, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Electrochemistry; Fluphenazine; Male; Mesencephalon; Mice; Neurons; Nucleic Acid Hybridization; RNA Probes; RNA, Messenger; Substantia Nigra; Tyrosine 3-Monooxygenase

1992
Regional distribution and regulation of preprosomatostatin messenger RNA in the striatum, as revealed by in situ hybridization histochemistry.
    Brain research. Molecular brain research, 1989, Volume: 5, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Fluphenazine; Male; Mice; Nucleic Acid Hybridization; Protein Precursors; RNA, Messenger; Somatostatin

1989
Differential effects of fluphenazine-N-mustard, on calmodulin activity and on D1 and D2 dopaminergic responses.
    Psychopharmacology, 1987, Volume: 92, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Calmodulin; Corpus Striatum; Ergolines; Fluphenazine; Male; Mice; Quinpirole; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior

1987
Alkylation of the bovine anterior pituitary D2-dopamine receptor: inconsistency with predictions of the ternary complex model.
    Biochemical and biophysical research communications, 1987, Sep-30, Volume: 147, Issue:3

    Topics: Alkylation; Animals; Apomorphine; Binding, Competitive; Cattle; Cell Membrane; Computer Simulation; Dopamine Antagonists; Fluphenazine; GTP-Binding Proteins; In Vitro Techniques; Ligands; Pituitary Gland, Anterior; Receptors, Dopamine; Spiperone; Structure-Activity Relationship

1987
Comparison of the effects of fluphenazine-N-mustard on dopamine binding sites and on behavior induced by apomorphine in supersensitive mice.
    Neuropharmacology, 1987, Volume: 26, Issue:10

    Topics: Animals; Apomorphine; Binding, Competitive; Fluphenazine; Hydroxydopamines; Male; Mice; Oxidopamine; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1987
Pharmacological properties of fluphenazine-mustard, an irreversible calmodulin antagonist.
    Molecular pharmacology, 1987, Volume: 32, Issue:3

    Topics: Alkylating Agents; Calcium; Calmodulin; Cell Division; Chemical Phenomena; Chemistry; DNA Damage; DNA-Binding Proteins; DNA, Neoplasm; Fluphenazine; Humans; Phenothiazines; Tumor Cells, Cultured

1987
D2 dopamine receptor antisense oligodeoxynucleotide inhibits the synthesis of a functional pool of D2 dopamine receptors.
    Molecular pharmacology, 1995, Volume: 48, Issue:4

    Topics: Animals; Behavior, Animal; Catalepsy; Corpus Striatum; Fluphenazine; Male; Mice; Oligonucleotides, Antisense; Protein Synthesis Inhibitors; Receptors, Dopamine D2

1995
Irreversible blockade of D2 dopamine receptors by fluphenazine-N-mustard increases D2 dopamine receptor mRNA and proenkephalin mRNA and decreases D1 dopamine receptor mRNA and mu and delta opioid receptors in rat striatum.
    Neurochemistry international, 1994, Volume: 25, Issue:4

    Topics: Animals; Base Sequence; Corpus Striatum; Dopamine D2 Receptor Antagonists; Enkephalins; Fluphenazine; Male; Molecular Sequence Data; Protein Precursors; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger

1994
Dopamine receptor blockade increases dopamine D2 receptor and glutamic acid decarboxylase mRNAs in mouse substantia nigra.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: Analysis of Variance; Animals; Autoradiography; Benzazepines; Binding, Competitive; Dopamine Antagonists; Fluphenazine; Gene Expression Regulation, Enzymologic; Glutamate Decarboxylase; Image Processing, Computer-Assisted; In Situ Hybridization; Male; Mice; Oligonucleotide Probes; Quinolines; Receptors, Dopamine D2; RNA, Messenger; Substantia Nigra

1994
D2 dopamine receptor messenger RNA is altered to a greater extent by blockade of glutamate receptors than by blockade of dopamine receptors.
    Neuroscience, 1994, Volume: 60, Issue:1

    Topics: Animals; Autoradiography; Basal Ganglia; Brain Chemistry; Dizocilpine Maleate; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; In Situ Hybridization; Male; Mice; Quinolines; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger

1994
Irreversible blockade of D2 dopamine receptors by fluphenazine-N-mustard increases glutamic acid decarboxylase mRNA in rat striatum.
    Neuroscience letters, 1993, Feb-19, Volume: 150, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Base Sequence; Blotting, Northern; Clozapine; Corpus Striatum; Depression, Chemical; Dopamine D2 Receptor Antagonists; Fluphenazine; Glutamate Decarboxylase; Haloperidol; In Vitro Techniques; Male; Molecular Sequence Data; Oligodeoxyribonucleotides; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA Probes; RNA, Messenger

1993
Dopaminergic and glutamatergic blocking drugs differentially regulate glutamic acid decarboxylase mRNA in mouse brain.
    Brain research. Molecular brain research, 1994, Volume: 21, Issue:3-4

    Topics: Animals; Brain; Dizocilpine Maleate; Dopamine Antagonists; Fluphenazine; Glutamate Decarboxylase; In Situ Hybridization; Male; Mice; Oligonucleotide Probes; Quinolines; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; RNA, Messenger

1994
Inhibition of agonist-mediated calcium entry by calmodulin antagonists and by the Ca2+/calmodulin kinase II inhibitor KN-62. Studies with thyroid FRTL-5 cells.
    The Journal of endocrinology, 1996, Volume: 148, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Barium; Biological Transport; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calcium-Transporting ATPases; Calmodulin; Cell Line; Depression, Chemical; Fluphenazine; Imidazoles; Isoquinolines; Membrane Potentials; Phenoxybenzamine; Piperazines; Rats; Sulfonamides; Terpenes; Thapsigargin; Thyroid Gland

1996
D2 dopamine antisense RNA expression vector, unlike haloperidol, produces long-term inhibition of D2 dopamine-mediated behaviors without causing Up-regulation of D2 dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Catalepsy; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Tolerance; Fluphenazine; Genetic Vectors; Grooming; Haloperidol; Male; Mice; Quinpirole; Receptors, Dopamine D2; RNA, Antisense; Stereotyped Behavior; Up-Regulation

1998
Calmodulin inhibition contributes to sensitize TRAIL-induced apoptosis in human lung cancer H1299 cells.
    Biochemistry and cell biology = Biochimie et biologie cellulaire, 2009, Volume: 87, Issue:6

    Topics: Apoptosis; Calmodulin; CASP8 and FADD-Like Apoptosis Regulating Protein; Caspases; Cell Line, Tumor; Enzyme Activation; Fluphenazine; Humans; Lung Neoplasms; Molecular Structure; Proto-Oncogene Proteins c-akt; RNA, Small Interfering; TNF-Related Apoptosis-Inducing Ligand

2009
Stimulation of neuronal KATP channels by cGMP-dependent protein kinase: involvement of ROS and 5-hydroxydecanoate-sensitive factors in signal transduction.
    American journal of physiology. Cell physiology, 2010, Volume: 298, Issue:4

    Topics: Animals; Anti-Arrhythmia Agents; Catalase; Cell Line; Cricetinae; Cricetulus; Cyclic GMP-Dependent Protein Kinases; Decanoic Acids; Enzyme Activation; Fluphenazine; Glycine; Humans; Hydrogen Peroxide; Hydroxy Acids; KATP Channels; Mice; Neurons; Nitric Oxide Donors; Oxidants; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Potassium Channels, Inwardly Rectifying; Purinones; Reactive Oxygen Species; Signal Transduction; Sulfhydryl Compounds

2010