flunitrazepam and triazoles

flunitrazepam has been researched along with triazoles in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19903 (18.75)18.7374
1990's12 (75.00)18.2507
2000's1 (6.25)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beer, B; Benson, DI; Klepner, CA; Lippa, AS; Sano, MC1
Barbaz, BS; Bernard, PS; Braunwalder, AF; Cash, WD; Francis, JE; Friedmann, RC; Hyun, JL; Loo, PS; Lovell, RA; Mazzenga, GC1
Kabuto, M; Namura, I; Saitoh, Y1
Beer, B; Lippa, AS; Meyerson, LR1
Catarzi, D; Cecchi, L; Colotta, V; Giusti, L; Lucacchini, A; Martini, C; Valle, G1
Catarzi, D; Cecchi, L; Colotta, V; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C; Melani, F2
Bain, C; Wafford, KA; Whiting, PJ; Wingrove, PB1
Biagi, G; Giorgi, I; Livi, O; Lucacchini, A; Martini, C; Scartoni, V1
Ambrogi, V; Giusti, L; Grandolini, G; Lucacchini, A; Martini, C; Perioli, L1
Barton, JM; Olson, MS; Svetlov, SI1
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G1
Friend, JM; Gee, KW; Xue, BG1
Braun, D; Chmielewski, PA; Kane, JM; Miller, JA1
Simmonds, MA; Zhong, Y1
Bostwick, R; Chen, T; Huston, J; Knappenberger, K; Liu, J; Norris, T; Wood, M1

Reviews

1 review(s) available for flunitrazepam and triazoles

ArticleYear
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
    Life sciences, 1982, Oct-04, Volume: 31, Issue:14

    Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles

1982

Other Studies

15 other study(ies) available for flunitrazepam and triazoles

ArticleYear
Resolution of two biochemically and pharmacologically distinct benzodiazepine receptors.
    Pharmacology, biochemistry, and behavior, 1979, Volume: 11, Issue:4

    Topics: Animals; Benzodiazepines; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Membranes; Rats; Receptors, Drug; Synaptosomes; Triazoles

1979
Synthesis and benzodiazepine binding activity of a series of novel [1,2,4]triazolo[1,5-c]quinazolin-5(6H)-ones.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Indicators and Reagents; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Triazoles

1991
Nocturnal enhancement of plasma melatonin could be suppressed by benzodiazepines in humans.
    Endocrinologia japonica, 1986, Volume: 33, Issue:3

    Topics: Adult; Benzodiazepines; Circadian Rhythm; Flunitrazepam; Growth Hormone; Humans; Male; Melatonin; Prolactin; Sleep; Triazoles

1986
Tricyclic heteroaromatic systems. 2-Phenyl-1,2,4-triazolo[1,5-c][1,3]benzoxazin-5-one: a novel benzodiazepine receptor ligand.
    Farmaco (Societa chimica italiana : 1989), 1994, Volume: 49, Issue:2

    Topics: Animals; Benzoxazines; Binding, Competitive; Brain; Cattle; Crystallography, X-Ray; Flunitrazepam; In Vitro Techniques; Ligands; Magnetic Resonance Spectroscopy; Oxazines; Receptors, GABA-A; Triazoles

1994
Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor.
    Journal of medicinal chemistry, 1994, Sep-02, Volume: 37, Issue:18

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Flunitrazepam; Imidazoles; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Structure-Activity Relationship; Triazoles

1994
The modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunit.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, May-10, Volume: 91, Issue:10

    Topics: Allosteric Site; Amino Acid Sequence; Animals; Anticonvulsants; Base Sequence; DNA Primers; DNA, Complementary; Dose-Response Relationship, Drug; Female; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Macromolecular Substances; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Point Mutation; Polymerase Chain Reaction; Receptors, GABA-A; Recombinant Fusion Proteins; Triazoles; Xenopus

1994
Tricyclic heteroaromatic systems 1,2,4-triazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Triazoles

1993
Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives.
    Journal of pharmaceutical sciences, 1993, Volume: 82, Issue:9

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; GABA-A Receptor Antagonists; Hydrogen Bonding; In Vitro Techniques; Receptors, GABA-A; Triazoles

1993
Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. VII. Synthesis and inhibition of benzodiazepine receptor binding of some 4,5-dihydro-tetrazolo[5,1-d]-1,5-benzothiazepines and 5-phenyl-s-triazolo[3,4-d]-1,5-benzothiazepines.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:5

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Flunitrazepam; Receptors, GABA-A; Structure-Activity Relationship; Thiazepines; Triazoles

1993
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
    Life sciences, 1996, Volume: 58, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium

1996
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
    Biochemical pharmacology, 1996, Jun-14, Volume: 51, Issue:11

    Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium

1996
Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Drug Interactions; Flunitrazepam; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA; Triazoles

1996
The enhancement of muscimol-stimulated 36C1 influx by the antispastic 5-aryl-3-(alkylsulfonyl)-4H-1,2,4-triazole (MDL 27,531) in rat brain membrane vesicles.
    Neuroscience letters, 1995, Dec-08, Volume: 201, Issue:2

    Topics: Animals; Brain Chemistry; Chloride Channels; Chlorine; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles

1995
Interactions between loreclezole, chlormethiazole and pentobarbitone at GABA(A) receptors: functional and binding studies.
    British journal of pharmacology, 1997, Volume: 121, Issue:7

    Topics: Animals; Anticonvulsants; Bicuculline; Chlormethiazole; Flunitrazepam; In Vitro Techniques; Male; Medulla Oblongata; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; Triazoles

1997
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
    Assay and drug development technologies, 2008, Volume: 6, Issue:6

    Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium

2008