flunitrazepam and pk 11195

flunitrazepam has been researched along with pk 11195 in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199012 (30.77)18.7374
1990's19 (48.72)18.2507
2000's5 (12.82)29.6817
2010's2 (5.13)24.3611
2020's1 (2.56)2.80

Authors

AuthorsStudies
Bendinelli, S; Castellano, S; Cosconati, S; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; Martini, C; Milite, C; Novellino, E; Pugliesi, I; Rizzetto, E; Sbardella, G; Stefancich, G; Taliani, S1
Baglini, E; Barresi, E; Costa, B; Da Pozzo, E; Da Settimo, F; Martini, C; Robello, M; Salerno, S; Taliani, S1
Gavish, M; Katz, Y; Weizman, A; Weizman, R1
Brodie, MJ; Larkin, JG; Scobie, G; Thompson, GG1
Amiri, Z; Burstein, O; Edoute, Y; Gavish, M; Katz, Y; Lochner, A; Weizman, R1
De Luca, C; De Medici, D; Massotti, M1
Becker, DP; Black, KL; Ikezaki, K; Payne, BA; Santori, EM; Smith, ML; Toga, AW1
Calandra, RS; Calvo, DJ; Medina, JH; Ritta, MN1
Gavish, M; Katz, Y1
Gavish, M; Weizman, R1
Black, KL; Ikezaki, K; Toga, AW1
Fares, F; Gavish, M; Pick, CG; Weizman, A; Yanai, J1
Arbilla, S; Langer, SZ1
Ciliax, BJ; Mancini, WR; Olson, JM; Young, AB1
Becker, D; Gavish, M; Tanne, Z; Weizman, R1
Gavish, M; Okun, F; Weizman, A; Youdim, MB1
Ciliax, BJ; McKeever, P; Penney, JB; Starosta-Rubinstein, S; Young, AB1
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B1
Junck, L; Mancini, WR; Olson, JM; Penney, JB; Young, AB1
Haumont, J; Lenfant, M; Zavala, F1
Cascio, C; Guarneri, P; Guarneri, R; Papadopoulos, V; Piccoli, F1
Niles, LP; Tenn, CC1
Dalezios, Y; Matsokis, N; Valcana, T1
Ruggieri, MR; Smyth, RJ; Uhlman, EJ1
Beauchemin, V; Dennis, T; Lavoie, N1
Alenfall, J; Batra, S1
Amiri, Z; Bar-Ami, S; Fares, F; Gavish, M; Weizman, A1
Giannaccini, G; Lucacchini, A; Martini, C; Piccolino, M; Strettoi, E1
Nakamoto, Y; Shiotani, T; Watabe, S; Yoshii, M1
Anzini, M; Basile, AS; Bruni, G; Cappelli, A; Giorgi, G; Langer, T; Romeo, MR; Vomero, S1
Bessler, H; Caspi, B; Gavish, M; Rehavi, M; Weizman, A1
Chaki, S; Nagamine, M; Nakazato, A; Ogawa, S; Okubo, T; Okuyama, S; Suzuki, Y; Tomisawa, K; Yoshikawa, R1
Bono, F; Herbert, JM; Lamarche, I; Le Fur, G; Prabonnaud, V1
Biggio, G; Busonero, F; Mascia, MP; Mostallino, MC; Pisu, MG; Talani, G1
Biggio, G; Chiarelotto, G; Dall'Acqua, S; Ferlin, MG; Maciocco, E; Mascia, MP; Pisu, MG1
Hajós, G; Kardos, J; Nyikos, L; Riedl, Z; Szárics, E1
Lopes, DV; Mendonça-Silva, DL; Noël, F; Thibaut, JP1
Ducroc, R; Lacapere, JJ; Ostuni, MA; Papadopoulos, V; Péranzi, G; Tonon, MC1
Elbim, C; Fasseu, M; Issop, L; Lacapere, JJ; Ostuni, MA; Papadopoulos, V; Péranzi, G; Walker, F1

Reviews

1 review(s) available for flunitrazepam and pk 11195

ArticleYear
An update into the medicinal chemistry of translocator protein (TSPO) ligands.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Anticonvulsants; Apoptosis; Benzimidazoles; Benzodiazepines; Cell Proliferation; Diazepam; Humans; Imidazoles; Membrane Potential, Mitochondrial; Mitochondria; Mitochondrial ADP, ATP Translocases; Mitochondrial Membranes; Mitochondrial Permeability Transition Pore; Oxidative Stress; Protein Binding; Pyridines; Quinolines; Receptors, GABA; Structure-Activity Relationship; Voltage-Dependent Anion Channels

2021

Other Studies

38 other study(ies) available for flunitrazepam and pk 11195

ArticleYear
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
    Journal of medicinal chemistry, 2012, May-10, Volume: 55, Issue:9

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cell Line, Tumor; Cell Survival; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship

2012
Disulfiram and diethyldithiocarbamate are competitive inhibitors at the peripheral benzodiazepine receptor.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Disulfiram; Ditiocarb; Flunitrazepam; Isoquinolines; Kidney; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
Central and peripheral benzodiazepine receptors in rat brain and platelets: effects of treatment with diazepam and clobazam.
    Seizure, 1992, Volume: 1, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Blood Platelets; Brain; Clobazam; Diazepam; Drug Tolerance; Flunitrazepam; Injections, Intraperitoneal; Isoquinolines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1992
Testosterone and cyproterone acetate modulate peripheral but not central benzodiazepine receptors in rats.
    Brain research, 1991, Jul-05, Volume: 553, Issue:1

    Topics: Androgen Antagonists; Animals; Central Nervous System; Cyproterone; Cyproterone Acetate; Down-Regulation; Flunitrazepam; Hypophysectomy; Isoquinolines; Male; Peripheral Nerves; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testosterone; Up-Regulation

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Three-dimensional comparison of peripheral benzodiazepine binding and histological findings in rat brain tumor.
    Neurosurgery, 1990, Volume: 27, Issue:1

    Topics: Animals; Brain Neoplasms; Female; Flunitrazepam; Glioma; Isoquinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tomography, Emission-Computed

1990
Peripheral-type benzodiazepine receptors are highly concentrated in mitochondrial membranes of rat testicular interstitial cells.
    Neuroendocrinology, 1990, Volume: 52, Issue:4

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Diazepam; Flunitrazepam; Intracellular Membranes; Isoquinolines; Kinetics; Leydig Cells; Male; Mitochondria; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Laudanosine does not displace receptor-specific ligands from the benzodiazepinergic or muscarinic receptors.
    Anesthesiology, 1989, Volume: 70, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Flunitrazepam; Isoquinolines; Kidney; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Muscarinic; Seizures

1989
Effects of chronic chlorpromazine treatment on peripheral benzodiazepine binding sites in heart, kidney, and cerebral cortex of rats.
    Journal of neurochemistry, 1989, Volume: 52, Issue:5

    Topics: Animals; Cerebral Cortex; Chlorpromazine; Flunitrazepam; Isoquinolines; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Imaging of brain tumors using peripheral benzodiazepine receptor ligands.
    Journal of neurosurgery, 1989, Volume: 71, Issue:1

    Topics: Animals; Autoradiography; Brain Neoplasms; Clonazepam; Female; Flunitrazepam; Glioma; Image Processing, Computer-Assisted; Isoquinolines; Ligands; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Chronic phenobarbital administration affects GABA and benzodiazepine receptors in the brain and periphery.
    European journal of pharmacology, 1989, Oct-10, Volume: 169, Issue:2-3

    Topics: Animals; Brain Chemistry; Flunitrazepam; Hippocampus; In Vitro Techniques; Isoquinolines; Kidney; Male; Membranes; Mice; Muscimol; Myocardium; Olfactory Bulb; Peripheral Nerves; Phenobarbital; Receptors, GABA-A

1989
Imidazopyridines as a tool for the characterization of benzodiazepine receptors: a proposal for a pharmacological classification as omega receptor subtypes.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Brain Chemistry; Flunitrazepam; GABA-A Receptor Antagonists; Imidazoles; In Vitro Techniques; Isoquinolines; Kidney; Ligands; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem

1988
Presence of peripheral-type benzodiazepine binding sites on human erythrocyte membranes.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: Benzodiazepinones; Clonazepam; Convulsants; Erythrocyte Membrane; Flunitrazepam; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Monoamine Oxidase; Receptors, GABA-A

1988
Effect of chronic haloperidol treatment on peripheral benzodiazepine binding sites in cerebral cortex of rats.
    Journal of neural transmission, 1988, Volume: 74, Issue:2

    Topics: Animals; Cerebral Cortex; Flunitrazepam; Haloperidol; Heart; Isoquinolines; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Modulatory effects of thyroxine treatment on central and peripheral benzodiazepine receptors in the rat.
    Journal of neurochemistry, 1986, Volume: 47, Issue:4

    Topics: Animals; Cerebral Cortex; Flunitrazepam; Hyperthyroidism; Isoquinolines; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Thyroxine

1986
Imaging of a glioma using peripheral benzodiazepine receptor ligands.
    Proceedings of the National Academy of Sciences of the United States of America, 1987, Volume: 84, Issue:3

    Topics: Adrenal Gland Neoplasms; Animals; Flunitrazepam; Glioma; Humans; Isoquinolines; Kidney; Mice; Mice, Nude; Neoplasm Transplantation; Neuroblastoma; Pheochromocytoma; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, GABA-A; Transplantation, Heterologous; Tritium

1987
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
    Life sciences, 1987, Apr-13, Volume: 40, Issue:15

    Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A

1987
Isoquinoline and peripheral-type benzodiazepine binding in gliomas: implications for diagnostic imaging.
    Cancer research, 1988, Oct-15, Volume: 48, Issue:20

    Topics: Benzodiazepines; Benzodiazepinones; Brain Neoplasms; Cells, Cultured; Flunitrazepam; Glioma; Humans; Isoquinolines; Kinetics; Tomography, Emission-Computed

1988
Interaction of benzodiazepines with mouse macrophages.
    European journal of pharmacology, 1984, Nov-27, Volume: 106, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antibody Formation; Female; Flunitrazepam; In Vitro Techniques; Isoquinolines; Macrophages; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Receptors, GABA-A

1984
gamma-Aminobutyric acid type A/benzodiazepine receptors regulate rat retina neurosteroidogenesis.
    Brain research, 1995, Jun-12, Volume: 683, Issue:1

    Topics: Animals; Flunitrazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Isoquinolines; Kinetics; Male; Neuroglia; Neurotransmitter Agents; Pregnenolone; Rats; Rats, Wistar; Receptors, GABA-A; Retina; Steroids; Synaptic Transmission

1995
Central-type benzodiazepine receptors mediate the antidopaminergic effect of clonazepam and melatonin in 6-hydroxydopamine lesioned rats: involvement of a GABAergic mechanism.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Bicuculline; Clonazepam; Corpus Striatum; Dopamine Agonists; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Isoquinolines; Male; Melatonin; Oxidopamine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1995
Interaction between [3H]flunitrazepam and [3H]GABA binding in the cerebellum of reeler mice.
    Neurochemistry international, 1995, Volume: 26, Issue:1

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cerebellum; Flunitrazepam; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Isoquinolines; Membrane Proteins; Membrane Transport Proteins; Mice; Mice, Neurologic Mutants; Models, Neurological; Nerve Tissue Proteins; Organic Anion Transporters; Protein Binding; Receptors, GABA-A; Up-Regulation

1995
Identification and characterization of a high-affinity peripheral-type benzodiazepine receptor in rabbit urinary bladder.
    The Journal of urology, 1994, Volume: 151, Issue:4

    Topics: Animals; Flumazenil; Flunitrazepam; GABA-A Receptor Antagonists; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth; Rabbits; Receptors, GABA-A; Urinary Bladder

1994
Quantitative autoradiographic studies of the effects of bilateral olfactory bulbectomy in the rat brain: central- and peripheral-type benzodiazepine receptors.
    Neuroscience, 1994, Volume: 58, Issue:3

    Topics: Animals; Autoradiography; Behavior, Animal; Brain Chemistry; Flumazenil; Flunitrazepam; Isoquinolines; Male; Olfactory Bulb; Peripheral Nervous System; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1994
Characterization of peripheral benzodiazepine receptors in rat prostatic adenocarcinoma.
    The Prostate, 1994, Volume: 24, Issue:5

    Topics: Adenocarcinoma; Animals; Benzodiazepinones; Binding, Competitive; Diazepam; Flunitrazepam; Isoquinolines; Male; Mesoporphyrins; Microsomes; Mitochondria; Neoplasm Transplantation; Prostatic Neoplasms; Rats; Receptors, GABA-A

1994
Long-term testosterone or diethylstilbestrol treatment affects gamma-aminobutyric acid and central-type benzodiazepine receptors but not peripheral-type benzodiazepine receptors in the female rat brain.
    Neuroendocrinology, 1993, Volume: 57, Issue:6

    Topics: Animals; Brain; Cerebellum; Diethylstilbestrol; Female; Flunitrazepam; In Vitro Techniques; Isoquinolines; Membranes; Muscimol; Parietal Lobe; Peripheral Nervous System; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Testosterone

1993
The peripheral-type benzodiazepine receptor ligands [3H]Ro 5-4864 and [3H]PK 11195 bind to the retina of rabbit, but not of turtle.
    Journal of neurochemistry, 1993, Volume: 61, Issue:4

    Topics: Animals; Benzodiazepinones; Flunitrazepam; Isoquinolines; Ligands; Rabbits; Receptors, GABA-A; Retina; Tritium; Turtles

1993
Peripheral-type benzodiazepine receptors in association with epileptic seizures in EL mice.
    Brain research, 1996, Apr-22, Volume: 717, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Cell Fractionation; Convulsants; Epilepsy; Flunitrazepam; GABA-A Receptor Agonists; Isoquinolines; Membrane Proteins; Mice; Mice, Mutant Strains; Mitochondria; Pentylenetetrazole; Prosencephalon; Receptors, GABA-A; Tritium

1996
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.
    Journal of medicinal chemistry, 1996, Oct-11, Volume: 39, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Drug Design; Flunitrazepam; Imidazoles; Isoquinolines; Models, Molecular; Protein Conformation; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship

1996
Significant inhibition of spontaneous IgA secretion by selective peripheral-type benzodiazepine receptor ligands.
    Clinical neuropharmacology, 1997, Volume: 20, Issue:3

    Topics: Anti-Anxiety Agents; Antibody-Producing Cells; B-Lymphocytes; Clonazepam; Diazepam; Flunitrazepam; GABA-A Receptor Antagonists; Humans; Immunoglobulin A; Immunoglobulin G; Immunoglobulin M; Isoquinolines; Lymphocyte Activation

1997
Neuropharmacological profile of peripheral benzodiazepine receptor agonists, DAA1097 and DAA1106.
    Life sciences, 1999, Volume: 64, Issue:16

    Topics: Acetamides; Anesthesia; Animals; Anti-Anxiety Agents; Benzodiazepinones; Brain; Buspirone; Cell Membrane; Diazepam; Exploratory Behavior; Flunitrazepam; GABA Modulators; GABA-A Receptor Agonists; Hexobarbital; Isoquinolines; Male; Mice; Mice, Inbred ICR; Mitochondria; Motor Activity; Phenyl Ethers

1999
Peripheral benzodiazepine receptor agonists exhibit potent antiapoptotic activities.
    Biochemical and biophysical research communications, 1999, Nov-19, Volume: 265, Issue:2

    Topics: Apoptosis; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Isoquinolines; Jurkat Cells; Kinetics; Ligands; Receptors, GABA-A; Transfection; Tumor Necrosis Factor-alpha; U937 Cells

1999
Inhibition by miltirone of up-regulation of GABAA receptor alpha4 subunit mRNA by ethanol withdrawal in hippocampal neurons.
    European journal of pharmacology, 2004, Jun-28, Volume: 494, Issue:2-3

    Topics: Animals; Binding, Competitive; Cells, Cultured; Central Nervous System Depressants; Cerebral Cortex; DNA, Complementary; Electrophysiology; Ethanol; Flunitrazepam; GABA Antagonists; Hippocampus; Isoquinolines; Male; Neurons; Oocytes; Patch-Clamp Techniques; Phenanthrenes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA Probes; RNA, Messenger; Substance Withdrawal Syndrome; Tranquilizing Agents; Xenopus laevis

2004
Novel anellated pyrazoloquinolin-3-ones: synthesis and in vitro BZR activity.
    Bioorganic & medicinal chemistry, 2005, May-16, Volume: 13, Issue:10

    Topics: Animals; Brain; Female; Flunitrazepam; GABA Modulators; Humans; Isoquinolines; Male; Oocytes; Pyrazoles; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; Structure-Activity Relationship; Xenopus laevis

2005
Interaction of novel condensed triazine derivatives with central and peripheral type benzodiazepine receptors: synthesis, in vitro pharmacology and modelling.
    European journal of medicinal chemistry, 2006, Volume: 41, Issue:4

    Topics: Animals; Binding, Competitive; Central Nervous System; Cerebral Cortex; Chromatography, Thin Layer; Flunitrazepam; GABA Modulators; In Vitro Techniques; Isoquinolines; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Peripheral Nervous System; Point Mutation; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA-A; Spectrophotometry, Infrared; Structure-Activity Relationship; Synaptic Membranes; Triazines

2006
Characterization of two classes of benzodiazepine binding sites in Schistosoma mansoni.
    Parasitology, 2007, Volume: 134, Issue:Pt 7

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Clonazepam; Diazepam; Flunitrazepam; GABA Agonists; GABA Modulators; Inhibitory Concentration 50; Isoquinolines; Ligands; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Schistosoma mansoni; Synaptosomes; Temperature; Time Factors; Tritium; Zolpidem

2007
Translocator protein (18 kDa) ligand PK 11195 induces transient mitochondrial Ca2+ release leading to transepithelial Cl- secretion in HT-29 human colon cancer cells.
    Biology of the cell, 2007, Volume: 99, Issue:11

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Calcium; Cell Line, Tumor; Chlorides; Colonic Neoplasms; Cyclosporine; Enzyme Inhibitors; Flunitrazepam; GABA Modulators; Gene Expression Regulation, Neoplastic; Humans; Isoquinolines; Ligands; Mitochondria; Mitochondrial Membranes; Mitochondrial Proteins; Neoplasm Proteins; Nitrobenzoates; Receptors, GABA; Sodium-Potassium-Chloride Symporters

2007
Overexpression of translocator protein in inflammatory bowel disease: potential diagnostic and treatment value.
    Inflammatory bowel diseases, 2010, Volume: 16, Issue:9

    Topics: Animals; Antineoplastic Agents; Benzodiazepinones; Carrier Proteins; Case-Control Studies; Colitis; Colon; Colonic Neoplasms; Cytokines; Dextran Sulfate; Enterocytes; Flunitrazepam; GABA Modulators; Humans; Hypolipidemic Agents; Immunoenzyme Techniques; Inflammatory Bowel Diseases; Isoquinolines; Male; Mitochondria; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2010