flunitrazepam and picrotoxin

flunitrazepam has been researched along with picrotoxin in 43 studies

Research

Studies (43)

TimeframeStudies, this research(%)All Research%
pre-199018 (41.86)18.7374
1990's17 (39.53)18.2507
2000's6 (13.95)29.6817
2010's2 (4.65)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Haefely, W; Polc, P1
Karobath, M; Supavilai, P1
Bertolini, A; Marrama, D; Sandrini, M; Vergoni, AV1
Allan, AM; Draski, LJ; Mayes, GG1
David, JA; Pinnock, RD; Sattelle, DB; Wafford, KA1
Ho, IK; Ito, Y; Lim, DK; Nabeshima, T1
Bowen, DM; Cross, AJ; Francis, PT; Green, AR; Robinson, TN; Stirling, JM1
Chang, YF; Gao, XM1
Ticku, MK1
Koe, BK; Kondratas, E; Russo, LL1
Kempner, ES; Paul, SM; Schwartz, RD; Skolnick, P; Thomas, JW1
Chweh, AY; Swinyard, EA; Ulloque, RA; Wolf, HH1
Maĭmets, MO; Nurk, AM; Riago, LK; Soosaar, AKh; Vasar, EE1
Crabbe, JC; Feller, DJ; Harris, RA1
Drexler, G; Sieghart, W1
Hamon, M; Hery, F; Jobert, A; Montastruc, JL; Soubrie, P; Thiebot, MH1
Drexler, G; Karobath, M; Supavilai, P1
Collins, JF; Karobath, M; Mannonen, A; Supavilai, P1
Saederup, E; Squires, RF1
Olsen, RW; Stephenson, FA1
Bormann, J; Feigenspan, A1
Nabeshima, A; Saito, T; Takahata, N; Toki, S1
Bormann, J; Feigenspan, A; Wässle, H1
Boksa, P; Chaudieu, I; Quirion, R; St-Pierre, JA1
Belelli, D; Chen, R; Lambert, JJ; Lan, NC; Peters, JA; Reyes, A1
Kikuchi de Beltrán, K; Kobayashi, M; Koshikawa, N; Miwa, Y; Stephenson, JD1
Dunn, SM; Thuynsma, RP1
Albin, RL; Caspary, DM; Milbrandt, JC; Turgeon, SM1
Davies, PA; Hales, TG; Hanna, MC; Kirkness, EF1
Belachew, S; Coucke, P; Goffin, F; Lefebvre, PP; Malgrange, B; Moonen, G; Rigo, JM; Van de Water, TR; Xhauflaire, G1
Buckingham, SD; Rauh, J; Sattelle, DB; Schnee, M1
Dunwiddie, TV; Proctor, WR; Soldo, BL1
Hartmann, J; Kettenmann, H; Labrakakis, C; Patt, S1
Higashi, H; Nagata, K; Park, JS; Yoshimura, M1
Ai, J; Kahnberg, P; Nielsen, M; Saederup, E; Squires, RF; Sterner, O; Witt, MR1
Findlay, GS; Harris, RA; Harrison, NL; Ueno, S2
Baufreton, J; Bioulac, B; Dovero, S; Dufy, B; Garret, M; Taupignon, A1
Baur, R; Senn, M; Séquin, U; Sigel, E; Simmen, U1
Jembrek, MJ; Pericić, D; Strac, DS; Vlainić, J1
Ebert, B; Klaerke, D; Søgaard, R; Werge, T1
Andreatini, R; Baretta, IP; Chioca, LR; Ferreira, J; Ferro, MM; Losso, EM; Oliveira, SM; Silva, CR1
Ferreri, MC; Gravielle, MC; Gutiérrez, ML1

Reviews

1 review(s) available for flunitrazepam and picrotoxin

ArticleYear
Biochemical pharmacology of the GABA receptor-ionophore protein complex.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Animals; Brain; Chlorides; Flunitrazepam; Humans; Ion Channels; Ionophores; Kinetics; Muscimol; Nerve Tissue Proteins; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sesterterpenes

1983

Other Studies

42 other study(ies) available for flunitrazepam and picrotoxin

ArticleYear
Effects of two benzodiazepines, phenobarbitone, and baclofen on synaptic transmission in the cat cuneate nucleus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 294, Issue:2

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Cats; Diazepam; Drug Interactions; Evoked Potentials; Flunitrazepam; Glutamate Decarboxylase; Medulla Oblongata; Neural Inhibition; Phenobarbital; Picrotoxin; Propionates; Semicarbazides; Synapses; Synaptic Transmission

1976
Stimulation of benzodiazepine receptor binding by SQ 20009 is chloride-dependent and picrotoxin-sensitive.
    European journal of pharmacology, 1979, Nov-23, Volume: 60, Issue:1

    Topics: Animals; Benzodiazepines; Brain; Chlorides; Etazolate; Flunitrazepam; In Vitro Techniques; Membranes; Nicotinic Acids; Picrotoxin; Rats; Receptors, Drug; Sodium Chloride; Stimulation, Chemical

1979
Repeated administration of triiodothyronine enhances the susceptibility of rats to isoniazid- and picrotoxin-induced seizures.
    Life sciences, 1992, Volume: 51, Issue:10

    Topics: Animals; Binding Sites; Cerebral Cortex; Flunitrazepam; Hippocampus; Hyperthyroidism; Isoniazid; Male; Picrotoxin; Rats; Rats, Inbred Strains; Seizures; Triiodothyronine

1992
gamma-Aminobutyric acid-activated chloride channels in rats selectively bred for differential acute sensitivity to alcohol.
    Alcoholism, clinical and experimental research, 1991, Volume: 15, Issue:2

    Topics: Alcohol Drinking; Animals; Chloride Channels; Diazepam; Female; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Proteins; Muscimol; Pentobarbital; Phenobarbital; Phenotype; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Selection, Genetic

1991
GABA receptors on the cell-body membrane of an identified insect motor neuron.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1988, Jan-22, Volume: 232, Issue:1269

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Chlorides; Cockroaches; Dibenzazepines; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Nipecotic Acids; Periplaneta; Picrotoxin; Receptors, GABA-A

1988
Effects of picrotoxin treatment on GABAA receptor supramolecular complexes in rat brain.
    Journal of neurochemistry, 1989, Volume: 52, Issue:4

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Flunitrazepam; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Tissue Distribution

1989
The modulation by chlormethiazole of the GABAA-receptor complex in rat brain.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Animals; Baclofen; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlormethiazole; CLC-2 Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Picrotoxin; Rats; Receptors, GABA-A

1989
Enhancement of benzodiazepine receptor binding by L-lysine is chloride-dependent and due to increase in binding affinity.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: Animals; Cattle; Chlorides; Flunitrazepam; In Vitro Techniques; Kinetics; Lysine; Pentylenetetrazole; Picrotoxin; Receptors, GABA-A; Sesterterpenes; Synaptic Membranes

1989
Behavioral and functional studies indicate a role for GABAAergic transmission in the actions of ethanol.
    Alcohol and alcoholism (Oxford, Oxfordshire). Supplement, 1987, Volume: 1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Ethanol; Flunitrazepam; Male; Mice; Mice, Inbred C57BL; Picrotoxin; Rats; Receptors, GABA-A; Seizures; Spinal Cord

1987
[3H]Ro 15-1788 binding to benzodiazepine receptors in mouse brain in vivo: marked enhancement by GABA agonists and other CNS drugs.
    European journal of pharmacology, 1987, Oct-27, Volume: 142, Issue:3

    Topics: Animals; Antipsychotic Agents; Barbiturates; Brain; Buspirone; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intravenous; Male; Mice; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasodilator Agents

1987
Radiation inactivation studies of the benzodiazepine/gamma-aminobutyric acid/chloride ionophore receptor complex.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Flumazenil; Flunitrazepam; Ionophores; Male; Molecular Weight; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Effect of picrotoxinin on benzodiazepine receptor binding.
    Neurochemical research, 1985, Volume: 10, Issue:7

    Topics: Animals; Brain; Cerebellum; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Membranes; Mice; Pentobarbital; Picrotoxin; Receptors, GABA-A; Sesterterpenes

1985
[Modulating effect of cerulein on benzodiazepine receptors].
    Biulleten' eksperimental'noi biologii i meditsiny, 1985, Volume: 100, Issue:12

    Topics: Animals; Brain; Ceruletide; Dose-Response Relationship, Drug; Drug Interactions; Flunitrazepam; Male; Mice; Picrotoxin; Proglumide; Reaction Time; Receptors, GABA-A; Seizures

1985
Differences in GABA activity between ethanol withdrawal seizure prone and resistant mice.
    European journal of pharmacology, 1988, Nov-22, Volume: 157, Issue:2-3

    Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Ethanol; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Picrotoxin; Seizures; Substance Withdrawal Syndrome

1988
Evidence for association of a high affinity avermectin binding site with the benzodiazepine receptor.
    European journal of pharmacology, 1984, Jun-01, Volume: 101, Issue:3-4

    Topics: Animals; Binding Sites; Binding, Competitive; Cell Membrane; Cerebellar Cortex; Chlorides; Flunitrazepam; In Vitro Techniques; Ivermectin; Lactones; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, GABA-A; Sesterterpenes; Temperature

1984
Decreased convulsant potency of picrotoxin and pentetrazol and enhanced [3H]flunitrazepam cortical binding following stressful manipulations in rats.
    Brain research, 1980, May-12, Volume: 189, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Diazepam; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Isoniazid; Male; Muscimol; Pentylenetetrazole; Picrotoxin; Rats; Seizures; Stress, Physiological; Thiosemicarbazones

1980
Modulation by picrotoxin and IPTBO of 3H-flunitrazepam binding to the GABA/benzodiazepine receptor complex of rat cerebellum.
    Life sciences, 1981, Jan-19, Volume: 28, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membranes; Organophosphorus Compounds; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Temperature

1981
Anion-dependent modulation of [3H]muscimol binding and of GABA-stimulated [3H]flunitrazepam binding by picrotoxin and related CNS convulsants.
    European journal of pharmacology, 1982, Jul-30, Volume: 81, Issue:4

    Topics: Animals; Anions; Anti-Anxiety Agents; Cerebral Cortex; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Oxazoles; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Strychnine; Tubocurarine

1982
gamma-aminobutyric acid receptors modulate cation binding sites coupled to independent benzodiazepine, picrotoxin, and anion binding sites.
    Molecular pharmacology, 1982, Volume: 22, Issue:2

    Topics: Animals; Binding Sites; Brain; Calcium Chloride; Electrolytes; Flunitrazepam; In Vitro Techniques; Isoxazoles; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Sodium Chloride

1982
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction

1994
[Changes in GABAA/benzodiazepine receptor complex function in the pentobarbital-dependent rat. II: Strain differences between Lewis and Wistar-Kyoto rats].
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1995, Volume: 15, Issue:4

    Topics: Animals; Bicuculline; Brain; Chlorine; Ethanol; Female; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Lew; Rats, Inbred WKY; Receptors, GABA-A; Substance-Related Disorders

1995
Pharmacology of GABA receptor Cl- channels in rat retinal bipolar cells.
    Nature, 1993, Jan-14, Volume: 361, Issue:6408

    Topics: Animals; Animals, Newborn; Bicuculline; Cells, Cultured; Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Membrane Potentials; Membrane Proteins; Neurons; Pentobarbital; Photoreceptor Cells; Picrotoxin; Pregnanediones; Rats; Receptors, GABA-A; Sesterterpenes; Strychnine

1993
GABAA receptor-mediated inhibition of N-methyl-D-aspartate-evoked [3H]dopamine release from mesencephalic cell cultures.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Baclofen; Cells, Cultured; Dopamine; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kainic Acid; Mesencephalon; Muscimol; N-Methylaspartate; Picrotoxin; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA; Ventral Tegmental Area

1994
Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Jun-21, Volume: 91, Issue:13

    Topics: Amino Acid Sequence; Animals; Base Sequence; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; Convulsants; DNA Primers; DNA, Complementary; Drosophila melanogaster; Female; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression; Macromolecular Substances; Molecular Sequence Data; Muscimol; Oocytes; Pentobarbital; Picrotoxin; Polymerase Chain Reaction; Receptors, GABA; Receptors, GABA-A; Transcription, Genetic; Xenopus laevis

1994
Further evidence for a functional dorsal-ventral division of the rat striatum: GABAergic involvement in oral movements.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Animals; Apomorphine; Behavior, Animal; Benzamides; Benzazepines; Carbachol; Corpus Striatum; Dopamine; Flunitrazepam; gamma-Aminobutyric Acid; Jaw; Male; Muscimol; N-Methylscopolamine; Picrotoxin; Pilocarpine; Rats; Rats, Sprague-Dawley; Scopolamine Derivatives

1993
Reconstitution of purified GABAA receptors: ligand binding and chloride transporting properties.
    Biochemistry, 1994, Jan-25, Volume: 33, Issue:3

    Topics: Animals; Bicuculline; Biological Transport; Brain Chemistry; Cattle; Chlorides; Chromatography, Affinity; Dose-Response Relationship, Drug; Flow Injection Analysis; Flunitrazepam; Ligands; Liposomes; Membrane Proteins; Muscimol; Picrotoxin; Quinolinium Compounds; Receptors, GABA-A

1994
GABAA receptor binding in the aging rat inferior colliculus.
    Neuroscience, 1996, Volume: 73, Issue:2

    Topics: Aged; Aging; Animals; Autoradiography; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Inferior Colliculi; Ligands; Muscimol; Picrotoxin; Rats; Rats, Inbred F344; Receptors, GABA-A; Tritium

1996
Insensitivity to anaesthetic agents conferred by a class of GABA(A) receptor subunit.
    Nature, 1997, Feb-27, Volume: 385, Issue:6619

    Topics: Amino Acid Sequence; Anesthetics, Intravenous; Animals; Bicuculline; Brain; Cell Line; Consensus Sequence; DNA, Complementary; Flumazenil; Flunitrazepam; GABA Agents; gamma-Aminobutyric Acid; Humans; Molecular Sequence Data; Muscimol; Pentobarbital; Picrotoxin; Pregnanolone; Propofol; Rats; Receptors, GABA-A; Recombinant Proteins; RNA, Messenger; Transfection

1997
Diazepam-insensitive GABAA receptors on postnatal spiral ganglion neurones in culture.
    Neuroreport, 1997, Feb-10, Volume: 8, Issue:3

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Carbolines; Cells, Cultured; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Spiral Ganglion; Zinc

1997
Pharmacology of skeletal muscle GABA-gated chloride channels in the cockroach Periplaneta americana.
    The Journal of experimental biology, 1997, Volume: 200, Issue:Pt 23

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Isonicotinic Acids; Male; Motor Neurons; Muscle, Skeletal; Periplaneta; Picrotoxin; Receptors, GABA; Sesterterpenes

1997
Ethanol selectively enhances the hyperpolarizing component of neocortical neuronal responses to locally applied GABA.
    Brain research, 1998, Aug-03, Volume: 800, Issue:2

    Topics: Animals; Central Nervous System Depressants; Electrophysiology; Ethanol; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neocortex; Neurons; Pentobarbital; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

1998
Functional GABA(A) receptors on human glioma cells.
    The European journal of neuroscience, 1998, Volume: 10, Issue:1

    Topics: Anti-Bacterial Agents; Calcium; Calcium Channel Blockers; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Glioblastoma; Gramicidin; Humans; Membrane Potentials; Muscimol; Oligodendroglioma; Patch-Clamp Techniques; Picrotoxin; Potassium; Receptors, GABA-A; Tumor Cells, Cultured; Verapamil

1998
Bicuculline-resistant, Cl- dependent GABA response in the rat spinal dorsal horn.
    Neuroscience research, 1999, Volume: 33, Issue:4

    Topics: Animals; Bicuculline; Chloride Channels; Evoked Potentials; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Neurons; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Gelatinosa; Thiopental

1999
Honokiol and magnolol increase the number of [3H] muscimol binding sites three-fold in rat forebrain membranes in vitro using a filtration assay, by allosterically increasing the affinities of low-affinity sites.
    Neurochemical research, 1999, Volume: 24, Issue:12

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Binding Sites; Biphenyl Compounds; Cell Membrane; Central Nervous System Depressants; Cerebellum; Diflunisal; Drugs, Chinese Herbal; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Lignans; Muscimol; Picrotoxin; Propofol; Prosencephalon; Rats; Receptors, GABA-A; Tritium

1999
Allosteric modulation in spontaneously active mutant gamma-aminobutyric acid(A) receptors [corrected].
    Neuroscience letters, 2000, Nov-03, Volume: 293, Issue:3

    Topics: Allosteric Regulation; Amino Acid Substitution; Animals; Bicuculline; Cells, Cultured; Female; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Mutagenesis, Site-Directed; Oocytes; Pentobarbital; Picrotoxin; Protein Structure, Tertiary; Receptors, GABA-A; Steroids; Xenopus laevis

2000
Allosteric modulation in spontaneously active mutant gamma-aminobutyric acidA receptors.
    Neuroscience letters, 2001, Jun-01, Volume: 305, Issue:1

    Topics: Allosteric Regulation; Animals; Bicuculline; Electric Conductivity; Female; Flunitrazepam; GABA Antagonists; GABA Modulators; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pregnanolone; Protein Isoforms; Receptors, GABA-A; Xenopus laevis

2001
Activation of GABA(A) receptors in subthalamic neurons in vitro: properties of native receptors and inhibition mechanisms.
    Journal of neurophysiology, 2001, Volume: 86, Issue:1

    Topics: Animals; Bicarbonates; Bicuculline; Chlorides; Diazepam; Electrophysiology; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; Organ Culture Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Subthalamic Nucleus

2001
Novel plant substances acting as beta subunit isoform-selective positive allosteric modulators of GABAA receptors.
    Molecular pharmacology, 2005, Volume: 68, Issue:3

    Topics: Allosteric Regulation; Animals; Araliaceae; Bicuculline; Flumazenil; Flunitrazepam; GABA Modulators; Picrotoxin; Plant Extracts; Receptors, GABA-A; Xenopus laevis

2005
Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Diazepam; Flumazenil; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Protein Subunits; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Transfection; Up-Regulation

2007
Triton X-100 inhibits agonist-induced currents and suppresses benzodiazepine modulation of GABA(A) receptors in Xenopus oocytes.
    Biochimica et biophysica acta, 2009, Volume: 1788, Issue:5

    Topics: Animals; Biophysical Phenomena; Electrophysiological Phenomena; Female; Flunitrazepam; GABA Modulators; GABA-A Receptor Agonists; Humans; In Vitro Techniques; Lipid Bilayers; Octoxynol; Oocytes; Picrotoxin; Receptors, GABA-A; Recombinant Proteins; Surface-Active Agents; Xenopus laevis

2009
Anxiolytic-like effect of lavender essential oil inhalation in mice: participation of serotonergic but not GABAA/benzodiazepine neurotransmission.
    Journal of ethnopharmacology, 2013, May-20, Volume: 147, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Inhalation; Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Diazepam; Flunitrazepam; GABA-A Receptor Antagonists; Lavandula; Male; Mice; Motor Activity; Oils, Volatile; Picrotoxin; Piperazines; Plant Oils; Pyridines; Rats; Receptors, GABA-A; Serotonin Antagonists; Serotonin Receptor Agonists; Serotonin Syndrome; Synaptic Transmission

2013
GABA-induced uncoupling of GABA/benzodiazepine site interactions is mediated by increased GABAA receptor internalization and associated with a change in subunit composition.
    Neuroscience, 2014, Jan-17, Volume: 257

    Topics: Animals; Benzodiazepines; Binding Sites; Cells, Cultured; Cerebral Cortex; Embryo, Mammalian; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression Regulation; Neurons; Picrotoxin; Protein Binding; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors; Tritium

2014